YU30403A - 2-, 3-, 4- ili 5-supstituisani-n1-(benzensulfonil)indoli i njihova upotreba u terapiji - Google Patents
2-, 3-, 4- ili 5-supstituisani-n1-(benzensulfonil)indoli i njihova upotreba u terapijiInfo
- Publication number
- YU30403A YU30403A YU30403A YUP30403A YU30403A YU 30403 A YU30403 A YU 30403A YU 30403 A YU30403 A YU 30403A YU P30403 A YUP30403 A YU P30403A YU 30403 A YU30403 A YU 30403A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- benzensulfonyl
- substituted
- indoles
- therapy
- receptor
- Prior art date
Links
- 150000002475 indoles Chemical class 0.000 title 1
- 238000002560 therapeutic procedure Methods 0.000 title 1
- 108091005435 5-HT6 receptors Proteins 0.000 abstract 1
- -1 5-substituted-N1-(benzensulfonyl)indoles compounds Chemical class 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 208000015114 central nervous system disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- 108020003175 receptors Proteins 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0003810A SE0003810D0 (sv) | 2000-10-20 | 2000-10-20 | Novel compounds their use and preparations |
| US24311500P | 2000-10-25 | 2000-10-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| YU30403A true YU30403A (sh) | 2006-03-03 |
Family
ID=20281502
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YU30403A YU30403A (sh) | 2000-10-20 | 2001-10-19 | 2-, 3-, 4- ili 5-supstituisani-n1-(benzensulfonil)indoli i njihova upotreba u terapiji |
Country Status (5)
| Country | Link |
|---|---|
| JP (2) | JP4343527B2 (sv) |
| CN (2) | CN101298433A (sv) |
| SE (1) | SE0003810D0 (sv) |
| YU (1) | YU30403A (sv) |
| ZA (1) | ZA200301693B (sv) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007098418A1 (en) * | 2006-02-17 | 2007-08-30 | Memory Pharmaceuticals Corporation | Compounds having 5-ht6 receptor affinity |
| RU2470011C2 (ru) | 2007-05-31 | 2012-12-20 | Сепракор Инк. | Циклоалкиламины, содержащие в качестве заместителя фенил, как ингибиторы обратного захвата моноаминов |
| UA100192C2 (en) * | 2008-11-11 | 2012-11-26 | УАЙТ ЭлЭлСи | 1-(arylsulfonyl)-4-(piperazin-1-yl)-1h-benzimidazoles as 5-hydroxytryptamine-6 ligands |
| CN105367472B (zh) * | 2014-08-12 | 2020-04-21 | 广东东阳光药业有限公司 | 吲哚啉类衍生物及其在药物上的应用 |
| CN105367473B (zh) * | 2014-08-12 | 2020-02-11 | 广东东阳光药业有限公司 | 吲哚啉类衍生物及其在药物上的应用 |
| CN111362858B (zh) * | 2020-03-16 | 2021-05-11 | 东莞市东阳光新药研发有限公司 | 芳杂环类衍生物的盐及其用途 |
| CN111362859B (zh) * | 2020-03-16 | 2021-05-11 | 东莞市东阳光新药研发有限公司 | 芳杂环类衍生物的盐及其用途 |
| CN111233737B (zh) * | 2020-03-16 | 2021-05-11 | 东莞市东阳光新药研发有限公司 | 芳杂环类衍生物的盐及其用途 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6100291A (en) * | 1998-03-16 | 2000-08-08 | Allelix Biopharmaceuticals Inc. | Pyrrolidine-indole compounds having 5-HT6 affinity |
| US6133287A (en) * | 1998-03-24 | 2000-10-17 | Allelix Biopharmaceuticals Inc. | Piperidine-indole compounds having 5-HT6 affinity |
| US6251893B1 (en) * | 1998-06-15 | 2001-06-26 | Nps Allelix Corp. | Bicyclic piperidine and piperazine compounds having 5-HT6 receptor affinity |
| JP2002518331A (ja) * | 1998-06-19 | 2002-06-25 | イーライ・リリー・アンド・カンパニー | セロトニン再取り込みの阻害 |
-
2000
- 2000-10-20 SE SE0003810A patent/SE0003810D0/sv unknown
-
2001
- 2001-10-19 CN CNA2008100742241A patent/CN101298433A/zh active Pending
- 2001-10-19 YU YU30403A patent/YU30403A/sh unknown
- 2001-10-19 CN CNB018174078A patent/CN100378074C/zh not_active Expired - Fee Related
- 2001-10-19 JP JP2002536047A patent/JP4343527B2/ja not_active Expired - Fee Related
- 2001-10-19 ZA ZA200301693A patent/ZA200301693B/en unknown
-
2009
- 2009-02-25 JP JP2009042453A patent/JP2009185031A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| JP2004524276A (ja) | 2004-08-12 |
| SE0003810D0 (sv) | 2000-10-20 |
| ZA200301693B (en) | 2004-03-01 |
| CN101298433A (zh) | 2008-11-05 |
| CN1714077A (zh) | 2005-12-28 |
| CN100378074C (zh) | 2008-04-02 |
| JP4343527B2 (ja) | 2009-10-14 |
| JP2009185031A (ja) | 2009-08-20 |
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