TNSN98194A1 - Derives nouveaux de 6-o-methylerythromycine a, procede pour leur preparation et compositions pharmaceutiques les contenant - Google Patents
Derives nouveaux de 6-o-methylerythromycine a, procede pour leur preparation et compositions pharmaceutiques les contenantInfo
- Publication number
- TNSN98194A1 TNSN98194A1 TNTNSN98194A TNSN98194A TNSN98194A1 TN SN98194 A1 TNSN98194 A1 TN SN98194A1 TN TNSN98194 A TNTNSN98194 A TN TNSN98194A TN SN98194 A TNSN98194 A TN SN98194A TN SN98194 A1 TNSN98194 A1 TN SN98194A1
- Authority
- TN
- Tunisia
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions containing
- methylerythromycin
- derivatives
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- AGOYDEPGAOXOCK-KCBOHYOISA-N clarithromycin Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@](C)([C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)OC)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 AGOYDEPGAOXOCK-KCBOHYOISA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 208000035143 Bacterial infection Diseases 0.000 abstract 1
- 208000022362 bacterial infectious disease Diseases 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
L'INVENTION CONCERNE DES COMPOSES DE FORMULE I DANS LAQUELLE R1, R2, R3, R4 ET X REPRESENTENT DIVERS RADICAUX. ELLE CONCERNE EGALEMENT DES PROCEDES POUR LA PREPARATION DE CES COMPOSES, AINSI QUE DES COMPOSITIONS PHARMACEUTIQUES LES CONTENANT. APPLICATION : UTILISATION DE CES COMPOSES ET COMPOSITIONS POUR LE TRAITEMENT OU LA PREVENTION D'INFECTIONS BACTERIENNES.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6367697P | 1997-10-29 | 1997-10-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TNSN98194A1 true TNSN98194A1 (fr) | 2005-03-15 |
Family
ID=22050768
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TNTNSN98194A TNSN98194A1 (fr) | 1997-10-29 | 1998-10-26 | Derives nouveaux de 6-o-methylerythromycine a, procede pour leur preparation et compositions pharmaceutiques les contenant |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US6159945A (fr) |
| AP (1) | AP9801378A0 (fr) |
| AR (1) | AR017177A1 (fr) |
| AU (1) | AU9277698A (fr) |
| CO (1) | CO4810375A1 (fr) |
| GT (1) | GT199800163A (fr) |
| HN (1) | HN1998000159A (fr) |
| HR (1) | HRP980571A2 (fr) |
| MA (1) | MA26558A1 (fr) |
| PA (1) | PA8461701A1 (fr) |
| PE (1) | PE122499A1 (fr) |
| TN (1) | TNSN98194A1 (fr) |
| WO (1) | WO1999021866A1 (fr) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6710033B1 (en) | 1996-08-14 | 2004-03-23 | Vanderbilt University | Methods and treatment of multiple sclerosis |
| US6890526B2 (en) | 1997-05-06 | 2005-05-10 | Vanderbilt University | Methods and reagents for the treatment of multiple sclerosis |
| AP9801420A0 (en) * | 1998-01-02 | 1998-12-31 | Pfizer Prod Inc | Novel macrolides. |
| AU3439899A (en) | 1998-06-03 | 1999-12-20 | Pfizer Products Inc. | Tricyclic 3-keto derivatives of 6-o-methylerythromycin |
| WO2000034297A1 (fr) * | 1998-12-10 | 2000-06-15 | Pfizer Products Inc. | Antibiotiques a base de cetolides de carbamate et de carbazate |
| EP1298138B1 (fr) * | 1998-12-10 | 2006-11-02 | Pfizer Products Inc. | Dérivés anitiobiotiques de Carbamate et de Carbazate Kètolides |
| SI1147121T1 (en) | 1999-01-27 | 2004-04-30 | Pfizer Products Inc. | Ketolide antibiotics |
| SK15162001A3 (sk) * | 1999-05-24 | 2003-02-04 | Pfizer Products Inc. | Deriváty 13-metylerytromycínu |
| ID27331A (id) * | 1999-09-29 | 2001-03-29 | Pfizer Prod Inc | Pembuatan antibiotik-antibiotik ketolida karbamat |
| US6498146B1 (en) * | 1999-10-28 | 2002-12-24 | Pfizer Inc | Erythromycin derivatives |
| EP1146051A3 (fr) * | 2000-04-10 | 2001-10-31 | Pfizer Products Inc. | Dérivées de l' érythromycine A |
| US20020115621A1 (en) * | 2000-08-07 | 2002-08-22 | Wei-Gu Su | Macrolide antibiotics |
| US20070003508A1 (en) * | 2005-07-01 | 2007-01-04 | Wooley Richard E | Methods and compositions for promoting wound healing |
| US20040151765A1 (en) * | 2001-09-18 | 2004-08-05 | Ritchie Branson W. | Methods and compositions for wound management |
| US20040208842A1 (en) * | 2001-09-18 | 2004-10-21 | Ritchie Branson W. | Antimicrobial cleansing compositions and methods of use |
| ES2552682T3 (es) | 2003-03-10 | 2015-12-01 | Merck Sharp & Dohme Corp. | Agentes antibacterianos novedosos |
| WO2005091967A2 (fr) * | 2004-03-03 | 2005-10-06 | University Of Georgia Research Foundation, Inc. | Procedes et compositions destines au traitement ophtalmique d'infections fongiques et bacteriennes |
| DE602005019786D1 (de) * | 2004-12-21 | 2010-04-15 | Pfizer Prod Inc | Makrolide |
| AU2008316830B2 (en) | 2007-10-25 | 2016-03-17 | Cempra Pharmaceuticals, Inc. | Process for the preparation of macrolide antibacterial agents |
| AU2009308181B2 (en) | 2008-10-24 | 2015-12-03 | Cempra Pharmaceuticals, Inc. | Methods for treating resistant diseases using triazole containing macrolides |
| US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
| ES2608285T3 (es) | 2009-09-10 | 2017-04-07 | Cempra Pharmaceuticals, Inc. | Procedimientos para el tratamiento de paludismo, tuberculosis y enfermedades por MAC |
| NZ602544A (en) | 2010-03-22 | 2014-11-28 | Cempra Pharmaceuticals Inc | Crystalline forms of a macrolide, and uses therefor |
| SI2571506T1 (sl) | 2010-05-20 | 2017-12-29 | Cempra Pharmaceuticals, Inc. | Postopki za pripravo makrolidov in ketolidov ter njihovih intermediatov |
| US9815863B2 (en) | 2010-09-10 | 2017-11-14 | Cempra Pharmaceuticals, Inc. | Hydrogen bond forming fluoro ketolides for treating diseases |
| SG11201405895UA (en) | 2012-03-27 | 2014-10-30 | Cempra Pharmaceuticals Inc | Parenteral formulations for administering macrolide antibiotics |
| CN105163785A (zh) | 2013-03-14 | 2015-12-16 | 森普拉制药公司 | 用于治疗呼吸道疾病的方法及其制剂 |
| JP6675973B2 (ja) | 2013-03-15 | 2020-04-08 | センプラ ファーマシューティカルズ,インコーポレイテッド | マクロライド抗菌薬を調製するための集束的な方法 |
| US9982005B2 (en) * | 2013-04-04 | 2018-05-29 | President And Fellows Of Harvard College | Macrolides and methods of their preparation and use |
| JP2017531663A (ja) | 2014-10-08 | 2017-10-26 | プレジデント アンド フェローズ オブ ハーバード カレッジ | 14員ケトライドならびにそれらの調製および使用の方法 |
| JP2018509452A (ja) | 2015-03-25 | 2018-04-05 | プレジデント アンド フェローズ オブ ハーバード カレッジ | 修飾デソサミン糖をもつマクロライドおよびその使用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL114589A (en) * | 1990-11-21 | 1999-12-22 | Roussel Uclaf | Intermediates for the preparation of erythromycin derivatives |
| US6060234A (en) * | 1991-01-17 | 2000-05-09 | Abbott Laboratories | Polyketide derivatives and recombinant methods for making same |
| EP0638585B1 (fr) * | 1992-04-22 | 1996-11-13 | Taisho Pharmaceutical Co. Ltd | Derive de 5-o-desosaminylerythronolide a |
| US6162794A (en) * | 1997-05-09 | 2000-12-19 | Pfizer Inc. | Erythromycin derivatives |
| CA2293335A1 (fr) * | 1997-06-11 | 1998-12-17 | Pfizer Products Inc., | Derives de 9-oxime erythromycine |
-
1998
- 1998-10-08 HN HN1998000159A patent/HN1998000159A/es unknown
- 1998-10-09 US US09/402,338 patent/US6159945A/en not_active Expired - Fee Related
- 1998-10-09 AU AU92776/98A patent/AU9277698A/en not_active Abandoned
- 1998-10-09 WO PCT/IB1998/001578 patent/WO1999021866A1/fr not_active Ceased
- 1998-10-16 PA PA19988461701A patent/PA8461701A1/es unknown
- 1998-10-22 PE PE1998000993A patent/PE122499A1/es not_active Application Discontinuation
- 1998-10-23 GT GT199800163A patent/GT199800163A/es unknown
- 1998-10-26 MA MA25314A patent/MA26558A1/fr unknown
- 1998-10-26 TN TNTNSN98194A patent/TNSN98194A1/fr unknown
- 1998-10-27 AR ARP980105379A patent/AR017177A1/es not_active Application Discontinuation
- 1998-10-29 CO CO98063687A patent/CO4810375A1/es unknown
- 1998-10-29 AP APAP/P/1998/001378A patent/AP9801378A0/en unknown
- 1998-10-29 HR HR60/063,676A patent/HRP980571A2/hr not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MA26558A1 (fr) | 2004-12-20 |
| CO4810375A1 (es) | 1999-06-30 |
| HRP980571A2 (en) | 1999-08-31 |
| AP9801378A0 (en) | 2000-04-29 |
| US6159945A (en) | 2000-12-12 |
| WO1999021866A1 (fr) | 1999-05-06 |
| HN1998000159A (es) | 1999-02-09 |
| AU9277698A (en) | 1999-05-17 |
| PE122499A1 (es) | 1999-12-02 |
| PA8461701A1 (es) | 2000-05-24 |
| AR017177A1 (es) | 2001-08-22 |
| GT199800163A (es) | 2000-04-15 |
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