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SI1753748T1 - Derivati prolina in njihova uporaba kot inhibitorji dipeptidil-peptidaze IV - Google Patents

Derivati prolina in njihova uporaba kot inhibitorji dipeptidil-peptidaze IV

Info

Publication number
SI1753748T1
SI1753748T1 SI200530767T SI200530767T SI1753748T1 SI 1753748 T1 SI1753748 T1 SI 1753748T1 SI 200530767 T SI200530767 T SI 200530767T SI 200530767 T SI200530767 T SI 200530767T SI 1753748 T1 SI1753748 T1 SI 1753748T1
Authority
SI
Slovenia
Prior art keywords
inhibitors
dipeptidyl peptidase
proline derivatives
proline
derivatives
Prior art date
Application number
SI200530767T
Other languages
English (en)
Inventor
Bernard Hulin
David Walter Piotrowski
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34966115&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1753748(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SI1753748T1 publication Critical patent/SI1753748T1/sl

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/14—Nitrogen atoms not forming part of a nitro radical
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

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SI200530767T 2004-05-12 2005-04-29 Derivati prolina in njihova uporaba kot inhibitorji dipeptidil-peptidaze IV SI1753748T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US57030004P 2004-05-12 2004-05-12
US66430505P 2005-03-21 2005-03-21
EP05733750A EP1753748B1 (en) 2004-05-12 2005-04-29 Proline derivatives and their use as dipeptidyl peptidase iv inhibitors

Publications (1)

Publication Number Publication Date
SI1753748T1 true SI1753748T1 (sl) 2009-12-31

Family

ID=34966115

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200530767T SI1753748T1 (sl) 2004-05-12 2005-04-29 Derivati prolina in njihova uporaba kot inhibitorji dipeptidil-peptidaze IV

Country Status (36)

Country Link
US (4) US7291618B2 (sl)
EP (2) EP2116541B1 (sl)
JP (1) JP4227660B2 (sl)
KR (1) KR100869616B1 (sl)
AP (1) AP2320A (sl)
AR (1) AR049894A1 (sl)
AT (1) ATE437870T1 (sl)
AU (1) AU2005247684B2 (sl)
BR (1) BRPI0510284A (sl)
CA (1) CA2566108C (sl)
CR (1) CR8744A (sl)
CY (1) CY1109322T1 (sl)
DE (1) DE602005015699D1 (sl)
DK (1) DK1753748T3 (sl)
EA (1) EA011086B9 (sl)
EC (1) ECSP066985A (sl)
ES (1) ES2327857T3 (sl)
GE (1) GEP20084421B (sl)
HR (1) HRP20090471T1 (sl)
IL (1) IL178339A (sl)
MA (1) MA28578B1 (sl)
MX (1) MXPA06013114A (sl)
MY (1) MY139805A (sl)
NL (1) NL1029015C2 (sl)
NO (1) NO20064400L (sl)
NZ (1) NZ550229A (sl)
PA (1) PA8632701A1 (sl)
PE (1) PE20060316A1 (sl)
PL (1) PL1753748T3 (sl)
PT (1) PT1753748E (sl)
RS (1) RS51106B (sl)
SI (1) SI1753748T1 (sl)
SV (1) SV2006002110A (sl)
TW (1) TWI347322B (sl)
UY (1) UY28892A1 (sl)
WO (1) WO2005116014A1 (sl)

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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
PT1753748E (pt) 2004-05-12 2009-08-28 Pfizer Prod Inc Derivados de prolina e a sua utilização como inibidores de dipeptidil peptidase iv
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
WO2006071958A1 (en) 2004-12-29 2006-07-06 Millennium Pharmaceuticals, Inc. Compounds useful as chemokine receptor antagonists
US7880002B2 (en) 2004-12-29 2011-02-01 Millennium Pharmaceuticals, Inc. Substituted piperazinyl-pyrrolidine compounds useful as chemokine receptor antagonists
WO2006073167A1 (ja) * 2005-01-07 2006-07-13 Ono Pharmaceutical Co., Ltd. ピロリジン誘導体
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
PE20071221A1 (es) 2006-04-11 2007-12-14 Arena Pharm Inc Agonistas del receptor gpr119 en metodos para aumentar la masa osea y para tratar la osteoporosis y otras afecciones caracterizadas por masa osea baja, y la terapia combinada relacionada a estos agonistas
AU2007235876A1 (en) 2006-04-12 2007-10-18 Probiodrug Ag Enzyme inhibitors
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
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AP2320A (en) 2011-11-07
EA200601896A1 (ru) 2007-02-27
US20070161664A1 (en) 2007-07-12
US20070099897A1 (en) 2007-05-03
JP4227660B2 (ja) 2009-02-18
CA2566108C (en) 2010-04-06
EP1753748B1 (en) 2009-07-29
EA011086B1 (ru) 2008-12-30
UY28892A1 (es) 2005-12-30
SV2006002110A (es) 2006-05-25
AP2006003770A0 (en) 2006-10-31
NL1029015C2 (nl) 2006-05-16
EP2116541B1 (en) 2015-02-25
MXPA06013114A (es) 2007-02-28
NO20064400L (no) 2006-10-25
AR049894A1 (es) 2006-09-13
NL1029015A1 (nl) 2005-11-15
PE20060316A1 (es) 2006-05-08
US20050256310A1 (en) 2005-11-17
EP2116541A1 (en) 2009-11-11
KR100869616B1 (ko) 2008-11-21
RS51106B (sr) 2010-10-31
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ECSP066985A (es) 2006-12-29
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PL1753748T3 (pl) 2010-01-29
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US20060079498A1 (en) 2006-04-13
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ATE437870T1 (de) 2009-08-15
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MA28578B1 (fr) 2007-05-02
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US7465732B2 (en) 2008-12-16
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ES2327857T3 (es) 2009-11-04
IL178339A0 (en) 2007-02-11
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MY139805A (en) 2009-10-30
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AU2005247684B2 (en) 2008-10-23
DE602005015699D1 (de) 2009-09-10
AU2005247684A1 (en) 2005-12-08
PT1753748E (pt) 2009-08-28
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JP2007537231A (ja) 2007-12-20
PA8632701A1 (es) 2006-06-02

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