SMT201600141B - Boronati quali inibitori di arginasi - Google Patents

Boronati quali inibitori di arginasi

Info

Publication number: SMT201600141B
Authority: SM; San Marino
Prior art keywords: boronati; arginasi; inhibitors; arginasi inhibitors
Prior art date: 2010-10-26

Application number

SM201600141T

Other languages

English (en)

Inventor

Zandt Michael Van

Gunnar Erik Jagdmann Jr

Original Assignee

Mars Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2010-10-26

Filing date

2016-05-19

Publication date

2016-07-01

2016-05-19 Application filed by Mars Inc filed Critical Mars Inc

2016-07-01 Publication of SMT201600141B publication Critical patent/SMT201600141B/it

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Pulmonology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Epidemiology (AREA)
Urology & Nephrology (AREA)
Hematology (AREA)
Dermatology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Diabetes (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Gynecology & Obstetrics (AREA)
Vascular Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

SM201600141T 2010-10-26 2016-05-19 Boronati quali inibitori di arginasi SMT201600141B (it)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US40676010P	2010-10-26	2010-10-26
PCT/US2011/056844 WO2012058065A1 (en)	2010-10-26	2011-10-19	Boronates as arginase inhibitors

Publications (1)

Publication Number	Publication Date
SMT201600141B true SMT201600141B (it)	2016-07-01

Family

ID=44913403

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SM201600141T SMT201600141B (it)	2010-10-26	2016-05-19	Boronati quali inibitori di arginasi

Country Status (19)

Country	Link
US (5)	US9233985B2 (it)
EP (3)	EP3034509B1 (it)
JP (1)	JP5909239B2 (it)
CN (2)	CN103249737B (it)
AU (1)	AU2011320732B2 (it)
BR (1)	BR112013010099B1 (it)
CA (1)	CA2815536C (it)
DK (1)	DK2632927T3 (it)
ES (2)	ES2568680T3 (it)
HK (1)	HK1223104A1 (it)
HR (1)	HRP20160305T1 (it)
HU (1)	HUE027317T2 (it)
IL (1)	IL225926A (it)
MX (1)	MX336381B (it)
PL (1)	PL2632927T3 (it)
RS (1)	RS54750B1 (it)
SI (1)	SI2632927T1 (it)
SM (1)	SMT201600141B (it)
WO (1)	WO2012058065A1 (it)

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US12215116B2 (en) *	2018-03-13	2025-02-04	Merck Sharp & Dohme Llc	Arginase inhibitors and methods of use
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2011
- 2011-10-19 DK DK11779904.9T patent/DK2632927T3/en active
- 2011-10-19 HU HUE11779904A patent/HUE027317T2/en unknown
- 2011-10-19 MX MX2013004491A patent/MX336381B/es unknown
- 2011-10-19 EP EP16150285.1A patent/EP3034509B1/en active Active
- 2011-10-19 RS RS20160243A patent/RS54750B1/sr unknown
- 2011-10-19 JP JP2013536669A patent/JP5909239B2/ja active Active
- 2011-10-19 EP EP20162218.0A patent/EP3719024A1/en active Pending
- 2011-10-19 BR BR112013010099-0A patent/BR112013010099B1/pt not_active IP Right Cessation
- 2011-10-19 WO PCT/US2011/056844 patent/WO2012058065A1/en not_active Ceased
- 2011-10-19 EP EP11779904.9A patent/EP2632927B1/en active Active
- 2011-10-19 CN CN201180057717.4A patent/CN103249737B/zh not_active Expired - Fee Related
- 2011-10-19 AU AU2011320732A patent/AU2011320732B2/en not_active Ceased
- 2011-10-19 SI SI201130766A patent/SI2632927T1/sl unknown
- 2011-10-19 ES ES11779904.9T patent/ES2568680T3/es active Active
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- 2011-10-19 PL PL11779904.9T patent/PL2632927T3/pl unknown
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- 2011-10-19 HR HRP20160305TT patent/HRP20160305T1/hr unknown
2013
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2015
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2016
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- 2016-09-23 HK HK16111212.1A patent/HK1223104A1/en unknown
2018
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Also Published As

Publication number	Publication date
AU2011320732A1 (en)	2013-11-21
CN103249737B (zh)	2016-06-08
CN106008569B9 (zh)	2020-05-22
DK2632927T3 (en)	2016-04-11
JP2013542223A (ja)	2013-11-21
EP2632927B1 (en)	2016-02-10
AU2011320732B2 (en)	2018-07-05
EP3719024A1 (en)	2020-10-07
US10603330B2 (en)	2020-03-31
BR112013010099A2 (pt)	2016-09-06
EP3034509A1 (en)	2016-06-22
PL2632927T3 (pl)	2016-09-30
US20200246362A1 (en)	2020-08-06
US20120129806A1 (en)	2012-05-24
MX2013004491A (es)	2013-11-04
EP2632927A1 (en)	2013-09-04
JP5909239B2 (ja)	2016-04-26
HK1225390A1 (zh)	2017-09-08
CA2815536C (en)	2019-10-01
EP3034509B1 (en)	2020-04-22
HUE027317T2 (en)	2016-10-28
IL225926A (en)	2016-09-29
BR112013010099B1 (pt)	2021-08-10
MX336381B (es)	2016-01-18
CN106008569B (zh)	2020-04-03
HK1223104A1 (en)	2017-07-21
HRP20160305T1 (hr)	2016-07-01
CN103249737A (zh)	2013-08-14
CN106008569A (zh)	2016-10-12
US20150191492A1 (en)	2015-07-09
US10098902B2 (en)	2018-10-16
US20170000808A1 (en)	2017-01-05
ES2794006T3 (es)	2020-11-17
US11389464B2 (en)	2022-07-19
US9440995B2 (en)	2016-09-13
US9233985B2 (en)	2016-01-12
SI2632927T1 (sl)	2016-08-31
WO2012058065A1 (en)	2012-05-03
RS54750B1 (sr)	2016-10-31
IL225926A0 (en)	2013-06-27
ES2568680T3 (es)	2016-05-03
CA2815536A1 (en)	2012-05-03
US20190054101A1 (en)	2019-02-21

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SMT201600141B (it)	2016-07-01	Boronati quali inibitori di arginasi
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HRP20181786T1 (hr)	2019-02-08	Inhibitori aktivacije t-stanica
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EP2629616A4 (en)	2014-03-26	SUBSTITUTED AMINO-TRIAZOLYL-PDE10-HEMMER
BR112013014148A2 (pt)	2016-09-27	inibidores de corrosão
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