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TR200103576T2 - Üre ikameli/katkılı imidazokinolinler. - Google Patents

Üre ikameli/katkılı imidazokinolinler.

Info

Publication number
TR200103576T2
TR200103576T2 TR2001/03576T TR200103576T TR200103576T2 TR 200103576 T2 TR200103576 T2 TR 200103576T2 TR 2001/03576 T TR2001/03576 T TR 2001/03576T TR 200103576 T TR200103576 T TR 200103576T TR 200103576 T2 TR200103576 T2 TR 200103576T2
Authority
TR
Turkey
Prior art keywords
urea substituted
useful
substituted imidazoquinolines
imidazoquinolines
compounds
Prior art date
Application number
TR2001/03576T
Other languages
English (en)
Inventor
L. Crooks Stephen
A. Merrill Bryon
J. Rice Michael
Original Assignee
3M Innovative Properties Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 3M Innovative Properties Company filed Critical 3M Innovative Properties Company
Publication of TR200103576T2 publication Critical patent/TR200103576T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Toxicology (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

1-pozisyonunda üre, tioüre, asilüre, veya sülfonilüre fonksiyonalitesi içeren imidazokinolin ve tetrahidroimidazokinolin bilesikleri, immun cevap modifayerleri olarak faydalidir. Bu bulusun bilesikleri ve kompozisyonlari, muhtelif sitokinlerin biyosentezini indükleyebilir ve viral hastaliklar ve neoplastik hastaliklar da dahil olamak üzere muhtelif durumlarin tedavisinde faydali olur.
TR2001/03576T 1999-06-10 2000-06-08 Üre ikameli/katkılı imidazokinolinler. TR200103576T2 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13836599P 1999-06-10 1999-06-10
US09/589,236 US6541485B1 (en) 1999-06-10 2000-06-07 Urea substituted imidazoquinolines

Publications (1)

Publication Number Publication Date
TR200103576T2 true TR200103576T2 (tr) 2002-06-21

Family

ID=26836140

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2001/03576T TR200103576T2 (tr) 1999-06-10 2000-06-08 Üre ikameli/katkılı imidazokinolinler.

Country Status (26)

Country Link
US (2) US6541485B1 (tr)
EP (1) EP1198232B1 (tr)
JP (1) JP2003501473A (tr)
KR (1) KR20020008223A (tr)
CN (1) CN1181070C (tr)
AT (1) ATE337007T1 (tr)
AU (1) AU766565B2 (tr)
BR (1) BR0014214A (tr)
CA (1) CA2376296A1 (tr)
DE (1) DE60030293T2 (tr)
DK (1) DK1198232T3 (tr)
EE (1) EE05065B1 (tr)
ES (1) ES2270839T3 (tr)
HK (1) HK1047224A1 (tr)
HR (1) HRP20010889A2 (tr)
HU (1) HUP0201664A2 (tr)
IL (1) IL146572A0 (tr)
MX (1) MXPA01012598A (tr)
NO (1) NO320853B1 (tr)
NZ (1) NZ515968A (tr)
PL (1) PL352257A1 (tr)
PT (1) PT1198232E (tr)
RU (1) RU2265020C2 (tr)
SK (1) SK17972001A3 (tr)
TR (1) TR200103576T2 (tr)
WO (1) WO2000076518A1 (tr)

Families Citing this family (162)

* Cited by examiner, † Cited by third party
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