WO2001058920A3 - Procede de production selective d'un anomere derive d'un sucre 1-phosphoryle - Google Patents

Procede de production selective d'un anomere derive d'un sucre 1-phosphoryle Download PDF

Info

Publication number: WO2001058920A3
Authority: WO; WIPO (PCT)
Prior art keywords: producing; nucleoside; sugar derivative; phosphorylated sugar; anomer
Prior art date: 2000-02-10
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Ceased

Application number

PCT/JP2001/000968

Other languages

English (en)

French (fr)

Other versions

WO2001058920A2 (en

Inventor

Hironori Komatsu

Hirokazu Awano

Nobuyuki Fukazawa

Kiyoshi Ito

Ichirou Ikeda

Tadashi Araki

Takeshi Nakamura

Tamotsu Asano

Junya Fujiwara

Tomoyuki Ando

Katsutoshi Tsuchiya

Kyoko Maruyama

Hideki Umetani

Takahiro Yamauchi

Hitoki Miyake

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Mitsui Chemicals Inc

Original Assignee

Mitsui Chemicals Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-02-10

Filing date

2001-02-13

Publication date

2001-11-08

2001-02-13 Application filed by Mitsui Chemicals Inc filed Critical Mitsui Chemicals Inc

2001-02-13 Priority to BR0104461-3A priority Critical patent/BR0104461A/pt

2001-02-13 Priority to DE60134196T priority patent/DE60134196D1/de

2001-02-13 Priority to CA002366513A priority patent/CA2366513A1/en

2001-02-13 Priority to EP01904386A priority patent/EP1178051B1/en

2001-02-13 Priority to US09/958,305 priority patent/US7038039B2/en

2001-08-16 Publication of WO2001058920A2 publication Critical patent/WO2001058920A2/ja

2001-11-08 Publication of WO2001058920A3 publication Critical patent/WO2001058920A3/ja

2002-08-10 Anticipated expiration legal-status Critical

2005-11-28 Priority to US11/287,212 priority patent/US20060094869A1/en

Status Ceased legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H11/00—Compounds containing saccharide radicals esterified by inorganic acids; Metal salts thereof
- C07H11/04—Phosphates; Phosphites; Polyphosphates
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/06—Pyrimidine radicals
- C07H19/10—Pyrimidine radicals with the saccharide radical esterified by phosphoric or polyphosphoric acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
- C07H19/20—Purine radicals with the saccharide radical esterified by phosphoric or polyphosphoric acids

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Saccharide Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

PCT/JP2001/000968 2000-02-10 2001-02-13 Process for selectively producing 1-phosphorylated sugar derivative anomer and process for producing nucleoside Ceased WO2001058920A2 (en)

Priority Applications (6)

Application Number	Priority Date	Filing Date	Title
BR0104461-3A BR0104461A (pt)	2000-02-10	2001-02-13	Processo seletivo para produzir um anÈmero a partir de um derivado de sacarìdeo 1-fosforilado e processo para produzir um nucleosìdeo
DE60134196T DE60134196D1 (de)	2000-02-10	2001-02-13	Verfahren zur selektiven herstellung eines 1-phosphoryliertem zuckerderivativ-anomers und verfahren zur herstellung von nukleosiden
CA002366513A CA2366513A1 (en)	2000-02-10	2001-02-13	Process for selectively producing 1-phosphorylated sugar derivative anomer and process for producing a nucleoside
EP01904386A EP1178051B1 (en)	2000-02-10	2001-02-13	Process for selectively producing 1-phosphorylated sugar derivative anomer and process for producing nucleoside
US09/958,305 US7038039B2 (en)	2000-02-10	2001-02-13	Process for selectively producing 1-phosphorylated sugar derivative anomer and process for producing nucleoside
US11/287,212 US20060094869A1 (en)	2000-02-10	2005-11-28	Selective process for producing an anomer of a 1-phosphorylated saccharide derivative and process for producing a nucleoside

Applications Claiming Priority (6)

Application Number	Priority Date	Filing Date	Title
JP2000-33212		2000-02-10
JP2000033212		2000-02-10
JP2000067333		2000-03-10
JP2000-67333		2000-03-10
JP2000341960		2000-11-09
JP2000-341960		2000-11-09

Related Child Applications (1)

Application Number	Title	Priority Date	Filing Date
US11/287,212 Division US20060094869A1 (en)	2000-02-10	2005-11-28	Selective process for producing an anomer of a 1-phosphorylated saccharide derivative and process for producing a nucleoside

Publications (2)

Publication Number	Publication Date
WO2001058920A2 WO2001058920A2 (en)	2001-08-16
WO2001058920A3 true WO2001058920A3 (fr)	2001-11-08

Family

ID=27342316

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PCT/JP2001/000968 Ceased WO2001058920A2 (en)	2000-02-10	2001-02-13	Process for selectively producing 1-phosphorylated sugar derivative anomer and process for producing nucleoside

Country Status (10)

Country	Link
US (2)	US7038039B2 (ja)
EP (1)	EP1178051B1 (ja)
JP (1)	JP2010031037A (ja)
KR (1)	KR100517163B1 (ja)
CN (1)	CN1372564A (ja)
AT (1)	ATE397001T1 (ja)
BR (1)	BR0104461A (ja)
CA (1)	CA2366513A1 (ja)
DE (1)	DE60134196D1 (ja)
WO (1)	WO2001058920A2 (ja)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2002031176A1 (fr) *	2000-10-12	2002-04-18	Mitsui Chemicals, Inc.	Procédé permettant la production de nucléosides
WO2002051852A1 (fr) *	2000-12-27	2002-07-04	Mitsui Chemicals, Inc.	Procede de production d'un derive de saccharide non naturel
JP2003055392A (ja) *	2001-08-08	2003-02-26	Mitsui Chemicals Inc	１−リン酸化糖の製造法並びにヌクレオシドの製造法
EP1676853A4 (en) *	2003-10-24	2009-12-23	Yamasa Corp	ALPHA-1-PHOSPHORYL-2-DESOXY-2-FLUOROARABINOSIDE AND PROCESS FOR PRODUCING 2'-DESOXY-2'-FLUORO-BETA-D-ARABINONUCLEOSIDE
JP4518867B2 (ja) *	2004-08-18	2010-08-04	三井化学株式会社	２’−デオキシリボース−１−リン酸２アンモニウム塩の製造方法
PT1932918E (pt) *	2006-12-15	2010-01-05	Explora Lab Sa	Método para a produção de cladribina
SG10201600836PA (en) *	2011-02-03	2016-03-30	Mirna Therapeutics Inc	Synthetic mimics of mir-34
EP2679593B1 (en) *	2012-06-26	2018-03-21	Umicore AG & Co. KG	Method for preparation of a ruthenium indenylidene complex
WO2020014041A1 (en)	2018-07-09	2020-01-16	Merck Sharp & Dohme Corp.	Enzymatic synthesis of 4'-ethynyl nucleoside analogs
DE102023123718A1 (de)	2023-09-04	2025-03-06	CHIRACON Pharma GmbH	Verfahren zur Herstellung von Nukleosiden

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US5770407A (en) *	1996-12-10	1998-06-23	The Scripps Research Institute	Process for preparing nucleotide inhibitors of glycosyltransferases

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WO2002051852A1 (fr) *	2000-12-27	2002-07-04	Mitsui Chemicals, Inc.	Procede de production d'un derive de saccharide non naturel

2001
- 2001-02-13 US US09/958,305 patent/US7038039B2/en not_active Expired - Fee Related
- 2001-02-13 AT AT01904386T patent/ATE397001T1/de not_active IP Right Cessation
- 2001-02-13 BR BR0104461-3A patent/BR0104461A/pt not_active IP Right Cessation
- 2001-02-13 DE DE60134196T patent/DE60134196D1/de not_active Expired - Lifetime
- 2001-02-13 WO PCT/JP2001/000968 patent/WO2001058920A2/ja not_active Ceased
- 2001-02-13 EP EP01904386A patent/EP1178051B1/en not_active Expired - Lifetime
- 2001-02-13 CN CN01800874A patent/CN1372564A/zh active Pending
- 2001-02-13 CA CA002366513A patent/CA2366513A1/en not_active Abandoned
- 2001-02-13 KR KR10-2001-7012917A patent/KR100517163B1/ko not_active Expired - Fee Related
2005
- 2005-11-28 US US11/287,212 patent/US20060094869A1/en not_active Abandoned
2009
- 2009-11-02 JP JP2009252470A patent/JP2010031037A/ja active Pending

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Also Published As

Publication number	Publication date
DE60134196D1 (de)	2008-07-10
US20020193314A1 (en)	2002-12-19
ATE397001T1 (de)	2008-06-15
KR20020013524A (ko)	2002-02-20
EP1178051A4 (en)	2003-05-28
US20060094869A1 (en)	2006-05-04
BR0104461A (pt)	2002-08-06
KR100517163B1 (ko)	2005-09-26
WO2001058920A2 (en)	2001-08-16
US7038039B2 (en)	2006-05-02
JP2010031037A (ja)	2010-02-12
EP1178051A2 (en)	2002-02-06
EP1178051B1 (en)	2008-05-28
CA2366513A1 (en)	2001-08-16
CN1372564A (zh)	2002-10-02

Publication	Publication Date	Title
WO2001058920A3 (fr)	2001-11-08	Procede de production selective d'un anomere derive d'un sucre 1-phosphoryle
NZ323855A (en)	1999-11-29	Method and compositions for the synthesis of dioxolane nucleosides particularly the beta-configuration of the 1,3-dioxolane sugar rings
Yoshikawa et al.	1991	A new type of antisweet principles occurring in Gymnema sylvestre
AR036169A1 (es)	2004-08-18	Procedimiento para la elaboracion de tagatosa
WO1998040390A3 (de)	1999-01-14	Oligosaccharide und deren derivate sowie ein chemo-enzymatisches verfahren zu deren herstellung
DK0740706T3 (da)	2006-02-13	Fremstilling af acariogene sukkererstatningsstoffer
AzUMA et al.	1977	Transnucleosidation: an improved method for transglycosylation from pyrimidines to purines
AU2001284529A1 (en)	2002-03-26	Process for producing purified anthocyanin and crystalline anthocyanin
Tanimori et al.	2002	An efficient chemical synthesis of nicotinamide riboside (NAR) and analogues
PT1133511E (pt)	2003-06-30	Novos intermediarios e processo para preparar um agente antibiotico macrolido a partir deles
WO2005014608A3 (en)	2005-08-11	Process for preparing maltitol enriched products
Chida et al.	1999	Pd-catalyzed coupling reaction of glycosylamines with 6-chloropurines: synthesis of 6-(β-D-mannopyranosylamino)-9H-purine and its β-D-gluco isomer, N-glycoside models for spicamycin and septacidin
CA2027861A1 (en)	1991-04-18	Method for preparing cellobiose
CA2332974A1 (en)	1999-12-16	Morphine-6-glucuronide synthesis
WO2007027564A3 (en)	2007-06-07	Process for preparing gemcitabine and associated intermediates
Colombo et al.	2000	Glycoglycerolipid analogues active as anti-tumor-promoters: The influence of the anomeric configuration
CA2493724A1 (en)	2004-03-04	Process for the preparation of 9-beta-anomeric nucleoside analogs
Chen et al.	2015	Stereoselective glycosylation of D-galactals by diethyl phosphorochloridite-and AlCl3-assisted Ferrier rearrangement
Komatsu et al.	2003	Chemo-enzymatic syntheses of natural and unnatural 2′-deoxynucleosides
Chiba et al.	2003	Highly α-stereoselective one-pot sequential glycosylation using glucosyl thioformimidate derivatives
Ghosh et al.	2004	Synergistic enhancement of catalytic activity of InCl3-Me3SiCl combination towards carbon Ferrier rearrangement in glycal derivatives
NO20003890D0 (no)	2000-07-28	Glykosidering av 4,5-epoksymorfinan-6-oler
Kishida et al.	2004	Chemoenzymatic synthesis of n-hexyl and O-β-D-xylopyranosyl-(1→ 6)-β-D-glucopyranosides
WO2003057895A1 (fr)	2003-07-17	Procede de production de 2'-desoxyguanosine
OHSAWA et al.	1993	Synthesis of optically active nucleoside analogs containing 2, 3-dideoxyapiose in the presence of a catalytic amount of trimethylsilyl iodide

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