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WO2009030649A3 - Verfahren zur herstellung von teda-derivaten - Google Patents

Verfahren zur herstellung von teda-derivaten Download PDF

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Publication number
WO2009030649A3
WO2009030649A3 PCT/EP2008/061393 EP2008061393W WO2009030649A3 WO 2009030649 A3 WO2009030649 A3 WO 2009030649A3 EP 2008061393 W EP2008061393 W EP 2008061393W WO 2009030649 A3 WO2009030649 A3 WO 2009030649A3
Authority
WO
WIPO (PCT)
Prior art keywords
derivatives
teda
producing
producing teda
relates
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/EP2008/061393
Other languages
English (en)
French (fr)
Other versions
WO2009030649A2 (de
Inventor
Gunther Van Cauwenberge
Johann-Peter Melder
Joachim-Thierry Anders
Christoph Benisch
Rainer Klopsch
Gregor Daun
Christian Dully
Boris Buschhaus
Henning Boeckemeier
Evelyn Pox
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Priority to EP08803391A priority Critical patent/EP2197882A2/de
Priority to US12/676,254 priority patent/US20100204438A1/en
Priority to CN200880114421A priority patent/CN101842375A/zh
Publication of WO2009030649A2 publication Critical patent/WO2009030649A2/de
Publication of WO2009030649A3 publication Critical patent/WO2009030649A3/de
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Die vorliegende Erfindung betrifft ein Verfahren zur Herstellung von Triethylendiamin- (TEDA)-Derivaten umfassend die folgenden Schritte: a) Reaktion eines Dihydropyrazins mit einem Olefin, b) gegebenenfalls eine Hydrierung in Anschluss an Schritt a). Weiterhin betrifft die vorliegende Erfindung auch neue TEDA-Derivate als solche sowie deren Verwendung als einbaubare Polyurethan-Katalysatoren.
PCT/EP2008/061393 2007-09-03 2008-08-29 Verfahren zur herstellung von teda-derivaten Ceased WO2009030649A2 (de)

Priority Applications (3)

Application Number Priority Date Filing Date Title
EP08803391A EP2197882A2 (de) 2007-09-03 2008-08-29 Verfahren zur herstellung von teda-derivaten
US12/676,254 US20100204438A1 (en) 2007-09-03 2008-08-29 Method for producing teda derivatives
CN200880114421A CN101842375A (zh) 2007-09-03 2008-08-29 制备teda衍生物的方法

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07115513.9 2007-09-03
EP07115513 2007-09-03

Publications (2)

Publication Number Publication Date
WO2009030649A2 WO2009030649A2 (de) 2009-03-12
WO2009030649A3 true WO2009030649A3 (de) 2009-10-01

Family

ID=40130546

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2008/061393 Ceased WO2009030649A2 (de) 2007-09-03 2008-08-29 Verfahren zur herstellung von teda-derivaten

Country Status (4)

Country Link
US (1) US20100204438A1 (de)
EP (1) EP2197882A2 (de)
CN (1) CN101842375A (de)
WO (1) WO2009030649A2 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2295438T5 (pl) 2008-05-30 2025-07-07 Tosoh Corporation Sposób wytwarzania kompozycji zawierającej hydroksyalkilotrietylenodiaminę i kompozycja katalizatora do wytwarzania żywicy poliuretanowej z zastosowaniem kompozycji hydroksyalkilotrietylenodiaminy
MY150768A (en) 2008-12-19 2014-02-28 Basf Se Method for producing pure triethanolamine (teoa)
ES2955137T3 (es) 2013-03-14 2023-11-28 Alkermes Pharma Ireland Ltd Profármacos de fumaratos y su uso en el tratamiento de diversas enfermedades
US8669281B1 (en) 2013-03-14 2014-03-11 Alkermes Pharma Ireland Limited Prodrugs of fumarates and their use in treating various diseases
AU2015218587B2 (en) 2014-02-24 2017-04-27 Alkermes Pharma Ireland Limited Sulfonamide and sulfinamide prodrugs of fumarates and their use in treating various diseases

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3048031A1 (de) * 1979-12-21 1981-09-17 Firmenich S.A., 1211 Genève Verfahren zur herstellung substituierter pyrazine
WO1998024790A1 (fr) * 1996-12-04 1998-06-11 Synthelabo Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-ylmethyle, leur preparation et leur application en therapeutique
WO2001002404A2 (de) * 1999-07-05 2001-01-11 Performance Chemicals Handels Gmbh Verfahren zur herstellung von triethylendiamin unter einsatz von ethylendiamin
WO2003004499A1 (de) * 2001-07-05 2003-01-16 Basf Aktiengesellschaft Verfahren zur selektiven synthese von triethylendiamin
DE10321565A1 (de) * 2003-05-14 2004-12-02 Symrise Gmbh & Co. Kg Verfahren zur Herstellung von Alkyldihydro-1,4-diazinen und Alkyl-1,4-diazinen

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6147185A (en) * 1999-07-23 2000-11-14 Air Products And Chemicals, Inc. 1,4-diazabicyclo[2.2.2]octane compounds and their use for the production of polyurethanes

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3048031A1 (de) * 1979-12-21 1981-09-17 Firmenich S.A., 1211 Genève Verfahren zur herstellung substituierter pyrazine
WO1998024790A1 (fr) * 1996-12-04 1998-06-11 Synthelabo Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-ylmethyle, leur preparation et leur application en therapeutique
WO2001002404A2 (de) * 1999-07-05 2001-01-11 Performance Chemicals Handels Gmbh Verfahren zur herstellung von triethylendiamin unter einsatz von ethylendiamin
WO2003004499A1 (de) * 2001-07-05 2003-01-16 Basf Aktiengesellschaft Verfahren zur selektiven synthese von triethylendiamin
DE10321565A1 (de) * 2003-05-14 2004-12-02 Symrise Gmbh & Co. Kg Verfahren zur Herstellung von Alkyldihydro-1,4-diazinen und Alkyl-1,4-diazinen

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
TOHRU OISHI: "Synthesis of chiral 2,3-disubstituted 1,4-Diazabicyclo[2.2.2]octane.New ligand for the Osmium-catalyzed Asymmetric Dihydrohylation of Olefins.", TETRAHEDRON LETTERS, vol. 33, no. 5, 1992, NLELSEVIER, AMSTERDAM, pages 639 - 642, XP002512485 *

Also Published As

Publication number Publication date
EP2197882A2 (de) 2010-06-23
US20100204438A1 (en) 2010-08-12
CN101842375A (zh) 2010-09-22
WO2009030649A2 (de) 2009-03-12

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