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ZA200806871B - Dihydrodiazepines useful as inhibitors of protein kinases - Google Patents

Dihydrodiazepines useful as inhibitors of protein kinases

Info

Publication number
ZA200806871B
ZA200806871B ZA200806871A ZA200806871A ZA200806871B ZA 200806871 B ZA200806871 B ZA 200806871B ZA 200806871 A ZA200806871 A ZA 200806871A ZA 200806871 A ZA200806871 A ZA 200806871A ZA 200806871 B ZA200806871 B ZA 200806871B
Authority
ZA
South Africa
Prior art keywords
dihydrodiazepines
inhibitors
useful
protein kinases
kinases
Prior art date
Application number
ZA200806871A
Other languages
English (en)
Inventor
Damien-Charrier Jean
Kay David
Knegtel Ronald
Twin Heather
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of ZA200806871B publication Critical patent/ZA200806871B/xx

Links

ZA200806871A 2006-02-14 2007-02-13 Dihydrodiazepines useful as inhibitors of protein kinases ZA200806871B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US77299206P 2006-02-14 2006-02-14

Publications (1)

Publication Number Publication Date
ZA200806871B true ZA200806871B (en) 2009-10-28

Family

ID=40631373

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200806871A ZA200806871B (en) 2006-02-14 2007-02-13 Dihydrodiazepines useful as inhibitors of protein kinases

Country Status (3)

Country Link
CN (1) CN101420955B (es)
ES (1) ES2351367T3 (es)
ZA (1) ZA200806871B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2013505927A (ja) * 2009-09-25 2013-02-21 バーテックス ファーマシューティカルズ インコーポレイテッド プロテインキナーゼ阻害剤として有用なピリミジン誘導体の調製方法
CA2918910A1 (en) 2013-07-25 2015-01-29 Dana-Farber Cancer Institute, Inc. Inhibitors of transcription factors and uses thereof
US10793571B2 (en) 2014-01-31 2020-10-06 Dana-Farber Cancer Institute, Inc. Uses of diazepane derivatives
CN105940005A (zh) * 2014-01-31 2016-09-14 达纳-法伯癌症研究所股份有限公司 二氮杂环庚烷衍生物及其用途
CN106029653A (zh) 2014-01-31 2016-10-12 达纳-法伯癌症研究所股份有限公司 二氨基嘧啶苯砜衍生物及其用途
MX2017001757A (es) 2014-08-08 2017-05-30 Dana Farber Cancer Inst Inc Derivados de dihidropteridinona y sus usos.
MX2017001756A (es) 2014-08-08 2017-05-30 Dana Farber Cancer Inst Inc Derivados de diazepano y sus usos.
US10702527B2 (en) 2015-06-12 2020-07-07 Dana-Farber Cancer Institute, Inc. Combination therapy of transcription inhibitors and kinase inhibitors
HK1256417A1 (zh) 2015-09-11 2019-09-20 达纳-法伯癌症研究所股份有限公司 氰基噻吩並三唑並二氮雜環庚三烯及其用途
CR20180199A (es) 2015-09-11 2018-05-25 Dana Farber Cancer Inst Inc Acetamida tienotriazolodiazepinas y usos de las mismas
RU2742035C2 (ru) 2015-11-25 2021-02-01 Дана-Фарбер Кэнсер Инститьют, Инк. Бивалентные ингибиторы бромодоменов и пути их применения
WO2017191304A1 (en) * 2016-05-06 2017-11-09 Laboratorios Del Dr. Esteve, S.A. Tetrahydropyrimidodiazepine and tetrahydropyridodiazepine compounds for treating pain and pain related conditions

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3880855A (en) * 1973-04-16 1975-04-29 Bristol Myers Co 5,6-DIHYDRO-11-H-pyrimido{8 4,5-b{9 {8 1,4{9 benzodiazepines

Also Published As

Publication number Publication date
CN101420955A (zh) 2009-04-29
CN101420955B (zh) 2013-07-17
ES2351367T3 (es) 2011-02-03

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