TW201943687A - 包含4-苯丁酸衍生物及類鴉片的組成物 - Google Patents

包含4-苯丁酸衍生物及類鴉片的組成物 Download PDF

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Publication number: TW201943687A
Authority: TW; Taiwan
Prior art keywords: phenylbutyric acid; treatment; cancer; pharmaceutical composition; composition
Prior art date: 2018-04-09

Application number

TW108109828A

Other languages

English (en)

Chinese (zh)

Inventor

彼得特魯

Original Assignee

彼得特魯

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2018-04-09

Filing date

2019-03-21

Publication date

2019-11-16

2019-03-21 Application filed by 彼得特魯 filed Critical 彼得特魯

2019-11-16 Publication of TW201943687A publication Critical patent/TW201943687A/zh

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USSIQXCVUWKGNF-UHFFFAOYSA-N 6-(dimethylamino)-4,4-diphenylheptan-3-one Chemical group C=1C=CC=CC=1C(CC(C)N(C)C)(C(=O)CC)C1=CC=CC=C1 USSIQXCVUWKGNF-UHFFFAOYSA-N 0.000 claims abstract description 14
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OGWKCGZFUXNPDA-UHFFFAOYSA-N vincristine Natural products C1C(CC)(O)CC(CC2(C(=O)OC)C=3C(=CC4=C(C56C(C(C(OC(C)=O)C7(CC)C=CCN(C67)CC5)(O)C(=O)OC)N4C=O)C=3)OC)CN1CCC1=C2NC2=CC=CC=C12 OGWKCGZFUXNPDA-UHFFFAOYSA-N 0.000 description 1
239000000080 wetting agent Substances 0.000 description 1
108020001612 μ-opioid receptors Proteins 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents

Landscapes

Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Emergency Medicine (AREA)
Epidemiology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

TW108109828A 2018-04-09 2019-03-21 包含4-苯丁酸衍生物及類鴉片的組成物 TW201943687A (zh)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
WOPCT/EP2018/059032		2018-04-09
PCT/EP2018/059032 WO2019197015A1 (fr)	2018-04-09	2018-04-09	Composition comprenant des dérivés d'acide 4-phénylbutyrique et des opioïdes

Publications (1)

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TW201943687A true TW201943687A (zh)	2019-11-16

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TW108109828A TW201943687A (zh)	2018-04-09	2019-03-21	包含4-苯丁酸衍生物及類鴉片的組成物

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TW (1)	TW201943687A (fr)
WO (1)	WO2019197015A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2024256849A1 (fr) *	2023-06-13	2024-12-19	Phenotec Ag	Dérivés d'acide 4-phénylbutyrique destinés à être utilisés en traitement de fibrose

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2593341B1 (fr)	1986-01-20	1988-03-04	Alcatel Thomson Faisceaux	Dispositif de recuperation de rythme
ES2283220B1 (es) *	2006-04-12	2008-11-01	Consejo Superior Investig. Cientificas	Uso de agonistas del receptor opioide delta en la elaboracion de composiciones farmaceuticas, composiciones farmaceuticas que las contienen y sus aplicaciones en el tratamiento de tumores.
PT2149372E (pt)	2008-07-31	2014-07-25	Universität Ulm	Utilização de opióides do grupo da metadona para o tratamento de pacientes com cancros resistentes
EP2599767A1 (fr)	2011-11-30	2013-06-05	Lunamed AG	Dérivés de phénylbutyl
PT2716291T (pt) *	2012-10-08	2020-03-04	Univ Ulm	Associação de opióides e fármacos anticancerígenos para o tratamento de cancro

2018
- 2018-04-09 WO PCT/EP2018/059032 patent/WO2019197015A1/fr not_active Ceased
2019
- 2019-03-21 TW TW108109828A patent/TW201943687A/zh unknown

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Publication number	Publication date
WO2019197015A1 (fr)	2019-10-17

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