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TNSN07141A1 - Use of 4-(4-methylpiperazin-1-ylmethyl)-n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide to inhibit the tyrosine kinase receptor c-fms - Google Patents

Use of 4-(4-methylpiperazin-1-ylmethyl)-n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide to inhibit the tyrosine kinase receptor c-fms

Info

Publication number
TNSN07141A1
TNSN07141A1 TNP2007000141A TNSN07141A TNSN07141A1 TN SN07141 A1 TNSN07141 A1 TN SN07141A1 TN P2007000141 A TNP2007000141 A TN P2007000141A TN SN07141 A TNSN07141 A TN SN07141A TN SN07141 A1 TNSN07141 A1 TN SN07141A1
Authority
TN
Tunisia
Prior art keywords
methylpiperazin
ylamino
benzamide
pyrimidin
ylmethyl
Prior art date
Application number
TNP2007000141A
Other languages
English (en)
Inventor
Andrea Louis Dewar
Timothy Peter Hughes
Alan Bruce Lyons
Original Assignee
Medvet Science Pty Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medvet Science Pty Ltd filed Critical Medvet Science Pty Ltd
Publication of TNSN07141A1 publication Critical patent/TNSN07141A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
TNP2007000141A 2004-10-18 2007-04-17 Use of 4-(4-methylpiperazin-1-ylmethyl)-n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide to inhibit the tyrosine kinase receptor c-fms TNSN07141A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61974404P 2004-10-18 2004-10-18
PCT/AU2005/001602 WO2006042362A1 (fr) 2004-10-18 2005-10-17 Inhibition du récepteur à tyrosine kinase c-fms à l’aide du 4-(4-méthylpipérazin-1-ylméthyl)-n-[4-méthyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phényl]benzamide

Publications (1)

Publication Number Publication Date
TNSN07141A1 true TNSN07141A1 (en) 2008-11-21

Family

ID=36202610

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2007000141A TNSN07141A1 (en) 2004-10-18 2007-04-17 Use of 4-(4-methylpiperazin-1-ylmethyl)-n-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide to inhibit the tyrosine kinase receptor c-fms

Country Status (19)

Country Link
US (1) US20080255139A1 (fr)
EP (1) EP1804800B1 (fr)
JP (1) JP2008516898A (fr)
KR (1) KR20070083705A (fr)
CN (1) CN101035535A (fr)
AT (1) ATE492277T1 (fr)
AU (1) AU2005297321A1 (fr)
BR (1) BRPI0517083A (fr)
CA (1) CA2580976A1 (fr)
DE (1) DE602005025514D1 (fr)
IL (1) IL182419A0 (fr)
MA (1) MA28946B1 (fr)
MX (1) MX2007004660A (fr)
NO (1) NO20072501L (fr)
NZ (1) NZ554009A (fr)
RU (1) RU2007118420A (fr)
TN (1) TNSN07141A1 (fr)
WO (1) WO2006042362A1 (fr)
ZA (1) ZA200702316B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009058968A2 (fr) * 2007-10-31 2009-05-07 Janssen Pharmaceutica N.V. Biomarqueur utilisé pour évaluer une réponse à un traitement de fms
SG11201705767PA (en) * 2015-01-13 2017-08-30 Univ Kyoto Agent for preventing and/or treating amyotrophic lateral sclerosis

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4837237A (en) * 1985-07-09 1989-06-06 Fred Hutchinson Cancer Research Center Therapy using glucosidase processing inhibitors
AU2002342878A1 (en) * 2001-05-16 2002-11-25 Axxima Pharmaceuticals Ag Pyridylpyrimidine derivatives as effective compounds against prion diseases
WO2004026930A2 (fr) * 2002-06-26 2004-04-01 The Ohio State University Research Foundation Composes organiques

Also Published As

Publication number Publication date
MX2007004660A (es) 2007-10-17
CA2580976A1 (fr) 2006-04-27
DE602005025514D1 (de) 2011-02-03
EP1804800A4 (fr) 2008-03-19
RU2007118420A (ru) 2008-11-27
ATE492277T1 (de) 2011-01-15
MA28946B1 (fr) 2007-10-01
ZA200702316B (en) 2008-09-25
EP1804800A1 (fr) 2007-07-11
US20080255139A1 (en) 2008-10-16
JP2008516898A (ja) 2008-05-22
IL182419A0 (en) 2007-09-20
BRPI0517083A (pt) 2008-09-30
NO20072501L (no) 2007-05-15
AU2005297321A1 (en) 2006-04-27
KR20070083705A (ko) 2007-08-24
CN101035535A (zh) 2007-09-12
WO2006042362A1 (fr) 2006-04-27
EP1804800B1 (fr) 2010-12-22
NZ554009A (en) 2010-09-30

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