TW200637553A - Indlomorphinane derivatives having a carboxy group at 6' position - Google Patents
Indlomorphinane derivatives having a carboxy group at 6' positionInfo
- Publication number
- TW200637553A TW200637553A TW094144035A TW94144035A TW200637553A TW 200637553 A TW200637553 A TW 200637553A TW 094144035 A TW094144035 A TW 094144035A TW 94144035 A TW94144035 A TW 94144035A TW 200637553 A TW200637553 A TW 200637553A
- Authority
- TW
- Taiwan
- Prior art keywords
- group
- hydrogen atom
- indlomorphinane
- derivatives
- carboxy group
- Prior art date
Links
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 title 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 206010028813 Nausea Diseases 0.000 abstract 1
- 125000004423 acyloxy group Chemical group 0.000 abstract 1
- 125000005194 alkoxycarbonyloxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 230000008693 nausea Effects 0.000 abstract 1
- 230000000069 prophylactic effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
- 229940124597 therapeutic agent Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/20—Spiro-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2004360966 | 2004-12-14 | ||
| JP2005028927 | 2005-02-04 | ||
| JP2005111912 | 2005-04-08 | ||
| JP2005296033 | 2005-10-11 | ||
| JP2005296045 | 2005-10-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW200637553A true TW200637553A (en) | 2006-11-01 |
Family
ID=36587834
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW094144035A TW200637553A (en) | 2004-12-14 | 2005-12-13 | Indlomorphinane derivatives having a carboxy group at 6' position |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20080227803A1 (zh) |
| EP (1) | EP1837022A4 (zh) |
| JP (1) | JPWO2006064779A1 (zh) |
| CA (1) | CA2590182A1 (zh) |
| TW (1) | TW200637553A (zh) |
| WO (1) | WO2006064779A1 (zh) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2240022B1 (en) * | 2008-01-09 | 2016-12-28 | Charleston Laboratories, Inc. | Bilayered tablets comprising oxycodone and promethazine |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9401728D0 (sv) * | 1994-05-18 | 1994-05-18 | Astra Ab | New compounds II |
| CO5271697A1 (es) * | 2000-01-12 | 2003-04-30 | Pfizer Prod Inc | Composiciones y procedimientos para el tratamiento de afecciones que responden a un aumento de testosterona |
| US7105556B2 (en) * | 2001-05-30 | 2006-09-12 | Bristol-Myers Squibb Company | Conformationally constrained analogs useful as antidiabetic and antiobesity agents and method |
| AP1816A (en) * | 2001-10-22 | 2008-01-04 | Pfizer Prod Inc | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists. |
| JP2004099586A (ja) * | 2002-05-21 | 2004-04-02 | Sumitomo Pharmaceut Co Ltd | ジヒドロオロテートデヒドロゲナーゼ阻害剤 |
| EP1522542A1 (en) * | 2002-07-11 | 2005-04-13 | Toray Industries, Inc. | Therapeutic or preventive agent for nausea/vomiting |
| TW200407127A (en) * | 2002-08-21 | 2004-05-16 | Astrazeneca Ab | Chemical compounds |
| JP2004143164A (ja) * | 2002-10-03 | 2004-05-20 | Sankyo Co Ltd | 活性化血液凝固第x因子阻害剤 |
| JP2004346059A (ja) * | 2003-01-28 | 2004-12-09 | Takeda Chem Ind Ltd | 受容体作動薬 |
| JP2004238296A (ja) * | 2003-02-04 | 2004-08-26 | Kissei Pharmaceut Co Ltd | 新規なトリアゾロピリミジン誘導体、それを含有する医薬組成物およびそれらの用途 |
-
2005
- 2005-12-13 US US11/792,876 patent/US20080227803A1/en not_active Abandoned
- 2005-12-13 WO PCT/JP2005/022820 patent/WO2006064779A1/ja not_active Ceased
- 2005-12-13 EP EP05816773A patent/EP1837022A4/en not_active Withdrawn
- 2005-12-13 CA CA002590182A patent/CA2590182A1/en not_active Abandoned
- 2005-12-13 JP JP2006548840A patent/JPWO2006064779A1/ja not_active Abandoned
- 2005-12-13 TW TW094144035A patent/TW200637553A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPWO2006064779A1 (ja) | 2008-06-12 |
| EP1837022A4 (en) | 2009-12-16 |
| CA2590182A1 (en) | 2006-06-22 |
| WO2006064779A1 (ja) | 2006-06-22 |
| EP1837022A1 (en) | 2007-09-26 |
| US20080227803A1 (en) | 2008-09-18 |
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