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ZA200701820B - Substituted phenylaminothiazoles and use thereof - Google Patents

Substituted phenylaminothiazoles and use thereof

Info

Publication number
ZA200701820B
ZA200701820B ZA200701820A ZA200701820A ZA200701820B ZA 200701820 B ZA200701820 B ZA 200701820B ZA 200701820 A ZA200701820 A ZA 200701820A ZA 200701820 A ZA200701820 A ZA 200701820A ZA 200701820 B ZA200701820 B ZA 200701820B
Authority
ZA
South Africa
Prior art keywords
phenylaminothiazoles
substituted
substituted phenylaminothiazoles
Prior art date
Application number
ZA200701820A
Other languages
English (en)
Inventor
Ergueden Jens-Kerim
Karig Gunter
Rosentreter Ulrich
Albrecht Barbara
Henninger Kerstin
Huetter Joachim
Diedrichs Nicole
Nell Peter
Arndt Sabine
Huebsch Walter
Knorr Andreas
Schlemmer Karl-Heinz
Brohm Dirk
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of ZA200701820B publication Critical patent/ZA200701820B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA200701820A 2004-09-03 2007-03-01 Substituted phenylaminothiazoles and use thereof ZA200701820B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004042607A DE102004042607A1 (de) 2004-09-03 2004-09-03 Substituierte Phenylaminothiazole und ihre Verwendung

Publications (1)

Publication Number Publication Date
ZA200701820B true ZA200701820B (en) 2008-08-27

Family

ID=35852458

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200701820A ZA200701820B (en) 2004-09-03 2007-03-01 Substituted phenylaminothiazoles and use thereof

Country Status (24)

Country Link
US (1) US8691850B2 (xx)
EP (1) EP1812430B1 (xx)
JP (1) JP4999691B2 (xx)
KR (1) KR20070057235A (xx)
CN (1) CN101056875A (xx)
AR (1) AR050551A1 (xx)
AT (1) ATE428710T1 (xx)
AU (1) AU2005281941A1 (xx)
BR (1) BRPI0514833A (xx)
CA (1) CA2578596C (xx)
DE (2) DE102004042607A1 (xx)
EC (1) ECSP077296A (xx)
ES (1) ES2324049T3 (xx)
GT (1) GT200500238A (xx)
IL (1) IL181670A0 (xx)
MA (1) MA28869B1 (xx)
MX (1) MX2007002470A (xx)
NO (1) NO20071343L (xx)
PE (1) PE20060589A1 (xx)
SV (1) SV2006002218A (xx)
TW (1) TW200621765A (xx)
UY (1) UY29099A1 (xx)
WO (1) WO2006027142A1 (xx)
ZA (1) ZA200701820B (xx)

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DE102006042143A1 (de) * 2006-09-08 2008-03-27 Bayer Healthcare Aktiengesellschaft Neue substituierte Bipyridin-Derivate und ihre Verwendung
DE102006044696A1 (de) 2006-09-22 2008-03-27 Bayer Healthcare Ag 3-Cyano-5-thiazaheteroaryl-dihydropyridine und ihre Verwendung
DE102006056740A1 (de) 2006-12-01 2008-06-05 Bayer Healthcare Ag Cyclisch substituierte 3,5-Dicyano-2-thiopyridine und ihre Verwendung
DE102006056739A1 (de) 2006-12-01 2008-06-05 Bayer Healthcare Ag Substituierte 4-Amino-3,5-dicyano-2-thiopyridine und ihre Verwendung
DE102007035367A1 (de) * 2007-07-27 2009-01-29 Bayer Healthcare Ag Substituierte Aryloxazole und ihre Verwendung
DE102007036076A1 (de) 2007-08-01 2009-02-05 Bayer Healthcare Aktiengesellschaft Dipeptoid-Produgs und ihre Verwendung
DE102007061764A1 (de) * 2007-12-20 2009-06-25 Bayer Healthcare Ag Anellierte Cyanopyridine und ihre Verwendung
DE102007061763A1 (de) * 2007-12-20 2009-06-25 Bayer Healthcare Ag Substituierte azabicyclische Verbindungen und ihre Verwendung
DE102008008838A1 (de) * 2008-02-13 2009-08-20 Bayer Healthcare Ag Cycloalkoxy-substituierte 4-Phenyl-3,5-dicyanopyridine und ihre Verwendung
DE102008013587A1 (de) * 2008-03-11 2009-09-17 Bayer Schering Pharma Aktiengesellschaft Heteroaryl-substituierte Dicyanopyridine und ihre Verwendung
EP2297104B1 (de) * 2008-05-29 2013-08-07 Bayer Intellectual Property GmbH 2-alkoxy-substituierte dicyanopyridine und ihre verwendung
DE102008062567A1 (de) 2008-12-16 2010-06-17 Bayer Schering Pharma Aktiengesellschaft Dipeptoid-Prodrugs und ihre Verwendung
DE102009006602A1 (de) * 2009-01-29 2010-08-05 Bayer Schering Pharma Aktiengesellschaft Alkylamino-substituierte Dicyanopyridine und deren Aminosäureester-Prodrugs
DE102009022894A1 (de) * 2009-05-27 2010-12-02 Bayer Schering Pharma Aktiengesellschaft Substituierte Piperidine
DE102010030688A1 (de) 2010-06-30 2012-01-05 Bayer Schering Pharma Aktiengesellschaft Substituierte Dicyanopyridine und ihre Verwendung
KR20220147691A (ko) 2013-08-09 2022-11-03 알데릭스, 인코포레이티드 인산염 수송을 억제하기 위한 화합물 및 방법
WO2018153897A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit hcn-kanal-hemmern
WO2018153899A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit stimulatoren und/oder aktivatoren der löslichen guanylatcyclase (sgc)
WO2018153898A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit mineralocorticoid-rezeptor-antagonisten
WO2018153895A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit einem inhibitor der neutralen endopeptidase und/oder einem angiotensin ii rezeptor-antagonisten
WO2018153900A1 (de) 2017-02-22 2018-08-30 Bayer Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit sglt-2-hemmern
JP7323913B2 (ja) * 2019-04-12 2023-08-09 国立大学法人 筑波大学 睡眠誘導剤である複素環化合物

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DE102007036076A1 (de) 2007-08-01 2009-02-05 Bayer Healthcare Aktiengesellschaft Dipeptoid-Produgs und ihre Verwendung
DE102008013587A1 (de) 2008-03-11 2009-09-17 Bayer Schering Pharma Aktiengesellschaft Heteroaryl-substituierte Dicyanopyridine und ihre Verwendung
DE102008062567A1 (de) 2008-12-16 2010-06-17 Bayer Schering Pharma Aktiengesellschaft Dipeptoid-Prodrugs und ihre Verwendung
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Also Published As

Publication number Publication date
ATE428710T1 (de) 2009-05-15
DE502005007106D1 (de) 2009-05-28
EP1812430A1 (de) 2007-08-01
JP2008511614A (ja) 2008-04-17
CN101056875A (zh) 2007-10-17
DE102004042607A1 (de) 2006-03-09
SV2006002218A (es) 2006-10-04
ES2324049T3 (es) 2009-07-29
JP4999691B2 (ja) 2012-08-15
EP1812430B1 (de) 2009-04-15
AU2005281941A1 (en) 2006-03-16
UY29099A1 (es) 2006-04-28
KR20070057235A (ko) 2007-06-04
GT200500238A (es) 2006-04-10
US20080269300A1 (en) 2008-10-30
MX2007002470A (es) 2009-02-12
US8691850B2 (en) 2014-04-08
IL181670A0 (en) 2007-07-04
CA2578596C (en) 2012-10-23
MA28869B1 (fr) 2007-09-03
AR050551A1 (es) 2006-11-01
BRPI0514833A (pt) 2008-06-24
TW200621765A (en) 2006-07-01
WO2006027142A1 (de) 2006-03-16
ECSP077296A (es) 2007-04-26
NO20071343L (no) 2007-05-30
CA2578596A1 (en) 2006-03-16
PE20060589A1 (es) 2006-08-12

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