UY30247A1 - IMPROVEMENTS IN THE PREPARATION OF INTERMEDIATES THAT CONDUCT HYDROCLORIDE OF (4- (5-AMINOMETIL-2-FLUORO-PHENYL) -PIPERIDIN - 1-IL) - (4-BROMO-3-METIL-5-PROPOXI-TIOFEN-2 -IL) -METANONA. - Google Patents
IMPROVEMENTS IN THE PREPARATION OF INTERMEDIATES THAT CONDUCT HYDROCLORIDE OF (4- (5-AMINOMETIL-2-FLUORO-PHENYL) -PIPERIDIN - 1-IL) - (4-BROMO-3-METIL-5-PROPOXI-TIOFEN-2 -IL) -METANONA.Info
- Publication number
- UY30247A1 UY30247A1 UY30247A UY30247A UY30247A1 UY 30247 A1 UY30247 A1 UY 30247A1 UY 30247 A UY30247 A UY 30247A UY 30247 A UY30247 A UY 30247A UY 30247 A1 UY30247 A1 UY 30247A1
- Authority
- UY
- Uruguay
- Prior art keywords
- preparation
- intermediates
- metanona
- aminometil
- tiofen
- Prior art date
Links
- 239000000543 intermediate Substances 0.000 title abstract 2
- VEXZGXHMUGYJMC-UHFFFAOYSA-N Hydrochloric acid Chemical compound Cl VEXZGXHMUGYJMC-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C327/00—Thiocarboxylic acids
- C07C327/20—Esters of monothiocarboxylic acids
- C07C327/22—Esters of monothiocarboxylic acids having carbon atoms of esterified thiocarboxyl groups bound to hydrogen atoms or to acyclic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
- C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
La presente invencion se dirige a mejoras en la preparacion de compuestos de formula 7,8 y 13, que son intermedios utiles para la preparacion del compuesto de formula I.The present invention is directed to improvements in the preparation of compounds of formula 7,8 and 13, which are useful intermediates for the preparation of the compound of formula I.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74390806P | 2006-03-29 | 2006-03-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY30247A1 true UY30247A1 (en) | 2007-11-30 |
Family
ID=38283355
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY30247A UY30247A1 (en) | 2006-03-29 | 2007-03-29 | IMPROVEMENTS IN THE PREPARATION OF INTERMEDIATES THAT CONDUCT HYDROCLORIDE OF (4- (5-AMINOMETIL-2-FLUORO-PHENYL) -PIPERIDIN - 1-IL) - (4-BROMO-3-METIL-5-PROPOXI-TIOFEN-2 -IL) -METANONA. |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP2001839A1 (en) |
| CN (1) | CN101405262A (en) |
| AR (1) | AR060181A1 (en) |
| MX (1) | MX2008011259A (en) |
| PE (1) | PE20071148A1 (en) |
| TW (1) | TW200811093A (en) |
| UY (1) | UY30247A1 (en) |
| WO (1) | WO2007118010A1 (en) |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DOP2005000039A (en) * | 2004-03-26 | 2005-10-31 | Aventis Pharma Inc | HYDROCHLORIDE OF [4- (5-AMINOMETIL-2-FLUORO-PHENYL) - PIPERIDIN-1-IL] - (4-BOMO-3-METHYL-5-PROPOXI-TIOFEN-2-IL) -METANONE AS AN INHIBITOR OF THE MASTOCYT TRIPTASE |
-
2007
- 2007-03-27 PE PE2007000345A patent/PE20071148A1/en not_active Application Discontinuation
- 2007-03-28 AR ARP070101299A patent/AR060181A1/en not_active Application Discontinuation
- 2007-03-28 CN CNA2007800096074A patent/CN101405262A/en active Pending
- 2007-03-28 WO PCT/US2007/065339 patent/WO2007118010A1/en not_active Ceased
- 2007-03-28 MX MX2008011259A patent/MX2008011259A/en not_active Application Discontinuation
- 2007-03-28 EP EP07759555A patent/EP2001839A1/en not_active Withdrawn
- 2007-03-29 UY UY30247A patent/UY30247A1/en not_active Application Discontinuation
- 2007-03-29 TW TW096110910A patent/TW200811093A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AR060181A1 (en) | 2008-05-28 |
| WO2007118010A1 (en) | 2007-10-18 |
| CN101405262A (en) | 2009-04-08 |
| MX2008011259A (en) | 2008-09-10 |
| TW200811093A (en) | 2008-03-01 |
| EP2001839A1 (en) | 2008-12-17 |
| PE20071148A1 (en) | 2007-12-10 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CR9331A (en) | VEGF-R2 INHIBITORS AND METHODS | |
| ECSP10010582A (en) | AMINODIHYDROTIAZINE DERIVATIVES AS BACE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE | |
| GT201200046A (en) | CONJUGATES OF PIRROLO DIMMERS [1,4] BENZODIAZEPINA AS ANTI-TARGET AGENTS | |
| BRPI0908926A2 (en) | Polycarbonate-polyorganosiloxane and / or polyurethane-polyorganosiloxane compounds | |
| CY1109911T1 (en) | PYRROLOVENZODIAZEPINES | |
| GEP20156266B (en) | Spiroheterocyclic n-oxypiperidines as pesticides | |
| ECSP11010889A (en) | CMET INHIBITORS | |
| CR11861A (en) | ORGANIC COMPOUNDS | |
| CR10662A (en) | METHYLPIRIDOPIRIMIDINONE COMPOUNDS | |
| CY1113716T1 (en) | A NEW METHOD OF COMPOSITION OF AGOMELATIN | |
| ATE554066T1 (en) | ANTI-INFLAMMATORY SUBSTITUTED CYCLOBUTENDIONE COMPOUNDS | |
| UY30146A1 (en) | NEW RADIOLIGANDS | |
| PA8846901A1 (en) | AKT AND P70 S6 CINASE INHIBITORS. | |
| UY31688A1 (en) | PESTICIDES | |
| HN2009001436A (en) | NEW AGOMETATINE SYNTHESIS PROCEDURE | |
| EA200702464A1 (en) | METHODS OF OBTAINING PHENOL 4-BIPHENYLILAZETIDIN-2-ONES | |
| EA200900090A1 (en) | BENZYLAMINES, METHOD OF THEIR PRODUCTION AND THEIR APPLICATION AS ANTI-INFLAMMATORY MEANS | |
| PA8792101A1 (en) | NEW SYNTHESIS PROCEDURE OF (7-METOXI-1- NAFTIL) ACETO | |
| BR112013028368A2 (en) | new compounds of hexahydrocyclopyrpyrrolone, hexahydropyrrolpyrrolone, octahydropyrrolopyridinone and octahydropyridinone | |
| CY1111573T1 (en) | A NEW METHOD OF COMPOSITION OF AGOMELATIN | |
| UY32042A (en) | 2-AMINOPIRIMIDINE COMPOUNDS AS POWERFUL INHIBITORS OF HSP-90 | |
| ECSP088374A (en) | AEROSOL FORMULATION FOR INHALATION | |
| EA200801366A1 (en) | DERIVATIVES 3,6-DIGIDRO-2-OXO-6N-1,3,4-TIADIAZINA | |
| EA200801365A1 (en) | SUBSTITUTED 5-PHENYL-3,6-DIGIDRO-2-OXO-6H-1,3,4-TIADIAZINS | |
| BRPI0516602A (en) | compound and pharmaceutical composition |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20130206 |