[go: up one dir, main page]

WO2025079634A1 - Composé cyclique condensé et composition de lutte contre les arthropodes nuisibles le contenant - Google Patents

Composé cyclique condensé et composition de lutte contre les arthropodes nuisibles le contenant Download PDF

Info

Publication number
WO2025079634A1
WO2025079634A1 PCT/JP2024/036248 JP2024036248W WO2025079634A1 WO 2025079634 A1 WO2025079634 A1 WO 2025079634A1 JP 2024036248 W JP2024036248 W JP 2024036248W WO 2025079634 A1 WO2025079634 A1 WO 2025079634A1
Authority
WO
WIPO (PCT)
Prior art keywords
group
optionally substituted
substituents selected
halogen atoms
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
PCT/JP2024/036248
Other languages
English (en)
Japanese (ja)
Inventor
裕人 小幡
晃一郎 土田
美咲 西田
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Chemical Co Ltd
Original Assignee
Sumitomo Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Co Ltd filed Critical Sumitomo Chemical Co Ltd
Publication of WO2025079634A1 publication Critical patent/WO2025079634A1/fr
Pending legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01M—CATCHING, TRAPPING OR SCARING OF ANIMALS; APPARATUS FOR THE DESTRUCTION OF NOXIOUS ANIMALS OR NOXIOUS PLANTS
    • A01M29/00—Scaring or repelling devices, e.g. bird-scaring apparatus
    • A01M29/12—Scaring or repelling devices, e.g. bird-scaring apparatus using odoriferous substances, e.g. aromas, pheromones or chemical agents
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N65/00—Biocides, pest repellants or attractants, or plant growth regulators containing material from algae, lichens, bryophyta, multi-cellular fungi or plants, or extracts thereof
    • A01N65/08—Magnoliopsida [dicotyledons]
    • A01N65/12—Asteraceae or Compositae [Aster or Sunflower family], e.g. daisy, pyrethrum, artichoke, lettuce, sunflower, wormwood or tarragon
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/02—Acaricides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/04—Insecticides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Definitions

  • the present invention relates to a fused ring compound and a composition for controlling harmful arthropods that contains the same.
  • Patent Document 1 describes that certain compounds have a pest control effect.
  • the present invention aims to provide a compound that has excellent control effect against harmful arthropods.
  • Group A C1-C6 chain hydrocarbon group ⁇ the C1-C6 chain hydrocarbon group may be substituted with one or more substituents selected from the group consisting of a C3-C6 cycloalkyl group optionally substituted with one or more halogen atoms, a cyano group, and a halogen atom ⁇
  • a C3-C6 cycloalkyl group ⁇ the C3-C6 cycloalkyl group may be substituted with one or more substituents selected from the group consisting of a C1-C6 alkoxy group, a cyano group, and a halogen atom ⁇
  • a phenyl group optionally substituted with one or more substituents selected from Group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted with one or more substituents selected from Group B, OR 3a , SF 5 , NR 3d OR 3b , NR 3b C(O)R 3c , NR 3d
  • R 3a represents a C3-C6 cycloalkyl group optionally substituted with one or more substituents selected from the group consisting of a halogen atom and a cyano group, a C1-C6 chain hydrocarbon group optionally substituted with one or more halogen atoms, a phenyl group optionally substituted with one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted with one or more substituents selected from group B, C(O)R 3c , C(O)OR 3j , C(O)NR 3f R 3g , S(O) 2 R 3k , or a hydrogen atom;
  • R 3b represents a C1-C6 chain hydrocarbon group optionally substituted with one or more halogen atoms, or a hydrogen atom;
  • R 3c represents a C1-C6 chain hydrocarbon group optionally substituted with one or more halogen atoms, a C3-C6
  • Group B a group consisting of C1-C6 chain hydrocarbon groups optionally substituted with one or more halogen atoms, C3-C6 cycloalkyl groups optionally substituted with one or more halogen atoms, C1-C6 alkoxy groups optionally substituted with one or more halogen atoms, cyano groups, hydroxy groups, and halogen atoms.
  • Group C a C3-C6 cycloalkyl group optionally substituted by one or more substituents selected from group E, a phenyl group optionally substituted by one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted by one or more substituents selected from group B, OR 3a , NR 3d OR 3b , NR 3b C(O)R 3c , NR 3d NR 3b C(O)R 3c , NR 3b C(O)OR 3e , NR 3d NR 3b C(O)OR 3e , NR 3b C(O ) NR 3f R 3g , NR 3d NR 3b C(O)NR 3f R 3g , N ⁇ S(O) p R 3h R 3i , C(O)R 3c , C(O) OR the group consisting of C(O)NR 3f R 3g , S(O) m R 3k ,
  • Group F a group consisting of a C3-C6 cycloalkyl group optionally substituted with one or more substituents selected from Group E, a phenyl group optionally substituted with one or more substituents selected from Group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted with one or more substituents selected from Group B, OR 3a , S(O) mR 3k , C(O)R 3c , C(O)OR 3j , C(O)NR 3fR 3g , NR 3bR 3c , NR 3bC (O)R 3c , NR 3bC (O)NR 3fR 3g , N ⁇ S(O) pR 3hR 3i , a 3- to 6-membered non-aromatic heterocyclic group, a cyano group, and a halogen atom.
  • compound N of the present invention or an N-oxide thereof (hereinafter, compound N of the present invention or an N-oxide thereof will be referred to as compound of the present invention).
  • R 3a is a C3-C6 cycloalkyl group optionally substituted with one or more substituents selected from the group consisting of halogen atoms and cyano groups, a C1-C6 chain hydrocarbon group optionally substituted with one or more halogen atoms, a phenyl group optionally substituted with one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted with one or more substituents selected from group B, C(O)R 3c , C(O)OR 3j , C(O)NR 3f R 3g , or a hydrogen atom.
  • L is a single bond, R 1 is a methyl group;
  • Q is a group represented by formula A1, a group represented by formula A2, or a group represented by formula A3;
  • Q1 is CR3q1 , Q2 is CR3q2 , and
  • Q3 is CR3q3 ;
  • R 3q1 , R 3q2 , and R 3q3 are the same or different and each is a methyl group, a halogen atom, or a hydrogen atom;
  • the combination of Q 1a and Q 2a is A combination in which Q 1a is CR 3q4 and Q 2a is CR 3q5 ; a combination in which Q 1a is a nitrogen atom and Q 2a is CR 3q5 ; or a combination in which Q 1a is CR 3q4 and Q 2a is a nitrogen atom, R 3q4 , R 3q5 and R 4 are the same or different and each is a methyl group, a halogen atom,
  • L is a single bond;
  • R 1 is a methyl group;
  • Q is a group represented by formula A1 or a group represented by formula A2,
  • Q1 is CR3q1
  • Q2 is CR3q2
  • Q3 is CR3q3 ;
  • R 3q1 , R 3q2 , and R 3q3 are a hydrogen atom;
  • R 2 is a phenyl group, a pyrazolyl group, a pyridyl group, or a pyrimidinyl group ⁇ the phenyl group, the pyrazolyl group, the pyridyl group, and the pyrimidinyl group may be substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group optionally substituted with one or more halogen atoms, a cyano group, and a halogen atom ⁇
  • X is NR10C (Z) R11 or NR10C (
  • a harmful arthropod control composition comprising the compound according to any one of [1] to [4] or an N-oxide thereof and an inert carrier.
  • a composition comprising one or more components selected from the group consisting of group (a), group (b), group (c), and group (d), and a compound or an N-oxide thereof according to any one of [1] to [4]: Group (a): A group consisting of insecticidal active ingredients, acaricidal active ingredients and nematicidal active ingredients; Group (b): bactericidal active ingredient; Group (c): plant growth regulating ingredients; Group (d): repellent components.
  • a method for controlling harmful arthropods comprising applying an effective amount of the compound according to any one of [1] to [4] or an N-oxide thereof, or an effective amount of the composition according to claim 6 to harmful arthropods or a habitat of harmful arthropods.
  • a seed or a vegetative reproductive organ carrying an effective amount of the compound according to any one of [1] to [4] or an N-oxide thereof, or an effective amount of the composition according to claim 6.
  • the present invention makes it possible to control harmful arthropods.
  • a halogen atom means a fluorine atom, a chlorine atom, a bromine atom, or an iodine atom.
  • a substituent has two or more halogen atoms or substituents, those halogen atoms or substituents may be the same or different.
  • CX-CY means that the number of carbon atoms is X to Y.
  • C1-C6 means that the number of carbon atoms is 1 to 6.
  • the chain hydrocarbon group refers to an alkyl group, an alkenyl group, or an alkynyl group.
  • alkyl group examples include a methyl group, an ethyl group, a propyl group, an isopropyl group, a 1,1-dimethylpropyl group, a 1,2-dimethylpropyl group, a 1-ethylpropyl group, a butyl group, a sec-butyl group, a tert-butyl group, a pentyl group, and a hexyl group.
  • alkenyl group examples include a vinyl group, a 1-propenyl group, a 2-propenyl group, a 1-methyl-1-propenyl group, a 1-methyl-2-propenyl group, a 1,2-dimethyl-1-propenyl group, a 1-ethyl-2-propenyl group, a 3-butenyl group, a 4-pentenyl group, and a 5-hexenyl group.
  • alkynyl group examples include an ethynyl group, a 1-propynyl group, a 2-propynyl group, a 1-methyl-2-propynyl group, a 1,1-dimethyl-2-propynyl group, a 1-ethyl-2-propynyl group, a 2-butynyl group, a 4-pentynyl group, and a 5-hexynyl group.
  • alkoxy groups include methoxy, ethoxy, propoxy, isopropoxy, butoxy, tert-butoxy, pentyloxy, and hexyloxy groups.
  • Examples of the 5- or 6-membered aromatic heterocyclic group include a pyrazolyl group, an imidazolyl group, a triazolyl group, a tetrazolyl group, an oxazolyl group, an isoxazolyl group, a thiazolyl group, an isothiazolyl group, an oxadiazolyl group, a thiadiazolyl group, a pyridyl group, a pyridazinyl group, a pyrimidinyl group, and a pyrazinyl group.
  • Examples of the 9-membered aromatic heterocyclic group include a benzoxazolyl group, a benzoisoxazolyl group, a benzothiazolyl group, a benzoisothiazolyl group, and a triazolopyridyl group.
  • Examples of the 10-membered aromatic heterocyclic group include a quinolyl group, an isoquinolyl group, a quinazolinyl group, and a quinazolonyl group.
  • the (C3-C6 cycloalkyl)C1-C3 alkyl group optionally substituted with one or more halogen atoms refers to a group in which the (C3-C6 cycloalkyl) and/or (C1-C3 alkyl) may have one or more halogen atoms, and examples thereof include a cyclopropylmethyl group, a cyclopropylethyl group, a (2,2-difluorocyclopropyl)methyl group, a 2-cyclopropyl-1,1,2,2-tetrafluoroethyl group, and a 2-(2,2-difluorocyclopropyl)-1,1,2,2-tetrafluoroethyl group.
  • Examples of the phenyl C1-C3 alkyl group ⁇ the phenyl moiety in the phenyl C1-C3 alkyl group may be substituted with one or more substituents selected from group B ⁇ include a benzyl group, a 2-fluorobenzyl group, a 4-chlorobenzyl group, a 4-(trifluoromethyl)benzyl group, and a 2-[4-(trifluoromethyl)phenyl]ethyl group.
  • Examples of the 3- to 6-membered non-aromatic heterocyclic group include an oxetanyl group, a pyrrolidinyl group, a 2-oxopyrrolidinyl group, a 2-oxoimidazolidinyl group, a 3,4,5,6-tetrahydro-2-pyrimidinyl group, a tetrahydrofuranyl group, a piperidyl group, a tetrahydropyranyl group, an isoxazolidinyl group, and a morpholinyl group.
  • alkylsulfonyl group examples include a methylsulfonyl group, an ethylsulfonyl group, a propylsulfonyl group, and an isopropylsulfonyl group.
  • cycloalkylsulfonyl group examples include a cyclopropylsulfonyl group, a cyclobutylsulfonyl group, and a cyclohexylsulfonyl group.
  • Cycloalkyl groups include, for example, cyclopropyl, cyclobutyl, cyclopentyl, and cyclohexyl groups.
  • the N-oxide of the compound represented by formula (I) means a structure in which at least one nitrogen atom contained in the compound represented by formula (I) is substituted with an oxo group.
  • Compound N of the present invention may form an acid addition salt.
  • acids that form acid addition salts include inorganic acids such as hydrogen chloride, phosphoric acid, and sulfuric acid, and organic acids such as acetic acid, trifluoroacetic acid, benzoic acid, and p-toluenesulfonic acid. Acid addition salts can be obtained, for example, by mixing compound N of the present invention with an acid.
  • Q is a group represented by formula A1-1, a group represented by formula A1-2, a group represented by formula A2-1, a group represented by formula A2-2, a group represented by formula A2-3, a group represented by formula A3-1, a group represented by formula A3-2, a group represented by formula A4-1, a group represented by formula A4-2, or a group represented by formula A5-1 (# represents a bonding site to R2 , and ⁇ represents a bonding site to a carbon atom), and R 3q1 , R 3q2 , R 3q3 , R 3q4 , R 3q5 and R Compounds in which 4 is the same or different and is a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, a phenyl group optionally substituted with one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted with one or more substituent
  • a compound of the present invention N in which L is a single bond or -(CR 4a R 4b ) n -, R 4a and R 4b are the same or different and are a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, and n is 1, 2, or 3.
  • R 4a and R 4b are the same or different and are a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, and n is 1, 2, or 3.
  • n is 1, 2, or 3.
  • a compound of the present invention in which R 1 in compound N is a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, or a hydrogen atom.
  • R 1 in compound N is a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, or a hydrogen atom.
  • R 1 is a methyl group.
  • R 1 is a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, or a hydrogen atom.
  • Aspect 15 The compound according to aspect 2, wherein R 1 is a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, or a hydrogen atom.
  • R 2 is a phenyl group, a 5- or 6-membered aromatic heterocyclic group ⁇ the phenyl group and the 5- or 6-membered aromatic heterocyclic group are optionally substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom, a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, OR 3a , NR 3b C(O)R 3c , C(O)NR 3f R 3g , S(O) m R 3k , a cyano group, and a halogen atom ⁇ , C(O)NR 6 R 7 , NR 16 C(O)R 17 , NR 16 C(O)OR 17 , NR 16 C(O)NR 17 R 18 , OR 18 , a group represented by formula E1-1, a group represented by formula E1-2,
  • R 2 is a phenyl group, a pyrazolyl group, a pyridyl group, or a pyrimidinyl group ⁇ the phenyl group, the pyrazolyl group, the pyridyl group, and the pyrimidinyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom, a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, a C1-C3 alkoxy group optionally substituted with one or more halogen atoms, NR 3b C(O)R 3c , C(O)NR 3f R 3g , S(O) m R 3k , a cyano group, and a halogen atom ⁇ , C( ⁇ NOR 9 )R 5 , C( ⁇ NOR 9 )
  • R 2 is a phenyl group, a pyrazolyl group, a pyridyl group, or a pyrimidinyl group ⁇ the phenyl group, the pyrazolyl group, the pyridyl group, and the pyrimidinyl group are optionally substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom, a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, a C1-C3 alkoxy group optionally substituted with one or more halogen atoms, NR 3b C(O)R 3c , C(O)NR 3f R 3g , S(O) m R 3k , a cyano group, and a halogen atom ⁇ , C( ⁇ NOR 9 )R 5 , C( ⁇ NOR 9
  • R 2 is a phenyl group, a 5- or 6-membered aromatic heterocyclic group ⁇ the phenyl group and the 5- or 6-membered aromatic heterocyclic group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom, a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, OR 3a , NR 3b C(O)R 3c , C(O)NR 3f R 3g , S(O) m R 3k , a cyano group, and a halogen atom ⁇ , C(O)NR 6 R 7 , NR 16 C(O)R 17 , OR 18 , a group represented by formula E1-1, a group represented by formula E1-2, a group represented by formula E2-1, a group represented by formula E2-2, a group represented by formula E
  • X is NR 10 C(O)R 11 , NR 10 C(O)NR 11 R 12 , or NR 10 X 1
  • X 1 is a 9- or 10-membered aromatic heterocyclic group ⁇ the 9- or 10-membered aromatic heterocyclic group may be substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 , NR 10 C(O)NR 11 R 12 , or NR 10 X 1
  • X 1 is a 9- or 10-membered aromatic heterocyclic group ⁇ the 9- or 10-membered aromatic heterocyclic group is optionally substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 , NR 10 C(O)NR 11 R 12 , or NR 10 X 1
  • X 1 is a 9- or 10-membered aromatic heterocyclic group ⁇ the 9- or 10-membered aromatic heterocyclic group is optionally substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 , NR 10 C(O)NR 11 R 12 , or NR 10 X 1
  • X 1 is a 9- or 10-membered aromatic heterocyclic group ⁇ the 9- or 10-membered aromatic heterocyclic group is optionally substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 , NR 10 C(O)NR 11 R 12 , or NR 10 X 1
  • X 1 is a 9- or 10-membered aromatic heterocyclic group ⁇ the 9- or 10-membered aromatic heterocyclic group is optionally substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 , NR 10 C(O)NR 11 R 12 , or NR 10 X 1
  • X 1 is a 9- or 10-membered aromatic heterocyclic group ⁇ the 9- or 10-membered aromatic heterocyclic group is optionally substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 or NR 10 C(O)NR 11 R 12
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group or a pyrazolyl group ⁇ the phenyl group, the pyridyl group and the pyrazolyl group are optionally substituted with a cyclopropyl group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 or NR 10 C(O)NR 11 R 12
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group or a pyrazolyl group ⁇ the phenyl group, the pyridyl group and the pyrazolyl group are optionally substituted with a cyclopropyl group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 , or NR 10 C(O)NR 11 R 12
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are optionally substituted with a cyclopropyl group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen atom ⁇
  • X is NR 10 C(O)R 11 or NR 10 C(O)NR 11 R 12
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group or a pyrazolyl group ⁇ the phenyl group, the pyridyl group and the pyrazolyl group are optionally substituted with a cyclopropyl group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 or NR 10 C(O)NR 11 R 12
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group or a pyrazolyl group ⁇ the phenyl group, the pyridyl group and the pyrazolyl group are optionally substituted with a cyclopropyl group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11 or NR 10 C(O)NR 11 R 12
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group or a pyrazolyl group ⁇ the phenyl group, the pyridyl group and the pyrazolyl group are optionally substituted with a cyclopropyl group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group and a halogen atom ⁇
  • X is NR 10 C(O)R 11
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are a cyclopropyl group optionally substituted with a cyano group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen
  • X is NR 10 C(O)R 11
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are a cyclopropyl group optionally substituted with a cyano group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen atom ⁇
  • R 13 is a C1-C3 alkyl group
  • OR 14
  • X is NR 10 C(O)R 11
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are a cyclopropyl group optionally substituted with a cyano group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen atom ⁇
  • R 13 is a C1-C3 alkyl group
  • OR 14
  • X is NR 10 C(O)R 11
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are a cyclopropyl group optionally substituted with a cyano group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen atom ⁇
  • R 13 is a C1-C3
  • X is NR 10 C(O)R 11
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are a cyclopropyl group optionally substituted with a cyano group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen atom ⁇
  • R 13 is a C1-C3
  • X is NR 10 C(O)R 11
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are a cyclopropyl group optionally substituted with a cyano group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen atom ⁇
  • R 13 is a C1-C3
  • Aspect 66 A compound according to any one of Aspects 1 to 36 or compound N of the present invention, wherein R 2 is a 5- or 6-membered aromatic heterocyclic group optionally substituted with one or more substituents selected from group A, X is NR 11 C(O)R 12 , R 11 is a C1-C6 alkyl group optionally substituted with one or more substituents selected from group F, and R 12 is a phenyl group optionally substituted with one or more substituents selected from group A.
  • Q is a group represented by formula A3-3 (# represents the bonding site to R2 , and ⁇ represents the bonding site to a carbon atom), and R3q5 and R4 are the same or different and are a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, a halogen atom, or a hydrogen atom.
  • R3q5 and R4 are the same or different and are a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms, a halogen atom, or a hydrogen atom.
  • a compound in aspect A4, wherein R 2 is a phenyl group, a pyrazolyl group, a pyridyl group, or a pyrimidinyl group ⁇ the phenyl group, the pyrazolyl group, the pyridyl group, and the pyrimidinyl group may be substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group optionally substituted with one or more halogen atoms, NR 3b C(O)R 3c , C(O)NR 3f R 3g , a cyano group, and a halogen atom ⁇ .
  • X is NR 10 C(O)R 11
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are a cyclopropyl group optionally substituted with a cyano group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen atom ⁇
  • R 13 is a C1-C3
  • Aspect A7 The compound in Aspect A4, wherein X is NR 10 C(O)R 11 , R 10 is a C1-C3 alkyl group or a hydrogen atom, and R 11 is a phenyl group ⁇ the phenyl group may be substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group substituted with one or more halogen atoms, a C1-C3 alkoxy group substituted with one or more halogen atoms, a cyano group, and a halogen atom ⁇ .
  • X is NR 10 C(O)R 11
  • R 10 is a C1-C3 alkyl group
  • OR 14 C(O)R 13 , C(O)OR 13 , or a hydrogen atom
  • R 11 is a phenyl group, a pyridyl group, or a pyrazolyl group ⁇ the phenyl group, the pyridyl group, and the pyrazolyl group are a cyclopropyl group optionally substituted with a cyano group
  • a C1-C3 alkyl group ⁇ the C1-C3 alkyl group may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a cyano group, and a halogen atom ⁇
  • OR 3a S(O) m R 3k , a cyano group, and a halogen atom ⁇
  • R 13 is a C1-C3
  • A9 The compound in Aspect A5, wherein X is NR 10 C(O)R 11 , R 10 is a C1-C3 alkyl group or a hydrogen atom, and R 11 is a phenyl group ⁇ the phenyl group may be substituted with one or more substituents selected from the group consisting of a C1-C3 alkyl group substituted with one or more halogen atoms, a C1-C3 alkoxy group substituted with one or more halogen atoms, a cyano group, and a halogen atom ⁇ .
  • the compound represented by formula (I-1) (hereinafter referred to as compound (I-1)) can be produced by reacting a compound represented by formula (I-2) (hereinafter referred to as compound (I-2)) with a compound represented by formula (I-3) (hereinafter referred to as compound (I-3)).
  • a solvent for example, ethers such as tetrahydrofuran (hereinafter referred to as THF), 1,4-dioxane, 1,2-dimethoxyethane, methyl tert-butyl ether, diethyl ether, etc.
  • ethers halogenated hydrocarbons such as dichloromethane, chloroform, etc.
  • halogenated hydrocarbons such as dichloromethane, chloroform, etc.
  • nitriles such as acetonitrile, etc.
  • aromatic hydrocarbons such as toluene, xylene, etc.
  • aromatic hydrocarbons aprotic polar solvents such as N-methylpyrrolidone (hereinafter referred to as NMP), N,N-dimethylformamide (hereinafter referred to as DMF), etc.
  • NMP N-methylpyrrolidone
  • DMF N,N-dimethylformamide
  • aprotic polar solvents aprotic polar solvents
  • the reaction can be carried out using a base as necessary, for example, organic bases such as triethylamine, N,N-diisopropylethylamine, pyridine, 4-(dimethylamino)pyridine (hereinafter referred to as organic bases), and alkali metal carbonates such as sodium carbonate, potassium carbonate, cesium carbonate (hereinafter referred to as alkali metal carbonates).
  • organic bases such as triethylamine, N,N-diisopropylethylamine, pyridine, 4-(dimethylamino)pyridine (hereinafter referred to as organic bases), and alkali metal carbonates such as sodium carbonate, potassium carbonate, cesium carbonate (hereinafter referred to as alkali metal carbonates).
  • compound (I-3) is usually used in a ratio of 1 to 10 moles per mole of compound (I-2).
  • the reaction temperature is usually in the range of 0° C. to 200° C.
  • the reaction time is usually in
  • compound (I-3) is a commercially available compound or can be prepared using known methods.
  • the compound represented by formula (I) (i.e., compound N of the present invention) can be produced by reacting a compound represented by formula (I-8) (hereinafter referred to as compound (I-8)) with a compound represented by formula (IM) (hereinafter referred to as compound (IM)).
  • X a represents a chlorine atom, a bromine atom, or an iodine atom
  • M A represents a 9-borabicyclo[3.3.1]nonan-9-yl group, a borono group, a 4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl group, or a tributylstannyl group, and the other symbols have the same meanings as above.
  • the reaction is usually carried out in a solvent, such as ethers, aromatic hydrocarbons, aprotic polar solvents, water, and mixtures of two or more thereof.
  • the metal catalyst examples include palladium catalysts such as tetrakis(triphenylphosphine)palladium(0), 1,1'-bis(diphenylphosphino)ferrocenepalladium(II) dichloride, tris(dibenzylideneacetone)dipalladium(0), palladium(II) acetate, etc.; nickel catalysts such as bis(cyclooctadiene)nickel(0), nickel(II) chloride, etc.; iron catalysts such as iron(III) chloride, iron(III) acetylacetonate, etc.; copper catalysts such as copper(I) iodide, copper(I) chloride, etc.; and combinations of two or more of these.
  • palladium catalysts such as tetrakis(triphenylphosphine)palladium(0), 1,1'-bis(diphenylphosphino)ferrocenepalladium(II) dichloride, tris(di
  • the reaction may, if necessary, use a ligand, a base, and/or an inorganic halide.
  • the ligand include triphenylphosphine, xantphos, 2,2'-bis(diphenylphosphino)-1,1'-binaphthyl, 1,1'-bis(diphenylphosphino)ferrocene, 2-dicyclohexylphosphino-2',4',6'-triisopropylbiphenyl, 2-dicyclohexylphosphino-2',6'-dimethoxybiphenyl, 1,2-bis(diphenylphosphino)ethane, 2,2'-bipyridine, 2-aminoethanol, 8-hydroxyquinoline, and 1,10-phenanthroline.
  • the bases include alkali metal carbonates and organic bases.
  • Inorganic halides include alkali metal fluorides such as potassium fluoride and sodium fluoride; and alkali metal chlorides such as lithium chloride and sodium chloride.
  • compound (IM) is usually used in a ratio of 1 to 10 moles and metal catalyst is usually used in a ratio of 0.01 to 0.5 moles per mole of compound (I-8).
  • metal catalyst is usually used in a ratio of 0.01 to 0.5 moles per mole of compound (I-8).
  • the ligand is usually used in a ratio of 0.01 to 1 mole per mole of compound (I-8).
  • the base is usually used in a ratio of 0.1 to 5 moles per mole of compound (I-8).
  • the inorganic halide When an inorganic halide is used in the reaction, the inorganic halide is usually used in a ratio of 0.1 to 5 moles per mole of compound (I-8).
  • the reaction temperature is usually in the range of ⁇ 20° C. to 200° C.
  • the reaction time is usually in the range of 0.1 to 72 hours.
  • the compound N of the present invention can be obtained by carrying out post-treatment operations such as adding water to the reaction mixture, extracting with an organic solvent, drying and concentrating the organic layer.
  • Compounds (IM) are commercially available compounds or can be prepared using known methods.
  • the reaction can also be carried out in accordance with, for example, the method described in Example H2 of WO 2020/070049.
  • the compound represented by formula (I-1A) (hereinafter referred to as compound (I-1A)) can be produced by reacting a compound represented by formula (I-2A) (hereinafter referred to as compound (I-2A)) with a compound represented by formula (M-g) (hereinafter referred to as compound (M-g)) in the presence of an acid.
  • X represents a leaving group such as a chlorine atom
  • Boc represents a tert-butoxycarbonyl group
  • the other symbols have the same meanings as above.
  • the reaction is usually carried out in a solvent, which may include ethers, halogenated hydrocarbons, aromatic hydrocarbons, nitriles, aprotic polar solvents, water, and mixtures of two or more thereof.
  • the acid used in the reaction includes, for example, trifluoroacetic acid and hydrogen chloride.
  • hydrogen chloride a solution of hydrogen chloride such as hydrochloric acid or a hydrogen chloride/methanol solution may be used in the reaction.
  • the reaction can be carried out, for example, by first mixing compound (I-2A) with an acid, then distilling off the acid, and mixing compound (Mg).
  • a base can be used as necessary.
  • the base include organic bases.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (I-2A).
  • compound (Mg) is usually used in a ratio of 1 to 2 moles and acid is usually used in a ratio of 1 to 100 moles, relative to 1 mole of compound (I-2A).
  • the reaction temperature is usually within the range of ⁇ 20 to 200° C.
  • the reaction time is usually within the range of 0.1 to 24 hours.
  • Compound (Mg) is a commercially available compound or can be prepared using known methods.
  • Compound (I-1A) can also be produced by reacting compound (I-2A) with a compound represented by formula (Me) (hereinafter referred to as compound (Me)) in the presence of a condensing agent and an acid.
  • a condensing agent for reacting compound (I-2A) with a compound represented by formula (Me) (hereinafter referred to as compound (Me)) in the presence of a condensing agent and an acid.
  • a solvent which may include ethers, halogenated hydrocarbons, aromatic hydrocarbons, nitriles, esters such as ethyl acetate and butyl acetate (hereinafter referred to as esters), aprotic polar solvents, nitrogen-containing aromatic compounds such as pyridine, picoline, lutidine, and quinoline (hereinafter referred to as nitrogen-containing aromatic compounds), and mixtures of two or more of these.
  • a solvent which may include ethers, halogenated hydrocarbon
  • the acid used in the reaction includes, for example, trifluoroacetic acid and hydrogen chloride.
  • hydrogen chloride a solution of hydrogen chloride such as hydrochloric acid or a hydrogen chloride/methanol solution may be subjected to the reaction.
  • the reaction can be carried out, for example, by first mixing compound (I-2A) with an acid, then distilling off the acid, and mixing compound (Me) with a condensing agent.
  • Condensing agents used in the reaction include, for example, carbodiimides such as 1-ethyl-3-[3-(dimethylamino)propyl]carbodiimide hydrochloride and 1,3-dicyclohexylcarbodiimide.
  • a catalyst may be used in the reaction, if necessary.
  • An example of the catalyst is 1-hydroxybenzotriazole.
  • the catalyst is usually used in a ratio of 0.01 to 0.5 moles per mole of compound (I-2A).
  • a base can be used as necessary.
  • the base include organic bases.
  • the base is usually used in a ratio of 1 to 5 moles per mole of compound (I-2A).
  • compound (Me) is usually used in a ratio of 1 to 2 moles
  • a condensing agent is usually used in a ratio of 1 to 5 moles
  • an acid is usually used in a ratio of 1 to 100 moles, relative to 1 mole of compound (I-2A).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours.
  • the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (I-1A).
  • Compound (Me) is a commercially available compound or can be prepared using known methods.
  • Compound (I-1A) can also be produced by reacting a compound represented by formula (I-11) (hereinafter referred to as compound (I-11)) with compound (I-3). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 1, except that compound (I-11) is used in place of compound (I-2).
  • Compound (I-1A) can also be produced by reacting compound (I-11) with compound (Me) in the presence of a condensing agent.
  • a condensing agent In the formula, the symbols have the same meanings as defined above.
  • the reaction is usually carried out in a solvent.
  • the solvent used in the reaction include ethers, halogenated hydrocarbons, aromatic hydrocarbons, esters, nitriles, aprotic polar solvents, nitrogen-containing aromatic compounds, and mixtures of two or more of these.
  • Condensing agents used in the reaction include, for example, carbodiimides such as 1-ethyl-3-[3-(dimethylamino)propyl]carbodiimide hydrochloride and 1,3-dicyclohexylcarbodiimide.
  • a catalyst may be used in the reaction, if necessary.
  • An example of the catalyst is 1-hydroxybenzotriazole.
  • the catalyst is usually used in a ratio of 0.01 to 0.5 moles per mole of compound (I-11).
  • a base can be used as necessary. Examples of the base include organic bases. When a base is used in the reaction, the base is usually used in a ratio of 1 to 5 moles per mole of compound (I-11).
  • compound (Me) is usually used in a ratio of 1 to 2 moles and a condensing agent is usually used in a ratio of 1 to 5 moles, relative to 1 mole of compound (I-11).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (I-1A).
  • the compound represented by formula (I-1B) (hereinafter referred to as compound (I-1B)) can be produced by reacting a compound represented by formula (I-2B) (hereinafter referred to as compound (I-2B)) with compound (I-3). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 1, except that compound (I-2B) is used in place of compound (I-2).
  • Production method 8 Compound (I-1B) can also be produced by reacting compound (I-2B) with compound (Me) in the presence of a condensing agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 6, except for using compound (I-2B) instead of compound (I-11).
  • Production method 9 Compound (I-1) can also be produced by reacting a compound represented by formula (I-20) (hereinafter referred to as compound (I-20)) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (I-20) is used in place of compound (I-8).
  • the compound represented by formula (II-1) (hereinafter referred to as compound (II-1)) can be produced by reacting a compound represented by formula (II-2) (hereinafter referred to as compound (II-2)) with compound (I-3). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 1, except that compound (II-2) is used in place of compound (I-2).
  • Compound (II-1) can also be produced by reacting compound (II-2) with compound (Me) in the presence of a condensing agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 6, except that compound (II-2) is used in place of compound (I-11).
  • Compound (II-1) can also be produced by reacting a compound represented by formula (II-19) (hereinafter referred to as compound (II-19)) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (II-19) is used in place of compound (I-8).
  • the compound represented by formula (II-1A) (hereinafter referred to as compound (II-1A)) can be produced by reacting a compound represented by formula (II-3A) (hereinafter referred to as compound (II-3A)) with compound (I-3) in the presence of an acid.
  • a compound represented by formula (II-3A) (hereinafter referred to as compound (II-3A))
  • compound (I-3) in place of compound (Mg).
  • Compound (I-2) can be produced from a compound represented by formula (I-4) (hereinafter referred to as compound (I-4)). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out, for example, according to the method described in Green's PROTECTIVE GROUPS in ORGANIC SYNTHESIS FORTH EDITION, p. 727.
  • Compound (I-2) may form an acid addition salt.
  • acids that form acid addition salts include inorganic acids such as hydrochloric acid and sulfuric acid; and organic acids such as acetic acid, trifluoroacetic acid, benzoic acid, and p-toluenesulfonic acid.
  • Compound (I-4) can be produced by reacting a compound represented by formula (I-5) (hereinafter referred to as compound (I-5)) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (I-5) is used in place of compound (I-8).
  • Compound (I-5) can be produced by reacting a compound represented by formula (I-6) (hereinafter referred to as compound (I-6)) with a halogenating agent.
  • a compound represented by formula (I-6) hereinafter referred to as compound (I-6)
  • a halogenating agent for example, acetyl alcohol, acetyl ether, benzyl ether, benzyl ether, benzyl, nitriles, ethers, aromatic hydrocarbons, aprotic polar solvents, halogenated hydrocarbons, water, and mixtures thereof.
  • a solvent for example, alcohols such as methanol and ethanol (hereinafter referred to as alcohols), nitriles, ethers, aromatic hydrocarbons, aprotic polar solvents, halogenated hydrocarbons, water, and mixtures thereof.
  • halogenating agent examples include chlorine, bromine, iodine, N-chlorosuccinimide, N-bromosuccinimide, and N-iodosuccinimide (hereinafter referred to as NIS).
  • a base can be used as necessary.
  • the base include alkali metal carbonates.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (I-6).
  • the halogenating agent is usually used in a ratio of 1 to 10 moles per mole of compound (I-6).
  • the reaction temperature is usually in the range of ⁇ 20° C. to 200° C.
  • the reaction time is usually in the range of 0.1 to 72 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (I-5).
  • Compound (I-6) can be produced from a compound represented by formula (I-7) (hereinafter referred to as compound (I-7)). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out, for example, according to the method described in Intermediate 23 of WO 2007/147794 or Example 5 of WO 2003/037900.
  • Compound (I-7) is a commercially available compound or can be prepared using known methods.
  • Compound (I-9) can be produced from a compound represented by formula (I-7A) (hereinafter referred to as compound (I-7A)) and a compound represented by formula (IA) (hereinafter referred to as compound (IA)).
  • compound (I-7A) a compound represented by formula (IA)
  • the symbols have the same meanings as defined above.
  • the reaction can be carried out, for example, according to the method described in International Publication No. 2007/147794, Intermediate 23.
  • Reference Manufacturing Method 6 Compound (I-8) can be produced by reacting compound (I-10) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 3, except for using compound (I-10) instead of compound (I-6).
  • Compound (I-11) can be produced from a compound represented by formula (I-2A) (hereinafter referred to as compound (I-2A)). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out, for example, according to the method described in Green's PROTECTIVE GROUPS in ORGANIC SYNTHESIS FORTH EDITION, p. 727.
  • Compound (I-11) may form an acid addition salt.
  • acids that form acid addition salts include inorganic acids such as hydrochloric acid and sulfuric acid; and organic acids such as acetic acid, trifluoroacetic acid, benzoic acid, and p-toluenesulfonic acid.
  • Compound (I-2A) can be produced by reacting a compound represented by formula (I-12) (hereinafter referred to as compound (I-12)) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (I-12) is used in place of compound (I-8).
  • Compound (I-12) can be produced by reacting a compound represented by formula (I-13) (hereinafter referred to as compound (I-13)) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 3, except for using compound (I-13) instead of compound (I-6).
  • Compound (I-13) is a commercially available compound or can be prepared using known methods.
  • Compound (I-2) can also be produced from a compound represented by formula (I-4B) (hereinafter referred to as compound (I-4B)).
  • compound (I-4B) a compound represented by formula (I-4B)
  • Cbz represents a benzyloxycarbonyl group, and the other symbols have the same meanings as defined above.
  • the reaction can be carried out, for example, according to the method described in Green's PROTECTIVE GROUPS in ORGANIC SYNTHESIS FORTH EDITION p. 750.
  • Compound (I-2) may form an acid addition salt.
  • acids that form acid addition salts include inorganic acids such as hydrochloric acid and sulfuric acid; and organic acids such as acetic acid, trifluoroacetic acid, benzoic acid, and p-toluenesulfonic acid.
  • Compound (I-4B) can be produced by reacting a compound represented by formula (I-5B) (hereinafter referred to as compound (I-5B)) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (I-5B) is used in place of compound (I-8).
  • Reference Manufacturing Method 3-1 Compound (I-5B) can be produced by reacting a compound represented by formula (I-6B) (hereinafter referred to as compound (I-6B)) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 3, except for using compound (I-6B) instead of compound (I-6).
  • Compound (I-6B) can be produced from a compound represented by formula (I-7B) (hereinafter referred to as compound (I-7B)).
  • compound (I-7B) a compound represented by formula (I-7B) (hereinafter referred to as compound (I-7B)).
  • the reaction may be carried out, for example, according to the method described in WO 2007/147794 Intermediate 23, the method described in WO 2003/037900 Example 5, the method described in WO 2007/134362 Example 1, the method described in WO 2021/158634 Intermediate BMR step 1, or Huaxue Xuebao (2005), 63 (9), 855-860.
  • Compound (I-7B) can be produced from a compound represented by formula (I-14B) (hereinafter referred to as compound (I-14B)). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out, for example, in accordance with the method described in WO 2016/148145, Example 1-1, Step 1-1-3.
  • Compound (I-14B) can be produced from a compound represented by formula (I-14A) (hereinafter referred to as compound (I-14A)). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out, for example, according to the method described in Inventive Example 25 of US Patent Application Publication No. 2002/6387938. Compound (I-14A) is a commercially available compound or can be prepared using known methods.
  • Compound (I-2B) can be produced by reacting a compound represented by formula (I-15) (hereinafter, compound (I-15) with an amine or an ammonium salt, and a reducing agent.
  • a compound represented by formula (I-15) hereinafter, compound (I-15)
  • an amine or an ammonium salt and a reducing agent.
  • the reaction is usually carried out in a solvent.
  • the solvent used in the reaction include alcohols, ethers, aprotic polar solvents, and mixtures thereof.
  • the amines include methylamine and ethylamine.
  • the ammonium salt includes ammonium acetate and the like.
  • an acid can be used as necessary. Examples of the acid include organic acids such as acetic acid.
  • the acid When an acid is used in the reaction, the acid is usually used in a ratio of 0.1 to 10 moles per mole of compound (I-15).
  • the reducing agent In the reaction, the reducing agent is usually used in a ratio of 1 to 10 moles per mole of compound (I-15).
  • the reaction temperature is usually in the range of ⁇ 20° C. to 200° C.
  • the reaction time is usually in the range of 0.1 to 72 hours.
  • compound (I-2B) can be obtained by carrying out post-treatment operations such as adding water to the reaction mixture, extracting with an organic solvent, drying and concentrating the organic layer.
  • Compound (I-15) can be produced by reacting a compound represented by formula (I-16) (hereinafter referred to as compound (I-16)) with a compound represented by formula (M-f) (hereinafter referred to as compound (M-f)).
  • Xd represents a chlorine atom, a bromine atom, or an iodine atom, and the other symbols have the same meanings as defined above.
  • the reaction is usually carried out in a solvent, such as, for example, ethers, aromatic hydrocarbons, aprotic polar solvents, and mixtures of two or more thereof.
  • compound (Mf) is usually used in a ratio of 1 to 10 moles per mole of compound (I-16).
  • the reaction temperature is usually in the range of ⁇ 20° C. to 200° C.
  • the reaction time is usually in the range of 0.1 to 72 hours.
  • the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (I-15).
  • Compound (Mf) is a commercially available compound or can be prepared using known methods.
  • Compound (I-16) can be produced by reacting a compound represented by formula (I-17) (hereinafter referred to as compound (I-17)) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (I-17) is used in place of compound (I-8).
  • Compound (I-17) can be produced by reacting a compound represented by formula (I-18) (hereinafter referred to as compound (I-18)) with a compound represented by formula (M-g) (hereinafter referred to as compound (M-g)) in the presence of a condensing agent.
  • a compound represented by formula (I-18) hereinafter referred to as compound (I-18)
  • M-g compound represented by formula (M-g)
  • a condensing agent In the formula, the symbols have the same meanings as defined above.
  • the reaction is usually carried out in a solvent.
  • the solvent used in the reaction include ethers, halogenated hydrocarbons, aromatic hydrocarbons, esters, nitriles, aprotic polar solvents, nitrogen-containing aromatic compounds, and mixtures of two or more of these.
  • the condensing agent used in the reaction includes, for example, 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridinium 3-oxide hexafluorophosphate.
  • a base can be used as necessary.
  • the base include organic bases.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (I-18).
  • compound (Mg) is usually used in a ratio of 1 to 3 mol and a condensing agent is usually used in a ratio of 1 to 5 mol, relative to 1 mol of compound (I-18).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (I-17).
  • Compound (I-18) can be produced by subjecting a compound represented by formula (I-19) (hereinafter referred to as compound (I-19)) to hydrolysis reaction in the presence of a base.
  • a compound represented by formula (I-19) hereinafter referred to as compound (I-19)
  • the reaction is carried out in the presence of a base, water and an organic solvent, such as ethers, nitriles, alcohols, and mixtures thereof.
  • the base used in the reaction includes, for example, alkali metal hydroxides such as lithium hydroxide, sodium hydroxide, potassium hydroxide, etc.
  • the reaction time is usually in the range of 5 minutes to 72 hours, and the reaction temperature is usually in the range of 0° C. to 100° C.
  • the amount of the base used in the reaction can be any amount from 1 mole to an excess amount, and is preferably 1 to 5 moles, per mole of compound (I-19).
  • the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (I-18).
  • Compound (I-19) is a commercially available compound or can be prepared using known methods.
  • the compound represented by formula (I-20) (hereinafter referred to as compound (I-20)) can be produced by reacting a compound represented by formula (I-21) (hereinafter referred to as compound (I-21)) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 3, except for using compound (I-21) instead of compound (I-6).
  • Compound (I-21) can be produced by reacting a compound represented by formula (I-22) (hereinafter referred to as compound (I-22)) with compound (I-3). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 1, except that compound (I-22) is used in place of compound (I-2).
  • Reference Manufacturing Method 18 Compound (I-21) can also be produced by reacting compound (I-22) with compound (Me) in the presence of a condensing agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 6, except that compound (I-22) is used in place of compound (I-11).
  • Compound (I-22) can be produced by reacting a compound represented by formula (I-23) (hereinafter, compound (I-23) with an amine or an ammonium salt, and a reducing agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 11, except for using compound (I-23) instead of compound (I-15).
  • Compound (I-23) can be produced by reacting a compound represented by formula (I-24) (hereinafter referred to as compound (I-24)) with compound (Mf). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 12, except for using compound (I-24) instead of compound (I-16).
  • Compound (I-24) can be produced by reacting a compound represented by formula (I-25) (hereinafter referred to as compound (I-25)) with compound (Mg) in the presence of a Lewis acid.
  • a Lewis acid In the formula, the symbols have the same meanings as defined above.
  • the reaction is usually carried out in a solvent. Examples of the solvent used in the reaction include ethers, halogenated hydrocarbons, aromatic hydrocarbons, aprotic polar solvents, and mixtures of two or more of these.
  • the Lewis acid used in the reaction includes, for example, trimethylaluminum. In the reaction, the Lewis acid is usually used in a proportion of 0.1 to 5 moles per mole of compound (I-25).
  • compound (Mg) is usually used in a ratio of 1 to 5 moles per mole of compound (I-25).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours.
  • the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (I-24).
  • Compound (I-25) is a commercially available compound or can be prepared using known methods.
  • Compound (II-2) can be produced from a compound represented by formula (II-3) (hereinafter referred to as compound (II-3)).
  • compound (II-3) a compound represented by formula (II-3)
  • PG represents a tert-butoxycarbonyl group or a benzyloxycarbonyl group, and the other symbols have the same meanings as defined above.
  • the reaction can be carried out, for example, according to the method described in Green's PROTECTIVE GROUPS in ORGANIC SYNTHESIS FORTH EDITION, p. 727 or p. 750.
  • Compound (II-2) may form an acid addition salt.
  • acids that form acid addition salts include inorganic acids such as hydrochloric acid and sulfuric acid; and organic acids such as acetic acid, trifluoroacetic acid, benzoic acid, and p-toluenesulfonic acid.
  • Compound (II-3) can be produced by reacting a compound represented by formula (II-4) (hereinafter referred to as compound (II-4)) with a compound represented by formula (M-h) (hereinafter referred to as compound (M-h)) in the presence of an acid.
  • a compound represented by formula (II-4) hereinafter referred to as compound (II-4)
  • a compound represented by formula (M-h) hereinafter referred to as compound (M-h)
  • the reaction is usually carried out in a solvent.
  • the solvent used in the reaction include ethers, halogenated hydrocarbons, aromatic hydrocarbons, esters, nitriles, aprotic polar solvents, and mixtures of two or more of these.
  • the acid used in the reaction includes organic acids such as trifluoroacetic acid and acetic acid.
  • the acid is usually used in a proportion of 0.1 to 100 moles per mole of compound (II-4).
  • a base can be used as necessary. Examples of the base include organic bases.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (II-4).
  • compound (Mh) is usually used in an amount of 1 to 10 moles per mole of compound (II-4).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (II-3).
  • Compound (II-4) can be produced by reacting a compound represented by formula (II-5) (hereinafter referred to as compound (II-5)) with a hydrazine.
  • a compound represented by formula (II-5) hereinafter referred to as compound (II-5)
  • Xb represents a chlorine atom or a bromine atom, and the other symbols have the same meanings as defined above.
  • the reaction is usually carried out in a solvent, for example, ethers, halogenated hydrocarbons, aromatic hydrocarbons, alcohols, aprotic polar solvents, water, and mixtures of two or more of these.
  • the hydrazines used in the reaction include anhydrous hydrazine, hydrazine monohydrate, hydrazine monohydrochloride, and the like.
  • the hydrazine is usually used in an amount of 1 to 10 moles per mole of compound (II-5).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (II-4).
  • Compound (II-5) can be produced by reacting a compound represented by formula (II-6) (hereinafter referred to as compound (II-6)) with a halogenating agent.
  • a compound represented by formula (II-6) hereinafter referred to as compound (II-6)
  • the reaction is usually carried out in a solvent.
  • the solvent used in the reaction include ethers, halogenated hydrocarbons, aromatic hydrocarbons, nitriles, aprotic polar solvents, nitrogen-containing aromatic compounds, and mixtures of two or more of these.
  • the halogenating agent used in the reaction includes phosphorus oxychloride and the like.
  • the halogenating agent is usually used in a ratio of 1 to 10 moles per mole of compound (II-6).
  • a base can be used as necessary.
  • the base include organic bases.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (II-6).
  • a quaternary ammonium salt can be used as necessary.
  • the quaternary ammonium salt include triethylbenzylammonium chloride.
  • the quaternary ammonium salt is usually used in a ratio of 0.1 to 5 moles per mole of compound (II-6).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours.
  • Compound (II-6) can be produced by reacting a compound represented by formula (II-7) (hereinafter referred to as compound (II-7)) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (II-7) is used in place of compound (I-8).
  • Compound (II-7) can be produced by reacting a compound represented by formula (II-8) (hereinafter referred to as compound (II-8)) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 3, except that compound (II-8) is used in place of compound (I-6).
  • Compound (II-8) can be produced by reacting a compound represented by formula (II-9) (hereinafter referred to as compound (II-9)) with a compound represented by formula (Mi) (hereinafter referred to as compound (Mi)).
  • a compound represented by formula (Mi) hereinafter referred to as compound (Mi)
  • R y represents a C1-C4 alkyl group, and the other symbols have the same meanings as defined above.
  • the reaction is usually carried out in a solvent, such as alcohols, ethers, aromatic hydrocarbons, nitriles, aprotic polar solvents, halogenated hydrocarbons, and mixtures of two or more of these.
  • compound (Mi) is usually used in a ratio of 1 to 5 moles per mole of compound (II-9).
  • a base can be used as necessary.
  • the base include alkali metal alkoxides such as sodium methoxide and sodium ethoxide; alkali metal carbonates; and organic bases.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (II-9).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 24 hours.
  • the compound represented by formula (II-10) (hereinafter referred to as compound (II-10)) can be produced by reacting a compound represented by formula (II-11) (hereinafter referred to as compound (II-11)) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 3, except that compound (II-11) is used in place of compound (I-6).
  • Reference Manufacturing Method 30 Compound (II-11) can be produced by reacting a compound represented by formula (II-12) (hereinafter referred to as compound (II-12)) with compound (Mh) in the presence of an acid. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 23, except for using compound (II-12) instead of compound (II-4).
  • Compound (II-12) can be produced by reacting a compound represented by formula (II-13) (hereinafter referred to as compound (II-13)) with a hydrazine. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 24, except for using compound (II-13) instead of compound (II-5).
  • Reference Manufacturing Method 32 Compound (II-13) can be produced by reacting compound (II-8) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 25, except for using compound (II-8) instead of compound (II-6).
  • Compound (II-3A) can be produced by reacting a compound represented by formula (II-14) (hereinafter referred to as compound (II-14)) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (II-14) is used in place of compound (I-8).
  • Compound (II-14) can be produced by reacting a compound represented by formula (II-15) (hereinafter referred to as compound (II-15)) with a compound represented by formula (M-j) (hereinafter referred to as compound (M-j)).
  • Xc represents a chlorine atom, a bromine atom, or an iodine atom
  • Rz represents a C1-C3 alkyl group, and the other symbols have the same meanings as defined above.
  • the reaction is usually carried out in a solvent, such as ethers, aromatic hydrocarbons, aprotic polar solvents, halogenated hydrocarbons, and mixtures of two or more of these.
  • compound (Mj) is usually used in a ratio of 1 to 5 moles per mole of compound (II-15).
  • an acid can be used as necessary.
  • the acid include organic acids such as acetic acid and p-toluenesulfonic acid.
  • the acid is usually used in a ratio of 0.1 to 100 moles per mole of compound (II-15).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (II-14).
  • Compound (II-15) can be produced from a compound represented by formula (II-16) (hereinafter referred to as compound (II-16)).
  • PG 1 represents a 2,4,6-trimethoxyphenylmethyl group, a 2,4-dimethoxyphenylmethyl group, or a 4-methoxyphenylmethyl group, and the other symbols have the same meanings as above.
  • the reaction is usually carried out in a solvent, such as ethers, alcohols, aromatic hydrocarbons, aprotic polar solvents, halogenated hydrocarbons, water, and mixtures of two or more of these.
  • an acid can be used as necessary.
  • the acid examples include inorganic acids such as hydrochloric acid, and organic acids such as trifluoroacetic acid and p-toluenesulfonic acid.
  • the acid is usually used in a ratio of 0.1 to 100 moles per mole of compound (II-16).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 72 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (II-15).
  • Compound (II-16) can be produced by reacting a compound represented by formula (II-17) (hereinafter referred to as compound (II-17)) with a compound represented by formula (M-k) (hereinafter referred to as compound (M-k)).
  • a solvent such as ethers, aromatic hydrocarbons, aprotic polar solvents, nitriles, halogenated hydrocarbons, and mixtures of two or more of these.
  • compound (Mk) is usually used in a ratio of 1 to 5 moles per mole of compound (II-17).
  • a base can be used as necessary.
  • Examples of the base include alkali metal carbonates and organic bases.
  • the base is usually used in a ratio of 0.1 to 10 moles per mole of compound (II-17).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 48 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (II-16).
  • Reference Manufacturing Method 37 Compound (II-17) can be produced by reacting compound (II-7) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 25, except for using compound (II-7) instead of compound (II-6).
  • the compound represented by the formula (II-18) (hereinafter referred to as compound (II-18)) can be produced from compound (II-10). (In the formula, the symbols have the same meanings as defined above.)
  • the reaction can be carried out, for example, according to the method described in Green's PROTECTIVE GROUPS in ORGANIC SYNTHESIS FORTH EDITION, p. 727 or p. 750.
  • Compound (II-18) may form an acid addition salt.
  • acids that form acid addition salts include inorganic acids such as hydrochloric acid and sulfuric acid; and organic acids such as acetic acid, trifluoroacetic acid, benzoic acid, and p-toluenesulfonic acid.
  • Reference Manufacturing Method 39 Compound (II-19) can be produced by reacting compound (II-18) with compound (I-3). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 1, except that compound (II-18) is used in place of compound (I-2).
  • Reference Manufacturing Method 40 Compound (II-3) can be produced by reacting compound (II-10) with compound (IM). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 2, except that compound (II-10) is used in place of compound (I-8).
  • the compound of the present invention can be mixed or used in combination with one or more components (hereinafter referred to as the present components) selected from the group consisting of the following groups (a), (b), (c) and (d):
  • the above-mentioned mixed or concomitant use means that the compound of the present invention and the present ingredient are used simultaneously, separately or with an interval between them.
  • the compound of the present invention and this ingredient may be contained in separate preparations or may be contained in a single preparation.
  • composition A containing one or more components selected from the group consisting of Group (a), Group (b), Group (c), and Group (d) (i.e., the present components), and a compound of the present invention.
  • Group (a) includes acetylcholinesterase inhibitors (e.g., carbamate insecticides, organophosphate insecticides), GABAergic chloride channel blockers (e.g., phenylpyrazole insecticides), sodium channel modulators (e.g., pyrethroid insecticides), nicotinic acetylcholine receptor competitive modulators (e.g., neonicotinoid insecticides), nicotinic acetylcholine receptor allosteric modulators, glutamatergic chloride channel allosteric modulators (e.g., macrolide insecticides), juvenile hormone mimics, multisite inhibitors, chordotonal organ TRPV channel modulators, mite growth inhibitors, The group consists of microbial insect midgut membrane disruptors, mitochondrial ATP synthase inhibitors, oxidative phosphorylation uncouplers, nicotinic acetylcholine receptor channel blockers (e.g., ner
  • Group (b) consists of nucleic acid synthesis inhibitors (e.g., phenylamide fungicides, acylamino acid fungicides), cell division and cytoskeleton inhibitors (e.g., MBC fungicides), respiratory inhibitors (e.g., QoI fungicides, QiI fungicides), amino acid synthesis and protein synthesis inhibitors (e.g., anilinopyridine fungicides), signal transduction inhibitors, lipid synthesis and membrane synthesis inhibitors, sterol biosynthesis inhibitors (e.g., DMI fungicides such as triazoles), cell wall biosynthesis inhibitors, melanin synthesis inhibitors, plant defense inducers, multisite contact active fungicides, microbial fungicides, and other fungicidal active ingredients. These are described in the classification based on the mechanism of action of FRAC.
  • nucleic acid synthesis inhibitors e.g., phenylamide fungicides, acylamino
  • Group (c) is a group of plant growth regulators (including mycorrhizal fungi and rhizobia).
  • Group (d) is a group of repellent components.
  • alanycarb + SX means a combination of alanycarb and SX.
  • the abbreviation SX means any one of the compounds of the present invention selected from the compound group SX1 to SX1338 and the compounds of the present invention 1 to 58.
  • the present components described below are all known components and can be obtained from commercially available preparations or produced by known methods. When the present components are microorganisms, they can also be obtained from a bacterial depository institution.
  • the numbers in parentheses represent CAS RN (registered trademark).
  • Kurstaki strain EG2348 + SX Bacillus thuringiensis subsp. Kurstaki strain EG7841 + SX, Bacillus thuringiensis subsp. Kurstaki strain EVB113-19 + SX, Bacillus thuringiensis subsp. Kurstaki strain F810 + SX, Bacillus thuringiensis subsp. Kurstaki strain HD-1 + SX, Bacillus thuringiensis subsp. Kurstaki strain PB54 + SX, Bacillus thuringiensis subsp. Kurstaki strain SA-11 + SX, Bacillus thuringiensis subsp. Kurstaki strain SA-12 + SX, Bacillus thuringiensis subsp.
  • Amyloliquefaciens strain FZB24 + SX Bacillus subtilis strain Y1336 + SX, Burkholderia cepacia + SX, Burkholderia cepacia type strain Wisconsin J82 + SX, Burkholderia cepacia type Wisconsin strain M54 + SX, Candida oleophila strain O + SX, Candida saitoana + SX, Chaetomium cupreum + carotovora strain CGE234M403 + SX, Fusarium oxysporum strain Fo47 + SX, Gliocladium catenulatum strain J1446 + SX, Paenibacillus polymyxa strain AC-1 + SX, Paenibacillus polymyxa strain BS-0105 + SX, Pantoea agglomerans strain E325 + SX, Phlebiopsis gigantea strain VRA1992 + SX, Pseudomonas aureofaciens strain TX-1 + SX,
  • the ratio of the compound of the present invention to this component is not particularly limited, but examples of the ratio by weight (compound of the present invention: this component) include 1000:1 to 1:1000, 500:1 to 1:500, 100:1 to 1:100, 50:1, 20:1, 10:1, 9:1, 8:1, 7:1, 6:1, 5:1, 4:1, 3:1, 2:1, 1:1, 1:2, 1:3, 1:4, 1:5, 1:6, 1:7, 1:8, 1:9, 1:10, 1:20, and 1:50.
  • the compound of the present invention is effective against harmful arthropods such as harmful insects and harmful mites, harmful nematodes, and harmful mollusks.
  • harmful arthropods such as harmful insects and harmful mites, harmful nematodes, and harmful mollusks.
  • harmful arthropods, harmful nematodes, and harmful mollusks include the following:
  • Hemiptera Delphacids, such as Laodelphax striatellus, Nilaparvata lugens, Sogatella furcifera, Peregrinus maidis, Javesella pellucida, Perkinsiella saccharicida, Tagosodes orizicolus, and Stenocranus pacificus.
  • Aphis pomi, snow willow aphid (Aphis spiraecola), green peach aphid (Myzus persicae), strawberry aphid (Brachycaudus helichrysi), radish aphid (Brevicoryne brassicae), rosy apple aphid (Dysaphis plantaginea), false radish aphid (Lipaphis erysimi), tulip long-horn aphid (Macrosiphum euphorbiae), oats Aulacorthum solani, lettuce aphid (Nasonovia ribisnigri), wheat curl aphid (Rhopalosiphum padi), corn aphid (Rhopalosiphum maidis), citrus black aphid (Toxoptera citricida), peach buttercup aphid (Hyalopterus pruni), barnyard millet aphid (Melana
  • Aleyrodidae such as the whitefly (Pealius euryae); the family Coccinellidae, such as the palm scale insect (Abgrallaspis cyanophylli), the red scale insect (Aonidiella aurantii), the pear scale insect (Diaspidiotus perniciosus), the mulberry scale insect (Pseudaulacaspis pentagona), the Yanon scale insect (Unaspis yanonensis), and the false Yanon scale insect (Unaspis citri).
  • Lepidoptera Chilo suppressalis, Dark headed stem borer, Chilo polychrysus, White stem borer, Scirpophaga innotata, Scirpophaga incertulas, Rupela albina, Cnaphalocrocis medinalis, Marasmia patnalis, Marasmia exigua, Notarcha derogata, Ostrinia furnacalis, European corn borer, Hellula undalis, Herpetogramma luct Crambidae, such as the Japanese bush moth (Parapediasia teterrellus), the rice case worm (Nymphula depunctalis), the sugar cane borer (Diatraea saccharalis), and the eggplant fruit borer (Leucinodes orbonalis); Pyralidae, such as the corn moth (Elasmopalpus lignosellus), the Indian meal moth (Plodia interpunctella), the two-spotted moth (
  • Heliothis virescens such as Heliothis virescens, Helicoverpa spp. such as Helicoverpa armigera, corn earworm (Helicoverpa zea), Noctuidae such as Velvet bean caterpillar (Anticarsia gemmatalis), cotton leafworm (Alabama argillacea), hop wine borer (Hydraecia immanis), Pieridae such as Pieris rapae, pear fruit moth (Grapholita molesta), plum fruit moth (Grapholita dimorpha), bean cicada (Coleoptera pedunculidae), etc.
  • Heliothis virescens such as Helicoverpa armigera, corn earworm (Helicoverpa zea), Noctuidae such as Velvet bean caterpillar (Anticarsia gemmatalis), cotton leafworm (Alabama argillacea), hop wine borer (Hydraecia
  • Tortricidae such as the grass moth (Leguminivora glycinivorella), the bean pea moth (Matsumuraeses azukivora), the smaller apple tortrix moth (Adoxophyes orana fasciata), the smaller tea tortrix moth (Adoxophyes honmai), the tea tortrix moth (Homona magnima), the common tortrix moth (Archips fuscocupreanus), the codling moth (Cydia pomonella), the sugar candy moth (Tetramoera schistaceana), the bean shoot borer (Epinotia aporema), the citrus fruit borer (Citripestis sagittiferella), and the European grape wine moth (Lobesia botrana); the Gracilariidae family, such as the tea leaf moth (Caloptilia theivora) and the golden leaf moth (Phyllonorycter ringoniella); the Carposini
  • the family Plutellidae includes the diamondback moth (Plutella xylostella);
  • the family Gelechiidae includes the peach leaf moth (Anarsia lineatella), the potato leaf moth (Helcystogramma triannulella), the red cotton moth (Pectinophora gossypiella), the potato tuber moth (Pthorimaea operculella), and the tomato leaf moth (Tuta absolutea);
  • the family Arctiidae includes the fall webworm (Hyphantria cunea);
  • the family Castniidae includes the giant sugarcane borer (Telchin licus);
  • the family Cossidae includes the lesser cotton candy (Cossus insularis); the family Ascotis selenari Geometridae such as Parasa lepida; Limacodidae
  • Thysanoptera Thripidae, such as Frankliniella occidentalis, Thrips palmi, Scirtothrips dorsalis, Thrips tabaci, Frankliniella intonsa, Stenchaetothrips biformis, Echinothrips americanus, Scirtothrips perseae; Phlaeothripidae, such as Haplothrips aculeatus.
  • Diptera Anthomyiidae such as Delia platura, Delia antiqua, Pegomyia cunicularia, etc.; Ulidiidae such as Tetanops myopaeformis, etc.; Agromyza oryzae, Liriomyza sativae, Liriomyza trifolii, Chromatomyia horticola, etc.
  • Agromyzidae (Agromyzidae); Chloropidae (Chlorops oryzae), etc.; Bactrocera cucurbitae (Melon fly), Bactrocera dorsalis (Oriental fruit fly), Bactrocera latifrons (Eastern fruit fly), Bactrocera oleae (Olive fruit fly), Bactrocera tryoni (Queensland fruit fly), Ceratitis capitata (Mediterranean fruit fly), Rhagoletis pomonella (Apple maggot), Rhagoletis suzukii (Sugar apple fly), Rhagoletis japonica (Chrysocarpus japonica), Rhagoletis japonica (Rhagoletis ...
  • Tephritidae such as Hacochlaena japonica
  • Ephydridae such as Hydrellia griseola, Hydrellia philippina, and Hydrellia sasakii
  • Drosophilidae such as Drosophila suzukii and Drosophila melanogaster
  • Megaselia spiracularis Psychodidae, such as Clogmia albipunctata, Sciaridae, such as Bradysia difformis and Bradysia odoriphaga
  • Cecidomyiidae such as Mayetiola destructor and Orseolia oryzae
  • Diopsidae such as Diopsis macrophthalma
  • Glos Family Glossinidae such as Glossina sina palpalis and Glossina morsitans
  • Family Simuliidae such as Simulium japonicum and Simulium damnosum
  • Diabrotica spp. e.g. Western corn rootworm (Diabrotica virgifera virgifera), Southern corn rootworm (Diabrotica undecimpunctata howardi), Northern corn rootworm (Diabrotica barberi), Mexican corn rootworm (Diabrotica virgifera zeae), Banded cucumber beetle (Diabrotica balteata), Cucumber beetle (Diabrotica speciosa), etc.), Bean leaf beetle (Cerotoma trifurcata), Red-necked leaf beetle (Oulema melanopus), Cucumber leaf beetle (Aulacophora femoralis), Striped flea beetle (Phyllotreta striolat a), cabbage free beetle (Phyllotreta cruciferae), western black free beetle (Phyllotreta pusilla), cabbage stem free beetle (Psylliodes chry
  • fungus weevils such as Araecerus coffeee Family Anthriibidae; Family Aponidae such as sweet potato weevil (Cylas formicarius); Family Bruchidae such as Brazilian bean weevil (Zabrotes subfasciatus); Family Scolytidae such as pine bark beetle (Tomicus piniperda) and coffee berry borer (Hypothenemus hampei); Family Scolytidae such as potato weevil (Hypothenemus hampei); Bug (Euscepes postfasciatus), Alfalfa weevil (Hypera postica), Maize weevil (Sitophilus zeamais), Rice weevil (Sitophilus oryzae), Granary maize weevil (Sitophilus granarius), Rice weevil (Echinocnemus squameus), Rice water weevil (Lis
  • Aracanthus spp. such as the rust gourd weevil (Scepticus griseus), the brown gourd weevil (Scepticus uniformis), Aracanthus mourei, and the cotton root borer (Eutinobothrus brasiliensis); eum, Tribolium confusum, Alphitobius diaperinus and other Tenebrionidae; Epilachna vigintioctopunctata and other Coccinellidae; Lyctus brunneus, Rhizope rtha dominica; Ptinidae; Cerambycidae; Anoplophora malasiaca, Migdolus fryanus, Aromia bungii; Melanotus okinawensis, Brown-necked wire beetle; Elateridae, including Agriotes fuscicollis, Melanotus legatus, Anchastus spp., Conoderus spp.,
  • Hymenoptera Tenthredinidae such as Athalia rosae and Athalia japonica; Solenopsis spp. such as Solenopsis invicta and Solenopsis geminata; Atta spp.
  • Atta capiguara and Acrom yrmex spp. such as Atta capiguara and Acrom yrmex spp.), Paraponera clavata, Ochetellus glaber, Monomorium pharaonis, Argentine ant (Linepithema humile), Formica japonica, Pristomyrmex punctutus, Pheidole noda, Pheidole megacephala, Camponotus spp., such as the Japanese camponotus (Camponotus japonicus), Camponotus spp., such as the red-breasted camponotus (Camponotus obscuripes), Pogonomyrmex spp., such as Pogonomyrmex occidentalis, Wasmania spp., such as Wasmania auropunctata, and Anoplolepis gracilipinas.
  • Vespidae such as the giant hornet (Vespa mandarinia), the hairy hornet (Vespa simillima), the small hornet (Vespa analis), the red hornet (Vespa velutina), and the Japanese paper wasp (Polistes jokahamae); Siricidae (Wasps) such as the fir wasp (Urocerus gigas); and Bethylidae (Hornets).
  • Vespidae such as the giant hornet (Vespa mandarinia), the hairy hornet (Vespa simillima), the small hornet (Vespa analis), the red hornet (Vespa velutina), and the Japanese paper wasp (Polistes jokahamae); Siricidae (Wasps) such as the fir wasp (Urocerus gigas); and Bethylidae (Hornets).
  • Family Ectobiidae such as the German cockroach (Blattella germanica); Family Blattidae, such as the Siberian cockroach (Periplaneta fuliginosa), the American cockroach (Periplaneta americana), the American cockroach (Periplaneta australiae), the brown cockroach (Periplaneta brunnea), and the Asian cockroach (Blatta orientalis); Family Reticulitermes speratus, Formosan termite (Coptotermes formosanus), Formosan dry wood termite (Incisitermes minor), Formosan termite (Cryptotermes domesticus), Formosan termite (Odontotermes formosanus), and Formosan termite (Neotermes Termites of the family Termitidae, such as Glyptotermes satsumensis, Glyptotermes nakajimai, Glyptotermes fuscus,
  • Order Siphonaptera Family Pulicidae such as the human flea (Pulex irritans), cat flea (Ctenocephalides felis), dog flea (Ctenocephalides canis), rat flea (Xenopsylla cheopis), chicken flea (Echidnophaga gallinacea), etc.; Family Hectopsyllidae such as the sand flea (Tunga penetrans); Family Ceratophyllidae such as the European rat flea (Nosopsyllus fasciatus).
  • Family Pulicidae such as the human flea (Pulex irritans), cat flea (Ctenocephalides felis), dog flea (Ctenocephalides canis), rat flea (Xenopsylla cheopis), chicken flea (Echidnophaga gallinacea), etc.
  • Family Hectopsyllidae such as the sand flea (Tunga penetrans)
  • Psocodae Family Pediculidae such as head lice (Pediculus humanus capitis); Family Pthiridae such as pubic lice (Pthirus pubis); Family Haematopinidae such as cow lice (Haematopinus eurysternus) and pig lice (Haematopinus suis); Family Linognathus vituli, Sheep trunk lice Family Linognathidae, such as body lice (Linognathus ovillus) and cow lice (Solenopotes capillatus); Family Bovicoliidae, such as cow lice (Bovicola bovis), sheep lice (Bovicola ovis), Bovicola breviceps, Damalinia forficula, and Werneckiella spp.; Family Bovicoliidae, such as dog lice (T Family Trichodectidae, such as richodectes canis and Felicola subrostratus; Family Menoponi
  • Trogiidae such as Trogium pulsatorium
  • Liposcelidae or Liposcelididae such as Liposcelis corrodens, Liposcelis bostrychophila, Liposcelis pearmani, and Liposcelis entomophila.
  • Thysanura Family Lepismatidae, including the Japanese silverfish (Ctenolepisma villosa) and the European silverfish (Lepisma saccharina).
  • Eriophyidae such as Acarus carinatus, Acaphylla theavagrans, Eriophyes chibaensis, Aculus Louendali, Aceria diospyri, Aceria tosichella, Shevtchenkella sp.; Tarsonemidae, such as Polyphagotarsonemus latus; Deutzia purpurea, such as Brevipalpus phoenicis.
  • Order Araneae Family Eutichuridae such as Cheiracanthium japonicum; Family Theridiidae such as Latrodectus hasseltii.
  • Polydesmida Paradoxosomatidae, including Oxidus gracilis, Nedyopus tambanus, etc.
  • Isopoda Family Armadillidiidae, including Armadillidium vulgare.
  • Chilopoda Scutigeridae such as Thereuonema hilgendorfi; Scolopendridae such as Scolopendra subspinipes; Ethopolyidae such as Bothropolys rugosus.
  • Class Gastropoda Family Limacidae such as the brown slug (Limax marginatus) and the yellow slug (Limax flavus); Family Philomycidae such as the slug (Meghimatium bilineatum); Family Ampullariidae such as the apple snail (Pomacea canaliculata); Family Lymnaeidae such as the lymnae snail (Austropeplea ollula).
  • Nematoda Aphelenchoididae, such as Aphelenchoides besseyi; Pratylenchidae, such as Pratylenchus coffeee, Pratylenchus brachyurus, Pratylenchus neglectus, and Radopholus similis Java root-knot nematode (Meloidogyne javanica), sweet potato root-knot nematode (Meloidogyne incognita), guava root-knot nematodes (Meloidogyne enterolobii), northern root-knot nematode (Meloidogyne hapla), soybean cyst nematode (Heterodera glycines), potato cyst nematode (Globodera rostochien sis, Globodera pallida, Meloidogyne chitwoodi, etc.
  • Java root-knot nematode Java root-k
  • the harmful insects, harmful arthropods such as harmful mites, harmful mollusks, and harmful nematodes may be harmful insects, harmful arthropods such as harmful mites, harmful mollusks, and harmful nematodes that have reduced sensitivity to insecticides, acaricides, molluscicides, or nematocides, or that have developed resistance to the insecticides, acaricides, molluscicides, or nematocides.
  • the method for controlling harmful arthropods of the present invention is carried out by applying an effective amount of the compound of the present invention or composition A directly to the harmful arthropods and/or to the habitat of the harmful arthropods (plants, soil, inside a house, animals, etc.).
  • Examples of the method for controlling harmful arthropods of the present invention include foliage treatment, soil treatment, root treatment, shower treatment, fumigation treatment, water surface treatment and seed treatment.
  • the compound of the present invention or composition A is usually mixed with an inactivated carrier such as a solid carrier, a liquid carrier, or a gaseous carrier and a surfactant, and formulation auxiliary agents such as a binder, a dispersant, or a stabilizer are added as necessary to prepare an aqueous suspension preparation, an oil suspension preparation, an oil solution, an emulsion, an emulsion preparation, a microemulsion preparation, a microcapsule preparation, a wettable powder, a wettable granule, a dust, a granule, a tablet, an aerosol, a resin preparation, etc.
  • an inactivated carrier such as a solid carrier, a liquid carrier, or a gaseous carrier and a surfactant
  • formulation auxiliary agents such as a binder, a dispersant, or a stabilizer are added as necessary to prepare an aqueous suspension preparation, an oil suspension preparation, an oil solution, an emulsion, an emulsion preparation,
  • Solid carriers include, for example, clay (pyrophyllite clay, kaolin clay, etc.), talc, calcium carbonate, diatomaceous earth, zeolite, bentonite, acid clay, attapulgite, white carbon, ammonium sulfate, vermiculite, perlite, pumice, silica sand, fine powders and granules of chemical fertilizers (ammonium sulfate, ammonium phosphate, ammonium nitrate, urea, ammonium chloride, etc.), and resins (polyethylene, polypropylene, polyester, polyurethane, polyamide, polyvinyl chloride, etc.).
  • clay pyrophyllite clay, kaolin clay, etc.
  • talc calcium carbonate
  • diatomaceous earth zeolite
  • bentonite acid clay
  • attapulgite white carbon
  • ammonium sulfate vermiculite
  • perlite perlite
  • pumice pumice
  • Liquid carriers include, for example, water, alcohols (ethanol, cyclohexanol, benzyl alcohol, propylene glycol, polyethylene glycol, etc.), ketones (acetone, cyclohexanone, etc.), aromatic hydrocarbons (xylene, phenylxylylethane, methylnaphthalene, etc.), aliphatic hydrocarbons (hexane, cyclohexane, etc.), esters (ethyl acetate, methyl oleate, propylene carbonate, etc.), nitriles (acetonitrile, etc.), ethers (ethylene glycol dimethyl ether, etc.), amides (N,N-dimethylformamide, N,N-dimethyloctanamide, etc.), sulfoxides (dimethyl sulfoxide, etc.), lactams (N-methylpyrrolidone, N-octylpyrrolidone, etc.), fatty
  • Gaseous carriers include, for example, fluorocarbons, butane gas, LPG (liquefied petroleum gas), dimethyl ether, nitrogen, and carbon dioxide.
  • Surfactants include, for example, nonionic surfactants (polyoxyethylene alkyl ethers, polyoxyethylene alkylaryl ethers, polyethylene glycol fatty acid esters, etc.) and anionic surfactants (alkyl sulfonates, alkylaryl sulfonates, alkyl sulfates, etc.).
  • formulation adjuvants include binders, dispersants, colorants, and stabilizers, and specific examples include polysaccharides (starch, gum arabic, cellulose derivatives, alginic acid, etc.), lignin derivatives, synthetic water-soluble polymers (polyvinyl alcohol, polyvinylpyrrolidone, polyacrylic acids, etc.), acid isopropyl phosphate, and dibutylhydroxytoluene.
  • adjuvants can be used as components that enhance or support the efficacy of the compounds of the present invention.
  • Specific examples include Nimbus (registered trademark), Assist (registered trademark), Aureo (registered trademark), Iharol (registered trademark), Silwet L-77 (registered trademark), BreakThru (registered trademark), SundanceII (registered trademark), Induce (registered trademark), Penetrator (registered trademark), AgriDex (registered trademark), Lutensol A8 (registered trademark), NP-7 (registered trademark), Triton (registered trademark), Nufilm (registered trademark), Emulgator NP7 (registered trademark), Emulad (registered trademark), TRITON X 45 (registered trademark), AGRAL 90 (registered trademark), AGROTIN (registered trademark), ARPON (registered trademark), EnSpray N (registered trademark), and BANOLE (registered trademark).
  • plants include whole plants, stems and leaves, flowers, spikes, fruits, trunks, branches, crowns, seeds, vegetative reproductive organs, and seedlings.
  • a vegetative reproductive organ is a part of a plant, such as a root, stem, or leaf, that has the ability to grow when it is separated from the main body and placed in soil.
  • vegetative reproductive organs include tuberous roots, creeping roots, bulbs, corms (or solid bulbs), tubers, rhizomes, stolons, rhizophores, cane cuttings, propagules, and vine cuttings. Stolons are sometimes called runners, and bulbils are also called bulbils and are divided into broad buds and bulbils. Vines refer to shoots (a collective term for leaves and stems) of sweet potatoes, Chinese yams, etc. Bulbs are a collective term for bulbs, corms, tubers, rhizomes, stem fragments, rhizophores, or tuberous roots.
  • Potato cultivation begins with planting tubers in the soil, and the tubers used are generally called seed potatoes.
  • An example of a method for controlling harmful arthropods by applying an effective amount of the compound of the present invention or composition A to soil is a method of applying an effective amount of the compound of the present invention or composition A to the soil before or after planting a plant. More specifically, for example, planting hole treatment (spraying in planting holes, mixing soil for planting hole treatment), plant base treatment (spraying at the plant base, mixing soil at the plant base, irrigation at the plant base, plant base treatment in the latter half of the seedling raising period), planting furrow treatment (spraying in planting furrow, mixing soil in planting furrow), crop row treatment (spraying in crop row, mixing soil in crop row, crop row spray during the growing season), crop row treatment at the time of sowing (crop row spraying at the time of sowing, mixing soil in crop row at the time of sowing), overall treatment (overall soil spray, overall soil mixing), side row treatment, water surface treatment (water surface application, water surface application after flooding), other soil spray treatments (foliar spraying of granules during the growing season, spraying
  • irrigation treatments include (soil irrigation, seedling irrigation, chemical injection treatment, ground level irrigation, chemical drip irrigation, chemigation), seedling box treatments (seedling box spraying, seedling box irrigation, seedling box flooding with chemicals), seedling tray treatments (seedling tray spraying, seedling tray irrigation, seedling tray flooding with chemicals), seedbed treatments (seedling bed spraying, seedling bed irrigation, water seedling bed spraying, seedling immersion), bed soil mixing treatments (bed soil mixing, bed soil mixing before sowing, spraying before soil cover at sowing, spraying after soil cover at sowing, soil cover mixing), and other treatments (mixing culture soil, plowing in, mixing topsoil, mixing soil from areas that have fallen off due to rain, planting position treatment, spraying granular inflorescences, mixing paste fertilizer).
  • Examples of seed treatment include treatment of seeds or vegetative reproductive organs with the compound of the present invention or composition A. More specifically, examples of the treatment include spraying treatment in which a suspension of the compound of the present invention or composition A is misted and sprayed onto the surface of a seed or vegetative reproductive organ, smearing treatment in which the compound of the present invention or composition A is applied to the seed or vegetative reproductive organ, immersion treatment in which the seed or vegetative reproductive organ is immersed in a liquid of the compound of the present invention or composition A for a certain period of time, and a method of coating the seed or vegetative reproductive organ with a carrier containing the compound of the present invention or composition A (film coating treatment, pellet coating treatment, etc.).
  • the above-mentioned vegetative reproductive organ particularly includes seed potatoes.
  • composition A When applying composition A to seeds or vegetative reproductive organs, composition A can be applied to the seeds or vegetative reproductive organs as one formulation, or composition A can be applied to the seeds or vegetative reproductive organs in multiple separate applications as different formulations.
  • Examples of the method of applying composition A in multiple separate applications as different formulations include a method of applying a formulation containing only the compound of the present invention as an active ingredient, air-drying the seeds or vegetative reproductive organs, and then applying a formulation containing this component; and a method of applying a formulation containing the compound of the present invention and this component as active ingredients, air-drying the seeds or vegetative reproductive organs, and then applying a formulation containing this component other than the component that has already been applied.
  • the seed or vegetative reproductive organ carrying the compound of the present invention or composition A means a seed or vegetative reproductive organ having the compound of the present invention or composition A attached to its surface.
  • the seed or vegetative reproductive organ carrying the compound of the present invention or composition A may have a material other than the compound of the present invention or composition A attached thereto before or after the compound of the present invention or composition A is attached to the seed or vegetative reproductive organ.
  • the layer may consist of one or more layers.
  • each layer may contain one or more active ingredients, or each layer may consist of a layer containing one or more active ingredients and a layer containing no active ingredients. Seeds or vegetative reproductive organs carrying the compound of the present invention or composition A can be obtained, for example, by applying a formulation containing the compound of the present invention or composition A to the seeds or vegetative reproductive organs by the seed treatment methods described above.
  • the application amount is usually 1 to 10,000 g of the compound of the present invention per 10,000 m2 .
  • the compound of the present invention is usually applied in an amount of 0.001 to 100 g per 1 kg of seeds or vegetative reproductive organs.
  • the compound of the present invention or composition A is formulated as an emulsifiable concentrate, wettable powder, flowable agent, or the like, it is usually applied after diluting with water so that the active ingredient concentration is 0.01 to 10,000 ppm, and granules, dusts, and the like are usually applied as is.
  • the compound or composition A of the present invention can also be applied by wrapping the resin preparation in a sheet or string shape around the crop, stretching it near the crop, or spreading it on the soil around the base of the plant.
  • the application amount is usually 0.01 to 1000 mg of the compound of the present invention per 1 m2 of treatment area when applied on a surface, and usually 0.01 to 500 mg of the compound of the present invention per 1 m3 of treatment space when applied in a space.
  • the compound of the present invention or composition A is formulated as an emulsifiable concentrate, wettable powder, flowable agent, etc., it is usually applied after diluting with water so that the active ingredient concentration is 0.1 to 10000 ppm, and when it is an oil agent, aerosol agent, fumigation agent, poison bait, etc., it is applied as it is.
  • the compound of the present invention or composition A When the compound of the present invention or composition A is used for controlling external parasites in livestock such as cows, horses, pigs, sheep, goats, and chickens, and small animals such as dogs, cats, rats, and mice, it can be administered to animals by methods known in veterinary medicine. Specific methods of use include, for example, administration by tablet, inclusion in feed, suppository, or injection (intramuscular, subcutaneous, intravenous, intraperitoneal, etc.) for systemic inhibition, and for non-systemic inhibition, for example, spraying an oil or aqueous liquid, pour-on treatment, or spot-on treatment, washing the animal with a shampoo preparation, or attaching a resin preparation to the animal as a collar or ear tag.
  • the amount of the compound of the present invention or composition A when administered to an animal is usually in the range of 0.1 to 1000 mg per 1 kg of the animal's body weight.
  • the compound of the present invention or composition A can be used as an agent for controlling harmful arthropods in agricultural land such as fields, paddy fields, lawns, orchards, etc.
  • agricultural land such as fields, paddy fields, lawns, orchards, etc.
  • plants include the following.
  • the above plants are not particularly limited as long as they are varieties that are commonly cultivated.
  • the above plants also include plants that can be produced by natural crossbreeding, plants that can be generated by mutation, F1 hybrid plants, and genetically modified crops.
  • genetically modified crops include plants that have been given resistance to herbicides such as HPPD (4-hydroxyphenylpyruvate dioxygenase enzyme) inhibitors such as isoxaflutole, ALS (acetolactate synthase) inhibitors such as imazethapyr and thifensulfuron methyl, EPSP (5-enolpyruvylshikimate-3-phosphate synthase) inhibitors, glutamine synthetase inhibitors, PPO (protoporphyrinogen oxidase) inhibitors, bromoxynil, or dicamba; plants that are able to synthesize selective toxins known from the Bacillus genus, such as Bacillus thuringiensis; and plants that can be given specific insecticid
  • Me represents a methyl group
  • Et represents an ethyl group
  • Boc represents a tert-butoxycarbonyl group
  • Cbz represents a benzyloxycarbonyl group.
  • LCMS liquid chromatography/mass spectrometry
  • MS mass spectrometry
  • Detector LCMS-2020 (Shimadzu Corporation)
  • Ionization method DUIS method (ESI, APCI)
  • Reference Manufacturing Example 1 0.41 g of 1,1,3,3-tetramethoxypropane and 8.3 mL of acetic acid were added to 0.50 g of tert-butyl [(1S)-1-(5-amino-1H-pyrazol-3-yl)ethyl] (methyl)carbamate produced according to the method described in Example 1-1 of JP 2018-76234 A, and the mixture was stirred under heating and reflux for 3 hours. The reaction solution was allowed to cool to room temperature, and 0.46 g of N-iodosuccinimide was added and stirred for another 16 hours. The resulting mixture was poured into an ice-cooled saturated aqueous sodium hydrogen carbonate solution and extracted with chloroform.
  • the resulting organic layer was washed successively with a saturated aqueous sodium thiosulfate solution, water, and saturated saline. The resulting organic layer was dried over sodium sulfate and concentrated. To the resulting residue, 0.52 g of 2-tributylstannylpyrimidine, 0.16 g of tetrakistriphenylphosphine palladium, 0.05 g of copper (I) iodide, 0.06 g of lithium chloride, and 7.1 mL of 1,4-dioxane were added and stirred at 100°C for 12 hours. The resulting mixture was allowed to cool to room temperature, water was added, and extraction was performed using chloroform.
  • Reference Manufacturing Example 12 2.0 mL of acetic acid, 2.0 mL of chloroform, and 0.325 g of N-iodosuccinimide were added to 0.485 g of intermediate 11, and the mixture was stirred at room temperature for 5 hours. Water was added to the resulting mixture, and the mixture was extracted with chloroform. The resulting organic layer was washed successively with a saturated aqueous solution of sodium hydrogen carbonate, a saturated aqueous solution of sodium thiosulfate, water, and saturated saline. The resulting organic layer was dried over sodium sulfate, filtered, and concentrated. The residue was subjected to silica gel column chromatography to obtain 0.500 g of intermediate 12 represented by the following formula.
  • Reference Manufacturing Example 13-1 293 mL of acetonitrile, 61.3 mL of triethylamine, and 55.9 g of magnesium chloride were added to 18.7 g of cyanoacetic acid in this order, and the mixture was stirred at room temperature for 23 hours to obtain mixture A. 28.5 g of 1,1'-carbonyldiimidazole and 3.58 g of 4-dimethylaminopyridine were added to a mixture of 34.8 g of N-methyl-N-(phenylmethoxycarbonyl)-L-alanine and 200 mL of THF in this order, and the mixture was stirred at room temperature for 4 hours to obtain mixture B.
  • Reference Production Example 18 The compound and its physical properties produced according to Reference Production Example 14 are shown below, except that acetylacetone was used instead of 1,1,3,3-tetramethoxypropane.
  • Intermediate 18 1 H-NMR (CDCl 3 ) ⁇ : 7.39-7.31 (5H, m), 6.52 (1H, s), 6.41 (1H, s), 5.78-5.65 (1H, m), 5.21 (2H, s), 2.79 (3H, s), 2.70 (3H, s), 2.54 (3H, s), 1.62 (3H, d).
  • Reference Production Example 20 A compound produced according to Reference Production Example 14 using 1,1,3,3-tetraethoxy-2-methylpropane instead of 1,1,3,3-tetramethoxypropane and its physical properties are shown below.
  • Intermediate 20 1 H-NMR (CDCl 3 ) ⁇ : 8.42 (1H, s), 8.33 (1H, d), 7.39-7.32 (5H, m), 6.52-6.47 (1H, m), 5.77-5.70 (1H, m), 5.21 (2H, s), 2.77 (3H, s), 2.36 (3H, s), 1.62 (3H, d).
  • Reference Production Example 45 The compound prepared according to Reference Production Example 4 using Intermediate 56 instead of Intermediate 3 and its physical properties are shown below.
  • Intermediate 57 1 H-NMR (CDCl 3 ) ⁇ : 9.45 (1H, s), 9.01 (2H, d), 8.46 (1H, s), 7.43 (1H, t), 7.33-7.31 (5H, m), 5.82 (1H, d), 5.38-5.37 (1H, m), 5.05-4.99 (2H, m), 1.57 (3H, d).
  • Reference Production Example 49 8.4 mL of hydrogen chloride (5-10 wt % methanol solution) was added to 0.50 g of intermediate 60, and the mixture was stirred at 90° C. for 15 hours. The resulting mixture was allowed to cool to room temperature and then concentrated, and 4.2 mL of DMF, 4.2 mL of bromoacetaldehyde dimethyl acetal, and 1.0 mL of acetic acid were added, and the mixture was stirred at 80° C. for 15 hours. Water was added to the resulting mixture, and the mixture was extracted with ethyl acetate. The resulting organic layer was washed with water and saturated saline in that order. The resulting organic layer was dried over sodium sulfate, filtered, and concentrated.
  • hydrogen chloride 5-10 wt % methanol solution
  • Reference Manufacturing Example 50 The compound prepared according to Reference Production Example 4 using Intermediate 61 instead of Intermediate 3 and its physical properties are shown below.
  • Intermediate 62 1 H-NMR (CDCl 3 ) ⁇ : 8.98 (2H, d), 7.72 (1H, d), 7.54 (1H, d), 7.37-7.37 (1H, m), 7.34-7.31 (5H, m), 6.00 (1H, d), 5.14-5.13 (1H, m), 5.05-5.03 (2H, m), 2.86 (3H, s), 1.49 (3H, d).
  • Reference Production Example 52 The compound and its physical properties are shown below, which were produced according to Reference Production Example 4, except that Intermediate 63 was used instead of Intermediate 3, and tributyl(1-ethoxyvinyl)stannane was used instead of 2-tributylstannylpyrimidine.
  • Intermediate 64 1 H-NMR (CDCl 3 ) ⁇ : 9.41 (1H, s), 8.44 (1H, s), 8.25 (2H, s), 8.02 (1H, s), 7.30 (1H, d), 5.87-5.84 (1H, m), 4.87 (1H, d), 4.81 (1H, d), 4.13-4.09 (2H, m), 1.64 (3H, d), 1.45 (3H, t).
  • Reference Manufacturing Example 66 A mixture of 0.30 g of Intermediate 66 and 5.0 mL of a hydrogen chloride/1,4-dioxane solution (4 mol/L) was stirred at room temperature for 15 hours, and the resulting mixture was concentrated. To a mixed solution of the obtained residue and 5.0 mL of THF, 0.37 mL of triethylamine and 0.27 mL of 3,5-bis(trifluoromethyl)benzoyl chloride were added in that order, and the mixture was stirred at room temperature for 1 hour. Water was added to the obtained mixture, and the mixture was extracted with ethyl acetate. The obtained organic layer was washed with water and saturated saline in that order.
  • Production Example 6 2.9 mL of THF, 2.3 ⁇ L of DMF, and 0.061 mL of oxalyl chloride were added to 0.165 g of 3,5-bis(difluoromethoxy)benzoic acid in this order, and the mixture was stirred at room temperature for 1 hour. The resulting mixture was concentrated, and 0.5 mL of THF was added to the residue to obtain mixture C. Mixture C was added to a mixture of 0.15 g of intermediate 17, 0.164 mL of triethylamine, and 1.2 mL of THF, and the mixture was stirred at room temperature for 1 hour. Water was added to the resulting mixture, and the mixture was extracted with chloroform.
  • Production Example 9 A compound produced according to Production Example 2 using Intermediate 36 instead of Intermediate 6 and its physical properties are shown below.
  • Production Example 15-1 A compound prepared according to Preparation Example 15 using 2-tributylstannylpyridine instead of 2-tributylstannylthiazole and its physical properties are shown below.
  • Compound 40 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 9.47 (1H, s), 8.85-8.84 (1H, m), 8.45 (1H, s), 8.22 (2H, s), 8.01-8.00 (2H, m), 7.97-7.96 (1H, m), 7.51 (1H, d), 7.47-7.46 (1H, m), 5.80-5.77 (1H, m), 1.67 (3H, d).
  • Production Example 17 A mixture of 0.20 g of the present compound 41, 0.10 g of methoxyamine hydrochloride, 0.074 g of sodium acetate, and 4.5 mL of ethanol was stirred at 50° C. for 3 hours. The resulting mixture was allowed to cool to room temperature, water was added, and extraction was performed using ethyl acetate. The resulting organic layer was washed successively with water and saturated saline. The resulting organic layer was dried over sodium sulfate, filtered, and concentrated. The residue was subjected to silica gel column chromatography to obtain 0.20 g of the present compound 42.
  • Production Example 17-1 A compound prepared according to Preparation Example 17 using hydroxylamine hydrochloride instead of methoxyamine hydrochloride and its physical properties are shown below.
  • Compound 43 of the present invention 1 H-NMR (DMSO-D 6 ) ⁇ : 9.30 (1H, d), 9.20 (1H, s), 8.80 (1H, s), 8.45 (2H, s), 8.30 (1H, s), 5.16 (1H, s), 2.29 (3H, s), 1.50 (3H, d).
  • Formula (L-1) (hereinafter, referred to as compound (L-1)), in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T1-1 (# 4 represents the bonding site to the carbon atom of the carbonyl group), and R 2 is any of the substituents described in [Table L1] to [Table L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX1).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX2).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX3).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX4).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX5).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX6).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX8).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX9).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX10).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX11).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX12).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX14).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX15).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX16).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX18).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX19).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX20).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX21).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX22).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX23).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX24).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX26).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX27).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX28).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX29).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX30).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX31).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX32).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX33).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX34).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX35).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX36).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX37).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX38).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX39).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX40).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX41).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX42).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX43).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX44).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX45).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX46).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX47).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX48).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX49).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX50).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX51).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX52).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX53).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX54).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX55).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX56).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX57).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX58).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX59).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX60).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX61).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX62).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX63).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX64).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX65).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX66).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX67).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX68).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX69).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX70).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX71).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX72).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX73).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX74).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX75).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX76).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX77).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX78).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX79).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX80).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX81).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX82).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX83).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX84).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX85).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX86).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX87).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX88).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX89).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX90).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX91).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX92).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX93).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX94).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX95).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX96).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX97).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX98).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX99).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX100).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX101).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX102).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX103).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX104).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX105).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX106).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX107).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX108).
  • Formula (L-2) (hereinafter, referred to as compound (L-2)), in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T1-1 (# 4 represents a bonding site to the carbon atom of the carbonyl group), and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents a bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX109).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX110).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX111).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX112).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX113).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX114).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX115).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX116).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX117).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX118).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX119).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX120).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX121).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX122).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX123).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX124).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX125).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX126).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX127).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX128).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX129).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX130).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX131).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX132).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX133).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX134).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX135).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX136).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX137).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX138).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX139).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX140).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX141).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX142).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX143).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX144).
  • compound group SX145 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX145).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX146).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX147).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX148).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX149).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX150).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX151).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX152).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX153).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX154).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX155).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX156).
  • compound group SX157 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX157).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX158).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX159).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX160).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX161).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX162).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX163).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX164).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX165).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX166).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX167).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX168).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX169).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX170).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX171).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX172).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX173).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX174).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX175).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX176).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX177).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX178).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX179).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX180).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX181).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX182).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX183).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX184).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX185).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX186).
  • compound group SX187 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX187).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX188).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX189).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX190).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX191).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX192).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX193).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX194).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX195).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX196).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX197).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX198).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX199).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX200).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX201).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX202).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX203).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX204).
  • compound group SX205 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX205).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX206).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX207).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX208).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX209).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX210).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX211).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX212).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX213).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX214).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX215).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX216).
  • Formula (L-3) (hereinafter, referred to as compound (L-3)), in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T1-1 (# 4 represents the bonding site to the carbon atom of the carbonyl group), and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX217).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX218).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX219).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX220).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX221).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX222).
  • compound group SX222 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX223).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX224).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX225).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX226).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX227).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX228).
  • compound group SX229 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX229).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX230).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX231).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX232).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX233).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX234)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX235).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX236).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX237).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX238).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX239).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX240).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX241).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX242).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX243).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX244)
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX245).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX246).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX247).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX248).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX249).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX250).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX251).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX252).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX253).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX254)
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX255).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX256).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX257).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX258).
  • compound group SX259 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX259).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX260).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX261).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX262).
  • compound group SX263 a compound in which R 1 is a hydrogen atom, R 10 is an ethyl group, R 11 is T1-8, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX263).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX264).
  • compound group SX264 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX265).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX266).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX267).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX268).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX269).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX270).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX271).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX272).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX273).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX274)
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX275).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX278).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX279).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX280).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX281).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX282).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX283).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX284)
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX285).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX286).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX287).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX290).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX291).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX300).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX301).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX302).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX303).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX306).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX307).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX308).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX309).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX310).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX311).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX312).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX313).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX314).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX315).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX316).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX317).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX320).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX321).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX326).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX327).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX332).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX333).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX336).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX337).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX338).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX339).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX340).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX341).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX342).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX343).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX344)
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX345).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX348).
  • compound group SX349 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX349).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX352).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX353).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX358).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX359).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX360).
  • compound group SX361 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX361).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX362).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX363).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX364)
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX365).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX370).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX371).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX372).
  • compound group SX373 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX373).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX374)
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX375).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX378).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX379).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX380).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX381).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX382).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX383).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX384)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX385).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX388).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX389).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX390).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX391).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX392).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX393).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX394)
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX395).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX396).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX397).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX398).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX399).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX400).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX401).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX406).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX407).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX412).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX413).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX414)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX415).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX418).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX419).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX420).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX421).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX422).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX423).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX428).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX429).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX436).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX437).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX438).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX439).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX440).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX441).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX442).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX443).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX444)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX445).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX446).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX447).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX448).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX449).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX458).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX459).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX460).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX461).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX464).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX465).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX466).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX467).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX472).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX473).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX474).
  • compound group SX475 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX475).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX476).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX477).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX478).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX479).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX482).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX483).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX484)
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX485).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX490).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-10
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX491).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX500).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX501).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX502).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX503).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX504)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX505).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX508).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX509).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX512).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX513).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX514)
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX515).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX518).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX519).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX520).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX521).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX522).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX523).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX528).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX529).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX532).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX533).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX534)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX535).
  • Formula (L-6) (hereinafter, referred to as compound (L-6)), in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T1-1 (# 4 represents a bonding site to the carbon atom of the carbonyl group), and R 2 is any of the substituents described in [Table L1] to [Table L20] (# 3 represents a bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX541).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX546)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX547).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX548).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX549).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX562).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX563).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX566)
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX567).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX570).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX571).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX572).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX573).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX582).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX583).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX588).
  • compound group SX589 a compound in which R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX589).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX590).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX591).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX592).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX593).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX604).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX605).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-11
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX606).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX607).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX608).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX609).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX610).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX611).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX612).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX613).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX618).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX619).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX620).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX621).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX622).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX623).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX628).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX629).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX632).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX633).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX634)
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX635).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX640).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX641).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX642).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-18
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX643).
  • R 1 is a hydrogen atom
  • R 11 is T2-3, and R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX653).
  • R 1 is a methyl group
  • R 11 is T2-3, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX654).
  • compound SX655 is any of the substituents described in [Tables L1] to [Tables L20].
  • R 1 is a methyl group, R 11 is T2-4, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX656).
  • R 1 is a hydrogen atom, R 11 is T2-5, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX657).
  • R 1 is a methyl group, R 11 is T2-5, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX658).
  • R 1 is a hydrogen atom
  • R 11 is T2-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX661).
  • R 1 is a methyl group
  • R 11 is T2-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX662).
  • R 1 is a hydrogen atom
  • R 11 is T2-8, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX663).
  • R 1 is a methyl group
  • R 11 is T2-8, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX664).
  • R 1 is a hydrogen atom
  • R 11 is T2-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX665).
  • R 1 is a methyl group
  • R 11 is T2-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX666).
  • R 1 is a hydrogen atom
  • R 11 is T2-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX667).
  • R 1 is a methyl group
  • R 11 is T2-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX668).
  • R 1 is a hydrogen atom
  • R 11 is T2-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX669).
  • R 1 is a methyl group, R 11 is T2-11, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX670).
  • R 1 is a hydrogen atom
  • R 11 is T2-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX671).
  • R 1 is a methyl group
  • R 11 is T2-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX672).
  • R 1 is a methyl group
  • R 11 is T2-14, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX676).
  • R 1 is a hydrogen atom
  • R 11 is T2-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX677).
  • R 1 is a methyl group
  • R 11 is T2-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX678).
  • Formula (L-8) (hereinafter, referred to as compound (L-8)), in which R 1 is a hydrogen atom, R 11 is T2-1 (# 5 represents a bonding site to the nitrogen atom), and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents a bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX683).
  • R 1 is a methyl group, R 11 is T2-1, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX684).
  • R 1 is a hydrogen atom, R 11 is T2-2, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX685).
  • R 1 is a methyl group, R 11 is T2-2, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX686).
  • compound (L-8) a compound in which R 1 is a hydrogen atom, R 11 is T2-3, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX687).
  • R 1 is a methyl group
  • R 11 is T2-3, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX688).
  • R 1 is a hydrogen atom
  • R 11 is T2-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX689).
  • R 1 is a methyl group
  • R 11 is T2-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX690).
  • R 1 is a hydrogen atom
  • R 11 is T2-5
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX691).
  • R 1 is a hydrogen atom
  • R 11 is T2-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX695).
  • R 1 is a methyl group
  • R 11 is T2-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX696).
  • R 1 is a hydrogen atom
  • R 11 is T2-8, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX697).
  • R 1 is a methyl group
  • R 11 is T2-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX704).
  • compound group SX704 a compound in which R 1 is a hydrogen atom
  • R 11 is T2-12
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX705)
  • R 1 is a methyl group
  • R 11 is T2-12
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX706).
  • R 1 is a hydrogen atom
  • R 11 is T2-14, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX709).
  • R 1 is a methyl group
  • R 11 is T2-14, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX710).
  • R 1 is a hydrogen atom
  • R 11 is T2-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX711).
  • R 1 is a methyl group
  • R 11 is T2-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX718).
  • R 1 is a hydrogen atom
  • R 11 is T2-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX719).
  • R 1 is a methyl group
  • R 11 is T2-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX720).
  • R 1 is a hydrogen atom
  • R 11 is T2-3, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX721).
  • R 1 is a methyl group
  • R 11 is T2-3, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX722).
  • R 1 is a hydrogen atom
  • R 11 is T2-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX723).
  • R 1 is a methyl group
  • R 11 is T2-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX724).
  • compound group SX725 a compound in which R 1 is a hydrogen atom, R 11 is T2-5, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX725).
  • R 1 is a methyl group
  • R 11 is T2-14, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX744).
  • R 1 is a hydrogen atom
  • R 11 is T2-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX745).
  • R 1 is a methyl group
  • R 11 is T2-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX746).
  • R 1 is a methyl group
  • R 11 is T2-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX752).
  • R 1 is a hydrogen atom
  • R 11 is T2-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX753).
  • R 1 is a methyl group
  • R 11 is T2-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX754).
  • compound (L-10) a compound in which R 1 is a hydrogen atom, R 11 is T2-4, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX757).
  • compound (L-10) R 1 is a methyl group, R 11 is T2-4, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX758).
  • R 1 is a hydrogen atom
  • R 11 is T2-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX767).
  • R 1 is a methyl group
  • R 11 is T2-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX768).
  • R 1 is a hydrogen atom
  • R 11 is T2-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX769).
  • compound (L-10) a compound in which R 1 is a hydrogen atom, R 11 is T2-15, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX779).
  • R 1 is a methyl group
  • R 11 is T2-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX780).
  • R 1 is a hydrogen atom
  • R 11 is T2-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX781).
  • R 1 is a methyl group
  • R 11 is T2-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX782).
  • R 1 is a hydrogen atom
  • R 11 is T2-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX783).
  • Formula (L-11) (hereinafter, referred to as compound (L-11)), in which R 1 is a hydrogen atom, R 11 is T2-1 (# 5 represents a bonding site to the nitrogen atom), and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents a bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX785).
  • R 1 is a methyl group, R 11 is T2-1, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX786).
  • R 1 is a hydrogen atom, R 11 is T2-2, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX787).
  • R 1 is a methyl group, R 11 is T2-2, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX788).
  • R 1 is a hydrogen atom
  • R 11 is T2-6, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX795).
  • R 1 is a methyl group
  • R 11 is T2-6, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX796).
  • R 1 is a hydrogen atom
  • R 11 is T2-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX797).
  • R 1 is a hydrogen atom
  • R 11 is T2-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX801).
  • R 1 is a methyl group
  • R 11 is T2-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX802).
  • R 1 is a hydrogen atom
  • R 11 is T2-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX803).
  • R 1 is a methyl group
  • R 11 is T2-13
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX810).
  • R 1 is a hydrogen atom
  • R 11 is T2-14
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX811).
  • R 1 is a methyl group
  • R 1 is a hydrogen atom
  • R 11 is T2-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX813).
  • R 1 is a methyl group
  • R 11 is T2-15
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX814).
  • R 1 is a hydrogen atom
  • R 11 is T2-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX815).
  • R 1 is a methyl group
  • R 11 is T2-16
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX816).
  • R 1 is a hydrogen atom
  • R 11 is T2-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX817).
  • R 1 is a methyl group
  • R 11 is T2-17
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX818).
  • R 1 is a methyl group
  • R 11 is T2-10
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX838).
  • R 1 is a hydrogen atom
  • R 11 is T2-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX839).
  • R 1 is a methyl group
  • R 11 is T2-11
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX840).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-1
  • # 6 represents the bonding site to the carbon atom of the carbonyl group
  • R 2 is any of the substituents described in [Table L1] to [Table L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX853).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX860).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX861).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX864)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX865).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX868).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX869).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX872).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX873).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX874)
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX875).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX878).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX879).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX880).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX881).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX882).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX883).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX890).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX891).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX896).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX897).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX898).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX899).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX900).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX901).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX913).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX914).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX933).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX934).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX935)
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX936).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX949).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX950).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX953).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX954).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX965)
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX966).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX967).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX968).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX971).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX972).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX973).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX974).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX975).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX976).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX977).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX978).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX985)
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX986).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX987).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX988).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX991).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX992).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX993).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX994).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX997).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX998).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1001).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1002).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1007).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1008).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1011).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1012).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1017).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1018).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1021).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1022).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1023).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1024).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1031).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1032).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1037).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1038).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1041).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1042).
  • compound (L-4) a compound in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T3-6, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1045).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1046).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1049).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1050).
  • compound (L-4) a compound in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T3-7, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1051).
  • compound group SX1052 a compound in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T3-7, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1052).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1055)
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1056).
  • compound (L-4) a compound in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T3-8, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1057).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1058).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1059).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1060).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1065).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1066).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1071).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1072).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1075).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1076).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1077).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1078).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1079).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1080).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1095)
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1096).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1097).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1098).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1101).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1102).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1107).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1108).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1113).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1114).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1115)
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1116).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-1
  • # 6 represents the bonding site to the carbon atom of the carbonyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX1123).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1124).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1129).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1130).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1139).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1140).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1141).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1142).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1147).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1148).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1149).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1150).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1153).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1154).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1155).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1156).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1157).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1158).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1159).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1160).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1167).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1168).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1169).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1170).
  • compound (L-6) a compound in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T3-9, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1171).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1172).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1173).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1174).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1175)
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T3-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1176).
  • Formula (L-13) (hereinafter, referred to as compound (L-13)), in which R 1 is a hydrogen atom, R 10 is a hydrogen atom, R 11 is T1-1 (# 4 represents the bonding site to the carbon atom of the carbonyl group), and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX1177).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1178).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1179).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1180).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-1
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1181).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1184).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1185).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1186).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-2
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1187).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1190).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1191).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1192).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1193).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-3
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1194).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1195).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-4
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1200).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1201).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-5
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1206).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1207).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1208).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1209).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-6
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1212).
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1213).
  • R 1 is a methyl group
  • R 10 is a hydrogen atom
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1214).
  • R 1 is a hydrogen atom
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1215).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1216).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-7
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1217).
  • R 1 is a methyl group
  • R 10 is a methyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1222).
  • R 1 is a hydrogen atom
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1223).
  • R 1 is a methyl group
  • R 10 is an ethyl group
  • R 11 is T1-8
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1224)
  • R 1 is a hydrogen atom
  • R 10 is a hydrogen atom
  • R 11 is T1-9
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1225).

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Organic Chemistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Insects & Arthropods (AREA)
  • Dentistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Public Health (AREA)
  • Toxicology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Botany (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne un composé ayant un excellent effet de lutte contre les arthropodes nuisibles. L'invention concerne un composé représenté par la formule (I) [dans laquelle L représente une liaison simple, ou similaire ; R1 représente un groupe hydrocarboné linéaire en C1-C6, ou similaire ; R2 représente un groupe hétérocyclique aromatique à 5 ou 6 chaînons, ou similaire ; X représente NR11C(Z)R12, ou similaire ; Z représente un atome d'oxygène, ou similaire ; R11 représente un groupe hydrocarboné linéaire en C1-C6, ou similaire ; R12 représente un groupe phényle qui peut être substitué par un ou plusieurs substituants, ou similaire ; et Q représente un groupe représenté par la formule A1 (dans laquelle # représente une position de liaison à 2, et ● représente une position de liaison à un atome de carbone)] ou un N-oxyde de celui-ci qui a un excellent effet de lutte contre les arthropodes nuisibles.
PCT/JP2024/036248 2023-10-12 2024-10-10 Composé cyclique condensé et composition de lutte contre les arthropodes nuisibles le contenant Pending WO2025079634A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2023176517 2023-10-12
JP2023-176517 2023-10-12

Publications (1)

Publication Number Publication Date
WO2025079634A1 true WO2025079634A1 (fr) 2025-04-17

Family

ID=95395760

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2024/036248 Pending WO2025079634A1 (fr) 2023-10-12 2024-10-10 Composé cyclique condensé et composition de lutte contre les arthropodes nuisibles le contenant

Country Status (1)

Country Link
WO (1) WO2025079634A1 (fr)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014200882A1 (fr) * 2013-06-11 2014-12-18 Janssen Pharmaceutica Nv Inhibiteurs de pde10a pour le traitement du diabète de type ii
WO2016148145A1 (fr) * 2015-03-16 2016-09-22 大正製薬株式会社 COMPOSÉ DE PYRAZOLO [1,5-a] PYRIMIDINE
WO2022233777A1 (fr) * 2021-05-06 2022-11-10 Bayer Aktiengesellschaft Imidazoles annelés substitués par alkylamide et leur utilisation comme insecticides

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014200882A1 (fr) * 2013-06-11 2014-12-18 Janssen Pharmaceutica Nv Inhibiteurs de pde10a pour le traitement du diabète de type ii
WO2016148145A1 (fr) * 2015-03-16 2016-09-22 大正製薬株式会社 COMPOSÉ DE PYRAZOLO [1,5-a] PYRIMIDINE
WO2022233777A1 (fr) * 2021-05-06 2022-11-10 Bayer Aktiengesellschaft Imidazoles annelés substitués par alkylamide et leur utilisation comme insecticides

Similar Documents

Publication Publication Date Title
JP7442463B2 (ja) 複素環化合物及びそれを含有する有害節足動物防除組成物
JP7667745B2 (ja) 複素環化合物及びそれを含有する有害節足動物防除組成物
WO2019131575A1 (fr) Composé hétérocyclique, et agent de lutte contre des arthropodes nuisibles comprenant celui-ci
JP7492946B2 (ja) 複素環化合物及びそれを含有する有害節足動物防除組成物
JP7253498B2 (ja) 複素環化合物及びそれを含有する有害節足動物防除剤
JP7675087B2 (ja) 複素環化合物及びそれを含有する有害節足動物防除組成物
JP7301042B2 (ja) 複素環化合物及びそれを含有する有害節足動物防除組成物
US20240228472A1 (en) Heterocyclic compound and harmful-arthropod-controlling composition containing same
JP7704770B2 (ja) 複素環化合物及びそれを含有する有害節足動物防除組成物
JP7428693B2 (ja) エーテル化合物及びそれを含有する有害節足動物防除組成物
JP7489564B1 (ja) ２－（５－シクロプロピル－３－（エチルスルホニル）ピリジン－２－イル）－５－（（トリフルオロメチル）スルフィニル）ベンゾ［ｄ］オキサゾールの結晶
JP7489565B1 (ja) ２－（５－シクロプロピル－３－（エチルスルホニル）ピリジン－２－イル）－５－（（トリフルオロメチル）スルホニル）ベンゾ［ｄ］オキサゾールの結晶
WO2024096093A1 (fr) Composé hétérocyclique et composition de lutte contre les arthropodes nuisibles le contenant
WO2025079634A1 (fr) Composé cyclique condensé et composition de lutte contre les arthropodes nuisibles le contenant
WO2025089403A1 (fr) Composé hétérocyclique et composition de lutte contre les arthropodes nuisibles le contenant
WO2024080330A1 (fr) Composé de sulfonamide et composition de lutte contre les arthropodes nuisibles le contenant
WO2025079605A1 (fr) Composé hétérocyclique et composition de lutte contre les arthropodes nuisibles le contenant
WO2024080354A1 (fr) Composé de sulfonamide et composition de lutte contre les arthropodes nuisibles le contenant
WO2024071393A1 (fr) Composé hétérocyclique et composition de lutte contre les arthropodes nuisibles le contenant
WO2024122450A1 (fr) Composé amide et composition de lutte contre les arthropodes nuisibles le contenant
WO2024248015A1 (fr) Composé hétérocyclique et composition de lutte contre les arthropodes nuisibles le contenant
WO2024080355A1 (fr) Composition de sulfonamide et composition de lutte contre les arthropodes nuisibles la contenant
WO2024147306A1 (fr) Composé amide et composition de lutte contre les arthropodes nuisibles le contenant
WO2024071219A1 (fr) Composé de sulfonamide et composition pour l'extermination d'arthropodes nuisibles le contenant

Legal Events

Date Code Title Description
121 Ep: the epo has been informed by wipo that ep was designated in this application

Ref document number: 24877228

Country of ref document: EP

Kind code of ref document: A1