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ZA200806871B - Dihydrodiazepines useful as inhibitors of protein kinases - Google Patents

Dihydrodiazepines useful as inhibitors of protein kinases

Info

Publication number
ZA200806871B
ZA200806871B ZA200806871A ZA200806871A ZA200806871B ZA 200806871 B ZA200806871 B ZA 200806871B ZA 200806871 A ZA200806871 A ZA 200806871A ZA 200806871 A ZA200806871 A ZA 200806871A ZA 200806871 B ZA200806871 B ZA 200806871B
Authority
ZA
South Africa
Prior art keywords
dihydrodiazepines
inhibitors
useful
protein kinases
kinases
Prior art date
Application number
ZA200806871A
Other languages
English (en)
Inventor
Damien-Charrier Jean
Kay David
Knegtel Ronald
Twin Heather
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of ZA200806871B publication Critical patent/ZA200806871B/xx

Links

ZA200806871A 2006-02-14 2007-02-13 Dihydrodiazepines useful as inhibitors of protein kinases ZA200806871B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US77299206P 2006-02-14 2006-02-14

Publications (1)

Publication Number Publication Date
ZA200806871B true ZA200806871B (en) 2009-10-28

Family

ID=40631373

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200806871A ZA200806871B (en) 2006-02-14 2007-02-13 Dihydrodiazepines useful as inhibitors of protein kinases

Country Status (3)

Country Link
CN (1) CN101420955B (xx)
ES (1) ES2351367T3 (xx)
ZA (1) ZA200806871B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ599356A (en) * 2009-09-25 2013-08-30 Vertex Pharma Methods for preparing pyrimidine derivatives useful as protein kinase inhibitors
KR20160034379A (ko) 2013-07-25 2016-03-29 다나-파버 캔서 인스티튜트 인크. 전사 인자의 억제제 및 그의 용도
KR20160111036A (ko) * 2014-01-31 2016-09-23 다나-파버 캔서 인스티튜트 인크. 디아제판 유도체 및 그의 용도
US10793571B2 (en) 2014-01-31 2020-10-06 Dana-Farber Cancer Institute, Inc. Uses of diazepane derivatives
US10150756B2 (en) 2014-01-31 2018-12-11 Dana-Farber Cancer Institute, Inc. Diaminopyrimidine benzenesulfone derivatives and uses thereof
RU2017104897A (ru) 2014-08-08 2018-09-10 Дана-Фарбер Кэнсер Инститьют, Инк. Производные диазепана и их применения
EP3177147A4 (en) 2014-08-08 2018-01-24 Dana-Farber Cancer Institute, Inc. Dihydropteridinone derivatives and uses thereof
CA2986441A1 (en) 2015-06-12 2016-12-15 Dana-Farber Cancer Institute, Inc. Combination therapy of transcription inhibitors and kinase inhibitors
CN108472300A (zh) 2015-09-11 2018-08-31 达纳-法伯癌症研究所股份有限公司 氰基噻吩并三唑并二氮杂环庚三烯及其用途
KR20180051576A (ko) 2015-09-11 2018-05-16 다나-파버 캔서 인스티튜트 인크. 아세트아미드 티에노트리아졸로디아제핀 및 그의 용도
PE20181298A1 (es) 2015-11-25 2018-08-07 Dana Farber Cancer Inst Inc Inhibidores de bromodominio bivalentes y usos de los mismos
ES2789676T3 (es) * 2016-05-06 2020-10-26 Steve Pharmaceuticals S A Compuestos de tetrahidropirimidodiazepina y tetrahidropiridodiazepina para tratar el dolor y afecciones relacionadas con el dolor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3880855A (en) * 1973-04-16 1975-04-29 Bristol Myers Co 5,6-DIHYDRO-11-H-pyrimido{8 4,5-b{9 {8 1,4{9 benzodiazepines

Also Published As

Publication number Publication date
CN101420955B (zh) 2013-07-17
CN101420955A (zh) 2009-04-29
ES2351367T3 (es) 2011-02-03

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