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TNSN06366A1 - PROLINE DERIVATIVES AND THEIR USE AS INHIBITORS OF IV DIPEPTIDYL PEPTIDASE - Google Patents

PROLINE DERIVATIVES AND THEIR USE AS INHIBITORS OF IV DIPEPTIDYL PEPTIDASE

Info

Publication number
TNSN06366A1
TNSN06366A1 TNP2006000366A TNSN06366A TNSN06366A1 TN SN06366 A1 TNSN06366 A1 TN SN06366A1 TN P2006000366 A TNP2006000366 A TN P2006000366A TN SN06366 A TNSN06366 A TN SN06366A TN SN06366 A1 TNSN06366 A1 TN SN06366A1
Authority
TN
Tunisia
Prior art keywords
des
leurs
diabétique
médicamenteux
stéréoisomères
Prior art date
Application number
TNP2006000366A
Other languages
French (fr)
Inventor
David Walter Piotrowski
Bernard Hulin
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/IB2005/001194 external-priority patent/WO2005116014A1/en
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TNSN06366A1 publication Critical patent/TNSN06366A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyrrole Compounds (AREA)

Abstract

La présente invention propose des composés de formule (I), Leurs précurseurs médicamenteux et leurs et des stéréoisomères, et les sels pharmaceutiquement acceptables des composés, précurseurs médicamenteux et stéréoisomères, formule dans laquelle R1, R2, R3, HET, n, Q, X, Y, et Z répondent aux définitions figurant dans le présent mémoire ; des compositions les contenant ; et leurs utilisations pour le traitement des complications du diabète, comprenant la neuropathie diabétique, la néphropathie diabétique, la microangiopathie diabétique et des complications similaires.
TNP2006000366A 2004-05-12 2006-11-10 PROLINE DERIVATIVES AND THEIR USE AS INHIBITORS OF IV DIPEPTIDYL PEPTIDASE TNSN06366A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US57030004P 2004-05-12 2004-05-12
PCT/IB2005/001194 WO2005116014A1 (en) 2004-05-12 2005-04-29 Proline derivatives and their use as dipeptidyl peptidase iv inhibitors

Publications (1)

Publication Number Publication Date
TNSN06366A1 true TNSN06366A1 (en) 2008-02-22

Family

ID=38077110

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2006000366A TNSN06366A1 (en) 2004-05-12 2006-11-10 PROLINE DERIVATIVES AND THEIR USE AS INHIBITORS OF IV DIPEPTIDYL PEPTIDASE

Country Status (5)

Country Link
CN (1) CN1968949B (en)
HN (1) HN2005000205A (en)
TN (1) TNSN06366A1 (en)
UA (1) UA83133C2 (en)
ZA (1) ZA200608741B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016107832A1 (en) * 2014-12-30 2016-07-07 F. Hoffmann-La Roche Ag Novel tetrahydropyridopyrimidines and tetrahydropyridopyridines for the treatment and prophylaxis of hepatitis b virus infection
EP3292120B1 (en) * 2015-05-04 2019-06-19 H. Hoffnabb-La Roche Ag Tetrahydropyridopyrimidines and tetrahydropyridopyridines as inhibitors of hbsag (hbv surface antigen) and hbv dna production for the treatment of hepatitis b virus infections
CN114213504B (en) * 2021-12-24 2023-05-09 西南医科大学 A class of compounds with antidiabetic activity and their applications
CN118831080B (en) * 2024-09-24 2024-11-22 上海交通大学医学院附属仁济医院 Application of 5-oxyproline in preparing medicine for preventing or treating cardiomyopathy

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE411285T1 (en) * 2000-08-10 2008-10-15 Mitsubishi Tanabe Pharma Corp PROLINE DERIVATIVES AND THEIR USE AS MEDICATIONS
GB0115517D0 (en) * 2001-06-25 2001-08-15 Ferring Bv Novel antidiabetic agents

Also Published As

Publication number Publication date
ZA200608741B (en) 2008-07-30
HN2005000205A (en) 2009-10-30
UA83133C2 (en) 2008-06-10
CN1968949B (en) 2011-05-04
CN1968949A (en) 2007-05-23

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