[go: up one dir, main page]

MA56053A - Procédés de préparation d'acide 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylique - Google Patents

Procédés de préparation d'acide 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylique

Info

Publication number
MA56053A
MA56053A MA056053A MA56053A MA56053A MA 56053 A MA56053 A MA 56053A MA 056053 A MA056053 A MA 056053A MA 56053 A MA56053 A MA 56053A MA 56053 A MA56053 A MA 56053A
Authority
MA
Morocco
Prior art keywords
pyrazole
pyridin
bromo
chloro
preparing
Prior art date
Application number
MA056053A
Other languages
English (en)
Inventor
Yanchun Cao
Xin Liu
Jianhua Mao
Zhijian Xu
Original Assignee
Fmc Agro Singapore Pte Ltd
Fmc Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fmc Agro Singapore Pte Ltd, Fmc Corp filed Critical Fmc Agro Singapore Pte Ltd
Publication of MA56053A publication Critical patent/MA56053A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16Halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MA056053A 2019-10-18 2020-10-16 Procédés de préparation d'acide 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylique MA56053A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962916840P 2019-10-18 2019-10-18
US202062982248P 2020-02-27 2020-02-27

Publications (1)

Publication Number Publication Date
MA56053A true MA56053A (fr) 2022-04-20

Family

ID=73198483

Family Applications (2)

Application Number Title Priority Date Filing Date
MA056055A MA56055A (fr) 2019-10-18 2020-10-16 Procédés de préparation d'acide 5-bromo-2-(3chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylique
MA056053A MA56053A (fr) 2019-10-18 2020-10-16 Procédés de préparation d'acide 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylique

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MA056055A MA56055A (fr) 2019-10-18 2020-10-16 Procédés de préparation d'acide 5-bromo-2-(3chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylique

Country Status (16)

Country Link
US (2) US20220396560A1 (fr)
EP (5) EP4219455B1 (fr)
JP (2) JP2022552273A (fr)
KR (2) KR20220084347A (fr)
CN (3) CN114650987B (fr)
AU (2) AU2020366037A1 (fr)
BR (2) BR112022007215A2 (fr)
HU (4) HUE062237T2 (fr)
IL (5) IL298694B2 (fr)
MA (2) MA56055A (fr)
MX (2) MX2022004631A (fr)
PL (4) PL4043451T3 (fr)
TW (3) TWI875840B (fr)
UY (1) UY38925A (fr)
WO (2) WO2021076835A1 (fr)
ZA (2) ZA202204277B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2020366425A1 (en) * 2019-10-18 2022-04-21 Fmc Corporation Methods for the preparation of 5-Bromo-2-(3-chloro-pyridin-2-yl)-2H-pyrazole-3-carboxylic acid
KR20220084347A (ko) * 2019-10-18 2022-06-21 에프엠씨 코포레이션 5-브로모-2-(3-클로로-피리딘-2-일)-2h-피라졸-3-카복실산의 제조 방법
CN115557931B (zh) * 2022-10-20 2024-05-14 浙江新安化工集团股份有限公司 一种3-溴-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酸的合成方法
CN117024374A (zh) * 2023-08-08 2023-11-10 安庆百谊生物科技有限公司 一种3-甲基-1,2,4-噻二唑-5-碳酰肼或其盐的合成方法

Family Cites Families (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2060816C3 (de) * 1970-12-10 1980-09-04 Merck Patent Gmbh, 6100 Darmstadt 4-Phenylpiperidinderivate Verfahren zu ihrer Herstellung und pharmazeutische Zubereitungen enthaltend diese Verbindungen
DE3011084A1 (de) * 1980-03-22 1981-10-01 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von substituierten n-azolylmethyl-halogenacetaniliden
JPH07110867B2 (ja) * 1987-04-04 1995-11-29 株式会社トクヤマ ハロゲン化複素環式化合物の製造方法
TWI325302B (en) 2001-08-13 2010-06-01 Du Pont Benzoxazinone compounds
KR100921594B1 (ko) * 2003-01-28 2009-10-14 이 아이 듀폰 디 네모아 앤드 캄파니 시아노 안트라닐아미드 살충제
PE20060285A1 (es) * 2004-03-30 2006-05-08 Aventis Pharma Inc Piridonas sustituidas como inhibidores de pol(adp-ribosa)-polimerasa (parp)
MY140912A (en) * 2004-07-26 2010-01-29 Du Pont Mixtures of anthranilamide invertebrate pest control agents
US7087755B1 (en) * 2004-11-12 2006-08-08 Frontier Scientific, Inc. Substituted pyridines
WO2008072079A2 (fr) * 2006-12-13 2008-06-19 Pfizer Products Inc. Procédés de préparation de 3-(4-(2,4-difluorobenzyloxy)-3-bromo-6-méthyl-2-oxopyridin-1(2h)-yl)-n,4-diméthylbenzamide
CL2008000979A1 (es) * 2007-04-11 2008-10-17 Sumitomo Chemical Co Proceso para producir un compuesto derivado de 2-piridin-2-il-2h-pirazol-3-fenilamida; compuestos intermediarios; el compuesto en si; composicion plaguicida que contiene a dicho compuesto; uso de dicho compuesto como plaguicida; y metodo para control
JP2008280340A (ja) * 2007-04-12 2008-11-20 Sumitomo Chemical Co Ltd ヒドラジド化合物及びそれを含有する有害節足動物防除剤
JP2009023991A (ja) * 2007-06-20 2009-02-05 Ishihara Sangyo Kaisha Ltd アントラニルアミド系化合物の製造方法
WO2009022600A1 (fr) * 2007-08-14 2009-02-19 Sumitomo Chemical Company, Limited Procédé de fabrication d'un composé hydrazine, intermédiaire pour la production d'un composé hydrazine, et procédé de fabrication de l'intermédiaire
TW201245155A (en) * 2010-09-01 2012-11-16 Du Pont Fungicidal pyrazoles
CN102651485B (zh) * 2011-02-28 2016-03-30 丰田自动车株式会社 可充镁电池、电解液在可充镁电池中的应用、以及用于可充镁电池的电解液
US9475812B2 (en) * 2011-06-04 2016-10-25 Xuanzhu Pharma Co., Ltd. Pyridonaphthyridine type dual PI3K and mTOR inhibitor and its preparation and use
WO2013105100A1 (fr) * 2012-01-09 2013-07-18 Symed Labs Limited Procédés de préparation de 5-chloro-n-( {(5s)-2-oxo-3-[4-(3-oxo-4-morpholinyl)phényl]-1,3-oxazolidin-5-yl méthyl)-2-thiophène-carboxamide et de ses intermédiaires
DK2892891T3 (da) * 2012-09-07 2019-10-14 Boehringer Ingelheim Int Alkoxypyrazoler som opløselige guanylatcyklaseaktivatorer
CN105669643A (zh) * 2013-12-05 2016-06-15 江西天人生态股份有限公司 一类基于鱼泥丁受体的邻甲酰氨基苯甲酰胺衍生物及其制备方法和用途
JP6673850B2 (ja) * 2014-04-14 2020-03-25 グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング ヘテロアリール置換されたヘテロシクリルスルホン
TW201726128A (zh) * 2015-10-08 2017-08-01 歌林達有限公司 經吡唑基取代之四氫哌喃基碸
BR112018007673A2 (pt) * 2015-10-16 2018-11-06 Univ Rice William M ?análogos de epotilona, métodos de síntese, métodos de tratamento e conjugados de fármaco dos mesmos?
JP7128189B2 (ja) * 2016-12-21 2022-08-30 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 2-ピリジルエチルカルボキサミド誘導体を調製する方法
GB201721969D0 (en) * 2017-12-27 2018-02-07 Bp Oil Int Methods for preparing fuel additives
CN111825653A (zh) * 2019-04-19 2020-10-27 安道麦马克西姆有限公司 取代吡唑类化合物的制备及其作为邻氨基苯甲酰胺前体的用途
KR20220084347A (ko) 2019-10-18 2022-06-21 에프엠씨 코포레이션 5-브로모-2-(3-클로로-피리딘-2-일)-2h-피라졸-3-카복실산의 제조 방법

Also Published As

Publication number Publication date
IL299818B1 (en) 2024-10-01
CN114641471A (zh) 2022-06-17
IL292090B2 (en) 2023-06-01
TW202128631A (zh) 2021-08-01
HUE066520T2 (hu) 2024-08-28
TWI875840B (zh) 2025-03-11
IL291939A (en) 2022-06-01
IL291939B2 (en) 2023-04-01
US20220396560A1 (en) 2022-12-15
AU2020366212A1 (en) 2022-04-21
MX2022004631A (es) 2022-05-24
IL298694B1 (en) 2025-01-01
WO2021076835A8 (fr) 2021-11-04
BR112022007102A2 (pt) 2022-07-05
MA56055A (fr) 2022-04-06
TW202517625A (zh) 2025-05-01
BR112022007215A2 (pt) 2022-07-05
TW202116748A (zh) 2021-05-01
ZA202204278B (en) 2024-08-28
EP4219455B1 (fr) 2024-12-11
IL294551B1 (en) 2023-01-01
EP4253380A3 (fr) 2023-11-15
IL292090A (en) 2022-06-01
IL298694A (en) 2023-02-01
IL294551A (en) 2022-09-01
CN114641471B (zh) 2025-05-23
UY38925A (es) 2021-05-31
EP4253380A2 (fr) 2023-10-04
JP7667144B2 (ja) 2025-04-22
HUE062237T2 (hu) 2023-10-28
AU2020366037A1 (en) 2022-04-21
EP4043451B1 (fr) 2024-02-28
PL4219455T3 (pl) 2025-04-14
IL298694B2 (en) 2025-05-01
EP4219455A1 (fr) 2023-08-02
EP3976589A1 (fr) 2022-04-06
CN114650987B (zh) 2024-09-06
IL299818A (en) 2023-03-01
PL3976589T3 (pl) 2023-07-31
KR20220084347A (ko) 2022-06-21
IL299818B2 (en) 2025-02-01
HUE062047T2 (hu) 2023-09-28
IL291939B (en) 2022-12-01
CN119039270A (zh) 2024-11-29
MX2022004627A (es) 2022-05-26
WO2021076839A1 (fr) 2021-04-22
EP3976589B1 (fr) 2023-04-12
JP2022552272A (ja) 2022-12-15
EP3976591A1 (fr) 2022-04-06
HUE070680T2 (hu) 2025-06-28
ZA202204277B (en) 2024-08-28
PL3976591T3 (pl) 2023-07-31
JP2022552273A (ja) 2022-12-15
CN114650987A (zh) 2022-06-21
EP4043451A1 (fr) 2022-08-17
WO2021076835A1 (fr) 2021-04-22
TWI884994B (zh) 2025-06-01
PL4043451T3 (pl) 2024-06-10
KR20220086612A (ko) 2022-06-23
IL294551B2 (en) 2023-05-01
EP3976591B1 (fr) 2023-04-19
US20220259178A1 (en) 2022-08-18

Similar Documents

Publication Publication Date Title
MA56053A (fr) Procédés de préparation d'acide 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylique
EP3824096A4 (fr) Nouveaux anticorps et leurs procédés de préparation et d'utilisation
EP3840673A4 (fr) Système de guidance pour correction d'hallux valgus
EP3622080C0 (fr) Procédés améliorés pour la production d'isobutène à partir d'acide 3-méthylcrotonique
EP3402787A4 (fr) Procédés de préparation d'acide 2,5-furandicarboxylique et des intermédiaires et dérivés correspondants
EP3353278A4 (fr) Préparation d'échantillons pour des types d'échantillons compliqués
EP3529232A4 (fr) Dérivés d'acide sulfamique et procédés pour leur préparation
EP3390415A4 (fr) (r)- et (s)-1-(3-(3-n,n-diméthylaminocarbonyl)phénoxyl-4-nitrophényl)-1-éthyl-n,n'-bis(éthylène)phosphoramidate, compositions et procédés pour leur utilisation et préparation
EP3512947A4 (fr) Procédés de préparation d'échantillon d'acide nucléique
EP3775210C0 (fr) Molécules d'acide nucléique pour pseudouridylation
MA52204A (fr) Procédés de préparation de compositions protéiques stables
EP3969457A4 (fr) Procédés de préparation d'indoles macrocycliques
MA45183A (fr) Procédés de préparation d'oligomères morpholino de phosphorodiamidate
EP3784031A4 (fr) Procédés de génotypage d'embryons haploïdes
EP3564218A4 (fr) Procédé de préparation d'acide 1,4,7,10-tétraazacyclododécane-1,4,7,10-tétraacétique
MA56054A (fr) Procédés de préparation d'acide 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylique
MA56052A (fr) Procédés de préparation d'acide 5-bromo-2-(3-chloro-pyridin-2-yl)-2 h-pyrazole-3-carboxylique
IL292091A (en) Method for preparing 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyralose-3-carboxylic acid
EP3902792A4 (fr) Procédé de préparation d'anthranilamides
EP3781544C0 (fr) Procédé de préparation d'iloprost
EP3710595C0 (fr) Compositions et procédés pour détecter l'acide nucléique de c1orf43
IL304456A (en) Methods for preparing 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazol-3-carboxylic acid
EP3797104A4 (fr) Nouveaux procédés de préparation d'un dérivé de diaminopyrimidine ou d'un sel d'addition d'acide de celui-ci
IL288585A (en) Alternative process for the preparation of 4-phenyl-5-alkoxycarbonyl-2-thiazol-2-yl-1,4-dihydropyrimidin-6-yl]methyl]-3-oxo-5,6,8,8a-tetrahydro-1h-imidazo[1,5-a]pyrazin-2-yl]-carboxylic acid
MA45362A (fr) Procédés de préparation d'oligomères morpholino de phosphorodiamidate