UY30550A1 - Nuevos beta-agonistas enantioméricamente puros, procedimientos para su preparacion y su uso como medicamentos - Google Patents
Nuevos beta-agonistas enantioméricamente puros, procedimientos para su preparacion y su uso como medicamentosInfo
- Publication number
- UY30550A1 UY30550A1 UY30550A UY30550A UY30550A1 UY 30550 A1 UY30550 A1 UY 30550A1 UY 30550 A UY30550 A UY 30550A UY 30550 A UY30550 A UY 30550A UY 30550 A1 UY30550 A1 UY 30550A1
- Authority
- UY
- Uruguay
- Prior art keywords
- procedures
- preparation
- enantioméricamente
- aganistas
- puros
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
La presente invencion se refiere a compuestos enantioméricamente puros de la formula 1 en donde los radicales R1, R2, R3, m e Ym- pueden tener los significados mencionados en las reivindicaciones y la descripcion, a procedimientos para su preparacion, así como a su uso como medicamentos, en especial como medicamentos para el tratamiento de enfermedades de las vias aéreas.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06119273 | 2006-08-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY30550A1 true UY30550A1 (es) | 2008-03-31 |
Family
ID=38698758
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY30550A UY30550A1 (es) | 2006-08-22 | 2007-08-20 | Nuevos beta-agonistas enantioméricamente puros, procedimientos para su preparacion y su uso como medicamentos |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US7709474B2 (es) |
| EP (1) | EP2057134A1 (es) |
| JP (1) | JP2010501522A (es) |
| KR (1) | KR20090043586A (es) |
| CN (1) | CN101506182A (es) |
| AR (1) | AR062476A1 (es) |
| AU (1) | AU2007287537A1 (es) |
| BR (1) | BRPI0715690A2 (es) |
| CA (1) | CA2661143A1 (es) |
| CO (1) | CO6150169A2 (es) |
| EA (1) | EA200900268A1 (es) |
| EC (1) | ECSP099082A (es) |
| IL (1) | IL197124A0 (es) |
| MX (1) | MX2009001515A (es) |
| NO (1) | NO20090101L (es) |
| NZ (1) | NZ575567A (es) |
| PE (1) | PE20080610A1 (es) |
| TW (1) | TW200817347A (es) |
| UA (1) | UA96951C2 (es) |
| UY (1) | UY30550A1 (es) |
| WO (1) | WO2008023004A1 (es) |
| ZA (1) | ZA200810829B (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20080425A1 (es) * | 2006-08-22 | 2008-06-16 | Boehringer Ingelheim Int | Formulacion aerosol para la inhalacion de beta-agonistas |
| US20100233268A1 (en) * | 2006-08-22 | 2010-09-16 | Boehringer Ingelheim International Gmbh | Powder formulations for inhalation containing enantiomerically pure beta-agonists |
| EP2486936A1 (en) | 2007-06-13 | 2012-08-15 | CSL Behring GmbH | A composition comprising VWF and FVIII preparations for use in treating of bleeding disorders |
| EP2093219A1 (de) | 2008-02-22 | 2009-08-26 | Boehringer Ingelheim International Gmbh | Kristalline, enantiomerenreine Salzform eines Betamimetikums und dessen Verwendung als Arzneimittel |
| ES2657291T3 (es) | 2013-04-22 | 2018-03-02 | Csl Ltd. | Un complejo covalente de factor de von Willebrand y factor VIII asociado por un puente disulfuro |
Family Cites Families (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3026534A1 (de) * | 1980-07-12 | 1982-03-18 | C.H. Boehringer Sohn, 6507 Ingelheim | 3,1-benzoxazin-2-one, ihre herstellung und verwendung |
| US4460581A (en) * | 1982-10-12 | 1984-07-17 | Boehringer Ingelheim Kg | (1-Hydroxy-2-amino-alkyl)-substituted benzoxazinones and benzoxazolinones |
| US4570630A (en) * | 1983-08-03 | 1986-02-18 | Miles Laboratories, Inc. | Medicament inhalation device |
| SE453566B (sv) | 1986-03-07 | 1988-02-15 | Draco Ab | Anordning vid pulverinhalatorer |
| DE3609152A1 (de) * | 1986-03-19 | 1987-09-24 | Bayer Ag | Verfahren zur herstellung des (-)-antipoden des (e)-1-cyclohexyl-4,4-dimethyl- 3-hydroxy-2-(1,2,4-triazol-1-yl)-pent-1-ens |
| SG45171A1 (en) | 1990-03-21 | 1998-01-16 | Boehringer Ingelheim Int | Atomising devices and methods |
| IL107120A (en) | 1992-09-29 | 1997-09-30 | Boehringer Ingelheim Int | Atomising nozzle and filter and spray generating device |
| DE4318455A1 (de) | 1993-06-03 | 1994-12-08 | Boehringer Ingelheim Kg | Kapselhalterung |
| US5495054A (en) | 1994-05-31 | 1996-02-27 | Sepracor, Inc. | Tetrahydroindeno[1,2-D][1,3,2]oxazaboroles and their use as enantioselective catalysts |
| DE19536902A1 (de) | 1995-10-04 | 1997-04-10 | Boehringer Ingelheim Int | Vorrichtung zur Hochdruckerzeugung in einem Fluid in Miniaturausführung |
| DE19536903C2 (de) | 1995-10-04 | 1998-09-10 | Boehringer Ingelheim Int | Vorrichtung zum Haltern eines fluidischen Bauteils |
| DE19545226C1 (de) | 1995-12-05 | 1997-06-19 | Boehringer Ingelheim Int | Sperrspannwerk für einen federbetätigten Abtrieb |
| DE19742439C1 (de) | 1997-09-26 | 1998-10-22 | Boehringer Ingelheim Int | Mikrostrukturiertes Filter |
| AP1572A (en) | 2000-10-12 | 2006-02-13 | Boehringer Ingelheim Pharma | Crystalline monohydrate, method for producing the same and use thereof in the production of a medicament. |
| DE10050995A1 (de) | 2000-10-14 | 2002-04-18 | Boehringer Ingelheim Pharma | Neue Anticholinergika, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| PL208137B1 (pl) | 2001-06-22 | 2011-03-31 | Boehringer Ingelheim Pharma | Bezwodny krystaliczny bromek tiotropium, sposób jego wytwarzania i zastosowanie krystalicznego monohydratu bromku tiotropium do wytwarzania krystalicznego bezwodnego bromku tiotropium |
| DE10203753A1 (de) | 2002-01-31 | 2003-08-14 | Boehringer Ingelheim Pharma | Neue Xanthencarbonsäureester, Verfahren zu deren Herstellung sowie deren Verwendung als Arzneimittel |
| DE10203749A1 (de) | 2002-01-31 | 2003-08-14 | Boehringer Ingelheim Pharma | Neue Anticholinergika, Verfahren zu deren Herstellung sowie deren Verwendung als Arzneimittel |
| DE10203741A1 (de) | 2002-01-31 | 2003-08-14 | Boehringer Ingelheim Pharma | Neue Fluorencarbonsäureester, Verfahren zu deren Herstellung sowie deren Verwendung als Arzneimittel |
| WO2004087142A1 (en) | 2003-04-04 | 2004-10-14 | Novartis Ag | Quinoline-2-one-derivatives for the treatment of airways diseases |
| DE102004003428A1 (de) | 2004-01-23 | 2005-08-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue langwirksame Beta-2-Agonisten, und deren Verwendung als Arzneimittel |
| DE102004024454A1 (de) | 2004-05-14 | 2005-12-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Enantiomerenreine Betaagonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| US7220742B2 (en) * | 2004-05-14 | 2007-05-22 | Boehringer Ingelheim International Gmbh | Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments |
| DE102005008921A1 (de) * | 2005-02-24 | 2006-08-31 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Arzneimittel zur Behandlung von Atemwegserkrankungen |
| US7423146B2 (en) * | 2005-11-09 | 2008-09-09 | Boehringer Ingelheim International Gmbh | Process for the manufacturing of pharmaceutically active 3,1-benzoxazine-2-ones |
| PE20080425A1 (es) * | 2006-08-22 | 2008-06-16 | Boehringer Ingelheim Int | Formulacion aerosol para la inhalacion de beta-agonistas |
| PE20081358A1 (es) * | 2006-08-22 | 2008-10-31 | Boehringer Ingelheim Int | Combinaciones farmacologicas para el tratamiento de enfermedades de la vias aereas |
-
2007
- 2007-08-20 UY UY30550A patent/UY30550A1/es not_active Application Discontinuation
- 2007-08-20 PE PE2007001125A patent/PE20080610A1/es not_active Application Discontinuation
- 2007-08-21 WO PCT/EP2007/058654 patent/WO2008023004A1/de not_active Ceased
- 2007-08-21 CN CNA2007800311865A patent/CN101506182A/zh active Pending
- 2007-08-21 EA EA200900268A patent/EA200900268A1/ru unknown
- 2007-08-21 EP EP07802746A patent/EP2057134A1/de not_active Withdrawn
- 2007-08-21 BR BRPI0715690-1A2A patent/BRPI0715690A2/pt not_active IP Right Cessation
- 2007-08-21 TW TW096130900A patent/TW200817347A/zh unknown
- 2007-08-21 UA UAA200902356A patent/UA96951C2/ru unknown
- 2007-08-21 KR KR1020097005850A patent/KR20090043586A/ko not_active Withdrawn
- 2007-08-21 NZ NZ575567A patent/NZ575567A/en not_active IP Right Cessation
- 2007-08-21 AU AU2007287537A patent/AU2007287537A1/en not_active Abandoned
- 2007-08-21 MX MX2009001515A patent/MX2009001515A/es active IP Right Grant
- 2007-08-21 CA CA002661143A patent/CA2661143A1/en not_active Abandoned
- 2007-08-21 US US11/842,485 patent/US7709474B2/en active Active
- 2007-08-21 JP JP2009525052A patent/JP2010501522A/ja active Pending
- 2007-08-22 AR ARP070103721A patent/AR062476A1/es not_active Application Discontinuation
-
2008
- 2008-12-23 ZA ZA200810829A patent/ZA200810829B/xx unknown
-
2009
- 2009-01-08 NO NO20090101A patent/NO20090101L/no not_active Application Discontinuation
- 2009-01-20 EC EC2009009082A patent/ECSP099082A/es unknown
- 2009-02-19 CO CO09016428A patent/CO6150169A2/es unknown
- 2009-02-19 IL IL197124A patent/IL197124A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EA200900268A1 (ru) | 2009-08-28 |
| ECSP099082A (es) | 2009-02-27 |
| MX2009001515A (es) | 2009-02-18 |
| NZ575567A (en) | 2011-12-22 |
| IL197124A0 (en) | 2009-11-18 |
| CO6150169A2 (es) | 2010-04-20 |
| ZA200810829B (en) | 2009-11-25 |
| UA96951C2 (ru) | 2011-12-26 |
| WO2008023004A8 (de) | 2008-05-22 |
| JP2010501522A (ja) | 2010-01-21 |
| WO2008023004A1 (de) | 2008-02-28 |
| AR062476A1 (es) | 2008-11-12 |
| CN101506182A (zh) | 2009-08-12 |
| US20080070909A1 (en) | 2008-03-20 |
| EP2057134A1 (de) | 2009-05-13 |
| PE20080610A1 (es) | 2008-07-15 |
| NO20090101L (no) | 2009-01-29 |
| AU2007287537A1 (en) | 2008-02-28 |
| KR20090043586A (ko) | 2009-05-06 |
| CA2661143A1 (en) | 2008-02-28 |
| US7709474B2 (en) | 2010-05-04 |
| TW200817347A (en) | 2008-04-16 |
| BRPI0715690A2 (pt) | 2013-09-17 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ECSP077331A (es) | Nuevos betamiméticos para el tratamiento de enfermedades de vías respiratorias | |
| GT201300179A (es) | Derivados heterociclicos novedosos y su uso en el tratamiento de trastornos neurologicos | |
| ECSP099750A (es) | Imidazoquinolinas con propiedades inmunomoduladoras | |
| ECSP109903A (es) | Derivados de pirazinona y su uso en el tratamiento de enfermedades pulmonares | |
| CO6491058A2 (es) | Derivados de oxazina y su uso como inhibidores de bace para el tratamiento de trastornos neurológicos | |
| UY30578A1 (es) | Nuevos derivados de 2,4??- y 3, 4??-bipiridina sustituidos, procedimientos para su preparacion, medicamentos conteniéndolos y aplicaciones | |
| UY32648A (es) | Nuevos derivados de pirimidina y su uso en el tratamiento de enfermedades | |
| UY30641A1 (es) | Derivados de 2-[1h-pirazol-5-il] y de 2-[2h-pirazol-3-il]tieno[3,2-c]piridinas sustituidas, sus sales farmaceuticamente aceptables y aplicaciones | |
| UY30498A1 (es) | Nueva clase de compuestos de benzimidazolilo, sus sales, composiciones farmacéuticas conteniéndolos y aplicaciones | |
| CR20140392A (es) | Dihidropirazolonas sustituidas | |
| ECSP11011082A (es) | Compuestos, composición farmaceutica y métodos para utilizarse en el tratamiento de desórdenes metabólicos | |
| ECSP088082A (es) | Derivados de piridazina | |
| UY30098A1 (es) | Compuestos de tiazol y metodos de uso | |
| UY30282A1 (es) | Compuestos quimicos | |
| ECSP066734A (es) | Derivados de ácido 7-fenilamino-4-quinolona-3-carboxílico, métodos para su producción y su uso como medicamentos | |
| ECSP066948A (es) | Benzoxazinas para el tratamiento de enfermedades de las vías respiratorias | |
| CR10356A (es) | Derivados de 4-benzilphthalazinona 2-sustituidos como antagonistas de histamina h1 y h3 | |
| UY28861A1 (es) | Nuevas combinaciones farmacologicas para el tratamiento de enfermedades de las vias respiratorias | |
| UY31322A1 (es) | Amidas heterocíclicas y sus métodos de uso-975 | |
| UY32055A (es) | Derivados sustituidos de la 5-Halo-N2-[sustituido](1-metil-1H-imidazol-4-il)pirimidin-2,-diamina y sus sales farmacéuticamente aceptables, procesos de preparación, composiciones y aplicaciones. | |
| DOP2006000061A (es) | Derivados de pirimidina para el tratamiento de trastornos hiperproliferativos | |
| PA8627001A1 (es) | Compuestos para el tratamiento de enfermedades | |
| UY30550A1 (es) | Nuevos beta-agonistas enantioméricamente puros, procedimientos para su preparacion y su uso como medicamentos | |
| UY30865A1 (es) | Nuevos analogos de piridina x 161 | |
| AR057148A1 (es) | Combinaciones farmacologicas para el tratamiento de enfermedades de las vias respiratorias |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20170725 |