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UA122762C2 - Пероральна композиція 9-[(2,2-диметилпропіламіно)-метил]-міноцикліну або його солі, тверда пресована дозована форма, композиція для ін'єкцій, застосування та спосіб приготування фармацевтичної композиції - Google Patents

Пероральна композиція 9-[(2,2-диметилпропіламіно)-метил]-міноцикліну або його солі, тверда пресована дозована форма, композиція для ін'єкцій, застосування та спосіб приготування фармацевтичної композиції

Info

Publication number
UA122762C2
UA122762C2 UAA201505310A UAA201505310A UA122762C2 UA 122762 C2 UA122762 C2 UA 122762C2 UA A201505310 A UAA201505310 A UA A201505310A UA A201505310 A UAA201505310 A UA A201505310A UA 122762 C2 UA122762 C2 UA 122762C2
Authority
UA
Ukraine
Prior art keywords
composition
dimethylpropylamino
minocycline
methyl
injections
Prior art date
Application number
UAA201505310A
Other languages
English (en)
Inventor
Джонстон Шон
Original Assignee
Паратек Фармасьютікалз, Інк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41114256&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA122762(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Паратек Фармасьютікалз, Інк. filed Critical Паратек Фармасьютікалз, Інк.
Publication of UA122762C2 publication Critical patent/UA122762C2/uk

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/65Tetracyclines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Винахід стосується композиції для ін’єкцій, яка містить приблизно 90-110 мг 9-[(2,2-диметилпропіламіно)-метил]-міноцикліну та один або більше компонентів, вибраних з ліопротектора, де ліопротектор являє собою цукор, антиоксиданту, сполуки для регулювання рН, вибраної з соляної кислоти або гідроксиду натрію, та фармацевтично прийнятного носія, причому рН композиції знаходиться в межах від приблизно 4,0 до приблизно 4,5.
UAA201505310A 2008-03-28 2009-03-30 Пероральна композиція 9-[(2,2-диметилпропіламіно)-метил]-міноцикліну або його солі, тверда пресована дозована форма, композиція для ін'єкцій, застосування та спосіб приготування фармацевтичної композиції UA122762C2 (uk)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US4039808P 2008-03-28 2008-03-28

Publications (1)

Publication Number Publication Date
UA122762C2 true UA122762C2 (uk) 2021-01-06

Family

ID=41114256

Family Applications (2)

Application Number Title Priority Date Filing Date
UAA201012435A UA109627C2 (uk) 2008-03-28 2009-03-30 Композиції тетрациклінових сполук для орального введення та ін'єкцій
UAA201505310A UA122762C2 (uk) 2008-03-28 2009-03-30 Пероральна композиція 9-[(2,2-диметилпропіламіно)-метил]-міноцикліну або його солі, тверда пресована дозована форма, композиція для ін'єкцій, застосування та спосіб приготування фармацевтичної композиції

Family Applications Before (1)

Application Number Title Priority Date Filing Date
UAA201012435A UA109627C2 (uk) 2008-03-28 2009-03-30 Композиції тетрациклінових сполук для орального введення та ін'єкцій

Country Status (30)

Country Link
US (2) US9314475B2 (uk)
EP (3) EP3789030A1 (uk)
JP (8) JP2011515473A (uk)
KR (3) KR101893740B1 (uk)
CN (1) CN102046177B (uk)
AU (1) AU2009229174A1 (uk)
BR (2) BRPI0909211B8 (uk)
CA (2) CA2719751C (uk)
CL (1) CL2010000281A1 (uk)
CO (1) CO6300935A2 (uk)
CY (2) CY1120240T1 (uk)
DK (2) DK2271348T3 (uk)
EC (1) ECSP10010576A (uk)
ES (2) ES2836448T3 (uk)
HR (2) HRP20180836T1 (uk)
HU (2) HUE038257T2 (uk)
IL (1) IL208440A0 (uk)
LT (2) LT2271348T (uk)
MA (1) MA32275B1 (uk)
MX (1) MX2010010585A (uk)
NO (1) NO2271348T3 (uk)
NZ (1) NZ588428A (uk)
PL (2) PL3348258T3 (uk)
PT (2) PT2271348T (uk)
RU (1) RU2010144130A (uk)
SI (2) SI2271348T1 (uk)
TR (1) TR201806893T4 (uk)
UA (2) UA109627C2 (uk)
WO (1) WO2009120389A1 (uk)
ZA (1) ZA201007013B (uk)

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SMT202300467T1 (it) * 2019-12-30 2024-01-10 Deciphera Pharmaceuticals Llc Formulazioni di inibitori di chinasi amorfi e loro procedimenti d’uso
PT117254B (pt) 2021-05-26 2024-04-18 Hovione Farm S A Método de síntese de compostos 9-aminometil tetraciclinas

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Also Published As

Publication number Publication date
IL208440A0 (en) 2010-12-30
WO2009120389A1 (en) 2009-10-01
HK1257928A1 (en) 2019-11-01
PL3348258T3 (pl) 2021-03-08
ZA201007013B (en) 2013-11-27
LT3348258T (lt) 2020-12-10
HUE038257T2 (hu) 2018-10-29
SI3348258T1 (sl) 2020-12-31
HUE052201T2 (hu) 2021-04-28
TR201806893T4 (tr) 2018-06-21
PT3348258T (pt) 2020-11-25
BRPI0909211B1 (pt) 2020-08-25
DK3348258T3 (da) 2020-12-07
ES2674708T3 (es) 2018-07-03
CL2010000281A1 (es) 2012-03-30
NZ588428A (en) 2012-08-31
CN102046177B (zh) 2012-12-19
JP2016145260A (ja) 2016-08-12
CO6300935A2 (es) 2011-07-21
JP2014221820A (ja) 2014-11-27
LT2271348T (lt) 2018-06-25
HRP20180836T1 (hr) 2018-07-27
ECSP10010576A (es) 2010-12-30
KR20110008057A (ko) 2011-01-25
KR101893740B1 (ko) 2018-08-30
EP2271348B1 (en) 2018-03-28
CY1120240T1 (el) 2019-07-10
JP6412521B2 (ja) 2018-10-24
KR101835574B1 (ko) 2018-03-08
KR20160105532A (ko) 2016-09-06
BR122020011180B8 (pt) 2021-07-27
JP2025137721A (ja) 2025-09-19
JP5940119B2 (ja) 2016-06-29
JP2011515473A (ja) 2011-05-19
NO2271348T3 (uk) 2018-08-25
RU2010144130A (ru) 2012-05-10
ES2836448T3 (es) 2021-06-25
EP3348258B1 (en) 2020-09-09
EP2271348A4 (en) 2011-05-25
KR101746228B1 (ko) 2017-06-12
EP3789030A1 (en) 2021-03-10
JP6577645B2 (ja) 2019-09-18
US20160279151A1 (en) 2016-09-29
CA2984301C (en) 2020-10-27
HRP20201883T1 (hr) 2021-01-22
BRPI0909211B8 (pt) 2021-05-25
AU2009229174A1 (en) 2009-10-01
US20100056638A1 (en) 2010-03-04
WO2009120389A8 (en) 2010-05-14
DK2271348T3 (en) 2018-06-14
PL2271348T3 (pl) 2018-08-31
CA2719751C (en) 2018-01-02
PT2271348T (pt) 2018-04-16
CN102046177A (zh) 2011-05-04
CA2984301A1 (en) 2009-10-01
SI2271348T1 (en) 2018-08-31
MX2010010585A (es) 2010-11-09
UA109627C2 (uk) 2015-09-25
CY1123382T1 (el) 2021-12-31
BR122020011180B1 (pt) 2021-03-23
EP2271348A1 (en) 2011-01-12
EP3348258A1 (en) 2018-07-18
JP2021167355A (ja) 2021-10-21
JP2023144043A (ja) 2023-10-06
CA2719751A1 (en) 2009-10-01
KR20180026799A (ko) 2018-03-13
US9314475B2 (en) 2016-04-19
JP2018203778A (ja) 2018-12-27
JP2019196408A (ja) 2019-11-14
MA32275B1 (fr) 2011-05-02
BRPI0909211A2 (pt) 2016-11-29

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