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AR060181A1 - IMPROVEMENTS IN THE PREPARATION OF INTERMEDIATES THAT CONDUCT HYDROCLORIDE OF [4- (5-AMINOMETIL-2-FLUORO-PHENYL) -PIPERIDIN-1-IL] - (4-BROMO-3-METIL-5-PROPOXI-TIOFEN-2- IL) -METANONE - Google Patents

IMPROVEMENTS IN THE PREPARATION OF INTERMEDIATES THAT CONDUCT HYDROCLORIDE OF [4- (5-AMINOMETIL-2-FLUORO-PHENYL) -PIPERIDIN-1-IL] - (4-BROMO-3-METIL-5-PROPOXI-TIOFEN-2- IL) -METANONE

Info

Publication number
AR060181A1
AR060181A1 ARP070101299A ARP070101299A AR060181A1 AR 060181 A1 AR060181 A1 AR 060181A1 AR P070101299 A ARP070101299 A AR P070101299A AR P070101299 A ARP070101299 A AR P070101299A AR 060181 A1 AR060181 A1 AR 060181A1
Authority
AR
Argentina
Prior art keywords
aminometil
tiofen
propoxi
metanone
hydrocloride
Prior art date
Application number
ARP070101299A
Other languages
Spanish (es)
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of AR060181A1 publication Critical patent/AR060181A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C327/00—Thiocarboxylic acids
    • C07C327/20—Esters of monothiocarboxylic acids
    • C07C327/22—Esters of monothiocarboxylic acids having carbon atoms of esterified thiocarboxyl groups bound to hydrogen atoms or to acyclic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Reivindicacion 1: Un método para preparar un compuesto de formula (1), que comprende condensar el compuesto de formula (2) con acetona.Claim 1: A method of preparing a compound of formula (1), which comprises condensing the compound of formula (2) with acetone.

ARP070101299A 2006-03-29 2007-03-28 IMPROVEMENTS IN THE PREPARATION OF INTERMEDIATES THAT CONDUCT HYDROCLORIDE OF [4- (5-AMINOMETIL-2-FLUORO-PHENYL) -PIPERIDIN-1-IL] - (4-BROMO-3-METIL-5-PROPOXI-TIOFEN-2- IL) -METANONE AR060181A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US74390806P 2006-03-29 2006-03-29

Publications (1)

Publication Number Publication Date
AR060181A1 true AR060181A1 (en) 2008-05-28

Family

ID=38283355

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070101299A AR060181A1 (en) 2006-03-29 2007-03-28 IMPROVEMENTS IN THE PREPARATION OF INTERMEDIATES THAT CONDUCT HYDROCLORIDE OF [4- (5-AMINOMETIL-2-FLUORO-PHENYL) -PIPERIDIN-1-IL] - (4-BROMO-3-METIL-5-PROPOXI-TIOFEN-2- IL) -METANONE

Country Status (8)

Country Link
EP (1) EP2001839A1 (en)
CN (1) CN101405262A (en)
AR (1) AR060181A1 (en)
MX (1) MX2008011259A (en)
PE (1) PE20071148A1 (en)
TW (1) TW200811093A (en)
UY (1) UY30247A1 (en)
WO (1) WO2007118010A1 (en)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DOP2005000039A (en) * 2004-03-26 2005-10-31 Aventis Pharma Inc HYDROCHLORIDE OF [4- (5-AMINOMETIL-2-FLUORO-PHENYL) - PIPERIDIN-1-IL] - (4-BOMO-3-METHYL-5-PROPOXI-TIOFEN-2-IL) -METANONE AS AN INHIBITOR OF THE MASTOCYT TRIPTASE

Also Published As

Publication number Publication date
WO2007118010A1 (en) 2007-10-18
CN101405262A (en) 2009-04-08
MX2008011259A (en) 2008-09-10
EP2001839A1 (en) 2008-12-17
UY30247A1 (en) 2007-11-30
PE20071148A1 (en) 2007-12-10
TW200811093A (en) 2008-03-01

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal