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WO2025079605A1 - Composé hétérocyclique et composition de lutte contre les arthropodes nuisibles le contenant - Google Patents

Composé hétérocyclique et composition de lutte contre les arthropodes nuisibles le contenant Download PDF

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Publication number
WO2025079605A1
WO2025079605A1 PCT/JP2024/036103 JP2024036103W WO2025079605A1 WO 2025079605 A1 WO2025079605 A1 WO 2025079605A1 JP 2024036103 W JP2024036103 W JP 2024036103W WO 2025079605 A1 WO2025079605 A1 WO 2025079605A1
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group
optionally substituted
substituents selected
halogen atoms
substituted
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Japanese (ja)
Inventor
裕人 小幡
晃一郎 土田
佑介 南波
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Sumitomo Chemical Co Ltd
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Sumitomo Chemical Co Ltd
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01M—CATCHING, TRAPPING OR SCARING OF ANIMALS; APPARATUS FOR THE DESTRUCTION OF NOXIOUS ANIMALS OR NOXIOUS PLANTS
    • A01M1/00—Stationary means for catching or killing insects
    • A01M1/20—Poisoning, narcotising, or burning insects
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N65/00—Biocides, pest repellants or attractants, or plant growth regulators containing material from algae, lichens, bryophyta, multi-cellular fungi or plants, or extracts thereof
    • A01N65/08—Magnoliopsida [dicotyledons]
    • A01N65/12—Asteraceae or Compositae [Aster or Sunflower family], e.g. daisy, pyrethrum, artichoke, lettuce, sunflower, wormwood or tarragon
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/02—Acaricides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/04—Insecticides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56—One oxygen atom and one sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Definitions

  • Patent Document 1 describes that certain heterocyclic compounds are useful for treating inflammatory and immune diseases.
  • the present invention aims to provide a compound that has excellent control effect against harmful arthropods.
  • Formula (I) [Wherein, Z represents an oxygen atom or a sulfur atom; L represents a single bond or --(CR 4a R 4b ) n --; R 4a and R 4b are the same or different and represent a C1-C6 chain hydrocarbon group optionally substituted with one or more halogen atoms, a C3-C6 cycloalkyl group optionally substituted with one or more halogen atoms, a C1-C6 alkoxy group optionally substituted with one or more halogen atoms, a cyano group, a hydroxyl group, a halogen atom, or a hydrogen atom; n represents 1, 2, 3, 4, 5, or 6; R 1 represents a C1-C6 chain hydrocarbon group optionally substituted
  • Group A C1-C6 chain hydrocarbon group ⁇ the C1-C6 chain hydrocarbon group may be substituted with one or more substituents selected from the group consisting of a C3-C6 cycloalkyl group optionally substituted with one or more halogen atoms, a cyano group, and a halogen atom ⁇
  • a C3-C6 cycloalkyl group ⁇ the C3-C6 cycloalkyl group may be substituted with one or more substituents selected from the group consisting of a C1-C6 alkoxy group, a cyano group, and a halogen atom ⁇
  • a phenyl group optionally substituted with one or more substituents selected from Group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted with one or more substituents selected from Group B, OR 3a , SF 5 , NR 3d OR 3b , NR 3b1 C(O)R 3c1 , NR 3
  • Group C a C3-C6 cycloalkyl group optionally substituted by one or more substituents selected from group E, a phenyl group optionally substituted by one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted by one or more substituents selected from group B, OR 3a , NR 3d OR 3b , NR 3b C(O)R 3c , NR 3d NR 3b C(O)R 3c , NR 3b C(O)OR 3e , NR 3d NR 3b C(O)OR 3e , NR 3b C(O ) NR 3f R 3g , NR 3d NR 3b C(O)NR 3f R 3g , N ⁇ S(O) p R 3h R 3i , C(O)R 3c , C(O) OR the group consisting of C(O)NR 3f R 3g , S(O) m R 3k ,
  • Group F a group consisting of a C3-C6 cycloalkyl group optionally substituted by one or more substituents selected from group E, a phenyl group optionally substituted by one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted by one or more substituents selected from group B, OR 3a , S(O) mR 3k , C(O)R 3c , C(O)OR 3j , C(O)NR 3fR 3g , NR 3bR 3c , NR 3bC (O)R 3c , NR 3bC (O)NR 3fR 3g , N ⁇ S(O) pR 3hR 3i , a 3- to 6-membered non-aromatic heterocyclic group, a cyano group , and a halogen atom.
  • Group G a C3-C6 cycloalkyl group optionally substituted by one or more substituents selected from group E, a phenyl group optionally substituted by one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted by one or more substituents selected from group B, OR 3a , NR 3d OR 3b , NR 3b C(O)R 3c , NR 3d NR 3b C(O)R 3c , NR 3b C(O)OR 3e , NR 3d NR 3b C(O)OR 3e , NR 3b C(O ) NR 3f R 3g , NR 3d NR 3b C(O)NR 3f R 3g , N ⁇ S(O) p R 3h R 3i , C(O)R 3c , C(O) OR 3j , C(O)NR 3f R 3g , S(O) m R 3k ,
  • a harmful arthropod control composition comprising the compound according to any one of [1] to [4] or an N-oxide thereof and an inert carrier.
  • a composition comprising one or more components selected from the group consisting of group (a), group (b), group (c), and group (d), and a compound or an N-oxide thereof according to any one of [1] to [4]: Group (a): A group consisting of insecticidal active ingredients, acaricidal active ingredients and nematicidal active ingredients; Group (b): bactericidal active ingredient; Group (c): plant growth regulating ingredients; Group (d): repellent components.
  • the present invention makes it possible to control harmful arthropods.
  • Compound N of the present invention may form an acid addition salt.
  • acids that form acid addition salts include inorganic acids such as hydrogen chloride, phosphoric acid, and sulfuric acid, and organic acids such as acetic acid, trifluoroacetic acid, benzoic acid, and p-toluenesulfonic acid. Acid addition salts can be obtained, for example, by mixing compound N of the present invention with an acid.
  • R 3 is a C1-C3 open chain hydrocarbon group ⁇ the C1-C3 open chain hydrocarbon group is optionally substituted with one or more substituents selected from the group consisting of a C1-C3 alkoxy group optionally substituted with one or more halogen atoms, a C3-C6 cycloalkyl group optionally substituted with one or more halogen atoms or cyano groups, a phenyl group optionally substituted with one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group optionally substituted with one or more substituents selected from group B, a 3- to 6-membered non-aromatic heterocyclic group, a cyano group, and a halogen atom ⁇ , C(O)R 5 , a cyclopropyl group optionally substituted with one or more halogen atoms or cyano groups, or a hydrogen atom, and R 5 is
  • R 3 is a C1-C3 alkyl group, a 2-propenyl group, a 2-propynyl group, a C3-C6 cycloalkylmethyl group, a phenylmethyl group, a pyridylmethyl group, a cyanomethyl group, a tetrahydrofuranylmethyl group, a cyclopropyl group, or a hydrogen atom.
  • R 4 is a C1-C3 chain hydrocarbon group ⁇ which may be substituted with one or more substituents selected from the group consisting of a cyclopropyl group, a phenyl group which may be substituted with one or more substituents selected from group B, a 5- or 6-membered aromatic heterocyclic group which may be substituted with one or more substituents selected from group B, a cyano group, and a halogen atom ⁇ , OR 18 , S(O) m R 29 , NR 7b R 8b , C(O)NR 7b R 8b , NR 9b C(O)R 5b , NR 9b C(O)OR 6b , NR 9 C(O)NR 7 R 8 , a cyclopropyl group, a halogen atom, or a hydrogen atom; R 18 is a C1-C3 alkyl group which may be substituted with one or more halogen atom, or a hydrogen atom; R 18 is
  • R 3 is a C1-C3 alkyl group, a 2-propenyl group, a 2-propynyl group, a C3-C6 cycloalkylmethyl group, a phenylmethyl group, a pyridylmethyl group, a cyanomethyl group, a tetrahydrofuranylmethyl group, a cyclopropyl group, or a hydrogen atom.
  • R3 and R4 together with the nitrogen atom to which R3 is bonded and the carbon atom to which R4 is bonded, form a group represented by the following formula A1-1, A4-3, A5-2, A5-3, A6-1, or A7-1 (# represents the bonding site with R2 , and ⁇ represents the bonding site with the carbon atom to which R1 is bonded),
  • R 25 is a C1-C3 alkyl group optionally substituted with one or more halogen atoms, a C1-C3 alkoxy group optionally substituted with one or more halogen atoms, C(O)R 5 , C(O)OR 6 , C(O)NR 7 R 8 , NR 9C (O)R 5 , NR 9C (O)OR 6 , NR 9C (O)NR 7 R 8 , a cyano group, a halogen atom, or a hydrogen atom;
  • R 26 is a
  • R3 and R4 together with the nitrogen atom to which R3 is bonded and the carbon atom to which R4 is bonded, form a group represented by the following formula A1-1, A4-3, A5-2, A5-3, A6-2, or A7-2 (# represents the bonding site with R2 , and ⁇ represents the bonding site with the carbon atom to which R1 is bonded),
  • R 25 is a methyl group, a methoxy group, a trifluoromethyl group, a trifluoromethoxy group, a cyano group, a halogen atom, or a hydrogen atom
  • R 26 is a C1-C3 alkyl group or a hydrogen atom
  • R 2a , R 2b , R 2c , R 2d , R 2g , and R 2h are the same or different and are a methyl group, a methoxy group, a trifluoromethyl group, a
  • R 4a and R 4b are the same or different and are a C1-C3 chain hydrocarbon group optionally substituted with one or more halogen atoms or a hydrogen atom, and n is 1, 2, or 3.
  • X is NR 11 C(O)R 12 , NR 11 C(O)NR 12 R 13 , or NR 11 X 1
  • X 1 is a 9- or 10-membered aromatic heterocyclic group ⁇ the 9- or 10-membered aromatic heterocyclic group is a C1-C3 chain hydrocarbon group ⁇ the C1-C3 chain hydrocarbon group may be substituted with one or more substituents selected from the group consisting of cyano groups and halogen atoms ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of cyano groups and halogen atoms ⁇
  • X is NR 11 C(O)R 12 , NR 11 C(O)NR 12 R 13 , or NR 11 X 1
  • X 1 is a 9- or 10-membered aromatic heterocyclic group
  • the 9- or 10-membered aromatic heterocyclic group is a C1-C3 chain hydrocarbon group
  • the C1-C3 chain hydrocarbon group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • X is NR 11 C(O)R 12
  • R 11 is a C1-C6 chain hydrocarbon group optionally substituted with one or more substituents selected from group F, a C1-C3 alkylsulfonyl group optionally substituted with one or more halogen atoms
  • OR 15 C(O)R 14 , C(O)OR 14 , or a hydrogen atom
  • R 12 is a phenyl group or a pyridyl group ⁇ the phenyl group and the pyridyl group are a C1-C3 chain hydrocarbon group ⁇ the C1-C3 chain hydrocarbon group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a
  • X is NR 11 C(O)R 12
  • R 11 is a C1-C6 chain hydrocarbon group optionally substituted with one or more substituents selected from group F, a C1-C3 alkylsulfonyl group optionally substituted with one or more halogen atoms
  • OR 15 C(O)R 14 , C(O)OR 14 , or a hydrogen atom
  • R 12 is a phenyl group or a pyridyl group ⁇ the phenyl group and the pyridyl group are a C1-C3 chain hydrocarbon group ⁇ the C1-C3 chain hydrocarbon group may be substituted with one or more substituents selected from the group consisting of a cyano group and a halogen atom ⁇
  • a cyclopropyl group ⁇ the cyclopropyl group may be substituted with one or more substituents selected from the group consisting of a cyano group and a
  • reaction time is usually in the range of 0.1 to 48 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures are carried out to obtain compound (Ia).
  • Compound (Md) is a commercially available compound or can be prepared using known methods.
  • Condensing agents used in the reaction include, for example, carbodiimides such as 1-ethyl-3-[3-(dimethylamino)propyl]carbodiimide hydrochloride and 1,3-dicyclohexylcarbodiimide.
  • a catalyst may be used in the reaction, if necessary.
  • An example of the catalyst is 1-hydroxybenzotriazole.
  • the catalyst is usually used in a ratio of 0.01 to 0.5 moles per mole of compound (M-6).
  • a base can be used as necessary. Examples of the base include organic bases. When a base is used in the reaction, the base is usually used in a ratio of 1 to 5 moles per mole of compound (M-6).
  • the acid used in the reaction includes, for example, trifluoroacetic acid and hydrogen chloride.
  • hydrogen chloride a solution of hydrogen chloride such as hydrochloric acid or a hydrogen chloride/methanol solution may be used in the reaction.
  • the reaction can be carried out, for example, by first mixing the compound (M-5) with an acid, then distilling off the acid, and mixing the compound (Mg).
  • a base can be used as necessary. Examples of the base include organic bases. When a base is used in the reaction, the base is usually used in a ratio of 1 to 10 moles per mole of compound (M-5).
  • the compound (Mg) is usually used in a ratio of 1 to 2 moles and the acid is usually used in a ratio of 1 to 100 moles, relative to 1 mole of the compound (M-5).
  • the reaction temperature is usually within the range of ⁇ 20 to 200° C.
  • the reaction time is usually within the range of 0.1 to 24 hours.
  • the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures are carried out to obtain compound (Ia).
  • Compound (Mg) is a commercially available compound or can be prepared using known methods.
  • the reaction may, if necessary, use a ligand, a base, and/or an inorganic halide.
  • the ligand include triphenylphosphine, xantphos, 2,2'-bis(diphenylphosphino)-1,1'-binaphthyl, 1,1'-bis(diphenylphosphino)ferrocene, 2-dicyclohexylphosphino-2',4',6'-triisopropylbiphenyl, 2-dicyclohexylphosphino-2',6'-dimethoxybiphenyl, 1,2-bis(diphenylphosphino)ethane, 2,2'-bipyridine, 2-aminoethanol, 8-hydroxyquinoline, and 1,10-phenanthroline.
  • the inorganic halide When an inorganic halide is used in the reaction, the inorganic halide is usually used in a ratio of 0.1 to 5 moles per mole of the compound (M-10).
  • the reaction temperature is usually in the range of ⁇ 20° C. to 200° C.
  • the reaction time is usually in the range of 0.1 to 72 hours.
  • the compound N of the present invention can be obtained by carrying out post-treatment operations such as adding water to the reaction mixture, extracting with an organic solvent, drying and concentrating the organic layer.
  • Compound (Mc) is a commercially available compound or can be prepared using known methods.
  • the compound (M-6) can be produced from the compound (M-5). (In the formula, the symbols have the same meanings as defined above.)
  • the reaction can be carried out, for example, according to the method described in Green's PROTECTIVE GROUPS in ORGANIC SYNTHESIS FORTH EDITION, p. 727.
  • Compound (M-6) may form an acid addition salt.
  • acids that form acid addition salts include inorganic acids such as hydrochloric acid and sulfuric acid; and organic acids such as acetic acid, trifluoroacetic acid, benzoic acid, and p-toluenesulfonic acid.
  • Compound (M-5) can be produced by reacting a compound represented by formula (M-4) (hereinafter referred to as compound (M-4)) with compound (M-c) in the presence of a metal catalyst. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 5, except that compound (M-4) is used in place of compound (M-10).
  • Reference Manufacturing Method 3 Compound (M-4) can be produced by reacting a compound represented by formula (M-3a) (hereinafter referred to as compound (M-3a)) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction is usually carried out in a solvent, for example, alcohols such as methanol and ethanol (hereinafter referred to as alcohols), nitriles, ethers, aromatic hydrocarbons, aprotic polar solvents, halogenated hydrocarbons, acetic acid, water, and mixtures of two or more of these.
  • a solvent for example, alcohols such as methanol and ethanol (hereinafter referred to as alcohols), nitriles, ethers, aromatic hydrocarbons, aprotic polar solvents, halogenated hydrocarbons, acetic acid, water, and mixtures of two or more of these.
  • halogenating agent examples include chlorine, bromine, iodine, N-chlorosuccinimide, N-bromosuccinimide, and N-iodosuccinimide.
  • a base can be used as necessary.
  • the base include alkali metal carbonates.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (M-3a).
  • the halogenating agent is usually used in a ratio of 1 to 20 moles per mole of compound (M-3a).
  • the reaction temperature is usually in the range of ⁇ 20° C. to 200° C.
  • the reaction time is usually in the range of 0.1 to 72 hours. After the reaction is completed, the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (M-4).
  • Compound (M-3a) can be produced by reacting a compound represented by formula (M-2a) (hereinafter referred to as compound (M-2a)) with a compound represented by formula (M-b) (hereinafter referred to as compound (M-b)) in the presence of a base.
  • a compound represented by formula (M-2a) hereinafter referred to as compound (M-2a)
  • M-b a compound represented by formula (M-b)
  • X represents a leaving group such as a bromine atom or an iodine atom, and the other symbols have the same meanings as above.
  • the reaction is usually carried out in a solvent, such as ethers, aromatic hydrocarbons, nitriles, aprotic polar solvents, and mixtures of two or more of these.
  • Reference Manufacturing Method 5 Compound (M-4) can also be produced by reacting a compound represented by formula (M-3b) (hereinafter referred to as compound (M-3b)) with compound (M-b) in the presence of a base. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 4, except for using compound (M-3b) instead of compound (M-2a).
  • the halogenating agent is usually used in a ratio of 1 to 20 moles per mole of compound (M-2a).
  • the base include alkali metal hydrides, alkali metal carbonates, and organic bases. For example, alkali metal carbonates are included.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (M-2a).
  • the reaction temperature is usually in the range of ⁇ 20° C. to 200° C.
  • the reaction time is usually in the range of 0.1 to 72 hours.
  • the reaction may be carried out by reacting compound (M-2a) with a halogenating agent and then mixing the resulting mixture with compound (M-b); it may be carried out by reacting compound (M-2a) with compound (M-b) and then mixing the resulting mixture with a halogenating agent; or it may be carried out by mixing compound (M-2a), compound (M-b), and a halogenating agent.
  • the reaction mixture is added with water, extracted with an organic solvent, and the organic layer is dried and concentrated, and other post-treatment procedures can be carried out to obtain compound (M-4).
  • Reference Manufacturing Method 7 Compound (M-3b) can be produced by reacting compound (M-2a) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 3, except for using compound (M-2a) instead of compound (M-3a).
  • the compound represented by formula (M-2b) (hereinafter referred to as compound (M-2b)) can be produced by reacting a compound represented by formula (M-2) (hereinafter referred to as compound (M-2)) with a sulfurizing agent.
  • R y represents a C1-C4 alkyl group, a cyano group, a halogen atom, or a hydrogen atom
  • R z represents a C1-C4 alkyl group, a C3-C6 cycloalkyl group, or a hydrogen atom
  • the other symbols have the same meanings as above.
  • the reaction is carried out in a solvent or in the absence of a solvent, such as ethers, halogenated hydrocarbons, aromatic hydrocarbons, nitriles, nitrogen-containing aromatic compounds, and mixtures of two or more of these.
  • the sulfurizing agent examples include diphosphorus pentasulfide and Lawesson's reagent (2,4-bis(4-methoxyphenyl)-1,3-dithia-2,4-diphosphetane-2,4-disulfide).
  • the sulfurizing agent is usually used in a ratio of 1 to 3 moles per mole of compound (M-2).
  • the reaction temperature is usually in the range of 0° C. to 200° C.
  • the reaction time is usually in the range of 1 to 48 hours.
  • the compound (M-2b) can be obtained by carrying out post-treatment operations such as adding water to the reaction mixture, extracting with an organic solvent, and drying and concentrating the organic layer.
  • Compound (M-2) can be produced by reacting a compound represented by formula (M-1) (hereinafter referred to as compound (M-1)) with a compound represented by formula (Ma) (hereinafter referred to as compound (Ma)).
  • compound (Ma) a compound represented by formula (Ma)
  • R x represents a C1-C4 alkyl group, and the other symbols have the same meanings as defined above.
  • the reaction is usually carried out in a solvent, such as alcohols, ethers, aromatic hydrocarbons, nitriles, aprotic polar solvents, halogenated hydrocarbons, and mixtures of two or more of these.
  • the compound (Ma) is usually used in a ratio of 1 to 5 moles per mole of the compound (M-1).
  • a base can be used as necessary.
  • the base include alkali metal alkoxides such as sodium methoxide and sodium ethoxide; alkali metal hydrides; alkali metal carbonates; and organic bases.
  • the base is usually used in a ratio of 1 to 10 moles per mole of compound (M-1).
  • the reaction temperature is usually in the range of ⁇ 20 to 200° C.
  • the reaction time is usually in the range of 0.1 to 24 hours.
  • the compound (M-2) can be obtained by carrying out post-treatment operations such as adding water to the reaction mixture, extracting with an organic solvent, drying and concentrating the organic layer.
  • the compound (Ma) is a commercially available compound or can be prepared using known methods.
  • Compound (M-1) is publicly known, or can be produced according to a known method described in Tetrahedron (2013) 69, 11092-11108.
  • the compound represented by formula (M-7) (hereinafter referred to as compound (M-7)) can be produced by reacting a compound represented by formula (M-1) (hereinafter referred to as compound (M-1)) with compound (M-g). (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Production Method 3, except that compound (M-1) is used in place of compound (M-5).
  • Reference Manufacturing Method 12 The compound represented by formula (M-8b) (hereinafter referred to as compound (M-8b)) can be produced by reacting compound (M-8a) with a sulfurizing agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 8, except for using compound (M-8a) instead of compound (M-2).
  • the compound (M-10) can be produced by reacting the compound (M-9) with a halogenating agent. (In the formula, the symbols have the same meanings as defined above.) The reaction can be carried out according to Reference Production Method 3, except that compound (M-9) is used in place of compound (M-3a).
  • composition A containing one or more components selected from the group consisting of Group (a), Group (b), Group (c), and Group (d) (i.e., the present component) and a compound of the present invention.
  • Group (a) includes acetylcholinesterase inhibitors (e.g., carbamate insecticides, organophosphate insecticides), GABAergic chloride channel blockers (e.g., phenylpyrazole insecticides), sodium channel modulators (e.g., pyrethroid insecticides), nicotinic acetylcholine receptor competitive modulators (e.g., neonicotinoid insecticides), nicotinic acetylcholine receptor allosteric modulators, glutamatergic chloride channel allosteric modulators (e.g., macrolide insecticides), juvenile hormone mimics, multisite inhibitors, chordotonal organ TRPV channel modulators, mite growth inhibitors, The group consists of microbial insect midgut membrane disruptors, mitochondrial ATP synthase inhibitors, oxidative phosphorylation uncouplers, nicotinic acetylcholine receptor channel blockers (e.g., ner
  • Group (b) consists of nucleic acid synthesis inhibitors (e.g., phenylamide fungicides, acylamino acid fungicides), cell division and cytoskeleton inhibitors (e.g., MBC fungicides), respiratory inhibitors (e.g., QoI fungicides, QiI fungicides), amino acid synthesis and protein synthesis inhibitors (e.g., anilinopyrimidine fungicides), signal transduction inhibitors, lipid synthesis and membrane synthesis inhibitors, sterol biosynthesis inhibitors (e.g., DMI fungicides such as triazoles), cell wall biosynthesis inhibitors, melanin synthesis inhibitors, plant defense inducers, multisite contact active fungicides, microbial fungicides, and other fungicidal active ingredients. These are described in the classification based on the mechanism of action of FRAC.
  • nucleic acid synthesis inhibitors e.g., phenylamide fungicides, acylamin
  • Group (c) is a group of plant growth regulators (including mycorrhizal fungi and rhizobia).
  • Group (d) is a group of repellent components.
  • the ratio of the compound of the present invention to this component is not particularly limited, but examples of the ratio by weight (compound of the present invention: this component) include 1000:1 to 1:1000, 500:1 to 1:500, 100:1 to 1:100, 50:1, 20:1, 10:1, 9:1, 8:1, 7:1, 6:1, 5:1, 4:1, 3:1, 2:1, 1:1, 1:2, 1:3, 1:4, 1:5, 1:6, 1:7, 1:8, 1:9, 1:10, 1:20, and 1:50.
  • the compound of the present invention is effective against harmful arthropods such as harmful insects and harmful mites, harmful nematodes, and harmful mollusks.
  • harmful arthropods such as harmful insects and harmful mites, harmful nematodes, and harmful mollusks.
  • harmful arthropods, harmful nematodes, and harmful mollusks include the following:
  • Hemiptera Small brown planthopper (Laodelphax striatellus), brown planthopper (Nilaparvata lugens), white-backed planthopper (Sogatella furcifera), corn planthopper (Peregrinus maidis), yellow horned planthopper (Javesella pellucida), black horned planthopper (Perkinsiella saccharicida), Tagosodes orizicolus, Stenocranus pacificus, etc.
  • Tuna leafhopper (Nephotettix cincticeps), Taiwan green leafhopper (Nephotettix virescens), Black-striped green leafhopper (Nephotettix nigropictus), Lightning leafhopper (Recilia dorsalis), Tea green leafhopper (Empoasca onukii), Potato leafhopper (Empoasca fabae), Corn leafhopper (Dalbulus maidis), White giant leafhopper (Cofana spectrum), Amrasca biguttul Cicadellidae (Cicadellidae), such as A.
  • Aphrophoridae such as the European spittlebug (Philaenus spumaris); Geisha distinctissima (Geisha distinctissima); Ricania shantungensis (Ricania shantungensis); Cercopidae (Cercopidae), such as Mahanarva posticata and Mahanarva fimbriolata; Aphis fabae), soybean aphid (Aphis glycines), cotton aphid (Aphis gossypii), European apple aphid (Aphis pomi), snow willow aphid (Aphis spiraecola), peach aphid (Myzus persicae), strawberry aphid (Brachycaudus helichrysi), radish aphid (Brevicoryne brassicae), rosy apple aphid (Dysaphis plantaginea),
  • Pseudococcidae such as Pseudococcus kraunhiae, Pseudococcus comstocki, Planococcus citri, Pseudococcus calceolariae, Pseudococcus longispinus, and Brevennia rehi; treae), pear psylla (Cacopsylla pyrisuga), Chinese pear psylla (Cacopsylla chinensis), potato psylla (Bactericera cockerelli), and cacopsylla (Cacopsylla pyricola); Tingidae family such as Cimex pyrioides; Cimicidae family such as Cimex lectularius and Cimex hempterus; Cicadidae family such as Quesada gigas; Reduviidae family such as Triatoma infestans, Triatoma rubrofasciata, Triatoma dimidiata
  • Lepidoptera Chilo suppressalis, Dark headed stem borer, Chilo polychrysus, White stem borer, Scirpophaga innotata, Scirpophaga incertulas, Rupela albina, Cnaphalocrocis medinalis, Marasmia patnalis, Rice leaf moth Cotton moth (Marasmia exigua), cotton borer (Notarcha derogata), corn borer (Ostrinia furnacalis), European corn borer (Ostrinia nubilalis), grey spotted moth (Hellula undalis), black-eared moth (Herpetogramma luctuosale), grass moth (Parapediasia teterrellus), rice case worm (Nymph Crambidae, such as the sugar cane borer (Diatraea saccharalis), the eggplant fruit borer (Leucinodes orbonalis), and the peach moth (Conogethes
  • Pyralidae family including Euzophera batangensis and Cadra cautella; Spodoptera litura, Spodoptera exigua, Mythimna separata, Mamestra brassicae, Sesamia inferens, Spodoptera mauritia), Naranga aenescens, Spodoptera frugiperda, Spodoptera exempta, Spodoptera cosmioides, Semi-tropical armyworm (Spodoptera eridania), Agrotis ipsilon, Agrotis segetum, Aut ographa nigrisigna, rice looper (Plusia festucae), soybean looper (Chrysodeixis includens), fig looper (Chrysodeixis eriosoma), three-leaf looper (Ctenoplusia agnata), nettle looper (Trichoplusia ni), etc.; Heliothis spp.
  • Thysanoptera Thripidae, such as Frankliniella occidentalis, Thrips palmi, Scirtothrips dorsalis, Thrips tabaci, Frankliniella intonsa, Stenchaetothrips biformis, Echinothrips americanus, Scirtothrips perseae; Phlaeothripidae, such as Haplothrips aculeatus.
  • Agromyzidae (Agromyzidae); Chloropidae (Chlorops oryzae), etc.; Bactrocera cucurbitae (Melon fly), Bactrocera dorsalis (Oriental fruit fly), Bactrocera latifrons (Eastern fruit fly), Bactrocera oleae (Olive fruit fly), Bactrocera tryoni (Queensland fruit fly), Ceratitis capitata (Mediterranean fruit fly), Rhagoletis pomonella (Apple maggot), Rhagoletis suzukii (Sugar apple fly), Rhagoletis japonica (Chrysocarpus japonica), Rhagoletis japonica (Rhagoletis ...
  • Cerambycidae Melanotus okina wensis, Agriotes fuscicollis, Melanotus legatus, Anchastus spp., Conoderus spp., Ctenicera spp., Limonius spp., Aeolus spp.
  • the family Staphylinidae such as Paederus fuscipes
  • the family Dermestidae such as Anthrenus verbasci, Dermestes maculates, and Trogoderma granarium
  • the family Lasioderma serricorne Ste gobium paniceum and other Anobiidae
  • Brassicogethes aeneus and other Blossom Beetles (Nitidulidae).
  • Hymenoptera Tenthredinidae such as Athalia rosae and Athalia japonica; Solenopsis spp. such as Solenopsis invicta and Solenopsis geminata; Atta spp.
  • Atta capiguara and Acrom yrmex spp. such as Atta capiguara and Acrom yrmex spp.), Paraponera clavata, Ochetellus glaber, Monomorium pharaonis, Argentine ant (Linepithema humile), Formica japonica, Pristomyrmex punctutus, Pheidole noda, Pheidole megacephala, Camponotus spp., such as the Japanese camponotus (Camponotus japonicus), Camponotus spp., such as the red-breasted camponotus (Camponotus obscuripes), Pogonomyrmex spp., such as Pogonomyrmex occidentalis, Wasmania spp., such as Wasmania auropunctata, and Anoplolepis gracilipinas.
  • Family Ectobiidae such as the German cockroach (Blattella germanica); Family Blattidae, such as the Siberian cockroach (Periplaneta fuliginosa), the American cockroach (Periplaneta americana), the American cockroach (Periplaneta australiae), the brown cockroach (Periplaneta brunnea), and the Asian cockroach (Blatta orientalis); Family Reticulitermes speratus, Formosan termite (Coptotermes formosanus), Formosan dry wood termite (Incisitermes minor), Formosan termite (Cryptotermes domesticus), Formosan termite (Odontotermes formosanus), and Formosan termite (Neotermes Termites of the family Termitidae, such as Glyptotermes satsumensis, Glyptotermes nakajimai, Glyptotermes fuscus,
  • Order Siphonaptera Family Pulicidae such as the human flea (Pulex irritans), cat flea (Ctenocephalides felis), dog flea (Ctenocephalides canis), rat flea (Xenopsylla cheopis), chicken flea (Echidnophaga gallinacea), etc.; Family Hectopsyllidae such as the sand flea (Tunga penetrans); Family Ceratophyllidae such as the European rat flea (Nosopsyllus fasciatus).
  • Family Pulicidae such as the human flea (Pulex irritans), cat flea (Ctenocephalides felis), dog flea (Ctenocephalides canis), rat flea (Xenopsylla cheopis), chicken flea (Echidnophaga gallinacea), etc.
  • Family Hectopsyllidae such as the sand flea (Tunga penetrans)
  • Psocodae Family Pediculidae such as head lice (Pediculus humanus capitis); Family Pthiridae such as pubic lice (Pthirus pubis); Family Haematopinidae such as cow lice (Haematopinus eurysternus) and pig lice (Haematopinus suis); Family Linognathus vituli, Sheep trunk lice Family Linognathidae, such as body lice (Linognathus ovillus) and cow lice (Solenopotes capillatus); Family Bovicoliidae, such as cow lice (Bovicola bovis), sheep lice (Bovicola ovis), Bovicola breviceps, Damalinia forficula, and Werneckiella spp.; Family Bovicoliidae, such as dog lice (T Family Trichodectidae, such as richodectes canis and Felicola subrostratus; Family Menoponi
  • Trogiidae such as Trogium pulsatorium
  • Liposcelidae or Liposcelididae such as Liposcelis corrodens, Liposcelis bostrychophila, Liposcelis pearmani, and Liposcelis entomophila.
  • Solid carriers include, for example, clay (pyrophyllite clay, kaolin clay, etc.), talc, calcium carbonate, diatomaceous earth, zeolite, bentonite, acid clay, attapulgite, white carbon, ammonium sulfate, vermiculite, perlite, pumice, silica sand, fine powders and granules of chemical fertilizers (ammonium sulfate, ammonium phosphate, ammonium nitrate, urea, ammonium chloride, etc.), and resins (polyethylene, polypropylene, polyester, polyurethane, polyamide, polyvinyl chloride, etc.).
  • clay pyrophyllite clay, kaolin clay, etc.
  • talc calcium carbonate
  • diatomaceous earth zeolite
  • bentonite acid clay
  • attapulgite white carbon
  • ammonium sulfate vermiculite
  • perlite perlite
  • pumice pumice
  • Liquid carriers include, for example, water, alcohols (ethanol, cyclohexanol, benzyl alcohol, propylene glycol, polyethylene glycol, etc.), ketones (acetone, cyclohexanone, etc.), aromatic hydrocarbons (xylene, phenylxylylethane, methylnaphthalene, etc.), aliphatic hydrocarbons (hexane, cyclohexane, etc.), esters (ethyl acetate, methyl oleate, propylene carbonate, etc.), nitriles (acetonitrile, etc.), ethers (ethylene glycol dimethyl ether, etc.), amides (N,N-dimethylformamide, N,N-dimethyloctanamide, etc.), sulfoxides (dimethyl sulfoxide, etc.), lactams (N-methylpyrrolidone, N-octylpyrrolidone, etc.), fatty
  • Gaseous carriers include, for example, fluorocarbons, butane gas, LPG (liquefied petroleum gas), dimethyl ether, nitrogen, and carbon dioxide.
  • formulation adjuvants include binders, dispersants, colorants, and stabilizers, and specific examples include polysaccharides (starch, gum arabic, cellulose derivatives, alginic acid, etc.), lignin derivatives, synthetic water-soluble polymers (polyvinyl alcohol, polyvinylpyrrolidone, polyacrylic acids, etc.), acid isopropyl phosphate, and dibutylhydroxytoluene.
  • plants include whole plants, stems and leaves, flowers, spikes, fruits, trunks, branches, crowns, seeds, vegetative reproductive organs, and seedlings.
  • irrigation treatments include (soil irrigation, seedling irrigation, chemical injection treatment, ground level irrigation, chemical drip irrigation, chemigation), seedling box treatments (seedling box spraying, seedling box irrigation, seedling box flooding with chemicals), seedling tray treatments (seedling tray spraying, seedling tray irrigation, seedling tray flooding with chemicals), seedbed treatments (seedling bed spraying, seedling bed irrigation, water seedling bed spraying, seedling immersion), bed soil mixing treatments (bed soil mixing, bed soil mixing before sowing, spraying before soil cover at sowing, spraying after soil cover at sowing, soil cover mixing), and other treatments (mixing culture soil, plowing in, mixing topsoil, mixing soil from areas that have fallen off due to rain, planting position treatment, spraying granular inflorescences, mixing paste fertilizer).
  • Examples of seed treatment include treatment of seeds or vegetative reproductive organs with the compound of the present invention or composition A. More specifically, examples of the treatment include spraying treatment in which a suspension of the compound of the present invention or composition A is misted and sprayed onto the surface of a seed or vegetative reproductive organ, smearing treatment in which the compound of the present invention or composition A is applied to the seed or vegetative reproductive organ, immersion treatment in which the seed or vegetative reproductive organ is immersed in a liquid of the compound of the present invention or composition A for a certain period of time, and a method of coating the seed or vegetative reproductive organ with a carrier containing the compound of the present invention or composition A (film coating treatment, pellet coating treatment, etc.).
  • the above-mentioned vegetative reproductive organ particularly includes seed potatoes.
  • composition A When applying composition A to seeds or vegetative reproductive organs, composition A can be applied to the seeds or vegetative reproductive organs as one formulation, or composition A can be applied to the seeds or vegetative reproductive organs in multiple separate applications as different formulations.
  • Examples of the method of applying composition A in multiple separate applications as different formulations include a method of applying a formulation containing only the compound of the present invention as an active ingredient, air-drying the seeds or vegetative reproductive organs, and then applying a formulation containing this component; and a method of applying a formulation containing the compound of the present invention and this component as active ingredients, air-drying the seeds or vegetative reproductive organs, and then applying a formulation containing this component other than the component that has already been applied.
  • the seed or vegetative reproductive organ carrying the compound of the present invention or composition A means a seed or vegetative reproductive organ having the compound of the present invention or composition A attached to its surface.
  • the seed or vegetative reproductive organ carrying the compound of the present invention or composition A may have a material other than the compound of the present invention or composition A attached thereto before or after the compound of the present invention or composition A is attached to the seed or vegetative reproductive organ.
  • the layer may consist of one or more layers.
  • each layer may contain one or more active ingredients, or each layer may consist of a layer containing one or more active ingredients and a layer containing no active ingredients. Seeds or vegetative reproductive organs carrying the compound of the present invention or composition A can be obtained, for example, by applying a formulation containing the compound of the present invention or composition A to the seeds or vegetative reproductive organs by the seed treatment methods described above.
  • the application amount is usually 1 to 10,000 g of the compound of the present invention per 10,000 m2 .
  • the compound of the present invention is usually applied in an amount of 0.001 to 100 g per 1 kg of seeds or vegetative reproductive organs.
  • the compound of the present invention or composition A is formulated as an emulsifiable concentrate, wettable powder, flowable agent, or the like, it is usually applied after diluting with water so that the active ingredient concentration is 0.01 to 10,000 ppm, and granules, dusts, and the like are usually applied as is.
  • the compound of the present invention or composition A can be used as an agent for controlling harmful arthropods in agricultural land such as fields, paddy fields, lawns, orchards, etc.
  • agricultural land such as fields, paddy fields, lawns, orchards, etc.
  • plants include the following.
  • the above plants are not particularly limited as long as they are varieties that are commonly cultivated.
  • the above plants also include plants that can be produced by natural crossbreeding, plants that can be generated by mutation, F1 hybrid plants, and genetically modified crops.
  • genetically modified crops include plants that have been given resistance to herbicides such as HPPD (4-hydroxyphenylpyruvate dioxygenase enzyme) inhibitors such as isoxaflutole, ALS (acetolactate synthase) inhibitors such as imazethapyr and thifensulfuron methyl, EPSP (5-enolpyruvylshikimate-3-phosphate synthase) inhibitors, glutamine synthetase inhibitors, PPO (protoporphyrinogen oxidase) inhibitors, bromoxynil, or dicamba; plants that are able to synthesize selective toxins known from the Bacillus genus, such as Bacillus thuringiensis; and plants that can be given specific insecticid
  • Me represents a methyl group
  • Et represents an ethyl group
  • Boc represents a tert-butoxycarbonyl group
  • Cbz represents a benzyloxycarbonyl group.
  • LCMS liquid chromatography/mass spectrometry
  • MS mass spectrometry
  • Production Example 4 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 2-4-1 was used instead of Intermediate 2-4-4, and 2-(trifluoromethyl)benzoyl chloride was used instead of 3,5-bis(trifluoromethyl)benzoyl chloride.
  • Compound 4 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.90(2H, d), 8.22(1H, s), 7.62(1H, d), 7.52(1H, t), 7.44(1H, t), 7.30(2H, t), 5.99(1H, d), 3.59(3H, s), 2.57(3H, s), 1.47(3H, d).
  • Production Example 5 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 2-4-1 was used instead of Intermediate 2-4-4, and 4-(trifluoromethyl)benzoyl chloride was used instead of 3,5-bis(trifluoromethyl)benzoyl chloride.
  • Compound 5 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.84(2H, d), 8.23(1H, s), 7.60(2H, d), 7.42(2H, d), 7.24(1H, s), 5.90-5.88(1H, m), 3.60(3H, s), 2.74(3H, s), 1.52(3H, d).
  • Production Example 7 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 2-4-2 was used instead of Intermediate 2-4-4, and 3-(trifluoromethyl)benzoyl chloride was used instead of 3,5-bis(trifluoromethyl)benzoyl chloride.
  • Production Example 9 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 2-4-1 was used instead of Intermediate 2-4-4, and 4-(trifluoromethyl)benzoyl chloride was used instead of 3,5-bis(trifluoromethyl)benzoyl chloride.
  • Compound 9 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.89-8.82(2H, m), 8.25(1H, d), 7.65-7.61(3H, m), 7.52(1H, d), 7.30-7.29(1H, m), 4.69(1H, s), 4.28(1H, s), 3.60(3H, s), 3.01-2.91(3H, m).
  • Production Example 12 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 2-4-3 was used instead of Intermediate 2-4-4.
  • Compound 12 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.86(2H, s), 8.52(1H, s), 7.88(1H, s), 7.75(2H, s), 5.89(1H, s), 2.81(3H, s), 2.51(3H, s), 1.54(3H, d).
  • Production Example 13 A compound produced according to Production Example 2 using 3-(trifluoromethyl)benzoyl chloride instead of 3,5-bis(trifluoromethyl)benzoyl chloride and its physical properties are shown below.
  • Invention compound 13 1 H-NMR (CDCl 3 ) ⁇ : 8.83(2H, d), 7.61-7.60(1H, m), 7.51-7.47(3H, m), 7.21(1H, s), 5.87-5.86(1H, m), 3.59(3H, s), 2.75(3H, s), 2.62(3H, s), 1.50(3H, d).
  • Production Example 19 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 2-4-9 was used instead of Intermediate 2-4-4.
  • Compound 19 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.92(2H, d), 8.22(2H, s), 8.00(1H, s), 7.67(1H, d), 7.33(1H, dd), 5.18(1H, m), 4.19-4.10(2H, m), 2.69(3H,t), 1.44(3H, d), 1.40(3H, t).
  • Production Example 23 The compound and its physical properties are shown below, which were produced according to Production Example 22 using Intermediate 2-4-10 instead of Intermediate 2-4-8.
  • Compound 23 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.92(2H, d), 8.73(1H, s), 8.24(1H, s), 8.18(1H, s), 7.76(1H, d), 7.34(1H, t), 5.50-5.45(1H, m), 3.79(3H, s), 2.17-2.14(1H, m), 1.42-1.33(4H, m), 1.41(3H, d).
  • reaction liquid A 0.15 g of triphosgene and 0.14 mL of triethylamine were added to a mixture of 0.12 g of 2,4-bis(trifluoromethyl)aniline and 5.1 mL of THF, and the mixture was stirred under ice cooling for 1 hour to obtain a mixture. Reaction liquid A was added to the mixture, and the mixture was stirred at room temperature for 3 hours.
  • Production Example 25 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 2-4-12 was used instead of Intermediate 2-4-4.
  • Compound 25 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.93(2H, d), 8.28(1H, s), 8.21(2H, s), 8.00(1H, s), 7.48(1H, d), 7.36(1H, t), 5.22-5.17(1H, m), 4.11-4.02(2H, m), 1.48-1.46(6H, m).
  • Production Example 26 The compound and its physical properties are shown below, which were produced according to Production Example 10 using Intermediate 2-4-8 instead of Intermediate 2-4-2 and 3,5-diiodobenzoic acid instead of 3,5-dibromobenzoic acid.
  • Compound 26 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.90(2H, d), 8.16(1H, t), 8.02(2H, d), 7.36(1H, d), 7.31(1H, t), 5.12(1H, m), 3.60(3H, s), 2.66(3H, s), 1.41(3H, d).
  • Production Example 27 The compound and its physical properties are shown below, which were produced according to Production Example 10 using Intermediate 2-4-8 instead of Intermediate 2-4-2 and 3,5-bis(difluoromethoxy)benzoic acid instead of 3,5-dibromobenzoic acid.
  • Compound 27 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.90(2H, d), 7.53(1H, d), 7.37(2H, d), 7.31(1H, t), 7.04(1H, d), 6.56(2H, t), 5.15(1H, m), 3.60(3H, s), 2.65(3H, s), 1.42(3H, d).
  • Production Example 28 The compound and its physical properties are shown below, which were produced according to Production Example 10 using Intermediate 2-4-8 instead of Intermediate 2-4-2 and 3-chloro-5-trifluoromethoxybenzoic acid instead of 3,5-dibromobenzoic acid.
  • Compound 28 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.90(2H, d), 7.67(1H, t), 7.51-7.48(2H, m), 7.35(1H, s), 7.32(1H, t), 5.18-5.14(1H, m), 3.60(3H, s), 2.66(3H, s), 1.42(3H, d).
  • Production Example 29 The compound and its physical properties are shown below, which were produced according to Production Example 10, except that Intermediate 2-4-1 was used instead of Intermediate 2-4-2.
  • Compound 29 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.86(2H, d), 8.23(1H, s), 7.65(1H, s), 7.36(2H, s), 7.26-7.25(1H, m), 5.84-5.82(1H, m), 3.60(3H, s), 2.74(3H, s), 1.49(3H, d).
  • Production Example 30 The compound and its physical properties are shown below, which were produced according to Production Example 10 using Intermediate 2-4-1 instead of Intermediate 2-4-2 and 3,5-dichlorobenzoic acid instead of 3,5-dibromobenzoic acid.
  • Production Example 31 Compounds and their physical properties are shown below, which were produced according to Production Example 10 using Intermediate 2-4-1 instead of Intermediate 2-4-2 and 1-methyl-3-trifluoromethyl-1H-pyrazole-5-carboxylic acid instead of 3,5-dibromobenzoic acid.
  • Production Example 33 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 5-2 was used instead of Intermediate 2-4-4.
  • Compound 33 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.88(2H, d), 8.25(2H, s), 8.07(1H, d), 8.00(1H, s), 7.25-7.24(1H, m), 5.28-5.27(1H, m), 4.96(1H, s), 3.47(3H, s), 3.17(3H, d), 1.41(3H, d).
  • Production Example 34 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 6-2 was used instead of Intermediate 2-4-4.
  • Compound 34 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.88(2H, d), 8.24(2H, s), 8.01(2H, d), 7.26-7.24(1H, m), 5.28-5.23(1H, m), 4.87(1H, s), 3.70-3.59(2H, m), 3.46(3H, s), 1.41-1.37(6H, m).
  • Production Example 35 The compound and its physical properties are shown below, which were produced according to Production Example 2, except that Intermediate 7-4-1 was used instead of Intermediate 2-4-4.
  • Compound 35 of the present invention 1 H-NMR (CDCl 3 ) ⁇ : 8.90(2H, d), 8.21(2H, s), 8.01(1H, s), 7.74(1H, d), 7.32(1H, t), 5.30-5.25(1H, m), 3.60(3H, s), 2.70(3H, s), 1.45(3H, d).
  • Reference production example 1-2-1 To a mixture of 6.0 g of intermediate 1-1-1 and 50 mL of methanol, 4.68 g of formamidine acetate was added, followed by the addition of 8.68 g of sodium methoxide (28 wt % methanol solution), and the mixture was stirred at room temperature for 18 hours. The resulting mixture was concentrated, water was added, and the mixture was extracted with chloroform. The resulting organic layer was washed successively with water and saturated saline, dried over sodium sulfate, filtered, and concentrated. The residue was subjected to silica gel column chromatography to obtain 1.93 g of intermediate 1-2-1 represented by the following formula.
  • Reference production example 4-3-1 To a mixture of 0.66 g of intermediate 2-1-4 and 14 mL of THF, 1.39 g of iodine and 0.79 g of potassium carbonate were added and stirred under heating and reflux for 7 hours. The resulting mixture was allowed to cool to room temperature, and 0.41 g of methyl iodide was added and stirred at 50°C for 5 hours. Water was added to the resulting mixture and extracted with chloroform. The resulting organic layer was washed successively with water and saturated saline. The resulting organic layer was dried over sodium sulfate, filtered and concentrated. The residue was subjected to silica gel column chromatography to obtain 0.88 g of intermediate 4-3-1 represented by the following formula.
  • Reference production example 2-4-3 The compounds and their physical properties are shown below, which were produced according to Reference Production Example 2-4-1 using Intermediate 3-2-1 instead of Intermediate 2-3-1.
  • Intermediate 2-4-3 1 H-NMR (CDCl 3 ) ⁇ : 12.35(1H, s), 8.86(2H, d), 7.23-7.21(1H, m), 5.47-5.13(1H, m), 2.79-2.63(3H, m), 2.43(3H, s), 1.37-1.35(3H, m), 1.28-1.26(9H, m).
  • Reference production example 2-4-5 The compound and its physical properties are shown below, which were produced according to Reference Production Example 2-4-1 using Intermediate 3-3-2 instead of Intermediate 2-3-1.
  • Intermediate 2-4-5 1 H-NMR (CDCl 3 ) ⁇ : 8.86(2H, d), 8.18(1H, s), 7.26-7.24(1H, m), 5.28(1H, d), 4.15-3.94(2H, m), 2.67(3H, s), 1.43-1.42(6H, m), 1.27-1.25(9H, m).
  • Reference production example 2-4-9 The compound and its physical properties are shown below, which were produced according to Reference Production Example 2-4-1 using Intermediate 4-3-4 instead of Intermediate 2-3-1.
  • Reference production example 2-4-10 The compound and its physical properties are shown below, which were produced according to Reference Production Example 2-4-1 using Intermediate 4-3-5 instead of Intermediate 2-3-1.
  • Intermediate 2-4-10 1 H-NMR (CDCl 3 ) ⁇ : 8.86(2H, d), 7.26-7.24(1H, m), 5.38-5.36(1H, m), 4.64(1H, s), 3.73(3H, s), 2.06-2.00(1H, m), 1.39-1.27(14H, m), 1.18-1.16(2H,m).
  • Reference production example 2-4-11 The compound and its physical properties are shown below, which were produced according to Reference Production Example 2-4-1 using Intermediate 4-3-6 instead of Intermediate 2-3-1.
  • Intermediate 2-4-11 1 H-NMR (CDCl 3 ) ⁇ : 8.87(2H, d), 7.28-7.27(1H, m), 5.60-5.59(1H, m), 4.68-4.67(1H, m), 3.57(3H, s), 2.84(2H, q), 1.40-1.29(15H, m).
  • Reference production example 3-2-3 The compound and its physical properties are shown below, which were produced according to Reference Production Example 3-2-1, except that Intermediate 2-1-4 was used instead of Intermediate 2-1-3.
  • Intermediate 3-2-3 1 H-NMR (CDCl 3 ) ⁇ : 8.12 (1H, s), 5.51 (1H, d), 5.15-5.14 (1H, m), 1.44 (9H, s), 1.37 (3H, d).
  • Reference production example 2-4-12 The compound and its physical properties are shown below, which were produced according to Reference Production Example 2-4-1 using Intermediate 3-3-3 instead of Intermediate 2-3-1.
  • Intermediate 2-4-12 1 H-NMR (CDCl 3 ) ⁇ : 8.89 (2H, d), 8.19 (1H, s), 7.30 (1H, t), 5.48 (1H, d), 4.67-4.65 (1H, m), 4.06-3.99 (2H, m), 1.43 (3H, t), 1.39 (9H, s), 1.35 (3H, d).
  • the resulting mixture was concentrated, water was added, and the mixture was extracted with ethyl acetate.
  • the resulting organic layer was washed successively with a saturated aqueous solution of sodium thiosulfate, water, and saturated saline, dried over sodium sulfate, filtered, and concentrated.
  • the resulting residue was dissolved in 22 mL of THF, and 1.90 g of methyl iodide and 2.32 g of potassium carbonate were added and stirred at 50° C. for 2 hours. Further, 1.90 g of methyl iodide was added and stirred at 50° C. for 6 hours.
  • the resulting mixture was concentrated, water was added, and extraction was performed using ethyl acetate.
  • Reference Manufacturing Example 8-2 The compounds and their physical properties are shown below, which were produced according to Reference Production Example 3-2-1, except that Intermediate 8-1 was used instead of Intermediate 2-1-3.
  • Intermediate 8-2 1 H-NMR (CDCl 3 ) ⁇ : 7.36-7.32 (5H, m), 5.90 (1H, d), 5.19-5.11 (3H, m), 2.47 (3H, s), 1.37 (3H, d).
  • Reference Manufacturing Example 8-3 The compounds and their physical properties are shown below, which were produced according to Reference Production Example 3-3-1 using Intermediate 8-2 instead of Intermediate 3-2-1.
  • Intermediate 8-3 1 H-NMR (CDCl 3 ) ⁇ : 7.37-7.32 (5H, m), 5.89 (1H, d), 5.12-5.10 (3H, m), 3.58 (3H, s), 2.51 (3H, s), 1.36 (3H, d).
  • Reference Manufacturing Example 8-4 A mixture of 0.50 g of intermediate 8-3, 0.29 g of 1-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-H-pyrazole, 0.14 g of tetrakistriphenylphosphine palladium(0), 0.75 g of potassium phosphate, and 11.7 mL of toluene was stirred at 110° C. for 9 hours. The resulting mixture was allowed to cool to room temperature, water was added, and the mixture was extracted with chloroform. The resulting organic layer was washed successively with water and saturated saline. The resulting organic layer was dried over sodium sulfate, filtered, and concentrated.
  • Intermediate 8-4 1 H-NMR (CDCl 3 ) ⁇ : 7.40 (1H, d), 7.34-7.31 (5H, m), 6.59 (1H, d), 5.97 (1H, d), 5.20-5.15 (1H, m), 5.09-5.03 (2H, m), 3.93 (3H, s), 3.54 (3H, s), 2.54 (3H, s), 1.40 (3H, d).
  • T 1 is T1-1, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX32).
  • compound group SX33 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX33).
  • T 1 is T1-1, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX34).
  • compound group SX35 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX35).
  • T 1 is T1-2, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX62).
  • compound group SX63 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX63).
  • T 1 is T1-3, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX84).
  • compound group SX84 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX84).
  • T 1 is T1-3, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX85).
  • T 1 is T1-3, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX92).
  • compound group SX92 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX92).
  • compound group SX93 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-3, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX94).
  • compound group SX95 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX95).
  • T 1 is T1-3, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX98).
  • compound group SX99 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX99).
  • T 1 is T1-3, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX100).
  • compound group SX101 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX101).
  • T 1 is T1-3, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX102).
  • compound group SX102 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX102).
  • T 1 is T1-3, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX103).
  • T 1 is T1-3, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX104).
  • compound group SX104 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX104).
  • compound group SX105 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-3, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX108).
  • T 1 is T1-4, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX109).
  • T 1 is T1-4, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX110).
  • compound group SX111 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX111).
  • T 1 is T1-4, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX112).
  • compound group SX112 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX113).
  • T 1 is T1-4, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX114).
  • compound group SX115 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX115).
  • T 1 is T1-4, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX116).
  • compound group SX116 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX116).
  • compound group SX117 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX117).
  • T 1 is T1-4, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX118).
  • compound group SX118 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX118).
  • compound group SX118 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX119).
  • T 1 is T1-4, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX120).
  • compound group SX120 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX120).
  • compound group SX121 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-4, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX122).
  • compound group SX122 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX122).
  • compound group SX123 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX123).
  • T 1 is T1-4, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX124).
  • compound group SX124 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX124).
  • T 1 is T1-4, and R 3 is a methyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX125).
  • T 1 is T1-4, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX126).
  • compound group SX126 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX126).
  • compound group SX127 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX127).
  • T 1 is T1-4, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX128).
  • T 1 is T1-4, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX129).
  • T 1 is T1-4, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX130).
  • compound group SX130 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX131).
  • T 1 is T1-4, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX132).
  • compound group SX133 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX133).
  • T 1 is T1-4, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX134).
  • compound group SX134 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX135).
  • T 1 is T1-4, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX136).
  • compound group SX136 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX136).
  • compound group SX137 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-4, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX138).
  • compound group SX138 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX138).
  • compound group SX139 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-4, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX140).
  • compound group SX141 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX141).
  • T 1 is T1-4, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX142).
  • compound group SX142 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX142).
  • compound group SX143 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-4, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX144).
  • T 1 is T1-5, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX145).
  • T 1 is T1-5, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX146).
  • compound group SX147 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX147).
  • T 1 is T1-5, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX148).
  • compound group SX149 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX149).
  • T 1 is T1-5, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX150).
  • compound group SX150 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX151).
  • T 1 is T1-5, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX152).
  • compound group SX152 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX152).
  • compound group SX153 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-5, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX154).
  • compound group SX154 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX154).
  • compound group SX154 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX154).
  • T 1 is T1-5, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX156).
  • compound group SX156 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX156).
  • compound group SX157 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX157).
  • T 1 is T1-5, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX158).
  • compound group SX158 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX158).
  • T 1 is T1-5, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX159).
  • T 1 is T1-5, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX160).
  • compound group SX160 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX161).
  • T 1 is T1-5, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX162).
  • compound group SX163 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX163).
  • T 1 is T1-5, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX164).
  • compound group SX164 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX164).
  • compound group SX165 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX165).
  • T 1 is T1-5, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX166).
  • compound group SX166 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX167).
  • T 1 is T1-5, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX168).
  • compound group SX168 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX169).
  • T 1 is T1-5, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX170).
  • compound group SX171 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX171).
  • T 1 is T1-5, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX172).
  • compound group SX172 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX172).
  • compound group SX172 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX173).
  • T 1 is T1-5, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX174).
  • compound group SX174 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX175).
  • T 1 is T1-5, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX176).
  • compound group SX177 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX177).
  • T 1 is T1-5, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX178).
  • compound group SX179 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX179).
  • T 1 is T1-5, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX180).
  • T 1 is T1-6, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX181).
  • T 1 is T1-6, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX182).
  • compound group SX183 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX183).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX184).
  • compound group SX184 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX184).
  • compound group SX185 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX185).
  • T 1 is T1-6, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX186).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX187).
  • T 1 is T1-6, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX188).
  • T 1 is T1-6, and R 3 is an ethyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX189).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX190).
  • T 1 is T1-6, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX191).
  • T 1 is T1-6, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX192).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX193).
  • T 1 is T1-6, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX194).
  • T 1 is T1-6, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX195).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX196).
  • compound group SX197 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX197).
  • T 1 is T1-6, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX198).
  • T 1 is T1-6, and R 3 and R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX199).
  • T 1 is T1-6, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX200).
  • compound group SX200 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX200).
  • compound group SX201 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX202).
  • compound group SX203 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX203).
  • T 1 is T1-6, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX204).
  • compound group SX204 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX204).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX205).
  • T 1 is T1-6, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX206).
  • compound group SX207 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX207).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX208).
  • compound group SX208 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX208).
  • T 1 is T1-6, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX209).
  • T 1 is T1-6, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX210).
  • compound group SX210 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX210).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX211).
  • T 1 is T1-6, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX212).
  • compound group SX212 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX212).
  • compound group SX213 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX213).
  • T 1 is T1-6, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX214).
  • compound group SX214 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX214).
  • compound group SX214 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX215).
  • T 1 is T1-6, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX216).
  • T 1 is T1-7, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX217).
  • T 1 is T1-7, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX218).
  • T 1 is T1-7, and R 3 is an ethyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX219).
  • T 1 is T1-7, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX220).
  • compound group SX220 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX220).
  • compound group SX220 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX221).
  • T 1 is T1-7, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX222).
  • compound group SX222 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX222).
  • compound group SX223 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX223).
  • T 1 is T1-7, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX224).
  • compound group SX224 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX224).
  • compound group SX225 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX225).
  • T 1 is T1-7, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX226).
  • T 1 is T1-7, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX227).
  • T 1 is T1-7, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX228).
  • T 1 is T1-7, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX229).
  • T 1 is T1-7, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX230).
  • compound group SX230 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX230).
  • compound group SX230 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX231).
  • T 1 is T1-7, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX232).
  • compound group SX233 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX233).
  • T 1 is T1-7, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX234).
  • T 1 is T1-7, and R 3 and R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX235).
  • T 1 is T1-7, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX238).
  • T 1 is T1-7, and R 3 , R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX239).
  • T 1 is T1-7, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX242).
  • compound group SX243 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX243).
  • T 1 is T1-7, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX244).
  • compound group SX245 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX245).
  • T 1 is T1-7, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX246).
  • T 1 is T1-7, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX247).
  • T 1 is T1-7, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX248).
  • T 1 is T1-7, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX249).
  • T 1 is T1-7, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter referred to as compound group SX250).
  • compound group SX250 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX251).
  • T 1 is T1-7, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX252).
  • T 1 is T1-8, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX253).
  • T 1 is T1-8, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX254).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX255).
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX256).
  • compound group SX257 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX257).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX258).
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX259).
  • T 1 is T1-8, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX260).
  • compound group SX260 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX260).
  • compound group SX261 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX261).
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX262).
  • compound group SX263 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX263).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX264).
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX265).
  • T 1 is T1-8, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX266).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX267).
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX268).
  • T 1 is T1-8, and R 3 is a methyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX269).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX270).
  • compound group SX270 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX270).
  • compound group SX271 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX274).
  • T 1 is T1-8, and R 3 , R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX275).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX276).
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX277).
  • T 1 is T1-8, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX278).
  • compound group SX279 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX279).
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX280).
  • compound group SX280 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX280).
  • compound group SX280 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX281).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX282).
  • compound group SX283 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX283).
  • T 1 is T1-8, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX284).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX285).
  • T 1 is T1-8, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX286).
  • compound group SX287 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX287).
  • T 1 is T1-8, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX288).
  • T 1 is T1-9, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX289).
  • T 1 is T1-9, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX290).
  • compound group SX290 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX291).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX292).
  • compound group SX293 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX293).
  • T 1 is T1-9, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX294).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX295).
  • T 1 is T1-9, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX296).
  • T 1 is T1-9, and R 3 is an ethyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX297).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX298).
  • T 1 is T1-9, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX299).
  • T 1 is T1-9, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX300).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX301).
  • T 1 is T1-9, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX302).
  • compound group SX303 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX303).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX304).
  • compound group SX305 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX305).
  • T 1 is T1-9, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX306).
  • T 1 is T1-9, and R 3 and R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX307).
  • T 1 is T1-9, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX308).
  • T 1 is T1-9, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX309).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX310).
  • compound group SX310 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX311).
  • T 1 is T1-9, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX312).
  • compound group SX313 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX313).
  • T 1 is T1-9, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX314).
  • compound group SX315 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX315).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX316).
  • compound group SX316 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX316).
  • T 1 is T1-9, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX317).
  • T 1 is T1-9, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX318).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX319).
  • T 1 is T1-9, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX320).
  • compound group SX320 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX320).
  • compound group SX320 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX321).
  • T 1 is T1-9, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX322).
  • compound group SX323 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX323).
  • T 1 is T1-9, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX324).
  • T 1 is T1-10, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX325).
  • T 1 is T1-10, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX326).
  • T 1 is T1-10, and R 3 is an ethyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX327).
  • T 1 is T1-10, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX328).
  • compound group SX328 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX328).
  • compound group SX328 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX329).
  • T 1 is T1-10, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX330).
  • compound group SX330 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX331).
  • T 1 is T1-10, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX332).
  • compound group SX333 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX333).
  • T 1 is T1-10, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX334).
  • T 1 is T1-10, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX335).
  • T 1 is T1-10, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX336).
  • T 1 is T1-10, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX337).
  • T 1 is T1-10, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX338).
  • T 1 is T1-10, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX339).
  • T 1 is T1-10, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX340).
  • compound group SX340 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX340).
  • compound group SX340 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX341).
  • T 1 is T1-10, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX342).
  • compound group SX343 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX343).
  • T 1 is T1-10, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX344).
  • compound group SX345 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX345).
  • T 1 is T1-10, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX346).
  • compound group SX347 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX347).
  • T 1 is T1-10, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX348).
  • compound group SX349 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX349).
  • T 1 is T1-10, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX350).
  • compound group SX350 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX351).
  • T 1 is T1-10, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX352).
  • compound group SX353 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX353).
  • T 1 is T1-10, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX356).
  • compound group SX357 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX357).
  • T 1 is T1-11, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX366).
  • compound group SX367 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX367).
  • T 1 is T1-11, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX368).
  • compound group SX369 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX369).
  • T 1 is T1-11, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX370).
  • compound group SX370 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX370).
  • compound group SX370 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX371).
  • T 1 is T1-11, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX372).
  • compound group SX373 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX373).
  • T 1 is T1-11, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX374).
  • T 1 is T1-11, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX375).
  • T 1 is T1-11, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX376).
  • T 1 is T1-11, and R 3 is a methyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX377).
  • T 1 is T1-11, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX378).
  • T 1 is T1-11, and R 3 and R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX379).
  • T 1 is T1-11, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX380).
  • compound group SX380 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX380).
  • compound group SX381 is any one of the substituents described in [Table L1] to [Table L20]
  • T 1 is T1-11, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX382).
  • compound group SX383 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX383).
  • T 1 is T1-11, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX384).
  • compound group SX385 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX385).
  • T 1 is T1-11, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX386).
  • compound group SX387 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX387).
  • T 1 is T1-11, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX388).
  • compound group SX389 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX389).
  • T 1 is T1-11, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX390).
  • compound group SX390 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX390).
  • T 1 is T1-11, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX391).
  • T 1 is T1-11, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX392).
  • compound group SX393 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX393).
  • T 1 is T1-11, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX394).
  • compound group SX395 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX395).
  • T 1 is T1-11, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX396).
  • T 1 is T1-12, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX397).
  • T 1 is T1-12, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX398).
  • T 1 is T1-12, and R 3 is an ethyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX399).
  • T 1 is T1-12, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX400).
  • compound group SX401 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX401).
  • T 1 is T1-12, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX402).
  • compound group SX403 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX403).
  • T 1 is T1-12, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX404).
  • compound group SX404 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX404).
  • compound group SX405 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX405).
  • T 1 is T1-12, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX406).
  • T 1 is T1-12, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX407).
  • T 1 is T1-12, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX408).
  • T 1 is T1-12, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX409).
  • T 1 is T1-12, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX410).
  • compound group SX410 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX410).
  • compound group SX410 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX411).
  • T 1 is T1-12, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX412).
  • compound group SX413 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX413).
  • T 1 is T1-12, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX414).
  • T 1 is T1-12, and R 3 and R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX415).
  • T 1 is T1-12, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX416).
  • T 1 is T1-12, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX417).
  • T 1 is T1-12, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX418).
  • compound group SX419 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX419).
  • T 1 is T1-12, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX420).
  • compound group SX420 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX421).
  • T 1 is T1-12, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX422).
  • compound group SX423 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX423).
  • T 1 is T1-12, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX424).
  • compound group SX425 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX425).
  • T 1 is T1-12, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX426).
  • compound group SX427 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX427).
  • T 1 is T1-12, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX428).
  • compound group SX429 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX429).
  • T 1 is T1-12, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX430).
  • compound group SX431 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX431).
  • T 1 is T1-12, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX432).
  • compound group SX433 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX433).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX434).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX435).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX436).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX437).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX438).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX439).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX440).
  • compound group SX441 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX441).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX442).
  • compound group SX443 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX443).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX444).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX445).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX446).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX447).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX448).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX449).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX450).
  • compound group SX450 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX450).
  • compound group SX451 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX451).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX452).
  • compound group SX453 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX453).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX454).
  • T 1 is T1-13, and R 3 , R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX455).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX456).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX457).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX458).
  • compound group SX459 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX459).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX460).
  • compound group SX460 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX460).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX461).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX462).
  • compound group SX463 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX463).
  • T 1 is T1-13, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX464).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX465).
  • T 1 is T1-13, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX466).
  • compound group SX467 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX467).
  • T 1 is T1-13, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX468).
  • T 1 is T1-14, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX469).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX470).
  • compound group SX470 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX471).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX472).
  • compound group SX473 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX473).
  • T 1 is T1-14, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX474).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX475).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX476).
  • T 1 is T1-14, and R 3 is an ethyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX477).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX478).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX479).
  • T 1 is T1-14, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX480).
  • compound group SX480 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX480).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX481).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX482).
  • compound group SX483 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX483).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX484).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX485).
  • T 1 is T1-14, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX486).
  • T 1 is T1-14, and R 3 and R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX487).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX488).
  • T 1 is T1-14, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX489).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX490).
  • compound group SX490 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX491).
  • T 1 is T1-14, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX492).
  • compound group SX493 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX493).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX494).
  • compound group SX495 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX495).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX496).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX497).
  • T 1 is T1-14, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX498).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX499).
  • T 1 is T1-14, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX500).
  • compound group SX501 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX501).
  • T 1 is T1-14, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX502).
  • compound group SX503 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX503).
  • T 1 is T1-14, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX504).
  • T 1 is T1-15, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX505).
  • T 1 is T1-15, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX508).
  • T 1 is T1-15, and R 3 is a methyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX509).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX510).
  • compound group SX510 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX511).
  • T 1 is T1-15, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX512).
  • compound group SX512 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX512).
  • compound group SX513 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX513).
  • T 1 is T1-15, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX514).
  • T 1 is T1-15, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX515).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX516).
  • T 1 is T1-15, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX517).
  • T 1 is T1-15, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX518).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX519).
  • T 1 is T1-15, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX520).
  • compound group SX520 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX520).
  • compound group SX520 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX521).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX522).
  • compound group SX523 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX523).
  • T 1 is T1-15, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX524).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX525).
  • T 1 is T1-15, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX526).
  • T 1 is T1-15, and R 3 , R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX527).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX528).
  • compound group SX529 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX529).
  • T 1 is T1-15, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX530).
  • compound group SX531 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX531).
  • T 1 is T1-15, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX532).
  • compound group SX533 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX533).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX534).
  • T 1 is T1-15, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX535).
  • T 1 is T1-15, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX536).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX537).
  • T 1 is T1-15, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX538).
  • compound group SX539 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX539).
  • T 1 is T1-15, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX540).
  • T 1 is T1-16, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX541).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX542).
  • compound group SX543 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX543).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX544).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX545).
  • T 1 is T1-16, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX546).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX547).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX548).
  • compound group SX549 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX549).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX550).
  • compound group SX550 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX550).
  • compound group SX551 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX551).
  • T 1 is T1-16, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX552).
  • compound group SX553 In the compound (L-1-1), T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX553).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX554).
  • T 1 is T1-16, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX555).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX556).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX557).
  • T 1 is T1-16, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX558).
  • T 1 is T1-16, and R 3 and R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX559).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX560).
  • compound group SX560 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX560).
  • T 1 is T1-16, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX561).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX562).
  • compound group SX563 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX563).
  • T 1 is T1-16, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX564).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX565).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX566).
  • compound group SX567 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX567).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX568).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX569).
  • T 1 is T1-16, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX570).
  • compound group SX570 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX570).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX571).
  • T 1 is T1-16, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX572).
  • compound group SX573 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX573).
  • T 1 is T1-16, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX574).
  • compound group SX575 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX575).
  • T 1 is T1-16, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX576).
  • T 1 is T1-17, and R 3 , R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX577).
  • T 1 is T1-17, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX578).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX579).
  • T 1 is T1-17, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX580).
  • compound group SX580 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX580).
  • compound group SX580 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX581).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX582).
  • compound group SX583 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX583).
  • T 1 is T1-17, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX584).
  • compound group SX585 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX585).
  • T 1 is T1-17, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX586).
  • T 1 is T1-17, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX587).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX588).
  • T 1 is T1-17, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX589).
  • T 1 is T1-17, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX590).
  • compound group SX590 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX590).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX591).
  • T 1 is T1-17, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX592).
  • compound group SX593 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX593).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX594).
  • T 1 is T1-17, and R 3 and R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX595).
  • T 1 is T1-17, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX596).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX597).
  • T 1 is T1-17, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX598).
  • T 1 is T1-17, and R 3 , R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX599).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX600).
  • compound group SX600 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX601).
  • T 1 is T1-17, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX602).
  • compound group SX603 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX603).
  • T 1 is T1-17, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX604).
  • compound group SX605 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX605).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX606).
  • T 1 is T1-17, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX607).
  • T 1 is T1-17, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX608).
  • compound group SX608 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX609).
  • T 1 is T1-17, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX610).
  • compound group SX610 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX610).
  • compound group SX610 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX611).
  • T 1 is T1-17, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX612).
  • compound group SX613 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX613).
  • T 1 is T1-18, and R 3 is a methyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX614).
  • T 1 is T1-18, and R 3 is an ethyl group, R 4 and R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX615).
  • T 1 is T1-18, and R 3 is a hydrogen atom, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX616).
  • T 1 is T1-18, and R 3 is a methyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX617).
  • T 1 is T1-18, and R 3 is an ethyl group, R 4 is a methyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX618).
  • T 1 is T1-18, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX619).
  • T 1 is T1-18, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX620).
  • compound group SX620 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX621).
  • T 1 is T1-18, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX622).
  • compound group SX623 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX623).
  • T 1 is T1-18, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX624).
  • T 1 is T1-18, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX625).
  • T 1 is T1-18, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX626).
  • T 1 is T1-18, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX627).
  • T 1 is T1-18, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX628).
  • T 1 is T1-18, and R 3 is a methyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX629).
  • T 1 is T1-18, and R 3 is an ethyl group, R 4 is a phenyl group, R 11 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX630).
  • compound group SX630 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX630).
  • compound group SX631 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX631).
  • T 1 is T1-18, and R 3 is a methyl group, R 4 is a hydrogen atom, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX632).
  • compound group SX633 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX633).
  • T 1 is T1-18, and R 3 is a hydrogen atom, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX634).
  • T 1 is T1-18, and R 3 , R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX635).
  • T 1 is T1-18, and R 3 is an ethyl group, R 4 and R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX636).
  • compound group SX636 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX636).
  • compound group SX637 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX637).
  • T 1 is T1-18, and R 3 is a methyl group, R 4 is an ethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX638).
  • compound group SX638 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX639).
  • T 1 is T1-18, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX640).
  • compound group SX640 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX641).
  • T 1 is T1-18, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX642).
  • compound group SX643 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX643).
  • T 1 is T1-18, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX644).
  • T 1 is T1-18, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX645).
  • T 1 is T1-18, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 11 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX646).
  • compound group SX647 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX647).
  • T 1 is T1-18
  • R 3 is an ethyl group
  • R 4 is a phenyl group
  • R 11 is a methyl group
  • R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX648).
  • Formula (L-1-2) (hereinafter, referred to as compound (L-1-2)), in which T2 is T2-1 (# 5 represents a bonding site to a nitrogen atom), R3 and R4 are hydrogen atoms, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents a bonding site to a carbon atom of a heterocycle) (hereinafter, referred to as compound group SX649).
  • T 2 is T2-1, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX650).
  • T 2 is T2-1, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX651).
  • T 2 is T2-1, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX652).
  • T 2 is T2-1, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX653).
  • T 2 is T2-1, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX654).
  • T 2 is T2-1, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX655).
  • T 2 is T2-1, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX656).
  • T 2 is T2-1, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX657).
  • T 2 is T2-1, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX658).
  • T 2 is T2-1, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX659).
  • T 2 is T2-1, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX660).
  • T 2 is T2-1, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX661).
  • T 2 is T2-1, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX662).
  • T 2 is T2-1, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX663).
  • T 2 is T2-1, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX664).
  • T 2 is T2-1, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX665).
  • T 2 is T2-1, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX666).
  • T 2 is T2-2, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX667).
  • T 2 is T2-2, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX668).
  • T 2 is T2-2, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX669).
  • T 2 is T2-2, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX672).
  • T 2 is T2-2, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX673).
  • T 2 is T2-2, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX674).
  • T 2 is T2-2, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX675).
  • T 2 is T2-2, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX676).
  • T 2 is T2-2, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX677).
  • T 2 is T2-2, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX678).
  • T 2 is T2-2, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX679).
  • T 2 is T2-2, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX680).
  • T 2 is T2-2, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX681).
  • T 2 is T2-2, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX682).
  • T 2 is T2-2, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX683).
  • T 2 is T2-2, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX684).
  • T 2 is T2-3, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX685).
  • T 2 is T2-3, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX686).
  • T 2 is T2-3, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX687).
  • T 2 is T2-3, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX688).
  • T 2 is T2-3, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX689).
  • T 2 is T2-3, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX690).
  • T 2 is T2-3, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX691).
  • T 2 is T2-3, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX692).
  • T 2 is T2-3, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX693).
  • T 2 is T2-3, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX694).
  • T 2 is T2-3, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX695).
  • T 2 is T2-3, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX696).
  • T 2 is T2-3, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX697).
  • T 2 is T2-3, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX698).
  • T 2 is T2-3, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX699).
  • T 2 is T2-3, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX700).
  • T 2 is T2-3, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX701).
  • T 2 is T2-3, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX702).
  • T 2 is T2-4, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX703).
  • T 2 is T2-4, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX704).
  • T 2 is T2-4, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX705).
  • T 2 is T2-4, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX706).
  • T 2 is T2-4, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX707).
  • T 2 is T2-4, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX708).
  • T 2 is T2-4, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX709).
  • T 2 is T2-4, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX710).
  • T 2 is T2-4, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX711).
  • T 2 is T2-4, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX712).
  • T 2 is T2-4, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX713).
  • T 2 is T2-4, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX714).
  • T 2 is T2-4, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX715).
  • T 2 is T2-4, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX716).
  • T 2 is T2-4, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX717).
  • T 2 is T2-4, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX718).
  • T 2 is T2-4, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX719).
  • T 2 is T2-4, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX720).
  • T 2 is T2-5, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX721).
  • T 2 is T2-5, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX722).
  • T 2 is T2-5, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX723).
  • T 2 is T2-5, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX724).
  • T 2 is T2-5, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX725).
  • T 2 is T2-5, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX726).
  • T 2 is T2-5, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX727).
  • T 2 is T2-5, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX728).
  • T 2 is T2-5, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX729).
  • T 2 is T2-5, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX730).
  • T 2 is T2-5, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX731).
  • T 2 is T2-5, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX732).
  • T 2 is T2-5, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX733).
  • T 2 is T2-5, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX734).
  • T 2 is T2-5, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX735).
  • T 2 is T2-5, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX736).
  • T 2 is T2-5, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX737).
  • T 2 is T2-5, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX738).
  • T 2 is T2-6, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX739).
  • T 2 is T2-6, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX740).
  • T 2 is T2-6, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX741).
  • T 2 is T2-6, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX742).
  • T 2 is T2-6, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX743).
  • T 2 is T2-6, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX744).
  • T 2 is T2-6, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX745).
  • T 2 is T2-6, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX746).
  • T 2 is T2-6, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX747).
  • T 2 is T2-6, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX748).
  • T 2 is T2-6, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX749).
  • T 2 is T2-6, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX750).
  • T 2 is T2-6, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX751).
  • T 2 is T2-6, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX752).
  • compound group SX753 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX753).
  • T 2 is T2-6, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX754).
  • T 2 is T2-6, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX755).
  • T 2 is T2-6, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX756).
  • T 2 is T2-7, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX757).
  • T 2 is T2-7, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX758).
  • T 2 is T2-7, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX759).
  • T 2 is T2-7, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX760).
  • T 2 is T2-7, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX761).
  • T 2 is T2-7, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX762).
  • T 2 is T2-7, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX763).
  • T 2 is T2-7, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX764).
  • T 2 is T2-7, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX765).
  • T 2 is T2-7, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX766).
  • T 2 is T2-7, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX767).
  • T 2 is T2-7, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX768).
  • T 2 is T2-7, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX769).
  • T 2 is T2-7, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX770).
  • T 2 is T2-7, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX771).
  • T 2 is T2-7, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX772).
  • T 2 is T2-7, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX773).
  • T 2 is T2-7, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX774).
  • T 2 is T2-8, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX775).
  • T 2 is T2-8, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX776).
  • T 2 is T2-8, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX777).
  • T 2 is T2-8, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX778).
  • T 2 is T2-8, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX779).
  • T 2 is T2-8, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX780).
  • T 2 is T2-8, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX781).
  • T 2 is T2-8, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX782).
  • T 2 is T2-8, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX783).
  • T 2 is T2-8, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX784).
  • T 2 is T2-8, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX785).
  • T 2 is T2-8, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX786).
  • T 2 is T2-8, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX787).
  • T 2 is T2-8, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX788).
  • T 2 is T2-8, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX789).
  • T 2 is T2-8, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX790).
  • T 2 is T2-8, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX791).
  • T 2 is T2-8, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX792).
  • T 2 is T2-9, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX793).
  • T 2 is T2-9, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX794).
  • T 2 is T2-9, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX795).
  • T 2 is T2-9, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX796).
  • T 2 is T2-9, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX797).
  • T 2 is T2-9, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX798).
  • T 2 is T2-9, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX799).
  • T 2 is T2-9, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter referred to as compound group SX800).
  • T 2 is T2-9, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX801).
  • T 2 is T2-9, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX802).
  • T 2 is T2-9, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX803).
  • T 2 is T2-9, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX804).
  • T 2 is T2-9, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX805).
  • T 2 is T2-9, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX806).
  • T 2 is T2-9, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX807).
  • T 2 is T2-9, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX808).
  • T 2 is T2-9, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX809).
  • T 2 is T2-9, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX810).
  • T 2 is T2-10, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX811).
  • T 2 is T2-10, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX812).
  • T 2 is T2-10, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX813).
  • T 2 is T2-10, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX814).
  • T 2 is T2-10, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX815).
  • T 2 is T2-10, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX816).
  • T 2 is T2-10, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX817).
  • T 2 is T2-10, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX818).
  • T 2 is T2-10, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX819).
  • T 2 is T2-10, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX820).
  • compound group SX820 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX821).
  • T 2 is T2-10, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX822).
  • T 2 is T2-10, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX823).
  • T 2 is T2-10, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX824).
  • T 2 is T2-10, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX825).
  • T 2 is T2-10, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX826).
  • T 2 is T2-10, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX827).
  • T 2 is T2-10, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX828).
  • T 2 is T2-11, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX829).
  • T 2 is T2-11, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX830).
  • T 2 is T2-11, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX831).
  • T 2 is T2-11, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX832).
  • T 2 is T2-11, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX833).
  • T 2 is T2-11, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX834).
  • T 2 is T2-11, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX835).
  • T 2 is T2-11, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX836).
  • T 2 is T2-11, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX837).
  • T 2 is T2-11, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX838).
  • T 2 is T2-11, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX839).
  • T 2 is T2-11, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX840).
  • T 2 is T2-11, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX841).
  • T 2 is T2-11, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX842).
  • T 2 is T2-11, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX843).
  • T 2 is T2-11, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX844).
  • T 2 is T2-11, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX845).
  • T 2 is T2-11, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX846).
  • T 2 is T2-12, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX847).
  • T 2 is T2-12, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX848).
  • T 2 is T2-12, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX849).
  • T 2 is T2-12, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX850).
  • T 2 is T2-12, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX851).
  • T 2 is T2-12, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX852).
  • T 2 is T2-12, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX853).
  • T 2 is T2-12, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX854).
  • T 2 is T2-12, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX855).
  • T 2 is T2-12, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX856).
  • T 2 is T2-12, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX857).
  • T 2 is T2-12, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX858).
  • T 2 is T2-12, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX859).
  • T 2 is T2-12, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX860).
  • T 2 is T2-12, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX861).
  • T 2 is T2-12, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX862).
  • T 2 is T2-12, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX863).
  • T 2 is T2-12, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX864).
  • T 2 is T2-13, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX865).
  • T 2 is T2-13, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX866).
  • T 2 is T2-13, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX867).
  • T 2 is T2-13, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX868).
  • T 2 is T2-13, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX869).
  • T 2 is T2-13, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX870).
  • T 2 is T2-13, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX871).
  • T 2 is T2-13, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX872).
  • T 2 is T2-13, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX873).
  • T 2 is T2-13, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX874).
  • T 2 is T2-13, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX875).
  • T 2 is T2-13, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX876).
  • T 2 is T2-13, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX877).
  • T 2 is T2-13, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX878).
  • T 2 is T2-13, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX879).
  • T 2 is T2-13, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX880).
  • T 2 is T2-13, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX881).
  • T 2 is T2-13, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX882).
  • T 2 is T2-14, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX883).
  • T 2 is T2-14, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX884).
  • T 2 is T2-14, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX885).
  • T 2 is T2-14, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX886).
  • T 2 is T2-14, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX887).
  • T 2 is T2-14, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX888).
  • T 2 is T2-14, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX889).
  • T 2 is T2-14, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX890).
  • T 2 is T2-14, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX891).
  • T 2 is T2-14, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX892).
  • T 2 is T2-14, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX893).
  • T 2 is T2-14, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX894).
  • T 2 is T2-14, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX895).
  • T 2 is T2-14, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX896).
  • T 2 is T2-14, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX897).
  • T 2 is T2-14, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX898).
  • T 2 is T2-14, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX899).
  • T 2 is T2-14, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX900).
  • T 2 is T2-15, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX901).
  • T 2 is T2-15, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX902).
  • T 2 is T2-15, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX903).
  • T 2 is T2-15, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX904).
  • T 2 is T2-15, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX905).
  • T 2 is T2-15, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX906).
  • T 2 is T2-15, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX907).
  • T 2 is T2-15, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX908).
  • T 2 is T2-15, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX909).
  • T 2 is T2-15, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX910).
  • T 2 is T2-15, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX911).
  • T 2 is T2-15, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX912).
  • T 2 is T2-15, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX913).
  • T 2 is T2-15, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX914).
  • T 2 is T2-15, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX915).
  • T 2 is T2-15, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX916).
  • T 2 is T2-15, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX917).
  • T 2 is T2-15, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX918).
  • T 2 is T2-16, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX919).
  • T 2 is T2-16, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX920).
  • T 2 is T2-16, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX921).
  • T 2 is T2-16, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX922).
  • T 2 is T2-16, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX923).
  • T 2 is T2-16, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX924).
  • T 2 is T2-16, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX925).
  • T 2 is T2-16, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX926).
  • T 2 is T2-16, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX927).
  • T 2 is T2-16, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX928).
  • T 2 is T2-16, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX929).
  • T 2 is T2-16, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX930).
  • T 2 is T2-16, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX931).
  • T 2 is T2-16, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX932).
  • T 2 is T2-16, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX933).
  • T 2 is T2-16, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX934).
  • T 2 is T2-16, and R 3 is a methyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX935).
  • T 2 is T2-16, and R 3 is an ethyl group, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX936).
  • T 2 is T2-17, and R 3 and R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX937).
  • T 2 is T2-17, and R 3 is a methyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX938).
  • T 2 is T2-17, and R 3 is an ethyl group, R 4 is a hydrogen atom, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX939).
  • T 2 is T2-17, and R 3 is a hydrogen atom, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX940).
  • T 2 is T2-17, and R 3 and R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX941).
  • T 2 is T2-17, and R 3 is an ethyl group, R 4 is a methyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX942).
  • T 2 is T2-17, and R 3 is a hydrogen atom, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX943).
  • T 2 is T2-17, and R 3 is a methyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX944).
  • T 2 is T2-17, and R 3 is an ethyl group, R 4 is an ethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX945).
  • T 2 is T2-17, and R 3 is a hydrogen atom, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX946).
  • T 2 is T2-17, and R 3 is a methyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX947).
  • T 2 is T2-17, and R 3 is an ethyl group, R 4 is a cyclopropyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX948).
  • T 2 is T2-17, and R 3 is a hydrogen atom, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX949).
  • T 2 is T2-17, and R 3 is a methyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX950).
  • T 2 is T2-17, and R 3 is an ethyl group, R 4 is a trifluoromethyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX951).
  • T 2 is T2-17, and R 3 is a hydrogen atom, R 4 is a phenyl group, R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX952).
  • compound group SX953 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX953).
  • T 2 is T2-17
  • R 3 is an ethyl group
  • R 4 is a phenyl group
  • R 2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX954).
  • Formula (L-1-3) (hereinafter, referred to as compound (L-1-3)), in which T3 is T3-1 (# 6 represents a bonding site to a nitrogen atom), R3 and R4 are hydrogen atoms, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents a bonding site to a carbon atom of a heterocycle) (hereinafter, referred to as compound group SX955).
  • T3 is T3-1, R3 is a methyl group, R4 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX956).
  • T3 is T3-1, R3 is an ethyl group, R4 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX957).
  • T3 is T3-1
  • R3 is a hydrogen atom
  • R4 is a methyl group
  • R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX958).
  • T3 is T3-1
  • R3 and R4 are methyl groups
  • R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX959).
  • T3 is T3-1, R3 is an ethyl group, R4 is a methyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX960).
  • T3 is T3-1, R3 is a hydrogen atom, R4 is an ethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX961).
  • T3 is T3-1, R3 is a methyl group, R4 is an ethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX962).
  • T3 is T3-1, R3 is an ethyl group, R4 is an ethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX963).
  • T3 is T3-1, R3 is a hydrogen atom, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX964).
  • T3 is T3-1, R3 is a methyl group, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX965).
  • T3 is T3-1
  • R3 is an ethyl group
  • R4 is a cyclopropyl group
  • R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX966).
  • T3 is T3-1
  • R3 is a hydrogen atom
  • R4 is a trifluoromethyl group
  • R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX967).
  • T3 is T3-1, R3 is a methyl group, R4 is a trifluoromethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX968).
  • T3 is T3-1, R3 is an ethyl group, R4 is a trifluoromethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX969).
  • T3 is T3-1
  • R3 is a hydrogen atom
  • R4 is a phenyl group
  • R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX970).
  • T3 is T3-1
  • R3 is a methyl group
  • R4 is a phenyl group
  • R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX971).
  • T3 is T3-1, R3 is an ethyl group, R4 is a phenyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX972).
  • T3 is T3-2, R3 and R4 are hydrogen atoms, and R2 is any one of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX973).
  • T3 is T3-2, R3 is a methyl group, R4 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX974).
  • T3 is T3-2, R3 is an ethyl group, R4 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX975).
  • T3 is T3-2, R3 is a hydrogen atom, R4 is a methyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX976).
  • T3 is T3-2, R3 and R4 are methyl groups, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX977).
  • T3 is T3-2, R3 is an ethyl group, R4 is a methyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX978).
  • T3 is T3-2, R3 is a hydrogen atom, R4 is an ethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX979).
  • T3 is T3-2, R3 is a methyl group, R4 is an ethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX980).
  • T3 is T3-2, R3 is an ethyl group, R4 is an ethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX981).
  • T3 is T3-2, R3 is a hydrogen atom, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX982).
  • T3 is T3-2, R3 is a methyl group, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX983).
  • T3 is T3-2, R3 is an ethyl group, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX984).
  • T3 is T3-2, R3 is a hydrogen atom, R4 is a trifluoromethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX985).
  • T3 is T3-2, R3 is a methyl group, R4 is a trifluoromethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX986).
  • T3 is T3-2, R3 is an ethyl group, R4 is a trifluoromethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX987).
  • T3 is T3-2, R3 is a hydrogen atom, R4 is a phenyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX988).
  • T3 is T3-2, R3 is a methyl group, R4 is a phenyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX989).
  • T3 is T3-2, R3 is an ethyl group, R4 is a phenyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX990).
  • T3 is T3-3, R3 and R4 are hydrogen atoms, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX991).
  • T3 is T3-3, R3 is a methyl group, R4 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX992).
  • T3 is T3-3, R3 is an ethyl group, R4 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX993).
  • T3 is T3-3, R3 is a hydrogen atom, R4 is a methyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX994).
  • T3 is T3-3, R3 and R4 are methyl groups, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX995).
  • T3 is T3-3, R3 is an ethyl group, R4 is a methyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX996).
  • T3 is T3-3, R3 is a hydrogen atom, R4 is an ethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX997).
  • T3 is T3-3, R3 is a methyl group, R4 is an ethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX998).
  • T3 is T3-3, R3 is an ethyl group, R4 is an ethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX999).
  • T3 is T3-3, R3 is a hydrogen atom, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1000).
  • T3 is T3-3, R3 is a methyl group, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1001).
  • T3 is T3-3, R3 is an ethyl group, R4 is a cyclopropyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1002).
  • T3 is T3-3, R3 is a hydrogen atom, R4 is a trifluoromethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1003).
  • T3 is T3-3, R3 is a methyl group, R4 is a trifluoromethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1004).
  • T3 is T3-3, R3 is an ethyl group, R4 is a trifluoromethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1005).
  • T3 is T3-3, R3 is a hydrogen atom, R4 is a phenyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1006).
  • T3 is T3-3, R3 is a methyl group, R4 is a phenyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1007).
  • T3 is T3-3, R3 is an ethyl group, R4 is a phenyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1008).
  • T3 is T3-4, R3 and R4 are hydrogen atoms, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1009).
  • T3 is T3-4, R3 is a methyl group, R4 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1010).
  • T3 is T3-4, R3 is an ethyl group, R4 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1011).
  • T3 is T3-4, R3 is a hydrogen atom, R4 is a methyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1012).
  • T3 is T3-4, R3 and R4 are methyl groups, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1013).
  • T3 is T3-4, R3 is an ethyl group, R4 is a methyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1014).
  • T3 is T3-4, R3 is a hydrogen atom, R4 is an ethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1015).
  • T3 is T3-4, R3 is a methyl group, R4 is an ethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1016).
  • T3 is T3-4, R3 is an ethyl group, R4 is an ethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1017).
  • T3 is T3-4, R3 is a hydrogen atom, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1018).
  • T3 is T3-4, R3 is a methyl group, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1019).
  • T3 is T3-4, R3 is an ethyl group, R4 is a cyclopropyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1020).
  • T3 is T3-4, R3 is a hydrogen atom, R4 is a trifluoromethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1021).
  • T3 is T3-4, R3 is a methyl group, R4 is a trifluoromethyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1022).
  • T3 is T3-4, R3 is an ethyl group, R4 is a trifluoromethyl group, and R2 is any one of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1023).
  • T3 is T3-4, R3 is a hydrogen atom, R4 is a phenyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1024).
  • T3 is T3-4, R3 is a methyl group, R4 is a phenyl group, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1025).
  • T3 is T3-4
  • R3 is an ethyl group
  • R4 is a phenyl group
  • R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1026).
  • Formula (L-3-1) (hereinafter, referred to as compound (L-3-1)), in which T1 is T1-1 (# 4 represents the bonding site to the carbon atom of the carbonyl group), R11 is a hydrogen atom, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX1027).
  • T 1 is T1-1
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1028).
  • T 1 is T1-2, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1029).
  • T 1 is T1-2, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1030).
  • T 1 is T1-3, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1031).
  • T 1 is T1-3, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1032).
  • T 1 is T1-4, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1033).
  • T 1 is T1-4, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1034).
  • T 1 is T1-5
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1035)
  • T 1 is T1-5
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1036).
  • T 1 is T1-6
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1037).
  • T 1 is T1-6
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1038).
  • T 1 is T1-7
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1039).
  • T 1 is T1-7
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1040).
  • T 1 is T1-8, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1041).
  • compound group SX1042 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1042).
  • T 1 is T1-9, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1043).
  • T 1 is T1-9, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1044).
  • T 1 is T1-10, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1045).
  • T 1 is T1-10, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1046).
  • T 1 is T1-11, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Table L1] to [Table L20] (hereinafter, referred to as compound group SX1047).
  • T 1 is T1-11, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1048).
  • T 1 is T1-12
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1049).
  • T 1 is T1-12
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1050).
  • T 1 is T1-13, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1051).
  • compound group SX1052 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1052).
  • T 1 is T1-14, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1053).
  • T 1 is T1-14, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1054).
  • T 1 is T1-15, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1055).
  • T 1 is T1-15, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1056).
  • T 1 is T1-16, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1057).
  • T 1 is T1-16, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1058).
  • T 1 is T1-17, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1059).
  • T 1 is T1-17, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1060).
  • T 1 is T1-18, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1061).
  • compound group SX1062 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1062).
  • Formula (L-3-2) (hereinafter, referred to as compound (L-3-2)), in which T2 is T2-1 (# 5 represents the bonding site to the nitrogen atom) and R2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX1063).
  • T2 is T2-1
  • # 5 represents the bonding site to the nitrogen atom
  • R2 is any of the substituents described in [Tables L1] to [Tables L20]
  • # 3 represents the bonding site to the carbon atom of the condensed ring
  • T 2 is T2-3, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1065).
  • T 2 is T2-4, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1066).
  • T 2 is T2-5, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1067).
  • T 2 is T2-6, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1068).
  • T 2 is T2-7, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1069).
  • T 2 is T2-8, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1070).
  • T 2 is T2-9, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1071).
  • T 2 is T2-10, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1072).
  • T2 is T2-11, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1073).
  • T 2 is T2-12, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1074).
  • T 2 is T2-13, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1075).
  • T 2 is T2-14, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1076).
  • T2 is T2-15, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1077).
  • T2 is T2-16, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1078).
  • T2 is T2-17, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1079).
  • Formula (L-4-1) (hereinafter, referred to as compound (L-4-1)), in which T 1 is T1-1 (# 4 represents the bonding site to the carbon atom of the carbonyl group), R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX1080).
  • T 1 is T1-1
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1081).
  • T 1 is T1-2, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1082).
  • T 1 is T1-2, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1083).
  • T 1 is T1-3, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1084).
  • T 1 is T1-3, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1085).
  • T 1 is T1-4, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1086).
  • T 1 is T1-4, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1087).
  • T 1 is T1-5
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1088).
  • T 1 is T1-5
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1089).
  • T 1 is T1-6, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1090).
  • T 1 is T1-6, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1091).
  • T 1 is T1-7, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1092).
  • T 1 is T1-7, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1093).
  • T 1 is T1-8, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1094).
  • T 1 is T1-8, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1095).
  • T 1 is T1-9, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1096).
  • T 1 is T1-9, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1097).
  • T 1 is T1-10, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1098).
  • T 1 is T1-10, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1099).
  • T 1 is T1-11, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1100).
  • T 1 is T1-11, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1101).
  • T 1 is T1-12, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1102).
  • T 1 is T1-12, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1103).
  • T 1 is T1-13, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1104).
  • T 1 is T1-13, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1105).
  • T 1 is T1-14, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1106).
  • T 1 is T1-14, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1107).
  • T 1 is T1-15, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1108).
  • T 1 is T1-15, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1109).
  • T 1 is T1-16, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1110).
  • T 1 is T1-16, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1111).
  • T 1 is T1-17, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1112).
  • T 1 is T1-17, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1113).
  • T 1 is T1-18, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1114).
  • T 1 is T1-18
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1115).
  • Formula (L-4-2) (hereinafter, referred to as compound (L-4-2)), in which T2 is T2-1 (# 5 represents the bonding site to the nitrogen atom) and R2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX1116).
  • T2 is T2-1
  • # 5 represents the bonding site to the nitrogen atom
  • R2 is any of the substituents described in [Tables L1] to [Tables L20]
  • # 3 represents the bonding site to the carbon atom of the condensed ring
  • T 2 is T2-3, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1118).
  • T 2 is T2-4, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1119).
  • T 2 is T2-5, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1120).
  • T 2 is T2-6 and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1121).
  • T 2 is T2-7, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1122).
  • T 2 is T2-8, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1123).
  • T 2 is T2-9, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1124).
  • T2 is T2-10, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1125).
  • T2 is T2-11, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1126).
  • T 2 is T2-12, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1127).
  • T 2 is T2-13, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1128).
  • T 2 is T2-14, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1129).
  • T2 is T2-15, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1130).
  • T2 is T2-16 and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1131).
  • T 2 is T2-16, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1132).
  • T2 is T2-17, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1133).
  • Formula (L-5-1) (hereinafter, referred to as compound (L-5-1)), in which T 1 is T1-1 (# 4 represents the bonding site to the carbon atom of the carbonyl group), R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the fused ring) (hereinafter, referred to as compound group SX1134).
  • T 1 is T1-1
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1135).
  • T 1 is T1-2, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1136).
  • T 1 is T1-2, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1137).
  • T 1 is T1-3, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1138).
  • T 1 is T1-3, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1139).
  • T 1 is T1-4, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1140).
  • T 1 is T1-4, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1141).
  • T 1 is T1-5
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1142).
  • T 1 is T1-5
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1143).
  • T 1 is T1-6
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1144)
  • T 1 is T1-6
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1145).
  • T 1 is T1-7
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1146)
  • T 1 is T1-7
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1147).
  • T 1 is T1-8, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1148).
  • T 1 is T1-8, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1149).
  • T 1 is T1-9
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1150).
  • T 1 is T1-9
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1151).
  • T 1 is T1-10, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1152).
  • compound group SX1153 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1153).
  • T 1 is T1-11, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1154).
  • T 1 is T1-11, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1155).
  • T 1 is T1-12
  • R 11 is a hydrogen atom
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1156)
  • T 1 is T1-12
  • R 11 is a methyl group
  • R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1157).
  • T 1 is T1-13, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1158).
  • T 1 is T1-13, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1159).
  • T 1 is T1-14, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1160).
  • T 1 is T1-14, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1161).
  • T 1 is T1-15, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1162).
  • compound group SX1163 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1163).
  • T 1 is T1-16, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1164).
  • T 1 is T1-16, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1165).
  • T 1 is T1-17, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1166).
  • T 1 is T1-17, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1167).
  • T 1 is T1-18, R 11 is a hydrogen atom, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1168).
  • T 1 is T1-18, R 11 is a methyl group, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1169).
  • T2 is T2-1 (# 4 represents the bonding site to the carbon atom of the carbonyl group) and R2 is any of the substituents described in [Tables L1] to [Tables L20] (# 3 represents the bonding site to the carbon atom of the condensed ring) (hereinafter, referred to as compound group SX1170).
  • T2 is T2-2 and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1171).
  • T2 is T2-3, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1172).
  • T 2 is T2-4, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1173).
  • T2 is T2-5 and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1174).
  • T2 is T2-6 and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1175).
  • T2 is T2-7 and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1176).
  • T 2 is T2-8, and R 2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1177).
  • T2 is T2-9, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1178).
  • T2 is T2-10, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1179).
  • T2 is T2-11, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1180).
  • T2 is T2-12, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1181).
  • T2 is T2-13, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1182).
  • T2 is T2-14, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1183).
  • T2 is T2-15, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1184).
  • T2 is T2-16, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1185).
  • T2 is T2-17, and R2 is any of the substituents described in [Tables L1] to [Tables L20] (hereinafter, referred to as compound group SX1186).
  • Compound S of the present invention refers to any of the compounds in compound group SX1 to SX1186 or compounds 1 to 37 of the present invention.
  • Formulation Example 1 A mixture of 35 parts of polyoxyethylene alkyl ether sulfate ammonium salt and silica (weight ratio 1:1), 10 parts of any one of the present compound S, and 55 parts of water are mixed and finely pulverized by a wet pulverization method to obtain a preparation.
  • Formulation Example 2 A preparation is obtained by grinding and mixing any one of the present compound S (50 parts), calcium lignosulfonate (3 parts), sodium lauryl sulfate (2 parts), and silica (45 parts).
  • Formulation Example 3 A preparation is obtained by mixing 5 parts of any one of the present compound S, 9 parts of polyoxyethylene styrylphenyl ether, 5 parts of polyoxyethylene decyl ether (number of ethylene oxide added: 5), 6 parts of calcium dodecylbenzenesulfonate, and 75 parts of xylene.
  • Formulation Example 4 2 parts of any one of the present compound S, 1 part of silica, 2 parts of calcium lignosulfonate, 30 parts of bentonite, and 65 parts of kaolin clay are pulverized and mixed, an appropriate amount of water is added, the mixture is kneaded, granulated in a granulator, and then dried to obtain a preparation.
  • Formulation Example 5 10 parts of any one of the present invention compounds S is mixed with a mixture of 18 parts of benzyl alcohol and 9 parts of DMSO, and 6.3 parts of GERONOL (registered trademark) TE250, 2.7 parts of Ethylan (registered trademark) NS-500LQ, and 54 parts of solvent naphtha are added thereto and mixed to obtain a formulation.
  • GERONOL registered trademark
  • TE250 2.3 parts of Ethylan (registered trademark) NS-500LQ
  • solvent naphtha 54 parts of solvent naphtha
  • Formulation Example 6 0.1 parts of any one of the present compound S and 39.9 parts of kerosene are mixed and dissolved, placed in an aerosol container, and filled with 60 parts of liquefied petroleum gas (a mixture of propane, butane and isobutane; saturated vapor pressure: 0.47 MPa (25° C.)) to obtain a formulation.
  • liquefied petroleum gas a mixture of propane, butane and isobutane; saturated vapor pressure: 0.47 MPa (25° C.
  • Formulation Example 7 0.2 parts of any one of the present compound S, 50 parts of pyrethrum extract residue powder, 30 parts of Tabu powder, and 19.8 parts of wood flour are mixed, an appropriate amount of water is added, and the mixture is kneaded. The mixture is then extruded into a plate-shaped sheet, and then wound into a spiral shape using a punching machine to obtain a preparation.
  • Test method 1 A test compound is formulated according to the method described in Formulation Example 1, and water containing 0.03% by volume of Syndyne (registered trademark) is added to the formulation to prepare a dilution containing the test compound at a predetermined concentration.
  • the diluted solution is sprayed at a rate of 20 mL per seedling on cabbage (Brassicaeoleracea) seedlings (at the second to third leaf stage) planted in a container.
  • the stems and leaves of the seedlings are then cut off and placed in a container lined with filter paper. Five second-instar diamondback moth larvae are released into the seedlings. After five days, the number of surviving insects is counted and the mortality rate is calculated using the following formula.
  • Mortality rate (%) (1-number of living insects/5) x 100
  • Test Example 1-1 The prescribed concentration was set at 500 ppm, and tests were carried out according to Test Method 1 using the following compounds of the present invention as test compounds. As a result, all of the following compounds of the present invention showed a mortality rate of 80% or more.
  • Compounds of the present invention 15, 17, 18, 19, 22, 23, 25, 26, 28, 35, 37
  • Test method 2 A test compound is formulated according to the method described in Formulation Example 1, and water containing 0.03% by volume of Syndyne (registered trademark) is added to the formulation to prepare a dilution containing the test compound at a predetermined concentration.
  • the diluted solution is sprayed at a rate of 20 mL per seedling on cabbage (Brassicaeoleracea) seedlings (at the second to third true leaf stage) planted in a container.
  • the stems and leaves of the seedlings are then cut off and placed in a container lined with filter paper. Five second-instar larvae of Spodoptera litura are released into the seedlings. After five days, the number of surviving insects is counted and the mortality rate is calculated using the following formula.
  • Mortality rate (%) (1-number of living insects/5) x 100
  • Test Example 2-1 Tests were carried out according to Test Method 2 using the compounds of the present invention as test compounds at a prescribed concentration of 500 ppm. As a result, all of the compounds of the present invention shown below showed a mortality rate of 80% or more.
  • Test method 3 A test compound is formulated according to the method described in Formulation Example 1, and water containing 0.03% by volume of Syndyne (registered trademark) is added to the formulation to prepare a dilution containing the test compound at a predetermined concentration. Approximately 30 cotton aphids (all stages) are inoculated onto cucumber (Cucumissativus) seedlings (at the second leaf stage) planted in a container. After one day, the diluted solution is sprayed onto the seedlings at a rate of 10 mL per seedling. After another five days, the number of surviving insects is counted, and the control value is calculated according to the following formula.
  • Syndyne registered trademark
  • Control value (%) ⁇ 1 - (Cb x Tai) / (Cai x Tb) ⁇ x 100
  • Cb Number of test insects in untreated area
  • Cai Number of surviving insects at the time of investigation in untreated area
  • Tb Number of test insects in treated area
  • Tai Number of surviving insects at the time of investigation in treated area
  • the untreated area means an area in which the same operation as the treated area is performed except that the test compound is not used.
  • Test Example 3-1 Tests were carried out according to Test Method 3 using the following compounds of the present invention as test compounds at a prescribed concentration of 500 ppm. As a result, all of the following compounds of the present invention showed a control value of 90% or more.
  • Compounds of the present invention 1, 2, 12, 14, 15, 17, 18, 19, 23, 24, 25, 26, 27, 28, 37
  • Test Example 4-1 The test was carried out according to Test Method 4, using the following compounds of the present invention as test compounds, with the given time being 1 hour. As a result, all of the following compounds of the present invention showed a mortality rate of 80% or more.
  • Compounds of the present invention 12, 17, 18, 19, 20, 22, 26, 28, 37
  • Test Example 4-2 The test was carried out according to Test Method 4 using the following compounds of the present invention as test compounds for a given period of 1 day. As a result, all of the following compounds of the present invention showed a mortality rate of 80% or more.
  • Compounds of the present invention 2, 4, 6, 12, 14, 15, 17, 18, 19, 20, 22, 23, 24, 25, 26, 27, 28, 34, 37
  • Test Example 5-1 The test was carried out according to Test Method 5, using the following compounds of the present invention as test compounds, with the given time being 1 hour. As a result, all of the following compounds of the present invention showed a mortality rate of 80% or more.
  • Test Example 5-2 The test was carried out according to Test Method 5 using the following compounds of the present invention as test compounds for a given period of 1 day. As a result, all of the following compounds of the present invention showed a mortality rate of 80% or more.
  • Compounds of the present invention 2, 14, 15, 17, 18, 19, 20, 22, 23, 26, 37
  • Test Example 6-1 The test was carried out according to Test Method 6 using the following compounds of the present invention as test compounds for a predetermined time of 1 hour. As a result, all of the following compounds of the present invention showed a mortality rate of 70% or more.
  • Compounds of the present invention 17, 19, 20
  • Test Example 6-2 The test was carried out according to Test Method 6 using the following compounds of the present invention as test compounds for a given period of 1 day. As a result, all of the following compounds of the present invention showed a mortality rate of 70% or more.
  • Compounds of the present invention 1, 2, 3, 6, 8, 10, 12, 13, 14, 15, 16, 17, 18, 19, 20, 22, 23, 24, 25, 26, 27, 28, 29, 30, 32, 33, 35, 37
  • Test Example 7-1 The prescribed time was set to 1 hour, and the test was carried out according to Test Method 7 using the following compounds of the present invention as test compounds. As a result, the following compounds of the present invention showed a mortality rate of 80% or more.
  • Compounds of the present invention 17, 22, 28
  • Test Example 7-2 The test was carried out for one day according to Test Method 7 using the following compounds of the present invention as test compounds. All of the following compounds of the present invention showed a mortality rate of 80% or more.
  • Compounds of the present invention 2, 17, 20, 22, 27, 28
  • Test Example 7-3 The test was carried out for a period of 3 days according to Test Method 7 using the following compounds of the present invention as test compounds. All of the following compounds of the present invention showed a mortality rate of 80% or more.
  • Compounds of the present invention 2, 17, 20, 22, 27, 28
  • Test Method 8 The test compound is formulated according to the method described in Formulation Example 5, and water is added to the formulation to prepare a diluent containing the test compound at a predetermined concentration.
  • the diluted solution is irrigated at the base of a cucumber (Cucumissativus) seedling (at the second true leaf stage) planted in a container at a rate of 5 mL per seedling. After 7 days, about 30 cotton aphids (all stages) are inoculated onto the leaf surface of the seedling. After another 6 days, the number of surviving insects is counted, and the control value is calculated according to the following formula.
  • Control value (%) ⁇ 1 - (Cb x Tai) / (Cai x Tb) ⁇ x 100
  • Cb Number of test insects in untreated area
  • Cai Number of surviving insects at the time of investigation in untreated area
  • Tb Number of test insects in treated area
  • Tai Number of surviving insects at the time of investigation in treated area
  • the untreated area means an area in which the same operation as the treated area is performed except that the test compound is not used.
  • Test Example 8-1 The effect can be confirmed by carrying out a test according to Test Method 8 using the compound of the present invention as a test compound at a predetermined concentration of 200 ppm.
  • Test Example 9-1 Tests were carried out according to Test Method 9 using the compounds of the present invention as test compounds at a prescribed concentration of 500 ppm. As a result, all of the compounds of the present invention shown below showed a mortality rate of 90% or more.
  • Test Method 10 The test compound is formulated according to the method described in Formulation Example 5, and water containing 0.03% by volume of Syndyne (registered trademark) is added to the formulation to prepare a dilution containing the test compound at a predetermined concentration.
  • Tomato (Lycopersicone sculentum) seedlings planted in a container are released with adult Bemisia tabaci and allowed to lay eggs for about 24 hours.
  • the seedlings are stored for 8 days, and larvae are allowed to hatch from the eggs that have been laid.
  • the diluted solution is sprayed onto the seedlings at a rate of 10 mL per seedling. After 7 days, the number of surviving insects is counted, and the control value is calculated using the following formula.
  • Control value (%) ⁇ 1 - (Cb x Tai) / (Cai x Tb) ⁇ x 100
  • Cb Number of insects in untreated area just before treatment
  • Cai Number of surviving insects at the time of investigation in untreated area
  • Tb Number of insects in treated area just before treatment
  • Tai Number of surviving insects at the time of investigation in treated area
  • the untreated area means an area where the same operation as the treated area is performed except that the test compound is not used.
  • Test Example 10-1 The effect can be confirmed by setting the predetermined concentration at 200 ppm and carrying out a test according to Test Method 10 using the compound of the present invention as a test compound.
  • Test Method 11 The test compound is formulated according to the method described in Formulation Example 1, and water containing 0.03% by volume of Syndyne (registered trademark) is added to the formulation to prepare a dilution containing the test compound at a predetermined concentration. About 40 adult female two-spotted spider mites are released onto a container of kidney bean (Phaseolus vulgaris) seedlings (at the first true leaf stage). After one day, the diluted solution is sprayed onto the seedlings at a rate of 10 mL per seedling. After another seven days, the number of surviving insects is counted, and the control value is calculated according to the following formula.
  • Syndyne registered trademark
  • Control value (%) ⁇ 1 - (Cb x Tai) / (Cai x Tb) ⁇ x 100
  • Cb Number of test insects in untreated area
  • Cai Number of surviving insects at the time of investigation in untreated area
  • Tb Number of test insects in treated area
  • Tai Number of surviving insects at the time of investigation in treated area
  • the untreated area means an area in which the same operation as the treated area is performed except that the test compound is not used.
  • Test Example 11-1 The effect can be confirmed by carrying out a test according to Test Method 11 using the compound of the present invention as a test compound at a predetermined concentration of 500 ppm.
  • Test Example 12-1 The effect can be confirmed by setting the predetermined concentration at 200 ppm and carrying out a test according to Test Method 12 using the compound of the present invention as a test compound.
  • Test Example 13-1 The effect can be confirmed by setting the predetermined concentration at 200 ppm and carrying out a test according to Test Method 13 using the compound of the present invention as a test compound.
  • Test Method 14 The test compound is formulated according to the method described in Formulation Example 5, and water is added to the formulation to prepare a dilution containing the test compound at a predetermined concentration.
  • the diluted solution is irrigated at the base of rice (Oryza sativa) seedlings (at the second leaf stage) planted in a container at a rate of 5 mL per seedling. After 7 days, 20 third-instar larvae of the brown planthopper are released. After another 6 days, the number of surviving insects is counted and the mortality rate is calculated using the following formula.
  • Mortality rate (%) ⁇ 1-number of living insects/20 ⁇ x 100
  • Test Example 14-1 The effect can be confirmed by carrying out a test according to Test Method 14 using the compound of the present invention as a test compound at a predetermined concentration of 500 ppm.
  • Test Method 15 The test compound is formulated according to the method described in Formulation Example 5, and water containing 0.03% by volume of Syndyne (registered trademark) is added to the formulation to prepare a dilution containing the test compound at a predetermined concentration.
  • 2.6 g of artificial feed (Silkmate 2S, Nippon Nosan Kogyo) is placed in a container lined with filter paper.
  • a net inoculated with 100 eggs of the peach fruit moth is placed on the artificial feed.
  • 0.5 mL of the diluted solution is poured onto the eggs. After 10 days, the number of surviving insects is counted and the mortality rate is calculated using the following formula.
  • Untreated group means a group in which the same procedures as those for the treated group are carried out except that the test compound is not used.
  • Test Example 15-1 The effect can be confirmed by setting the predetermined concentration at 200 ppm and carrying out a test according to Test Method 15 using the compound of the present invention as a test compound.
  • Test Example 16-1 The effect can be confirmed by setting the predetermined concentration at 3.5 ppm and carrying out a test according to Test Method 16 using the compound of the present invention as a test compound.
  • Test Example 17-1 The effect can be confirmed by carrying out the test according to Test Method 17 using the compound of the present invention as the test compound for a predetermined period of time of 2 days.
  • Cucumber cotyledonary leaf pieces (1.5 cm long) are placed in each well of a 24-well microplate, 2 wingless adults and 8 larvae of cotton aphids are released per well, and 20 ⁇ L of diluent C is sprayed per well. This is used as a treatment group.
  • 20 ⁇ L of water containing 0.02% by volume of a spreading agent was sprayed onto wells instead of diluent C to serve as an untreated group. After the diluent C has dried, the top of the microplate is covered with a film sheet. After 5 days, the number of surviving insects in each well is counted.
  • the control value is calculated according to the following formula.
  • Control value (%) ⁇ 1 - (Tai) / (Cai) ⁇ x 100
  • the symbols in the formula have the following meanings.
  • Cai Number of surviving insects at the time of investigation in the untreated area
  • Tai Number of surviving insects at the time of investigation in the treated area
  • CompX means any one compound selected from the compound group SX1 to SX1186 and the compounds of the present invention 1 to 37.
  • Dilution solution C in which the concentration of the compound of the present invention is 200 ppm and the concentration of this component is 200 ppm in the combination described in List A.
  • Dilution solution C in which the concentration of the compound of the present invention is 500 ppm and the concentration of this component is 50 ppm in the combination described in List A.
  • Dilution solution C in which the concentration of the compound of the present invention is 500 ppm and the concentration of this component is 5 ppm in the combination described in List A.
  • Dilution solution C in which the concentration of the compound of the present invention is 500 ppm and the concentration of this component is 0.5 ppm in the combination described in List A.
  • comparative test compound 12.01 described in WO 2007/002701.
  • Comparative Test Example 1 The test was carried out according to Test Method 4, with the prescribed time being 1 hour, and using Comparative Test Compound 12.01 as the test compound. As a result, the mortality rate was 20% or less.
  • Comparative Test Example 2 The test was carried out according to Test Method 4, using the comparative test compound 12.01 as the test compound for a predetermined period of time of 1 day, and the mortality rate was 20% or less.
  • Comparative Test Example 3 The test was carried out according to Test Method 5, with the prescribed time being 1 hour, and using Comparative Test Compound 12.01 as the test compound. As a result, the mortality rate was 20% or less.
  • Comparative Test Example 4 The prescribed time period was set to 1 day, and the test was carried out according to Test Method 5 using Comparative Test Compound 12.01 as the test compound. As a result, the mortality rate was 20% or less.
  • Comparative Test Example 5 The test was carried out according to Test Method 7, with the prescribed time being set at 1 hour, and using Comparative Test Compound 12.01 as the test compound. As a result, the mortality rate was 20% or less.
  • Comparative Test Example 6 The prescribed time period was set to 1 day, and the test was carried out according to Test Method 7 using Comparative Test Compound 12.01 as the test compound. As a result, the mortality rate was 20% or less.
  • Comparative Test Example 7 The test was carried out for a period of 3 days according to Test Method 7 using Comparative Test Compound 12.01 as the test compound, and the mortality rate was 20% or less.
  • the compound of the present invention exhibits excellent control effects against harmful arthropods.

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Abstract

L'invention concerne un composé ayant un excellent effet de lutte contre les arthropodes nuisibles. L'invention concerne un composé représenté par la formule (I) [dans laquelle Z représente un atome d'oxygène, ou similaire ; L représente une liaison simple, ou similaire ; R1 représente un groupe hydrocarboné linéaire en C1-C6, ou similaire ; R2 représente un groupe hétérocyclique aromatique à 5 à 6 chaînons, ou similaire ; R3 représente un groupe hydrocarboné linéaire en C1-C6, ou similaire ; R4 représente un atome d'hydrogène, ou similaire ; X représente NR11C(Z)R12, ou similaire ; R11 représente un groupe hydrocarboné linéaire en C1-C6, ou similaire ; et R12 représente un groupe phényle qui peut être substitué par un ou plusieurs substituants, ou similaire] ou un N-oxyde de celui-ci qui a un excellent effet de lutte contre les arthropodes nuisibles.
PCT/JP2024/036103 2023-10-11 2024-10-09 Composé hétérocyclique et composition de lutte contre les arthropodes nuisibles le contenant Pending WO2025079605A1 (fr)

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Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008546843A (ja) * 2005-06-27 2008-12-25 アムゲン インコーポレイティッド 抗炎症性アリールニトリル化合物
JP2012531435A (ja) * 2009-06-25 2012-12-10 アムジエン・インコーポレーテツド ＰＩ３Ｋ阻害剤としての４Ｈ−ピリド［１，２−ａ］ピリミジン−４−オン誘導体
JP2012532131A (ja) * 2009-06-29 2012-12-13 インサイト・コーポレイション Ｐｉ３ｋ阻害剤としてのピリミジノン
JP2022521644A (ja) * 2019-02-28 2022-04-11 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体
WO2023016278A1 (fr) * 2021-08-12 2023-02-16 贵州大学 Composé de pyridinopyrimidinone contenant un isoxazole, son procédé de préparation et son utilisation

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008546843A (ja) * 2005-06-27 2008-12-25 アムゲン インコーポレイティッド 抗炎症性アリールニトリル化合物
JP2012531435A (ja) * 2009-06-25 2012-12-10 アムジエン・インコーポレーテツド ＰＩ３Ｋ阻害剤としての４Ｈ−ピリド［１，２−ａ］ピリミジン−４−オン誘導体
JP2012532131A (ja) * 2009-06-29 2012-12-13 インサイト・コーポレイション Ｐｉ３ｋ阻害剤としてのピリミジノン
JP2022521644A (ja) * 2019-02-28 2022-04-11 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体
WO2023016278A1 (fr) * 2021-08-12 2023-02-16 贵州大学 Composé de pyridinopyrimidinone contenant un isoxazole, son procédé de préparation et son utilisation

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