TW200635932A - New pyridothienopyrimidine derivatives - Google Patents

New pyridothienopyrimidine derivatives

Info

Publication number: TW200635932A
Authority: TW; Taiwan
Prior art keywords: diseases; new; pde4; pyridothienopyrimidine; derivatives
Prior art date: 2004-11-30

Application number

TW094142175A

Other languages

English (en)

Inventor

Santacana Lluis Miquel Pages

Moll Joan Taltavull

Original Assignee

Almirall Prodesfarma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-11-30

Filing date

2005-11-30

Publication date

2006-10-16

2005-11-30 Application filed by Almirall Prodesfarma Sa filed Critical Almirall Prodesfarma Sa

2006-10-16 Publication of TW200635932A publication Critical patent/TW200635932A/zh

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Epidemiology (AREA)
Pulmonology (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pain & Pain Management (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

TW094142175A 2004-11-30 2005-11-30 New pyridothienopyrimidine derivatives TW200635932A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
ES200402876A ES2259891B1 (es)	2004-11-30	2004-11-30	Nuevos derivados de piridotienopirimidina.

Publications (1)

Publication Number	Publication Date
TW200635932A true TW200635932A (en)	2006-10-16

Family

ID=35064879

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
TW094142175A TW200635932A (en)	2004-11-30	2005-11-30	New pyridothienopyrimidine derivatives

Country Status (21)

Country	Link
US (1)	US20090029955A1 (zh)
EP (1)	EP1819710B1 (zh)
JP (1)	JP2008521855A (zh)
KR (1)	KR20070086869A (zh)
CN (1)	CN101068816A (zh)
AR (1)	AR051686A1 (zh)
AT (1)	ATE425167T1 (zh)
AU (1)	AU2005311423A1 (zh)
BR (1)	BRPI0518094A (zh)
CA (1)	CA2588741A1 (zh)
DE (1)	DE602005013278D1 (zh)
ES (2)	ES2259891B1 (zh)
IL (1)	IL183142A0 (zh)
MX (1)	MX2007006173A (zh)
NO (1)	NO20073283L (zh)
PE (1)	PE20061078A1 (zh)
RU (1)	RU2007124326A (zh)
TW (1)	TW200635932A (zh)
UY (1)	UY29239A1 (zh)
WO (1)	WO2006058724A1 (zh)
ZA (1)	ZA200703827B (zh)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7763609B2 (en)	2003-12-15	2010-07-27	Schering Corporation	Heterocyclic aspartyl protease inhibitors
ES2281251B1 (es) *	2005-07-27	2008-08-16	Laboratorios Almirall S.A.	Nuevos derivados de pirido (3',2':4,5) furo (3,2-d) pirimidina.
JP2009508966A (ja) *	2005-09-23	2009-03-05	シェーリングコーポレイション	治療薬としての縮合四環性ｍＧｌｕＲ１アンタゴニスト
BR112012026157A2 (pt) *	2010-04-14	2015-09-08	Bayer Cropscience Ag	processo para preparar ditiina-tetracarboximidas.
EP3474846B1 (en)	2016-06-22	2022-11-30	Vanderbilt University	Positive allosteric modulators of the muscarinic acetylcholine receptor m4
MA46899A (fr)	2016-11-07	2021-04-14	Univ Vanderbilt	Modulateurs allostériques positifs du récepteur muscarinique de l'acétylcholine m4
JP7099725B2 (ja)	2016-11-07	2022-07-12	ヴァンダービルトユニヴァーシティ	ムスカリン性アセチルコリンレセプターｍ４のポジティブアロステリック調節因子
EP3534901B1 (en)	2016-11-07	2022-06-22	Vanderbilt University	Positive allosteric modulators of the muscarinic acetylcholine receptor m4
TW201930311A (zh)	2017-12-05	2019-08-01	泛德比爾特大學	蕈毒鹼型乙醯膽鹼受體m4之正向別構調節劑
US11376254B2 (en)	2017-12-05	2022-07-05	Vanderbilt University	Positive allosteric modulators of the muscarinic acetylcholine receptor M4
US20230084927A1 (en) *	2019-11-13	2023-03-16	Metabomed Ltd.	Glucose uptake inhibitors and uses thereof
CN115684415B (zh) *	2022-11-02	2024-09-10	山东华泰新材料技术研发有限公司	一种高效液相色谱测定5,6-二氢环戊并[b]噻吩-4-酮含量的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE19644228A1 (de) *	1996-10-24	1998-04-30	Merck Patent Gmbh	Thienopyrimidine
DE19752952A1 (de) *	1997-11-28	1999-06-02	Merck Patent Gmbh	Thienopyrimidine
DE19819023A1 (de) *	1998-04-29	1999-11-04	Merck Patent Gmbh	Thienopyrimidine
KR20010105399A (ko) *	1999-03-30	2001-11-28	쓰끼하시 다미까따	티에노피리미딘 화합물 및 그의 염, 및 그들의 제조 방법

2004
- 2004-11-30 ES ES200402876A patent/ES2259891B1/es not_active Expired - Fee Related
2005
- 2005-11-28 AR ARP050104956A patent/AR051686A1/es unknown
- 2005-11-28 PE PE2005001379A patent/PE20061078A1/es not_active Application Discontinuation
- 2005-11-29 UY UY29239A patent/UY29239A1/es unknown
- 2005-11-30 KR KR1020077015102A patent/KR20070086869A/ko not_active Withdrawn
- 2005-11-30 BR BRPI0518094-5A patent/BRPI0518094A/pt not_active IP Right Cessation
- 2005-11-30 JP JP2007543767A patent/JP2008521855A/ja active Pending
- 2005-11-30 EP EP05814833A patent/EP1819710B1/en not_active Expired - Lifetime
- 2005-11-30 CA CA002588741A patent/CA2588741A1/en not_active Abandoned
- 2005-11-30 RU RU2007124326/04A patent/RU2007124326A/ru not_active Application Discontinuation
- 2005-11-30 AT AT05814833T patent/ATE425167T1/de not_active IP Right Cessation
- 2005-11-30 US US11/791,450 patent/US20090029955A1/en not_active Abandoned
- 2005-11-30 MX MX2007006173A patent/MX2007006173A/es not_active Application Discontinuation
- 2005-11-30 ES ES05814833T patent/ES2321966T3/es not_active Expired - Lifetime
- 2005-11-30 WO PCT/EP2005/012774 patent/WO2006058724A1/en not_active Ceased
- 2005-11-30 TW TW094142175A patent/TW200635932A/zh unknown
- 2005-11-30 AU AU2005311423A patent/AU2005311423A1/en not_active Abandoned
- 2005-11-30 DE DE602005013278T patent/DE602005013278D1/de not_active Expired - Fee Related
- 2005-11-30 CN CNA200580040992XA patent/CN101068816A/zh active Pending
2007
- 2007-05-10 IL IL183142A patent/IL183142A0/en unknown
- 2007-05-11 ZA ZA200703827A patent/ZA200703827B/xx unknown
- 2007-06-27 NO NO20073283A patent/NO20073283L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
EP1819710B1 (en)	2009-03-11
ZA200703827B (en)	2008-08-27
UY29239A1 (es)	2006-02-24
RU2007124326A (ru)	2009-01-10
AR051686A1 (es)	2007-01-31
NO20073283L (no)	2007-06-27
BRPI0518094A (pt)	2008-10-28
ES2259891A1 (es)	2006-10-16
DE602005013278D1 (de)	2009-04-23
ATE425167T1 (de)	2009-03-15
CN101068816A (zh)	2007-11-07
JP2008521855A (ja)	2008-06-26
KR20070086869A (ko)	2007-08-27
IL183142A0 (en)	2007-09-20
ES2321966T3 (es)	2009-06-15
US20090029955A1 (en)	2009-01-29
ES2259891B1 (es)	2007-11-01
AU2005311423A1 (en)	2006-06-08
WO2006058724A1 (en)	2006-06-08
HK1101638A1 (zh)	2007-10-18
CA2588741A1 (en)	2006-06-08
PE20061078A1 (es)	2006-11-10
MX2007006173A (es)	2007-07-09
EP1819710A1 (en)	2007-08-22

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WO2007076286A3 (en)	2007-11-29	Chemical compounds
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