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SK9502003A3 - Combinations of sterol absorption inhibitor(s) with blood modifier(s) for treating vascular conditions - Google Patents

Combinations of sterol absorption inhibitor(s) with blood modifier(s) for treating vascular conditions Download PDF

Info

Publication number
SK9502003A3
SK9502003A3 SK950-2003A SK9502003A SK9502003A3 SK 9502003 A3 SK9502003 A3 SK 9502003A3 SK 9502003 A SK9502003 A SK 9502003A SK 9502003 A3 SK9502003 A3 SK 9502003A3
Authority
SK
Slovakia
Prior art keywords
alkyl
group
aryl
substituted
independently selected
Prior art date
Application number
SK950-2003A
Other languages
English (en)
Slovak (sk)
Inventor
Teddy Kosoglou
Rudyard Joseph Ress
John Strony
Enrico P Veltri
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of SK9502003A3 publication Critical patent/SK9502003A3/sk

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
SK950-2003A 2001-01-26 2002-01-25 Combinations of sterol absorption inhibitor(s) with blood modifier(s) for treating vascular conditions SK9502003A3 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US26439601P 2001-01-26 2001-01-26
US26460001P 2001-01-26 2001-01-26
US26427501P 2001-01-26 2001-01-26
US32412301P 2001-09-21 2001-09-21
PCT/US2002/002013 WO2002058734A2 (en) 2001-01-26 2002-01-25 Combinations of sterol absorption inhibitor(s) with blood modifier(s) for treating vascular conditions

Publications (1)

Publication Number Publication Date
SK9502003A3 true SK9502003A3 (en) 2003-12-02

Family

ID=27500818

Family Applications (1)

Application Number Title Priority Date Filing Date
SK950-2003A SK9502003A3 (en) 2001-01-26 2002-01-25 Combinations of sterol absorption inhibitor(s) with blood modifier(s) for treating vascular conditions

Country Status (26)

Country Link
US (1) US20020147184A1 (de)
EP (2) EP1810693A3 (de)
JP (1) JP2004517920A (de)
KR (2) KR20040025890A (de)
CN (1) CN1658903A (de)
AR (1) AR032403A1 (de)
AT (1) ATE381347T1 (de)
AU (1) AU2002237927B2 (de)
BR (1) BR0206639A (de)
CA (1) CA2434504A1 (de)
CY (1) CY1107174T1 (de)
CZ (1) CZ20032039A3 (de)
DE (1) DE60224163T2 (de)
DK (1) DK1353694T3 (de)
ES (1) ES2296894T3 (de)
HU (1) HUP0303917A2 (de)
IL (1) IL156488A0 (de)
MX (1) MXPA03006728A (de)
NO (1) NO20033357L (de)
NZ (1) NZ542090A (de)
PL (1) PL364178A1 (de)
PT (1) PT1353694E (de)
RU (1) RU2314126C2 (de)
SI (1) SI1353694T1 (de)
SK (1) SK9502003A3 (de)
WO (1) WO2002058734A2 (de)

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US7053080B2 (en) 2001-09-21 2006-05-30 Schering Corporation Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors
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WO2002058734A3 (en) 2003-07-03
PT1353694E (pt) 2008-03-12
EP1810693A2 (de) 2007-07-25
NO20033357L (no) 2003-09-25
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CA2434504A1 (en) 2002-08-01
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RU2314126C2 (ru) 2008-01-10
AR032403A1 (es) 2003-11-05
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EP1353694B1 (de) 2007-12-19
EP1353694A2 (de) 2003-10-22
CY1107174T1 (el) 2012-10-24
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WO2002058734A2 (en) 2002-08-01
BR0206639A (pt) 2004-02-25
EP1810693A3 (de) 2007-10-17
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ATE381347T1 (de) 2008-01-15
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