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UY30206A1 - Derivados de diamina, composiciones farmacéuticas conteniéndolos, procesos de preparacion y aplicaciones - Google Patents

Derivados de diamina, composiciones farmacéuticas conteniéndolos, procesos de preparacion y aplicaciones

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Publication number
UY30206A1
UY30206A1 UY30206A UY30206A UY30206A1 UY 30206 A1 UY30206 A1 UY 30206A1 UY 30206 A UY30206 A UY 30206A UY 30206 A UY30206 A UY 30206A UY 30206 A1 UY30206 A1 UY 30206A1
Authority
UY
Uruguay
Prior art keywords
pharmaceutical compositions
compositions containing
applications
preparation processes
diamine derivatives
Prior art date
Application number
UY30206A
Other languages
English (en)
Inventor
Garry Pairaudeau
Andrew Lister
Lilian Alcaraz
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY30206A1 publication Critical patent/UY30206A1/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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Abstract

La presente invencion proporciona compuestos de formula (1):en donde Ar, R1, R2. T, A, X, Y, R51, R52, R y R3 y R4 son como se define en la memoira descriptiva, procesos para su preparacion, composiciones farmacéuticas que los contienen y su uso en terapia.
UY30206A 2006-03-14 2007-03-14 Derivados de diamina, composiciones farmacéuticas conteniéndolos, procesos de preparacion y aplicaciones UY30206A1 (es)

Applications Claiming Priority (2)

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US78273306P 2006-03-14 2006-03-14
US86265106P 2006-10-24 2006-10-24

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UY30206A1 true UY30206A1 (es) 2007-10-31

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UY30206A UY30206A1 (es) 2006-03-14 2007-03-14 Derivados de diamina, composiciones farmacéuticas conteniéndolos, procesos de preparacion y aplicaciones

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JP2009530272A (ja) 2009-08-27
US20090062259A1 (en) 2009-03-05
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WO2007106016A1 (en) 2007-09-20
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