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WO2008126797A1 - 微粉砕化有機化合物粒子の製造方法 - Google Patents

微粉砕化有機化合物粒子の製造方法 Download PDF

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Publication number
WO2008126797A1
WO2008126797A1 PCT/JP2008/056799 JP2008056799W WO2008126797A1 WO 2008126797 A1 WO2008126797 A1 WO 2008126797A1 JP 2008056799 W JP2008056799 W JP 2008056799W WO 2008126797 A1 WO2008126797 A1 WO 2008126797A1
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WO
WIPO (PCT)
Prior art keywords
organic compound
compound particle
poorly water
producing
medical use
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/JP2008/056799
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English (en)
French (fr)
Inventor
Takashi Hirokawa
Takahiro Tada
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Activus Pharma Co Ltd
Original Assignee
Activus Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to KR1020097014759A priority Critical patent/KR101369061B1/ko
Priority to CA2679929A priority patent/CA2679929C/en
Priority to JP2009509328A priority patent/JP5317960B2/ja
Priority to IL223087A priority patent/IL223087A/en
Priority to ES08739905.1T priority patent/ES2563979T3/es
Application filed by Activus Pharma Co Ltd filed Critical Activus Pharma Co Ltd
Priority to EP08739905.1A priority patent/EP2143423B1/en
Priority to CN2008800084620A priority patent/CN101636150B/zh
Publication of WO2008126797A1 publication Critical patent/WO2008126797A1/ja
Priority to US12/585,786 priority patent/US8226983B2/en
Priority to IL201169A priority patent/IL201169A/en
Anticipated expiration legal-status Critical
Priority to US13/484,460 priority patent/US20120237768A1/en
Ceased legal-status Critical Current

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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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Abstract

　本発明は、難水溶性であり、かつ、結晶性である有機化合物の微粉砕化粒子の製造方法、及び、該製造方法により製造された微粉砕化有機化合物粒子の提供することを目的とする。特に、本発明は、難水溶性医療用有機化合物を、生理学的に許容される塩及び生理学的に許容されるポリオールと混合して、前記有機化合物を湿式粉砕することを特徴とする、難水溶性医療用有機化合物微粒子の製造方法、及び該製造方法により得られる難水溶性医療用有機化合物微粒子を提供することを目的とする。
PCT/JP2008/056799 2007-04-06 2008-04-04 微粉砕化有機化合物粒子の製造方法 Ceased WO2008126797A1 (ja)

Priority Applications (10)

Application Number Priority Date Filing Date Title
EP08739905.1A EP2143423B1 (en) 2007-04-06 2008-04-04 Method for producing pulverized organic compound particle
CA2679929A CA2679929C (en) 2007-04-06 2008-04-04 Method for producing finely pulverized organic compound particle
JP2009509328A JP5317960B2 (ja) 2007-04-06 2008-04-04 微粉砕化有機化合物粒子の製造方法
IL223087A IL223087A (en) 2007-04-06 2008-04-04 Finely pulverized organic compound particles
ES08739905.1T ES2563979T3 (es) 2007-04-06 2008-04-04 Método para producción de partículas de compuesto orgánico pulverizadas
KR1020097014759A KR101369061B1 (ko) 2007-04-06 2008-04-04 미분쇄화 유기 화합물 입자의 제조 방법
CN2008800084620A CN101636150B (zh) 2007-04-06 2008-04-04 难水溶性医疗用有机化合物微粒子的制造方法
US12/585,786 US8226983B2 (en) 2007-04-06 2009-09-24 Method for producing pulverized organic compound particle
IL201169A IL201169A (en) 2007-04-06 2009-09-24 A method for producing crushed particles of organic compound
US13/484,460 US20120237768A1 (en) 2007-04-06 2012-05-31 Method for producing pulverized organic compound particle

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JP2007-100902 2007-04-06
JP2007100902 2007-04-06
JP2007210370 2007-08-10
JP2007-210370 2007-08-10

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EP (2) EP2143423B1 (ja)
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CN (1) CN101636150B (ja)
CA (1) CA2679929C (ja)
ES (1) ES2563979T3 (ja)
HU (1) HUE028529T2 (ja)
IL (2) IL223087A (ja)
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WO2010052896A1 (ja) * 2008-11-04 2010-05-14 日揮株式会社 プロピオン酸フルチカゾンを含む局所投与剤
WO2011001214A1 (en) * 2009-06-30 2011-01-06 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi Surface amorphization of phenprobamate
WO2011118960A2 (ko) 2010-03-22 2011-09-29 (주)바이오시네틱스 나노입자 제조방법
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