UY33097A - DERIVADOS DE (1h-PIRAZOL-5-IL)UREIDOARILO 1,3-DISUSTITUIDOS Y SUS USOS TERAPÉUTICOS - Google Patents
DERIVADOS DE (1h-PIRAZOL-5-IL)UREIDOARILO 1,3-DISUSTITUIDOS Y SUS USOS TERAPÉUTICOSInfo
- Publication number
- UY33097A UY33097A UY0001033097A UY33097A UY33097A UY 33097 A UY33097 A UY 33097A UY 0001033097 A UY0001033097 A UY 0001033097A UY 33097 A UY33097 A UY 33097A UY 33097 A UY33097 A UY 33097A
- Authority
- UY
- Uruguay
- Prior art keywords
- ureidoarilo
- disustituidos
- pirazol
- derivatives
- therapeutic uses
- Prior art date
Links
- 230000001225 therapeutic effect Effects 0.000 title 1
- 230000009385 viral infection Effects 0.000 abstract 2
- 208000036142 Viral infection Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
- 241000712461 unidentified influenza virus Species 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0921731.6A GB0921731D0 (en) | 2009-12-11 | 2009-12-11 | Theraputic uses |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY33097A true UY33097A (es) | 2011-06-30 |
Family
ID=41666983
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY0001033097A UY33097A (es) | 2009-12-11 | 2010-12-10 | DERIVADOS DE (1h-PIRAZOL-5-IL)UREIDOARILO 1,3-DISUSTITUIDOS Y SUS USOS TERAPÉUTICOS |
Country Status (4)
| Country | Link |
|---|---|
| GB (1) | GB0921731D0 (fr) |
| TW (1) | TW201130813A (fr) |
| UY (1) | UY33097A (fr) |
| WO (1) | WO2011070368A1 (fr) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0821227A2 (pt) | 2007-12-19 | 2015-06-16 | Cancer Rec Tech Ltd | Composto, composição farmacêutica, método para preparar a mesma, uso de um composto, método para tratar uma doença ou distúrbio, para inibir função de raf e para inibir proliferação celular, inibir progressão do ciclo celular, promover apoptose, ou uma combinação de um ou mais dos mesmos |
| GB0905955D0 (en) | 2009-04-06 | 2009-05-20 | Respivert Ltd | Novel compounds |
| EP2531502B1 (fr) | 2010-02-01 | 2014-04-02 | Cancer Research Technology Limited | 1-(5-tert-butyl-2-phényl-2h-pyrazol-3-yl)-3-[2-fluoro-4-(1-méthyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-7-yloxy)-phényl]-urée et composés associés, et leur utilisation dans des traitements |
| EP2582700B1 (fr) | 2010-06-17 | 2016-11-02 | Respivert Limited | Formulations respiratoires contenant inhibiteurs de p38 mapk |
| GB201010196D0 (en) * | 2010-06-17 | 2010-07-21 | Respivert Ltd | Methods |
| GB201010193D0 (en) * | 2010-06-17 | 2010-07-21 | Respivert Ltd | Medicinal use |
| PL2763984T3 (pl) | 2011-10-03 | 2016-10-31 | 1-pirazolilo-3-(4-((2-anilinopirymidyno-4-ilo)oksy)naftaleno-1-ilo)moczniki jako inhibitory kinazy p38 MAP | |
| EP2578582A1 (fr) | 2011-10-03 | 2013-04-10 | Respivert Limited | 1-Pyrazolyl-3-(4-((2-anilinopyrimidin-4-yl)oxy)napthtalèn-1-yl) urées comme inhibiteurs de la p38 MAP kinase |
| PE20141370A1 (es) | 2011-12-09 | 2014-10-17 | Chiesi Farma Spa | Inhibidores de quinasa |
| CA2860479A1 (fr) | 2011-12-09 | 2013-06-13 | Chiesi Farmaceutici S.P.A. | Inhibiteurs de kinases |
| GB201214750D0 (en) | 2012-08-17 | 2012-10-03 | Respivert Ltd | Compounds |
| GB201215357D0 (en) | 2012-08-29 | 2012-10-10 | Respivert Ltd | Compounds |
| WO2014033449A1 (fr) | 2012-08-29 | 2014-03-06 | Respivert Limited | Inhibiteurs de kinases |
| US20150225373A1 (en) | 2012-08-29 | 2015-08-13 | Respivert Limited | Kinase inhibitors |
| EP2890460B1 (fr) | 2012-08-29 | 2017-02-22 | Respivert Limited | Inhibiteurs de kinases |
| EP2925742B1 (fr) | 2012-11-16 | 2016-10-26 | Respivert Limited | Inhibiteurs de kinase |
| WO2014140582A1 (fr) | 2013-03-14 | 2014-09-18 | Respivert Limited | Inhibiteurs de kinases |
| EP2981535B8 (fr) | 2013-04-02 | 2021-03-10 | Oxular Acquisitions Limited | Dérivés d'urée utilisés en tant qu'inhibiteurs de kinase |
| WO2014162121A1 (fr) | 2013-04-02 | 2014-10-09 | Topivert Pharma Limited | Inhibiteurs de kinase à base de n-alkyl pyrazoles |
| GB201320729D0 (en) | 2013-11-25 | 2014-01-08 | Cancer Rec Tech Ltd | Therapeutic compounds and their use |
| GB201320732D0 (en) | 2013-11-25 | 2014-01-08 | Cancer Rec Tech Ltd | Methods of chemical synthesis |
| EP3083604A1 (fr) | 2013-12-20 | 2016-10-26 | Respivert Limited | Dérivés d'urée utiles comme inhibiteurs de kinase |
| JP6586098B2 (ja) | 2014-02-14 | 2019-10-02 | レスピバート・リミテツド | キナーゼ阻害剤としてのピラゾリル尿素 |
| MA40774A (fr) | 2014-10-01 | 2017-08-08 | Respivert Ltd | Dérivés de diaryle-urée en tant qu'inhibiteurs de kinase p38 |
| BR112018067552A2 (pt) | 2016-04-06 | 2019-01-08 | Topivert Pharma Ltd | inibidores de cinase |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA73492C2 (en) | 1999-01-19 | 2005-08-15 | Aromatic heterocyclic compounds as antiinflammatory agents | |
| WO2003072569A1 (fr) * | 2002-02-25 | 2003-09-04 | Boehringer Ingelheim Pharmaceuticals, Inc. | Composes de cycloalkyle uree benzofusionnes a disubstitution en position 1,4 utiles dans le traitement de maladies mediees par la cytokine |
| MX2007016311A (es) | 2005-06-20 | 2008-03-07 | Tibotec Pharm Ltd | Bencimidazoles sustituidos con heterociclilaminoalquilo. |
| ATE539748T1 (de) | 2006-01-27 | 2012-01-15 | Array Biopharma Inc | Glucokinaseaktivatoren |
| AU2007208156A1 (en) | 2006-01-30 | 2007-08-02 | Irm Llc | Spiro imidazole derivatives as PPAR modulators |
| WO2007096764A2 (fr) | 2006-02-27 | 2007-08-30 | Glenmark Pharmaceuticals S.A. | Dérivés d'hétéroaryles bicycliques en tant que modulateurs des récepteurs cannabinoïdes |
| EP2370428B1 (fr) * | 2008-12-11 | 2016-08-10 | Respivert Limited | Inhibiteur de kinase map p38 |
-
2009
- 2009-12-11 GB GBGB0921731.6A patent/GB0921731D0/en not_active Ceased
-
2010
- 2010-12-10 UY UY0001033097A patent/UY33097A/es unknown
- 2010-12-10 WO PCT/GB2010/052066 patent/WO2011070368A1/fr not_active Ceased
- 2010-12-10 TW TW099143134A patent/TW201130813A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB0921731D0 (en) | 2010-01-27 |
| TW201130813A (en) | 2011-09-16 |
| WO2011070368A1 (fr) | 2011-06-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| UY33097A (es) | DERIVADOS DE (1h-PIRAZOL-5-IL)UREIDOARILO 1,3-DISUSTITUIDOS Y SUS USOS TERAPÉUTICOS | |
| ECSP17084267A (es) | Pirazolo[1,5a]pirimidinas como agentes antivirales | |
| ECSP11011310A (es) | Análogos carba - nucleósido para tratamiento antiviral | |
| CL2019000271A1 (es) | Inhibidores de polimerasa hcv. (divisional solicitud 201600493) | |
| UA116083C2 (uk) | Похідні пурину для лікування вірусних інфекцій | |
| CL2017001426A1 (es) | Nuevos compuestos de 5-amino-6h-tiazolo[4,5-d]pirimidin-2,7-diona 3-sustituidos para el tratamiento y profilaxis de infecciones virales. | |
| ECSP10010210A (es) | Compuestos nucleósidos antivirales | |
| CA2807584C (fr) | Analogues de carba-nucleosides substitues par 2'-fluoro pour traitement antiviral | |
| ECSP099319A (es) | Analogos de tiofeno para el tratamiento o prevencion de las infecciones por flavivirus | |
| CO6561783A2 (es) | Inhibidores del virus flaviviridae | |
| PH12015500347A1 (en) | 6-amino acid heteroaryldihydropyrimidines for the treatment and prophylaxis of hepatitis b virus infection | |
| ECSP12011684A (es) | Inhibidores de los virus flaviviridae. | |
| CY1117200T1 (el) | Παραγωγα βενζυλαμινης ως αναστολεις καλλικρεϊνης πλασματος | |
| MX346264B (es) | Compuestos antivirales. | |
| ECSP10010609A (es) | Carba-nucleosidos analogos 1' - sustituidos para tratamiento antiviral | |
| NZ629996A (en) | 2’- substituted carba-nucleoside analogs for antiviral treatment | |
| IN2012DN01855A (fr) | ||
| ECSP11011389A (es) | Compuestos orgánicos y sus usos | |
| MX2012006026A (es) | Derivados de acido 5-alquinil-tiofen-2-carboxilico y usos para tratamiento o prevencion de infecciones por flavivirus. | |
| ECSP15035530A (es) | Compuestos tetracíclicos sustituidos con heterociclo y métodos de uso de los mismos para el tratamiento de enfermedades víricas | |
| MX2016001855A (es) | Nuevos aza-oxo-indoles para el tratamiento y profilaxis de la infeccion por virus sincitial respiratorio. | |
| CY1118399T1 (el) | Ενωσεις βενζοφουρανιου για την θεραπεια μολυνσεων ιου ηπατιτιδας c | |
| CL2008002291A1 (es) | Compuestos derivados del acido 4-fluor-benzoico, inhibidores de la polimerasa hcv, composicion farmaceutica, kit farmaceutico y su uso para el tratamiento de una infeccion viral por hepatitis c. | |
| ECSP13013075A (es) | Método de tratamiento de la fiebre dengue | |
| UY30545A1 (es) | Derivados sustituidos del acido acilamino-benzoico, composiciones que los contienen y aplicaciones |