TN2013000257A1 - Immunosuppressant formulations - Google Patents

Immunosuppressant formulations

Info

Publication number: TN2013000257A1
Authority: TN; Tunisia
Prior art keywords: api; immunosuppressant; formulations; compound; immunosuppressant formulations
Prior art date: 2011-01-07

Application number

TNP2013000257A

Other languages

English (en)

Inventor

Philippe Bouillot

Emeric Reynaud

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2011-01-07

Filing date

2013-06-14

Publication date

2014-11-10

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44022942&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2013000257(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2013-06-14 Application filed by Novartis Ag filed Critical Novartis Ag

2014-11-10 Publication of TN2013000257A1 publication Critical patent/TN2013000257A1/fr

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Organic Chemistry (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Immunology (AREA)
Rheumatology (AREA)
Transplantation (AREA)
Pain & Pain Management (AREA)
Oncology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Communicable Diseases (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

TNP2013000257A 2011-01-07 2013-06-14 Immunosuppressant formulations TN2013000257A1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP11150431		2011-01-07
PCT/EP2012/050151 WO2012093161A1 (fr)	2011-01-07	2012-01-05	Formulations d'immunosuppresseurs

Publications (1)

Publication Number	Publication Date
TN2013000257A1 true TN2013000257A1 (en)	2014-11-10

Family

ID=44022942

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
TNP2013000257A TN2013000257A1 (en)	2011-01-07	2013-06-14	Immunosuppressant formulations

Country Status (36)

Country	Link
US (4)	US20130273161A1 (fr)
EP (2)	EP2661261B1 (fr)
JP (2)	JP6111202B2 (fr)
KR (2)	KR102166885B1 (fr)
CN (1)	CN103458877B (fr)
AR (2)	AR084801A1 (fr)
AU (1)	AU2012204835B2 (fr)
BR (1)	BR112013017302B1 (fr)
CA (1)	CA2823616C (fr)
CL (1)	CL2013001979A1 (fr)
CO (1)	CO6761402A2 (fr)
CY (1)	CY1122182T1 (fr)
DK (1)	DK2661261T3 (fr)
EA (1)	EA026144B9 (fr)
EC (1)	ECSP13012812A (fr)
ES (1)	ES2751920T3 (fr)
GT (1)	GT201300178A (fr)
HR (1)	HRP20191842T1 (fr)
HU (1)	HUE045612T2 (fr)
IL (1)	IL227094B (fr)
JO (1)	JO3619B1 (fr)
LT (1)	LT2661261T (fr)
MA (1)	MA34897B1 (fr)
MX (2)	MX357304B (fr)
MY (1)	MY161162A (fr)
PE (1)	PE20140216A1 (fr)
PH (1)	PH12013501442B1 (fr)
PL (1)	PL2661261T3 (fr)
PT (1)	PT2661261T (fr)
SG (1)	SG191286A1 (fr)
SI (1)	SI2661261T1 (fr)
TN (1)	TN2013000257A1 (fr)
TW (2)	TWI610672B (fr)
UA (1)	UA114283C2 (fr)
WO (1)	WO2012093161A1 (fr)
ZA (1)	ZA201304465B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
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EP2661261B1 (fr)	2011-01-07	2019-07-31	Novartis AG	Formulations d'immunosuppresseurs
AU2015246038C1 (en) *	2014-04-10	2018-05-31	Novartis Ag	Immunosuppressant formulation
EP3129020A1 (fr) *	2014-04-10	2017-02-15	Novartis AG	Régime posologique de modulateur s1p à libération immédiate
CA2973540A1 (fr)	2015-02-26	2016-09-01	Novartis Ag	Traitement de maladie auto-immune chez un patient recevant en outre un betabloquant
HRP20230253T1 (hr) *	2015-07-03	2023-04-28	Astellas Pharma Inc.	Stabilna farmaceutska kompozicija za oralnu administraciju
US11629124B2 (en)	2017-03-09	2023-04-18	Novartis Ag	Solid forms comprising an oxime ether compound, compositions and methods of use thereof
US11434200B2 (en)	2017-03-09	2022-09-06	Novartis Ag	Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof
CN111107837A (zh)	2017-09-27	2020-05-05	诺华股份有限公司	包含西普尼莫德的肠胃外制剂
US20200306222A1 (en)	2017-09-29	2020-10-01	Novartis Ag	Dosing Regimen of Siponimod
JP2020535147A (ja)	2017-09-29	2020-12-03	ノバルティスアーゲー	シポニモドの投与レジメン
CN109908095A (zh) *	2019-04-08	2019-06-21	肇庆学院	一种西尼莫德片剂及制备方法
WO2021214717A1 (fr)	2020-04-23	2021-10-28	Novartis Ag	Schéma posologique pour l'utilisation de siponimod pour le traitement du syndrome de détresse respiratoire aiguë
IL315531A (en) *	2022-03-09	2024-11-01	Isp Investments Llc	The composition of an inactive substance for drugs, produced by joint processing of its components
EP4633611A1 (fr)	2022-12-12	2025-10-22	Synthon B.V.	Composition pharmaceutique contenant du siponimod

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JP2010526116A (ja)	2007-05-04	2010-07-29	ノバルティスアーゲー	Ｓ１ｐ受容体調節因子の使用
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CN102076335A (zh)	2008-06-20	2011-05-25	诺瓦提斯公司	用于治疗多发性硬化的儿科组合物
CN102105144B (zh)	2008-07-23	2013-11-13	诺华股份有限公司	鞘氨醇1磷酸酯受体调节剂以及它们用于制备治疗肌肉炎症的药物的用途
EP2326325B1 (fr) *	2008-08-18	2014-11-12	Novartis AG	Dérivé azétidine destinés au traitement de neuropathies périphériques
RS53041B (sr) *	2008-12-18	2014-04-30	Novartis Ag	Hemifumaratna so 1-[4-[1-(4-cikloheksil-3-trifluorometil-benziloksiimino)-etil]-2-etil-benzil]-azetidin-3-karboksilne kiseline
WO2010080455A1 (fr)	2008-12-18	2010-07-15	Novartis Ag	Nouveaux sels
EP2379498B1 (fr) *	2008-12-18	2015-01-21	Novartis AG	Forme polymorphe de l' acide 1-(4-{1-[(e)-4-cyclohexyl-3-trifluorométhyl-benzyloxyimino]-éthyl}-2-éthyl-benzyl)-azétidine-3-carboxylique
BRPI0922567A2 (pt)	2008-12-19	2015-12-15	Novartis Ag	boquilha para um inalador
HUE026400T2 (en)	2008-12-22	2016-06-28	Novartis Ag	Dosage Scheme for S1P Receptor Agonist
EP3677260A1 (fr)	2008-12-22	2020-07-08	Novartis AG	Posologie d'un agoniste du récepteur s1p
EP2482810A2 (fr)	2009-09-29	2012-08-08	Novartis AG	Schéma posologique d'un modulateur des récepteurs de s1p
EP2661261B1 (fr)	2011-01-07	2019-07-31	Novartis AG	Formulations d'immunosuppresseurs
WO2012095853A1 (fr)	2011-01-10	2012-07-19	Novartis Pharma Ag	Formulations à libération modifiée comprenant des modulateurs des récepteurs sip
TW201320994A (zh)	2011-10-11	2013-06-01	Novartis Ag	投藥療程
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AU2015246038C1 (en)	2014-04-10	2018-05-31	Novartis Ag	Immunosuppressant formulation

2012
- 2012-01-05 EP EP12700262.4A patent/EP2661261B1/fr active Active
- 2012-01-05 HR HRP20191842TT patent/HRP20191842T1/hr unknown
- 2012-01-05 MX MX2013007909A patent/MX357304B/es active IP Right Grant
- 2012-01-05 UA UAA201307576A patent/UA114283C2/uk unknown
- 2012-01-05 AU AU2012204835A patent/AU2012204835B2/en active Active
- 2012-01-05 HU HUE12700262A patent/HUE045612T2/hu unknown
- 2012-01-05 CN CN201280004869.2A patent/CN103458877B/zh active Active
- 2012-01-05 ES ES12700262T patent/ES2751920T3/es active Active
- 2012-01-05 SG SG2013047923A patent/SG191286A1/en unknown
- 2012-01-05 DK DK12700262.4T patent/DK2661261T3/da active
- 2012-01-05 EA EA201391018A patent/EA026144B9/ru active Protection Beyond IP Right Term
- 2012-01-05 PE PE2013001522A patent/PE20140216A1/es active IP Right Grant
- 2012-01-05 LT LT12700262T patent/LT2661261T/lt unknown
- 2012-01-05 PH PH1/2013/501442A patent/PH12013501442B1/en unknown
- 2012-01-05 MX MX2017007300A patent/MX371290B/es unknown
- 2012-01-05 JP JP2013547861A patent/JP6111202B2/ja active Active
- 2012-01-05 PL PL12700262T patent/PL2661261T3/pl unknown
- 2012-01-05 EP EP19188018.6A patent/EP3590507A1/fr active Pending
- 2012-01-05 CA CA2823616A patent/CA2823616C/fr active Active
- 2012-01-05 PT PT127002624T patent/PT2661261T/pt unknown
- 2012-01-05 JO JOP/2012/0005A patent/JO3619B1/ar active
- 2012-01-05 WO PCT/EP2012/050151 patent/WO2012093161A1/fr not_active Ceased
- 2012-01-05 SI SI201231683T patent/SI2661261T1/sl unknown
- 2012-01-05 BR BR112013017302-5A patent/BR112013017302B1/pt active IP Right Grant
- 2012-01-05 MA MA36170A patent/MA34897B1/fr unknown
- 2012-01-05 KR KR1020197004860A patent/KR102166885B1/ko not_active Expired - Fee Related
- 2012-01-05 KR KR1020137020755A patent/KR101951966B1/ko active Active
- 2012-01-06 TW TW101100702A patent/TWI610672B/zh active
- 2012-01-06 TW TW104142389A patent/TWI583380B/zh active
- 2012-01-06 MY MYPI2013002251A patent/MY161162A/en unknown
- 2012-01-06 AR ARP120100047A patent/AR084801A1/es not_active Application Discontinuation
2013
- 2013-06-14 US US13/917,730 patent/US20130273161A1/en not_active Abandoned
- 2013-06-14 TN TNP2013000257A patent/TN2013000257A1/fr unknown
- 2013-06-18 ZA ZA2013/04465A patent/ZA201304465B/en unknown
- 2013-06-20 IL IL227094A patent/IL227094B/en active IP Right Grant
- 2013-07-05 GT GT201300178A patent/GT201300178A/es unknown
- 2013-07-05 CL CL2013001979A patent/CL2013001979A1/es unknown
- 2013-07-16 CO CO13168667A patent/CO6761402A2/es unknown
- 2013-08-07 EC ECSP13012812 patent/ECSP13012812A/es unknown
2017
- 2017-03-13 JP JP2017047220A patent/JP6324569B2/ja active Active
2019
- 2019-10-22 CY CY20191101097T patent/CY1122182T1/el unknown
2020
- 2020-02-28 US US16/804,926 patent/US20200199069A1/en not_active Abandoned
2021
- 2021-04-14 US US17/230,175 patent/US12071402B2/en active Active
2022
- 2022-01-17 AR ARP220100086A patent/AR124662A2/es unknown
2024
- 2024-08-13 US US18/802,089 patent/US20250084034A1/en active Pending

Also Published As

Publication number	Publication date
ECSP13012812A (es)	2013-09-30
JO3619B1 (ar)	2020-08-27
CY1122182T1 (el)	2020-11-25
CO6761402A2 (es)	2013-09-30
HUE045612T2 (hu)	2020-01-28
US20200199069A1 (en)	2020-06-25
UA114283C2 (uk)	2017-05-25
US20220064110A1 (en)	2022-03-03
EP2661261A1 (fr)	2013-11-13
AR084801A1 (es)	2013-06-26
HRP20191842T1 (hr)	2019-12-27
US20250084034A1 (en)	2025-03-13
KR102166885B1 (ko)	2020-10-19
MX2013007909A (es)	2013-08-29
BR112013017302B1 (pt)	2021-12-07
ZA201304465B (en)	2014-02-26
CA2823616C (fr)	2019-01-29
MY161162A (en)	2017-04-14
EA026144B1 (ru)	2017-03-31
CL2013001979A1 (es)	2013-11-22
CN103458877A (zh)	2013-12-18
PT2661261T (pt)	2019-10-25
GT201300178A (es)	2014-12-30
MX371290B (es)	2020-01-24
TWI583380B (zh)	2017-05-21
JP2014501770A (ja)	2014-01-23
AU2012204835A1 (en)	2013-08-01
EP2661261B1 (fr)	2019-07-31
EA201391018A1 (ru)	2013-11-29
ES2751920T3 (es)	2020-04-02
PH12013501442B1 (en)	2018-04-20
BR112013017302A2 (pt)	2016-10-25
PH12013501442A1 (en)	2013-09-09
SG191286A1 (en)	2013-07-31
AR124662A2 (es)	2023-04-19
SI2661261T1 (sl)	2019-11-29
CN103458877B (zh)	2016-06-08
KR20140037815A (ko)	2014-03-27
WO2012093161A1 (fr)	2012-07-12
IL227094B (en)	2019-03-31
TWI610672B (zh)	2018-01-11
MX357304B (es)	2018-07-04
KR101951966B1 (ko)	2019-02-25
AU2012204835B2 (en)	2015-07-09
TW201609092A (zh)	2016-03-16
EP3590507A1 (fr)	2020-01-08
US12071402B2 (en)	2024-08-27
TW201249438A (en)	2012-12-16
EA026144B9 (ru)	2021-10-26
PE20140216A1 (es)	2014-03-01
NZ612420A (en)	2015-05-29
KR20190025727A (ko)	2019-03-11
JP2017141248A (ja)	2017-08-17
JP6324569B2 (ja)	2018-05-16
JP6111202B2 (ja)	2017-04-05
DK2661261T3 (da)	2019-10-21
US20130273161A1 (en)	2013-10-17
CA2823616A1 (fr)	2012-07-12
MA34897B1 (fr)	2014-02-01
PL2661261T3 (pl)	2020-01-31
LT2661261T (lt)	2019-10-25

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