SG166799A1 - Quinoline derivatives as antibacterial agents - Google Patents

Quinoline derivatives as antibacterial agents

Info

Publication number: SG166799A1
Authority: SG; Singapore
Prior art keywords: antibacterial agents; compound; quinoline derivatives; bacterial infection; compounds
Prior art date: 2005-06-28

Application number

SG201007977-0A

Other languages

English (en)

Inventor

Koenraad Jozef Lodewijk Marcel Andries

Anil Koul

Jerome Emile Georges Guillemont

Magali Madeline Simone Motte

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-06-28

Filing date

2006-06-26

Publication date

2010-12-29

2006-06-26 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2010-12-29 Publication of SG166799A1 publication Critical patent/SG166799A1/en

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
- C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/36—Sulfur atoms

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Epidemiology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Quinoline Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

SG201007977-0A 2005-06-28 2006-06-26 Quinoline derivatives as antibacterial agents SG166799A1 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP05105769		2005-06-28

Publications (1)

Publication Number	Publication Date
SG166799A1 true SG166799A1 (en)	2010-12-29

Family

ID=35445742

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SG201007977-0A SG166799A1 (en)	2005-06-28	2006-06-26	Quinoline derivatives as antibacterial agents

Country Status (33)

Country	Link
US (2)	US20100204270A1 (fr)
EP (1)	EP1898910B1 (fr)
JP (1)	JP5193859B2 (fr)
KR (1)	KR101423229B1 (fr)
CN (1)	CN101252928B (fr)
AP (1)	AP2733A (fr)
AR (1)	AR057654A1 (fr)
AU (1)	AU2006263884B2 (fr)
BR (1)	BRPI0612534B8 (fr)
CA (1)	CA2612623C (fr)
CY (1)	CY1118515T1 (fr)
DK (1)	DK1898910T3 (fr)
EA (1)	EA014163B1 (fr)
ES (1)	ES2606772T3 (fr)
HR (1)	HRP20161704T1 (fr)
HU (1)	HUE031268T2 (fr)
IL (1)	IL188394A (fr)
JO (1)	JO3270B1 (fr)
LT (1)	LT1898910T (fr)
ME (1)	ME02690B (fr)
MX (1)	MX2008000082A (fr)
MY (1)	MY151030A (fr)
NO (1)	NO341283B1 (fr)
NZ (1)	NZ564339A (fr)
PL (1)	PL1898910T3 (fr)
PT (1)	PT1898910T (fr)
RS (1)	RS55408B1 (fr)
SG (1)	SG166799A1 (fr)
SI (1)	SI1898910T1 (fr)
TW (1)	TWI392494B (fr)
UA (1)	UA91549C2 (fr)
WO (1)	WO2007000436A1 (fr)
ZA (1)	ZA200711149B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US9790186B2 (en)	2009-07-21	2017-10-17	Trustees Of Dartmouth College	Composition and method for prevention, mitigation or treatment of an enteropathogenic bacterial infection
JP6153603B2 (ja)	2012-04-27	2017-06-28	ヤンセンファーマシューティカエヌ．ベー．	抗菌性キノリン誘導体
EP2841425B1 (fr)	2012-04-27	2016-03-23	Janssen Pharmaceutica, N.V.	Dérivés de quinoléine antibactériens
CN105037497B (zh) *	2015-03-27	2018-06-26	中牧实业股份有限公司	一种恩拉霉素的提纯方法
WO2017035288A1 (fr) *	2015-08-27	2017-03-02	Trustees Of Dartmouth College	Composition et procédé destinés à prévenir, limiter ou traiter une infection à bactéries entéropathogènes

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6103905A (en) *	1997-06-19	2000-08-15	Sepracor, Inc.	Quinoline-indole antimicrobial agents, uses and compositions related thereto
DE19937116A1 (de) *	1999-08-06	2001-02-08	Bayer Ag	Moxifloxacin Kochsalzformulierung
BRPI0312927B8 (pt) *	2002-07-25	2021-05-25	Janssen Pharmaceutica Nv	"compostos, derivados de quinolina, composição, seu uso como inibidores micobacteriais, bem como processo para preparação dos referidos derivados".
ATE390925T1 (de) *	2004-05-28	2008-04-15	Janssen Pharmaceutica Nv	Verwendung von substituierten chinolin-derivaten zur behandlung von arzneimittelresistenten mycobakteriellen erkrankungen
EE05394B1 (et) *	2004-12-24	2011-04-15	Janssen Pharmaceutica N.V.	Kinoliinihendid kasutamiseks latentse tuberkuloosi ravis

2006
- 2006-06-25 JO JOP/2006/0189A patent/JO3270B1/ar active
- 2006-06-26 RS RS20161121A patent/RS55408B1/sr unknown
- 2006-06-26 NZ NZ564339A patent/NZ564339A/en not_active IP Right Cessation
- 2006-06-26 MX MX2008000082A patent/MX2008000082A/es active IP Right Grant
- 2006-06-26 EP EP06763891.6A patent/EP1898910B1/fr active Active
- 2006-06-26 ME MEP-2016-291A patent/ME02690B/fr unknown
- 2006-06-26 SI SI200632126A patent/SI1898910T1/sl unknown
- 2006-06-26 BR BRPI0612534A patent/BRPI0612534B8/pt not_active IP Right Cessation
- 2006-06-26 SG SG201007977-0A patent/SG166799A1/en unknown
- 2006-06-26 PT PT67638916T patent/PT1898910T/pt unknown
- 2006-06-26 WO PCT/EP2006/063556 patent/WO2007000436A1/fr not_active Ceased
- 2006-06-26 JP JP2008518812A patent/JP5193859B2/ja not_active Expired - Fee Related
- 2006-06-26 UA UAA200714716A patent/UA91549C2/ru unknown
- 2006-06-26 AP AP2008004300A patent/AP2733A/xx active
- 2006-06-26 LT LTEP06763891.6T patent/LT1898910T/lt unknown
- 2006-06-26 CA CA2612623A patent/CA2612623C/fr active Active
- 2006-06-26 ES ES06763891.6T patent/ES2606772T3/es active Active
- 2006-06-26 EA EA200800152A patent/EA014163B1/ru unknown
- 2006-06-26 HR HRP20161704TT patent/HRP20161704T1/hr unknown
- 2006-06-26 CN CN2006800313527A patent/CN101252928B/zh not_active Expired - Fee Related
- 2006-06-26 DK DK06763891.6T patent/DK1898910T3/en active
- 2006-06-26 PL PL06763891T patent/PL1898910T3/pl unknown
- 2006-06-26 AU AU2006263884A patent/AU2006263884B2/en not_active Ceased
- 2006-06-26 US US11/917,923 patent/US20100204270A1/en not_active Abandoned
- 2006-06-26 KR KR1020087002248A patent/KR101423229B1/ko not_active Expired - Fee Related
- 2006-06-26 HU HUE06763891A patent/HUE031268T2/en unknown
- 2006-06-27 TW TW095123051A patent/TWI392494B/zh not_active IP Right Cessation
- 2006-06-27 MY MYPI20063045 patent/MY151030A/en unknown
- 2006-06-27 AR ARP060102760A patent/AR057654A1/es unknown
2007
- 2007-12-20 ZA ZA200711149A patent/ZA200711149B/xx unknown
- 2007-12-25 IL IL188394A patent/IL188394A/en active IP Right Grant
2008
- 2008-01-25 NO NO20080481A patent/NO341283B1/no not_active IP Right Cessation
2012
- 2012-08-07 US US13/568,597 patent/US20130030017A1/en not_active Abandoned
2016
- 2016-12-20 CY CY20161101322T patent/CY1118515T1/el unknown

Also Published As

Publication number	Publication date
SI1898910T1 (sl)	2017-01-31
NZ564339A (en)	2011-02-25
IL188394A0 (en)	2008-08-07
EP1898910A1 (fr)	2008-03-19
NO341283B1 (no)	2017-10-02
AU2006263884A1 (en)	2007-01-04
CA2612623C (fr)	2016-09-27
CA2612623A1 (fr)	2007-01-04
ME02690B (fr)	2017-10-20
AR057654A1 (es)	2007-12-12
HRP20161704T1 (hr)	2017-02-10
AU2006263884B2 (en)	2013-01-10
HK1120734A1 (en)	2009-04-09
BRPI0612534A8 (pt)	2017-12-26
ZA200711149B (en)	2009-06-24
MY151030A (en)	2014-03-31
US20100204270A1 (en)	2010-08-12
TW200738237A (en)	2007-10-16
NO20080481L (no)	2008-02-29
KR20080028460A (ko)	2008-03-31
CN101252928B (zh)	2012-05-23
EP1898910B1 (fr)	2016-09-28
CN101252928A (zh)	2008-08-27
UA91549C2 (ru)	2010-08-10
MX2008000082A (es)	2008-03-24
ES2606772T3 (es)	2017-03-27
PT1898910T (pt)	2016-11-16
RS55408B1 (sr)	2017-04-28
US20130030017A1 (en)	2013-01-31
BRPI0612534B8 (pt)	2021-05-25
BRPI0612534B1 (pt)	2020-04-22
LT1898910T (lt)	2017-01-10
EA200800152A1 (ru)	2008-06-30
AP2733A (en)	2013-09-30
IL188394A (en)	2012-09-24
JP2008546825A (ja)	2008-12-25
HUE031268T2 (en)	2017-06-28
CY1118515T1 (el)	2017-07-12
BRPI0612534A2 (pt)	2010-11-23
JO3270B1 (ar)	2018-09-16
EA014163B1 (ru)	2010-10-29
DK1898910T3 (en)	2017-01-09
JP5193859B2 (ja)	2013-05-08
KR101423229B1 (ko)	2014-07-25
TWI392494B (zh)	2013-04-11
PL1898910T3 (pl)	2017-03-31
WO2007000436A1 (fr)	2007-01-04

Publication	Publication Date	Title
UA100972C2 (ru)	2013-02-25	Антибактериальные производные хинолина
UA90267C2 (ru)	2010-04-26	Применение замещенных хинолиновых производных для лечения заболеваний, вызванных микобактериями, резистентными к лекарственным средствам
EA200800501A1 (ru)	2008-10-30	Производные хинолина в качестве антибактериальных средств
CY1114318T1 (el)	2016-08-31	Παραγωγα κινολινης ως αντιβακτηριακοι παραγοντες
WO2010047737A3 (fr)	2010-06-17	Composés indoliniques antimicrobiens pour le traitement d'infections bactériennes
MY145924A (en)	2012-05-15	Antibacterial quinoline derivatives
MX2009005981A (es)	2009-06-16	Derivados de quinolina antibacterianos.
NO20080501L (no)	2008-02-28	Kinolinderivater som antibakterielle midler
MX2008000079A (es)	2008-03-19	Derivados de quinolina como agentes antibacterianos.
CY1114384T1 (el)	2016-08-31	Αντιβακτηριακα παραγωγα κινολινης
MX2009005980A (es)	2009-06-16	Derivados antibacterianos de quinolina.
SG166799A1 (en)	2010-12-29	Quinoline derivatives as antibacterial agents
MY145940A (en)	2012-05-31	Antibacterial quinoline derivatives
UA95911C2 (ru)	2011-09-26	Производные хинолина как антибактериальные средства