SI1885339T1 - Formulacije inhibitorja src/abl - Google Patents

Formulacije inhibitorja src/abl

Info

Publication number: SI1885339T1
Authority: SI; Slovenia
Prior art keywords: src; formulations; abl inhibitor; abl; inhibitor
Prior art date: 2005-05-05

Application number

SI200631971T

Other languages

English (en)

Inventor

Julia Zh Gao

Rajeshwar Motheram

Original Assignee

Bristol-Myers Squibb Holdings Ireland

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-05-05

Filing date

2006-05-04

Publication date

2015-10-30

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37076246&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1885339(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-05-04 Application filed by Bristol-Myers Squibb Holdings Ireland filed Critical Bristol-Myers Squibb Holdings Ireland

2015-10-30 Publication of SI1885339T1 publication Critical patent/SI1885339T1/sl

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Chemistry (AREA)
Immunology (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Inorganic Chemistry (AREA)
Hematology (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Plural Heterocyclic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

SI200631971T 2005-05-05 2006-05-04 Formulacije inhibitorja src/abl SI1885339T1 (sl)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US67803005P	2005-05-05	2005-05-05
PCT/US2006/017073 WO2006121742A2 (en)	2005-05-05	2006-05-04	Formulations of a src/abl inhibitor
EP06769997.5A EP1885339B1 (en)	2005-05-05	2006-05-04	Formulations of a src/abl inhibitor

Publications (1)

Publication Number	Publication Date
SI1885339T1 true SI1885339T1 (sl)	2015-10-30

Family

ID=37076246

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SI200631971T SI1885339T1 (sl)	2005-05-05	2006-05-04	Formulacije inhibitorja src/abl

Country Status (18)

Country	Link
US (2)	US20060251723A1 (sl)
EP (1)	EP1885339B1 (sl)
JP (1)	JP5173794B2 (sl)
CN (2)	CN102813655A (sl)
AR (1)	AR054445A1 (sl)
DK (1)	DK1885339T3 (sl)
ES (1)	ES2546847T3 (sl)
GE (1)	GEP20104927B (sl)
HR (1)	HRP20151051T1 (sl)
HU (1)	HUE026040T2 (sl)
NO (1)	NO343939B1 (sl)
PE (1)	PE20061373A1 (sl)
PL (1)	PL1885339T3 (sl)
PT (1)	PT1885339E (sl)
RS (1)	RS54258B1 (sl)
SI (1)	SI1885339T1 (sl)
TW (1)	TWI386205B (sl)
WO (1)	WO2006121742A2 (sl)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN1348370A (zh)	1999-04-15	2002-05-08	布里斯托尔-迈尔斯斯奎布公司	环状蛋白酪氨酸激酶抑制剂
SI1885339T1 (sl)	2005-05-05	2015-10-30	Bristol-Myers Squibb Holdings Ireland	Formulacije inhibitorja src/abl
CA2610157A1 (en) *	2005-06-09	2006-12-21	Bristol-Myers Squibb Company	Methods of identifying and treating individuals exhibiting mutant kit protein
WO2007035874A1 (en) *	2005-09-21	2007-03-29	Bristol-Myers Squibb Company	Oral administration of n-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-1,3-thiazole-5-carboxamide and salts thereof
US20090306094A1 (en) *	2006-03-17	2009-12-10	Bristol-Myers Squibb Company	Methods Of Identifying And Treating Individuals Exhibiting Mutant Bcr/Abl Kinase Polypeptides
US20090318560A1 (en) *	2007-02-26	2009-12-24	Wayne Parent	Formulations for cathepsin k inhibitors
EP2359813A1 (en)	2010-02-04	2011-08-24	Ratiopharm GmbH	Pharmaceutical composition comprising N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-5-thiazolecarboxamid
JP5589097B2 (ja) *	2010-02-08	2014-09-10	南京▲か▼文迪許生物工程技術有限公司	ダサチニブ多結晶体、並びにその調製方法及び薬物組成物
CN101891738B (zh)	2010-02-08	2011-09-28	南京卡文迪许生物工程技术有限公司	达沙替尼多晶型物及其制备方法和药用组合物
CN104274420B (zh) *	2013-07-11	2019-03-05	石药集团中奇制药技术（石家庄）有限公司	一种达沙替尼组合物及其制备方法
IN2013MU03610A (sl)	2013-12-18	2015-04-24	Dharmesh Mahendrabhai Shah
WO2017144109A1 (en)	2016-02-25	2017-08-31	Remedica Ltd	Dasatinib formulation
JP7166754B2 (ja)	2017-11-22	2022-11-08	沢井製薬株式会社	ダサチニブ無水物含有製剤
JP7249397B2 (ja) *	2017-12-27	2023-03-30	日本化薬株式会社	ダサチニブを有効成分とする医薬組成物
JP7000148B2 (ja) *	2017-12-27	2022-01-19	日本化薬株式会社	ダサチニブを有効成分とする医薬組成物
WO2020018053A2 (en) *	2018-05-25	2020-01-23	Arven Ilac Sanayi Ve Ticaret Anonim Sirketi	The tablet comprising dasatinib
CN113292537B (zh)	2018-06-15	2024-04-05	汉达癌症医药责任有限公司	激酶抑制剂的盐类及其组合物
GB2592680A (en)	2020-03-06	2021-09-08	Zentiva Ks	Pharmaceutical compositions comprising dasatinib anhydrous and uses thereof
EP4071248A1 (en)	2021-04-07	2022-10-12	Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts	Means and methods for enhancing receptor-targeted gene transfer

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3539380A (en)	1968-01-08	1970-11-10	Upjohn Co	Methylcellulose and polyalkylene glycol coating of solid medicinal dosage forms
US4543370A (en)	1979-11-29	1985-09-24	Colorcon, Inc.	Dry edible film coating composition, method and coating form
US5681382A (en)	1995-08-22	1997-10-28	Shin-Etsu Chemical Co., Ltd.	Rapidly soluble coating composition and method for preparing same
AR016827A1 (es) *	1997-08-22	2001-08-01	Smithkline Beecham Corp	PROCEDIMIENTO PARA LA PREPARACIoN DE UNA TABLETA FARMACÉUTICA
US7125875B2 (en) *	1999-04-15	2006-10-24	Bristol-Myers Squibb Company	Cyclic protein tyrosine kinase inhibitors
CN1348370A (zh)	1999-04-15	2002-05-08	布里斯托尔-迈尔斯斯奎布公司	环状蛋白酪氨酸激酶抑制剂
CN1679556A (zh) *	1999-12-08	2005-10-12	法马西亚公司	维得克西组合物
GB0209257D0 (en) *	2002-04-23	2002-06-05	Novartis Ag	Organic compounds
US20050215795A1 (en)	2004-02-06	2005-09-29	Bang-Chi Chen	Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
US7491725B2 (en)	2004-02-06	2009-02-17	Bristol-Myers Squibb Company	Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
TWI338004B (en)	2004-02-06	2011-03-01	Bristol Myers Squibb Co	Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
SI1885339T1 (sl)	2005-05-05	2015-10-30	Bristol-Myers Squibb Holdings Ireland	Formulacije inhibitorja src/abl

2006
- 2006-05-04 SI SI200631971T patent/SI1885339T1/sl unknown
- 2006-05-04 PT PT67699975T patent/PT1885339E/pt unknown
- 2006-05-04 ES ES06769997.5T patent/ES2546847T3/es active Active
- 2006-05-04 CN CN2012103135834A patent/CN102813655A/zh active Pending
- 2006-05-04 DK DK06769997.5T patent/DK1885339T3/en active
- 2006-05-04 WO PCT/US2006/017073 patent/WO2006121742A2/en not_active Ceased
- 2006-05-04 PL PL06769997T patent/PL1885339T3/pl unknown
- 2006-05-04 GE GEAP200610410A patent/GEP20104927B/en unknown
- 2006-05-04 HU HUE06769997A patent/HUE026040T2/en unknown
- 2006-05-04 RS RS20150635A patent/RS54258B1/sr unknown
- 2006-05-04 JP JP2008510188A patent/JP5173794B2/ja active Active
- 2006-05-04 AR ARP060101816A patent/AR054445A1/es not_active Application Discontinuation
- 2006-05-04 CN CNA2006800150680A patent/CN101170996A/zh active Pending
- 2006-05-04 EP EP06769997.5A patent/EP1885339B1/en not_active Revoked
- 2006-05-04 US US11/418,338 patent/US20060251723A1/en not_active Abandoned
- 2006-05-04 HR HRP20151051TT patent/HRP20151051T1/hr unknown
- 2006-05-05 PE PE2006000477A patent/PE20061373A1/es not_active Application Discontinuation
- 2006-05-05 TW TW095116078A patent/TWI386205B/zh active
2007
- 2007-10-10 NO NO20075154A patent/NO343939B1/no unknown
2013
- 2013-01-07 US US13/735,081 patent/US20130122093A1/en not_active Abandoned

Also Published As

Publication number	Publication date
JP2008540440A (ja)	2008-11-20
PL1885339T3 (pl)	2015-12-31
HUE026040T2 (en)	2016-05-30
PE20061373A1 (es)	2006-12-15
US20130122093A1 (en)	2013-05-16
NO20075154L (no)	2008-02-01
TW200716117A (en)	2007-05-01
ES2546847T3 (es)	2015-09-29
WO2006121742A2 (en)	2006-11-16
EP1885339A2 (en)	2008-02-13
TWI386205B (zh)	2013-02-21
EP1885339B1 (en)	2015-07-29
CN101170996A (zh)	2008-04-30
NO343939B1 (no)	2019-07-15
HRP20151051T1 (hr)	2015-11-06
PT1885339E (pt)	2015-10-12
US20060251723A1 (en)	2006-11-09
JP5173794B2 (ja)	2013-04-03
GEP20104927B (en)	2010-03-25
WO2006121742A3 (en)	2007-02-22
AR054445A1 (es)	2007-06-27
DK1885339T3 (en)	2015-10-19
RS54258B1 (sr)	2016-02-29
CN102813655A (zh)	2012-12-12

Publication	Publication Date	Title
ZA200802585B (en)	2009-02-25	Pyridopyrimidinone inhibitors of Pl3Kα
IL190292A0 (en)	2009-09-22	PYRIDOPYRIMIDINONE INHIBITORS OF P13Ka
PT1885339E (pt)	2015-10-12	Formulações de um inibidor src/abl
IL184303A0 (en)	2007-10-31	Amino-pyridines as inhibitors of ??-secretase
IL212841A0 (en)	2011-07-31	Dpp iv inhibitor formulations
PL2079727T3 (pl)	2016-08-31	Inhibitory kinazy
SI2402317T1 (sl)	2013-10-30	DGAT inhibitor
IL185185A0 (en)	2007-12-03	Azolylacylguanidines as ??-secretase inhibitors
PT2094708E (pt)	2014-01-07	Pirrolopirazina como inibidor da cinase syk
ZA200702394B (en)	2008-11-26	Indozolone derivatives as 11b-HSD1 inhibitors
ZA200700181B (en)	2009-03-25	Aryl-pyridine derivatives as 11-beta-HSD1 inhibitors
IL184569A0 (en)	2007-10-31	Intravenous formulations of pde-5 inhibitors
ZA200707070B (en)	2008-09-25	Analgesic compositions
EP2036894A4 (en)	2011-01-12	AURORA INHIBITOR
GB0504995D0 (en)	2005-04-20	Use of a compound
EP1941873A4 (en)	2012-09-26	METALLO-BETA-Lactamase INHIBITORS
EP2098544A4 (en)	2013-10-16	POLYMERIZABLE COMPOUNDS AND POLYMERIZABLE COMPOSITIONS
EP2036893A4 (en)	2011-04-13	ABL Kinase Inhibitor
AP2007004282A0 (en)	2007-12-31	Derivatives of A 1-phenyltriazole as antiparasiticagents
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GB0516967D0 (en)	2005-09-28	Inhibitors
GB0512626D0 (en)	2005-07-27	Inhibitor compounds
GB0517677D0 (en)	2005-10-05	Inhibitor compounds II
GB0522829D0 (en)	2005-12-21	Use of a compound
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