TR201002084A1 - Oral yolla dağılan donepezil tablet formülasyonları ve hazırlama yöntemi - Google Patents
Oral yolla dağılan donepezil tablet formülasyonları ve hazırlama yöntemiInfo
- Publication number
- TR201002084A1 TR201002084A1 TR2010/02084A TR201002084A TR201002084A1 TR 201002084 A1 TR201002084 A1 TR 201002084A1 TR 2010/02084 A TR2010/02084 A TR 2010/02084A TR 201002084 A TR201002084 A TR 201002084A TR 201002084 A1 TR201002084 A1 TR 201002084A1
- Authority
- TR
- Turkey
- Prior art keywords
- preparation
- tablet formulations
- oral dispersible
- donepezil
- donepezil tablet
- Prior art date
Links
- 239000007916 tablet composition Substances 0.000 title abstract 2
- ADEBPBSSDYVVLD-UHFFFAOYSA-N donepezil Chemical compound O=C1C=2C=C(OC)C(OC)=CC=2CC1CC(CC1)CCN1CC1=CC=CC=C1 ADEBPBSSDYVVLD-UHFFFAOYSA-N 0.000 title 2
- 229960003530 donepezil Drugs 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
- FBPFZTCFMRRESA-KVTDHHQDSA-N D-Mannitol Chemical compound OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)CO FBPFZTCFMRRESA-KVTDHHQDSA-N 0.000 abstract 1
- 229930195725 Mannitol Natural products 0.000 abstract 1
- WHNWPMSKXPGLAX-UHFFFAOYSA-N N-Vinyl-2-pyrrolidone Chemical compound C=CN1CCCC1=O WHNWPMSKXPGLAX-UHFFFAOYSA-N 0.000 abstract 1
- 239000004376 Sucralose Substances 0.000 abstract 1
- 229960000913 crospovidone Drugs 0.000 abstract 1
- 229960003135 donepezil hydrochloride Drugs 0.000 abstract 1
- XWAIAVWHZJNZQQ-UHFFFAOYSA-N donepezil hydrochloride Chemical compound [H+].[Cl-].O=C1C=2C=C(OC)C(OC)=CC=2CC1CC(CC1)CCN1CC1=CC=CC=C1 XWAIAVWHZJNZQQ-UHFFFAOYSA-N 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 235000010355 mannitol Nutrition 0.000 abstract 1
- 239000000594 mannitol Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 235000013809 polyvinylpolypyrrolidone Nutrition 0.000 abstract 1
- 229920000523 polyvinylpolypyrrolidone Polymers 0.000 abstract 1
- BAQAVOSOZGMPRM-QBMZZYIRSA-N sucralose Chemical compound O[C@@H]1[C@@H](O)[C@@H](Cl)[C@@H](CO)O[C@@H]1O[C@@]1(CCl)[C@@H](O)[C@H](O)[C@@H](CCl)O1 BAQAVOSOZGMPRM-QBMZZYIRSA-N 0.000 abstract 1
- 235000019408 sucralose Nutrition 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Zoology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2010/02084A TR201002084A1 (tr) | 2010-03-19 | 2010-03-19 | Oral yolla dağılan donepezil tablet formülasyonları ve hazırlama yöntemi |
| EP11719675A EP2547330A2 (fr) | 2010-03-19 | 2011-03-17 | Formulations de comprime delitant par voie orale de donepezil et procede pour preparer celui-ci |
| PCT/TR2011/000071 WO2011115599A2 (fr) | 2010-03-19 | 2011-03-17 | Formulations de comprimé délitant par voie orale de donépézil et procédé pour préparer celui-ci |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| TR2010/02084A TR201002084A1 (tr) | 2010-03-19 | 2010-03-19 | Oral yolla dağılan donepezil tablet formülasyonları ve hazırlama yöntemi |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR201002084A1 true TR201002084A1 (tr) | 2011-10-21 |
Family
ID=42668843
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2010/02084A TR201002084A1 (tr) | 2010-03-19 | 2010-03-19 | Oral yolla dağılan donepezil tablet formülasyonları ve hazırlama yöntemi |
Country Status (3)
| Country | Link |
|---|---|
| EP (1) | EP2547330A2 (fr) |
| TR (1) | TR201002084A1 (fr) |
| WO (1) | WO2011115599A2 (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2826465B1 (fr) * | 2013-07-19 | 2018-09-05 | Sanovel Ilac Sanayi ve Ticaret A.S. | Formulations de comprimé à désintégration orale de donépézil |
| CN114748435B (zh) * | 2022-05-18 | 2023-06-23 | 四川升和药业股份有限公司 | 一种盐酸多奈哌齐口崩片及其制备方法 |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020071864A1 (en) * | 1999-03-25 | 2002-06-13 | Yuhan Corporation | Rapidly disintegrable tablet for oral administration |
| WO2004066974A1 (fr) * | 2003-01-30 | 2004-08-12 | Ethypharm | Particules presentant un enrobage de masquage du gout, procede de preparation associe et comprimes orodispersibles contenant lesdites particules enrobees |
| EP1681048A1 (fr) * | 2005-01-14 | 2006-07-19 | Krka Tovarna Zdravil, D.D., Novo Mesto | Composition à désintégration orale à base d'olanzépine ou de donepézil |
| WO2007074472A2 (fr) * | 2005-12-27 | 2007-07-05 | Jubilant Organosys Limited | Composition pharmaceutique se dissolvant dans la bouche et son procede de preparation |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4642903A (en) | 1985-03-26 | 1987-02-17 | R. P. Scherer Corporation | Freeze-dried foam dosage form |
| US5188825A (en) | 1989-12-28 | 1993-02-23 | Iles Martin C | Freeze-dried dosage forms and methods for preparing the same |
| WO1995001782A2 (fr) | 1993-07-09 | 1995-01-19 | R.P. Scherer Corporation | Procede de fabrication de formes galeniques de medicaments lyophilises |
| GB9421836D0 (en) | 1994-10-28 | 1994-12-14 | Scherer Corp R P | Process for preparing solid pharmaceutical dosage forms of hydrophobic substances |
| US5976577A (en) | 1997-07-11 | 1999-11-02 | Rp Scherer Corporation | Process for preparing fast dispersing solid oral dosage form |
| EP1120109A3 (fr) | 2000-01-24 | 2002-07-10 | Pfizer Products Inc. | Formes posologiques solides à désintégration et dissolution rapide |
-
2010
- 2010-03-19 TR TR2010/02084A patent/TR201002084A1/xx unknown
-
2011
- 2011-03-17 EP EP11719675A patent/EP2547330A2/fr not_active Withdrawn
- 2011-03-17 WO PCT/TR2011/000071 patent/WO2011115599A2/fr not_active Ceased
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020071864A1 (en) * | 1999-03-25 | 2002-06-13 | Yuhan Corporation | Rapidly disintegrable tablet for oral administration |
| WO2004066974A1 (fr) * | 2003-01-30 | 2004-08-12 | Ethypharm | Particules presentant un enrobage de masquage du gout, procede de preparation associe et comprimes orodispersibles contenant lesdites particules enrobees |
| EP1681048A1 (fr) * | 2005-01-14 | 2006-07-19 | Krka Tovarna Zdravil, D.D., Novo Mesto | Composition à désintégration orale à base d'olanzépine ou de donepézil |
| WO2007074472A2 (fr) * | 2005-12-27 | 2007-07-05 | Jubilant Organosys Limited | Composition pharmaceutique se dissolvant dans la bouche et son procede de preparation |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011115599A3 (fr) | 2011-12-08 |
| EP2547330A2 (fr) | 2013-01-23 |
| WO2011115599A2 (fr) | 2011-09-22 |
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