ZA200806139B - Tricyclic N-heteroaryl-carboxamide derivatives containing a benzimidazole unit, method for preparing same and their therapeutic use - Google Patents

Tricyclic N-heteroaryl-carboxamide derivatives containing a benzimidazole unit, method for preparing same and their therapeutic use

Info

Publication number: ZA200806139B
Authority: ZA; South Africa
Prior art keywords: tricyclic; heteroaryl; therapeutic use; derivatives containing; preparing same
Prior art date: 2006-02-03

Application number

ZA200806139A

Other languages

English (en)

Inventor

Laurent Dubois

Yannick Evanno

Luc Even

Catherine Gille

Andre Malanda

David Machnik

Nathalie Rakotoarisoa

Original Assignee

Sanofi Aventis

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-02-03

Filing date

2007-02-01

Publication date

2010-05-26

2007-02-01 Application filed by Sanofi Aventis filed Critical Sanofi Aventis

2010-05-26 Publication of ZA200806139B publication Critical patent/ZA200806139B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4188—1,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
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- A61P11/08—Bronchodilators
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- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
- A61P31/22—Antivirals for DNA viruses for herpes viruses
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Diabetes (AREA)
Pain & Pain Management (AREA)
Reproductive Health (AREA)
Endocrinology (AREA)
Dermatology (AREA)
Virology (AREA)
Hematology (AREA)
Urology & Nephrology (AREA)
Pulmonology (AREA)
Gynecology & Obstetrics (AREA)
Psychiatry (AREA)
Communicable Diseases (AREA)
Ophthalmology & Optometry (AREA)
Hospice & Palliative Care (AREA)
Rheumatology (AREA)
Obesity (AREA)
Pregnancy & Childbirth (AREA)
Oncology (AREA)
Molecular Biology (AREA)
Biotechnology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

ZA200806139A 2006-02-03 2007-02-01 Tricyclic N-heteroaryl-carboxamide derivatives containing a benzimidazole unit, method for preparing same and their therapeutic use ZA200806139B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0601007A FR2897061B1 (fr)	2006-02-03	2006-02-03	Derives de n-heteroaryl-carboxamides tricycliques contenant un motif benzimidazole, leur preparation et leur application en therapeutique.

Publications (1)

Publication Number	Publication Date
ZA200806139B true ZA200806139B (en)	2010-05-26

Family

ID=36954977

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200806139A ZA200806139B (en)	2006-02-03	2007-02-01	Tricyclic N-heteroaryl-carboxamide derivatives containing a benzimidazole unit, method for preparing same and their therapeutic use

Country Status (32)

Country	Link
US (2)	US8143248B2 (xx)
EP (1)	EP1987010B1 (xx)
JP (1)	JP5136938B2 (xx)
KR (1)	KR20080090495A (xx)
CN (1)	CN101379041B (xx)
AR (1)	AR059279A1 (xx)
AT (1)	ATE463484T1 (xx)
AU (1)	AU2007211399B2 (xx)
BR (1)	BRPI0710480A2 (xx)
CA (1)	CA2637333C (xx)
CY (1)	CY1110168T1 (xx)
DE (1)	DE602007005779D1 (xx)
DK (1)	DK1987010T3 (xx)
DO (1)	DOP2007000022A (xx)
EA (1)	EA014450B1 (xx)
ES (1)	ES2344087T3 (xx)
FR (1)	FR2897061B1 (xx)
HR (1)	HRP20100327T1 (xx)
IL (1)	IL192648A (xx)
JO (1)	JO2602B1 (xx)
MA (1)	MA30229B1 (xx)
NO (1)	NO20083520L (xx)
NZ (1)	NZ569669A (xx)
PE (1)	PE20071325A1 (xx)
PL (1)	PL1987010T3 (xx)
PT (1)	PT1987010E (xx)
RS (1)	RS51366B (xx)
SI (1)	SI1987010T1 (xx)
TW (1)	TWI401256B (xx)
UY (1)	UY30130A1 (xx)
WO (1)	WO2007088277A1 (xx)
ZA (1)	ZA200806139B (xx)

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FR2888848B1 (fr) *	2005-07-22	2007-09-28	Sanofi Aventis Sa	Derives de n-(arylalkyl)-1h-pyrrrolopyridine-2-carboxamides, leur preparation et leur application en therapeutique
FR2911604B1 (fr) *	2007-01-19	2009-04-17	Sanofi Aventis Sa	Derives de n-(heteroaryl-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique
FR2911605B1 (fr) *	2007-01-19	2009-04-17	Sanofi Aventis Sa	Derives de pyrrolopyridine-2-carbowamides, leur preparation et leur application en therapeutique
FR2919610B1 (fr) *	2007-08-02	2009-10-16	Sanofi Aventis Sa	Derives de n-heteroaryl-carboxamides tricycliques,leur preparation et leur application en therapeutique
FR2926555B1 (fr) *	2008-01-22	2010-02-19	Sanofi Aventis	Derives bicycliques de carboxamides azabicycliques, leur preparation et leur application en therapeutique
FR2926556B1 (fr) *	2008-01-22	2010-02-19	Sanofi Aventis	Derives de carboxamides n-azabicycliques, leur preparation et leur application en therapeutique
FR2926554B1 (fr)	2008-01-22	2010-03-12	Sanofi Aventis	Derives de carboxamides azabicycliques, leur preparation et leur application en therapeutique
FR2926553B1 (fr) *	2008-01-23	2010-02-19	Sanofi Aventis	Derives d'indole-2-carboxamides et d'azaindole-2- carboxamides substitues par un groupe silanyle, leur preparation et leur application en therapeutique
WO2009108551A2 (en) *	2008-02-25	2009-09-03	H. Lundbeck A/S	Heteroaryl amide analogues
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AU2009308687A1 (en) *	2008-11-03	2010-05-06	Chemocentryx, Inc.	Compounds for the treatment of osteoporosis and cancers
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MX2012002827A (es) *	2009-09-11	2012-04-10	Sunovion Pharmaceuticals Inc	Agonistas inversos y antagonistas de histamina h3 y metodos para usar los mismos.
EA201291114A1 (ru) *	2010-04-27	2013-04-30	Астеллас Фарма Инк.	ПРОИЗВОДНЫЕ ИМИДАЗО[1,2-a]ПИРИДИНА
NZ629189A (en) *	2012-03-16	2016-08-26	Vitae Pharmaceuticals Inc	Liver x receptor modulators
KR102069912B1 (ko)	2012-03-16	2020-01-23	비타이 파마슈티컬즈, 엘엘씨	간 x 수용체 조절제
ES2904267T3 (es) *	2012-06-18	2022-04-04	Dart Neuroscience Llc	Composiciones farmacéuticas de derivados de 6H-pirido[3.2-e][1.2.4]triazolo[1,5-c]pirimidina-5-ona y[1.2.4]triazolo[1,5-c]pteridina-5(6H)-ona como inhibidores de PDE1 para el tratamiento, por ejemplo, de trastornosneurológicos
MX381819B (es)	2014-08-04	2025-03-13	Nuevolution As	Derivados de heterociclico opcionalmente condensados de pirimidina útiles para el tratamiento de enfermedades inflamatorias, metabólicas oncológicas y autoinmunitarias.
EP3313846B1 (en) *	2015-06-25	2020-05-06	Promega Corporation	Thienopyrrole compounds and uses thereof as inhibitors of oplophorus-derived luciferases
AU2017336074A1 (en) *	2016-09-30	2019-03-28	Epizyme, Inc.	Substituted fused bi- or tri- heterocyclic compounds as ehmt2 inhibitors
US10815247B2 (en)	2016-12-28	2020-10-27	Promega Corporation	Functionalized NANOLUC inhibitors
CN110621316B (zh)	2017-04-21	2024-01-26	Epizyme股份有限公司	用ehmt2抑制剂进行的组合疗法
CN109761974B (zh) *	2019-01-21	2021-05-14	河南大学	1,2,3,4-四氢-9H-吡啶并[3,4-b]吲哚类TRPV1拮抗剂及其应用
MX2022007265A (es)	2019-12-20	2022-09-09	Nuevolution As	Compuestos activos frente a receptores nucleares.
JP7746259B2 (ja)	2019-12-20	2025-09-30	ヌエヴォリューション・アクティーゼルスカブ	核内受容体に対して活性の化合物
EP4126875A1 (en)	2020-03-31	2023-02-08	Nuevolution A/S	Compounds active towards nuclear receptors
WO2021198955A1 (en)	2020-03-31	2021-10-07	Nuevolution A/S	Compounds active towards nuclear receptors
CN114276354B (zh) *	2022-01-07	2023-06-02	中山大学	1-氨基苯并[4,5]咪唑并[1,2-a]吡嗪-3-甲酰胺类化合物及其制备和应用
CN114539265B (zh) *	2022-03-02	2023-07-21	中山大学	靶向a2a的苯并咪唑并吡嗪-3-甲酰胺及其肿瘤免疫功能

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2006
- 2006-02-03 FR FR0601007A patent/FR2897061B1/fr not_active Expired - Fee Related
2007
- 2007-01-30 PE PE2007000106A patent/PE20071325A1/es not_active Application Discontinuation
- 2007-01-31 TW TW096103550A patent/TWI401256B/zh not_active IP Right Cessation
- 2007-02-01 DO DO2007000022A patent/DOP2007000022A/es unknown
- 2007-02-01 CA CA2637333A patent/CA2637333C/fr not_active Expired - Fee Related
- 2007-02-01 PT PT07730900T patent/PT1987010E/pt unknown
- 2007-02-01 BR BRPI0710480-4A patent/BRPI0710480A2/pt not_active IP Right Cessation
- 2007-02-01 AR ARP070100426A patent/AR059279A1/es not_active Application Discontinuation
- 2007-02-01 JP JP2008552848A patent/JP5136938B2/ja not_active Expired - Fee Related
- 2007-02-01 JO JO200729A patent/JO2602B1/en active
- 2007-02-01 EP EP07730900A patent/EP1987010B1/fr active Active
- 2007-02-01 NZ NZ569669A patent/NZ569669A/en not_active IP Right Cessation
- 2007-02-01 AU AU2007211399A patent/AU2007211399B2/en not_active Ceased
- 2007-02-01 RS RSP-2010/0301A patent/RS51366B/sr unknown
- 2007-02-01 HR HR20100327T patent/HRP20100327T1/hr unknown
- 2007-02-01 EA EA200870226A patent/EA014450B1/ru not_active IP Right Cessation
- 2007-02-01 SI SI200730254T patent/SI1987010T1/sl unknown
- 2007-02-01 PL PL07730900T patent/PL1987010T3/pl unknown
- 2007-02-01 ZA ZA200806139A patent/ZA200806139B/xx unknown
- 2007-02-01 ES ES07730900T patent/ES2344087T3/es active Active
- 2007-02-01 KR KR1020087019041A patent/KR20080090495A/ko not_active Ceased
- 2007-02-01 WO PCT/FR2007/000183 patent/WO2007088277A1/fr not_active Ceased
- 2007-02-01 DK DK07730900.3T patent/DK1987010T3/da active
- 2007-02-01 DE DE602007005779T patent/DE602007005779D1/de active Active
- 2007-02-01 CN CN2007800042835A patent/CN101379041B/zh not_active Expired - Fee Related
- 2007-02-01 AT AT07730900T patent/ATE463484T1/de active
- 2007-02-02 UY UY30130A patent/UY30130A1/es not_active Application Discontinuation
2008
- 2008-07-06 IL IL192648A patent/IL192648A/en not_active IP Right Cessation
- 2008-08-01 US US12/184,437 patent/US8143248B2/en not_active Expired - Fee Related
- 2008-08-13 NO NO20083520A patent/NO20083520L/no not_active Application Discontinuation
- 2008-08-26 MA MA31193A patent/MA30229B1/fr unknown
2010
- 2010-07-01 CY CY20101100609T patent/CY1110168T1/el unknown
2012
- 2012-01-24 US US13/357,015 patent/US8288376B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
JP2009525313A (ja)	2009-07-09
EP1987010B1 (fr)	2010-04-07
JP5136938B2 (ja)	2013-02-06
IL192648A (en)	2012-06-28
HRP20100327T1 (hr)	2010-08-31
EP1987010A1 (fr)	2008-11-05
HK1129670A1 (en)	2009-12-04
AU2007211399B2 (en)	2012-09-20
DOP2007000022A (es)	2007-09-15
US8143248B2 (en)	2012-03-27
NZ569669A (en)	2011-05-27
DE602007005779D1 (de)	2010-05-20
PE20071325A1 (es)	2008-02-21
CY1110168T1 (el)	2015-01-14
FR2897061A1 (fr)	2007-08-10
BRPI0710480A2 (pt)	2012-08-14
ATE463484T1 (de)	2010-04-15
CA2637333C (fr)	2015-12-29
IL192648A0 (en)	2009-02-11
NO20083520L (no)	2008-09-11
ES2344087T3 (es)	2010-08-17
AU2007211399A1 (en)	2007-08-09
TWI401256B (zh)	2013-07-11
CN101379041A (zh)	2009-03-04
US8288376B2 (en)	2012-10-16
FR2897061B1 (fr)	2010-09-03
MA30229B1 (fr)	2009-02-02
TW200738726A (en)	2007-10-16
CA2637333A1 (fr)	2007-08-09
KR20080090495A (ko)	2008-10-08
AR059279A1 (es)	2008-03-19
DK1987010T3 (da)	2010-08-02
CN101379041B (zh)	2012-08-29
EA200870226A1 (ru)	2009-02-27
RS51366B (sr)	2011-02-28
SI1987010T1 (sl)	2010-07-30
US20120122852A1 (en)	2012-05-17
PL1987010T3 (pl)	2010-09-30
PT1987010E (pt)	2010-06-25
JO2602B1 (en)	2011-11-01
UY30130A1 (es)	2007-09-28
WO2007088277A1 (fr)	2007-08-09
EA014450B1 (ru)	2010-12-30
US20090042873A1 (en)	2009-02-12

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