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WO2008111474A1 - インドール化合物の製造方法 - Google Patents

インドール化合物の製造方法 Download PDF

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Publication number
WO2008111474A1
WO2008111474A1 PCT/JP2008/054016 JP2008054016W WO2008111474A1 WO 2008111474 A1 WO2008111474 A1 WO 2008111474A1 JP 2008054016 W JP2008054016 W JP 2008054016W WO 2008111474 A1 WO2008111474 A1 WO 2008111474A1
Authority
WO
WIPO (PCT)
Prior art keywords
indole compound
oco
amount
active carbon
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/JP2008/054016
Other languages
English (en)
French (fr)
Inventor
Masahiko Hayashi
Yukiko Nomura
Juichi Yanagi
Tatsuo Fujii
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kobe University NUC
Japan Enviro Chemicals Ltd
Original Assignee
Kobe University NUC
Japan Enviro Chemicals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kobe University NUC, Japan Enviro Chemicals Ltd filed Critical Kobe University NUC
Publication of WO2008111474A1 publication Critical patent/WO2008111474A1/ja
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J21/00—Catalysts comprising the elements, oxides, or hydroxides of magnesium, boron, aluminium, carbon, silicon, titanium, zirconium, or hafnium
    • B01J21/18—Carbon
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2235/00—Indexing scheme associated with group B01J35/00, related to the analysis techniques used to determine the catalysts form or properties

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Indole Compounds (AREA)
  • Catalysts (AREA)
  • Carbon And Carbon Compounds (AREA)

Abstract

　本発明は、インドリン化合物を、式（Ｉ）を満たす活性炭からなる触媒の存在下酸素と接触させるインドール化合物の製造方法である。 ４０００<Ｓ×（Ｏｃｏ）　　　　　　　（Ｉ） 　但し、ＳはＢＥＴ比表面積（ｍ２／ｇ）を、Ｏｃｏは加熱により一酸化炭素として脱離する表面酸素量の活性炭に対する重量％を示す。 　この方法によれば、インドメタシンのような医薬品、または染料の骨格成分としても重要なインドール化合物を廉価、安全且つ効率よく製造することができる。
PCT/JP2008/054016 2007-03-09 2008-03-06 インドール化合物の製造方法 Ceased WO2008111474A1 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007059414A JP2008222576A (ja) 2007-03-09 2007-03-09 インドール化合物の製造方法
JP2007-059414 2007-03-09

Publications (1)

Publication Number Publication Date
WO2008111474A1 true WO2008111474A1 (ja) 2008-09-18

Family

ID=39759416

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2008/054016 Ceased WO2008111474A1 (ja) 2007-03-09 2008-03-06 インドール化合物の製造方法

Country Status (2)

Country Link
JP (1) JP2008222576A (ja)
WO (1) WO2008111474A1 (ja)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8889730B2 (en) 2012-04-10 2014-11-18 Pfizer Inc. Indole and indazole compounds that activate AMPK
US9394285B2 (en) 2013-03-15 2016-07-19 Pfizer Inc. Indole and indazole compounds that activate AMPK
CN106432040A (zh) * 2016-08-09 2017-02-22 中钢集团鞍山热能研究院有限公司 医药中间体5‑溴吲哚的一种绿色合成方法
CN106966950A (zh) * 2017-04-17 2017-07-21 兰州大学 药物中间体5‑溴吲哚的一种制备方法
CN119018891A (zh) * 2024-08-16 2024-11-26 福建省鑫森炭业股份有限公司 一种以农作物秸秆为原料制备活性炭的方法及其应用

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS51110561A (ja) * 1975-03-25 1976-09-30 Mitsui Toatsu Chemicals Indooruseizoho
JP2005145859A (ja) * 2003-11-13 2005-06-09 Nippon Steel Chem Co Ltd 脱水素化方法及び芳香族複素環化合物の製造方法
WO2006028035A1 (ja) * 2004-09-06 2006-03-16 Japan Envirochemicals, Ltd. 酸化反応触媒およびそれを用いた化合物の製法

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS51110561A (ja) * 1975-03-25 1976-09-30 Mitsui Toatsu Chemicals Indooruseizoho
JP2005145859A (ja) * 2003-11-13 2005-06-09 Nippon Steel Chem Co Ltd 脱水素化方法及び芳香族複素環化合物の製造方法
WO2006028035A1 (ja) * 2004-09-06 2006-03-16 Japan Envirochemicals, Ltd. 酸化反応触媒およびそれを用いた化合物の製法

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8889730B2 (en) 2012-04-10 2014-11-18 Pfizer Inc. Indole and indazole compounds that activate AMPK
US9394285B2 (en) 2013-03-15 2016-07-19 Pfizer Inc. Indole and indazole compounds that activate AMPK
CN106432040A (zh) * 2016-08-09 2017-02-22 中钢集团鞍山热能研究院有限公司 医药中间体5‑溴吲哚的一种绿色合成方法
CN106432040B (zh) * 2016-08-09 2019-02-19 中钢集团鞍山热能研究院有限公司 医药中间体5-溴吲哚的一种绿色合成方法
CN106966950A (zh) * 2017-04-17 2017-07-21 兰州大学 药物中间体5‑溴吲哚的一种制备方法
CN119018891A (zh) * 2024-08-16 2024-11-26 福建省鑫森炭业股份有限公司 一种以农作物秸秆为原料制备活性炭的方法及其应用

Also Published As

Publication number Publication date
JP2008222576A (ja) 2008-09-25

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