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PL2661261T3 - Formulacje immunosupresyjne - Google Patents

Formulacje immunosupresyjne

Info

Publication number
PL2661261T3
PL2661261T3 PL12700262T PL12700262T PL2661261T3 PL 2661261 T3 PL2661261 T3 PL 2661261T3 PL 12700262 T PL12700262 T PL 12700262T PL 12700262 T PL12700262 T PL 12700262T PL 2661261 T3 PL2661261 T3 PL 2661261T3
Authority
PL
Poland
Prior art keywords
immunosuppressant
formulations
immunosuppressant formulations
Prior art date
Application number
PL12700262T
Other languages
English (en)
Inventor
Philippe BOUILLOT
Emeric Reynaud
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44022942&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2661261(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PL2661261T3 publication Critical patent/PL2661261T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Transplantation (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
PL12700262T 2011-01-07 2012-01-05 Formulacje immunosupresyjne PL2661261T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11150431 2011-01-07
PCT/EP2012/050151 WO2012093161A1 (en) 2011-01-07 2012-01-05 Immunosuppressant formulations
EP12700262.4A EP2661261B1 (en) 2011-01-07 2012-01-05 Immunosuppressant formulations

Publications (1)

Publication Number Publication Date
PL2661261T3 true PL2661261T3 (pl) 2020-01-31

Family

ID=44022942

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12700262T PL2661261T3 (pl) 2011-01-07 2012-01-05 Formulacje immunosupresyjne

Country Status (36)

Country Link
US (4) US20130273161A1 (pl)
EP (2) EP3590507A1 (pl)
JP (2) JP6111202B2 (pl)
KR (2) KR102166885B1 (pl)
CN (1) CN103458877B (pl)
AR (2) AR084801A1 (pl)
AU (1) AU2012204835B2 (pl)
BR (1) BR112013017302B1 (pl)
CA (1) CA2823616C (pl)
CL (1) CL2013001979A1 (pl)
CO (1) CO6761402A2 (pl)
CY (1) CY1122182T1 (pl)
DK (1) DK2661261T3 (pl)
EA (1) EA026144B9 (pl)
EC (1) ECSP13012812A (pl)
ES (1) ES2751920T3 (pl)
GT (1) GT201300178A (pl)
HR (1) HRP20191842T1 (pl)
HU (1) HUE045612T2 (pl)
IL (1) IL227094B (pl)
JO (1) JO3619B1 (pl)
LT (1) LT2661261T (pl)
MA (1) MA34897B1 (pl)
MX (2) MX357304B (pl)
MY (1) MY161162A (pl)
PE (1) PE20140216A1 (pl)
PH (1) PH12013501442B1 (pl)
PL (1) PL2661261T3 (pl)
PT (1) PT2661261T (pl)
SG (1) SG191286A1 (pl)
SI (1) SI2661261T1 (pl)
TN (1) TN2013000257A1 (pl)
TW (2) TWI610672B (pl)
UA (1) UA114283C2 (pl)
WO (1) WO2012093161A1 (pl)
ZA (1) ZA201304465B (pl)

Families Citing this family (14)

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PT2661261T (pt) 2011-01-07 2019-10-25 Novartis Ag Formulações imunossupressoras.
CN106456552A (zh) * 2014-04-10 2017-02-22 诺华股份有限公司 S1p调节剂的立即释放剂量方案
CN106163502B (zh) 2014-04-10 2020-12-01 诺华股份有限公司 免疫抑制剂配方
US20180042895A1 (en) 2015-02-26 2018-02-15 Novartis Ag Treatment of autoimmune disease in a patient receiving additionally a beta-blocker
ES2940306T3 (es) 2015-07-03 2023-05-05 Astellas Pharma Inc Composición farmacéutica estable para administración oral
US11434200B2 (en) 2017-03-09 2022-09-06 Novartis Ag Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof
US11629124B2 (en) 2017-03-09 2023-04-18 Novartis Ag Solid forms comprising an oxime ether compound, compositions and methods of use thereof
ES3024636T3 (en) 2017-09-27 2025-06-04 Novartis Ag Parenteral formulation comprising siponimod
CN111107845A (zh) 2017-09-29 2020-05-05 诺华股份有限公司 西尼莫德的给药方案
KR20200062240A (ko) 2017-09-29 2020-06-03 노파르티스 아게 시포니모드의 투여 요법
CN109908095A (zh) * 2019-04-08 2019-06-21 肇庆学院 一种西尼莫德片剂及制备方法
WO2021214717A1 (en) 2020-04-23 2021-10-28 Novartis Ag Dosing regimen for the use of siponimod for the treatment of acute respiratory distress syndrome
IL315531A (en) * 2022-03-09 2024-11-01 Isp Investments Llc The composition of an inactive substance for drugs, produced by joint processing of its components
EP4633611A1 (en) 2022-12-12 2025-10-22 Synthon B.V. Pharmaceutical composition of siponimod

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MY150088A (en) 2003-05-19 2013-11-29 Irm Llc Immunosuppressant compounds and compositions
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CA2539033C (en) 2003-09-12 2013-03-05 Neuronova Ab Treatment of disease or injury of the nervous system with fty720
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CN102256942B (zh) * 2008-12-18 2013-07-24 诺瓦提斯公司 1-(4-{1-[(e)-4-环己基-3-三氟甲基-苄氧基亚氨基]-乙基}-2-乙基-苄基)-氮杂环丁烷-3-甲酸的多晶型物
US8486930B2 (en) 2008-12-18 2013-07-16 Novartis Ag Salts
HRP20131106T1 (hr) * 2008-12-18 2013-12-20 Novartis Ag Hemifumaratna sol od 1-[4-[1-(4-cikloheksil-3-trifluorometil-benziloksiimino)-etil]-2-etil-benzil]-azetidin-3-karboksilne kiseline
WO2010070083A1 (en) 2008-12-19 2010-06-24 Novartis Ag Mouthpiece for an inhaler
SI4098256T1 (sl) 2008-12-22 2025-06-30 Novartis Ag Režim odmerjanja za agonist receptorja s1p
PL2379069T3 (pl) 2008-12-22 2015-08-31 Novartis Ag Schemat dawkowania agonisty receptora S1P
EP3831371A1 (en) 2009-09-29 2021-06-09 Novartis AG Dosage regimen of an s1p receptor modulator
PT2661261T (pt) 2011-01-07 2019-10-25 Novartis Ag Formulações imunossupressoras.
WO2012095853A1 (en) 2011-01-10 2012-07-19 Novartis Pharma Ag Modified release formulations comprising sip receptor modulators
TW201320994A (zh) 2011-10-11 2013-06-01 Novartis Ag 投藥療程
EP4556908A3 (en) 2013-04-04 2025-07-30 Novartis AG Identifying patient response to s1p receptor modulator administration
CN106163502B (zh) 2014-04-10 2020-12-01 诺华股份有限公司 免疫抑制剂配方

Also Published As

Publication number Publication date
US20220064110A1 (en) 2022-03-03
EA201391018A1 (ru) 2013-11-29
TWI583380B (zh) 2017-05-21
ES2751920T3 (es) 2020-04-02
KR20140037815A (ko) 2014-03-27
MX371290B (es) 2020-01-24
AR084801A1 (es) 2013-06-26
KR102166885B1 (ko) 2020-10-19
GT201300178A (es) 2014-12-30
LT2661261T (lt) 2019-10-25
CN103458877A (zh) 2013-12-18
DK2661261T3 (da) 2019-10-21
CA2823616A1 (en) 2012-07-12
JP2017141248A (ja) 2017-08-17
ECSP13012812A (es) 2013-09-30
US20200199069A1 (en) 2020-06-25
PE20140216A1 (es) 2014-03-01
CO6761402A2 (es) 2013-09-30
KR20190025727A (ko) 2019-03-11
US12071402B2 (en) 2024-08-27
CA2823616C (en) 2019-01-29
US20130273161A1 (en) 2013-10-17
MY161162A (en) 2017-04-14
JP2014501770A (ja) 2014-01-23
EA026144B1 (ru) 2017-03-31
PH12013501442B1 (en) 2018-04-20
US20250084034A1 (en) 2025-03-13
EP3590507A1 (en) 2020-01-08
AR124662A2 (es) 2023-04-19
TW201249438A (en) 2012-12-16
PT2661261T (pt) 2019-10-25
CN103458877B (zh) 2016-06-08
BR112013017302B1 (pt) 2021-12-07
AU2012204835B2 (en) 2015-07-09
AU2012204835A1 (en) 2013-08-01
MA34897B1 (fr) 2014-02-01
CL2013001979A1 (es) 2013-11-22
TWI610672B (zh) 2018-01-11
UA114283C2 (uk) 2017-05-25
NZ612420A (en) 2015-05-29
JP6111202B2 (ja) 2017-04-05
ZA201304465B (en) 2014-02-26
HUE045612T2 (hu) 2020-01-28
TW201609092A (zh) 2016-03-16
KR101951966B1 (ko) 2019-02-25
PH12013501442A1 (en) 2013-09-09
MX2013007909A (es) 2013-08-29
JO3619B1 (ar) 2020-08-27
SG191286A1 (en) 2013-07-31
BR112013017302A2 (pt) 2016-10-25
CY1122182T1 (el) 2020-11-25
MX357304B (es) 2018-07-04
WO2012093161A1 (en) 2012-07-12
EA026144B9 (ru) 2021-10-26
IL227094B (en) 2019-03-31
TN2013000257A1 (en) 2014-11-10
EP2661261A1 (en) 2013-11-13
HRP20191842T1 (hr) 2019-12-27
EP2661261B1 (en) 2019-07-31
SI2661261T1 (sl) 2019-11-29
JP6324569B2 (ja) 2018-05-16

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