SE8704746D0 - Tricykliska ketoner - Google Patents

Tricykliska ketoner

Info

Publication number: SE8704746D0
Authority: SE; Sweden
Prior art keywords: ketons; tricyclic; compounds; image; formula
Prior art date: 1986-11-28

Application number

SE8704746A

Other languages

English (en)

Other versions

SE8704746L (sv

SE467255B (sv

Inventor

I H Coates

J Bradshaw

J A Bell

D C Humber

G B Ewan

W L Mitchell

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-11-28

Filing date

1987-11-27

Publication date

1987-11-27

1986-11-28 Priority claimed from GB868628473A external-priority patent/GB8628473D0/en

1987-11-12 Priority claimed from GB878726537A external-priority patent/GB8726537D0/en

1987-11-27 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

1987-11-27 Publication of SE8704746D0 publication Critical patent/SE8704746D0/sv

1988-05-29 Publication of SE8704746L publication Critical patent/SE8704746L/sv

1992-06-22 Publication of SE467255B publication Critical patent/SE467255B/sv

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

SE8704746A 1986-11-28 1987-11-27 3-imidazolylmetyl-4-karbazoloner, 3-imidazolylmetylen-4-karbazoloner och mellanprodukter SE467255B (sv)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB868628473A GB8628473D0 (en)	1986-11-28	1986-11-28	Chemical compounds
GB878726537A GB8726537D0 (en)	1987-11-12	1987-11-12	Tricyclic ketones

Publications (3)

Publication Number	Publication Date
SE8704746D0 true SE8704746D0 (sv)	1987-11-27
SE8704746L SE8704746L (sv)	1988-05-29
SE467255B SE467255B (sv)	1992-06-22

Family

ID=26291603

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE8704746A SE467255B (sv)	1986-11-28	1987-11-27	3-imidazolylmetyl-4-karbazoloner, 3-imidazolylmetylen-4-karbazoloner och mellanprodukter

Country Status (24)

Country	Link
US (1)	US4822881A (sv)
AT (1)	AT396933B (sv)
AU (1)	AU605805B2 (sv)
BE (1)	BE1001004A4 (sv)
CA (1)	CA1326032C (sv)
CH (1)	CH676120A5 (sv)
CZ (1)	CZ404591A3 (sv)
DE (1)	DE3740352A1 (sv)
DK (1)	DK169675B1 (sv)
ES (1)	ES2008360A6 (sv)
FI (1)	FI92062C (sv)
FR (1)	FR2611366B1 (sv)
GB (1)	GB2202530B (sv)
GR (1)	GR871809B (sv)
HK (1)	HK51591A (sv)
IE (1)	IE61510B1 (sv)
IL (1)	IL84635A (sv)
IT (1)	IT1211936B (sv)
NL (1)	NL8702851A (sv)
NO (1)	NO172581C (sv)
NZ (1)	NZ222725A (sv)
PH (1)	PH30436A (sv)
SE (1)	SE467255B (sv)
SG (1)	SG46591G (sv)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8518742D0 (en) *	1985-07-24	1985-08-29	Glaxo Group Ltd	Process
US5202343A (en) *	1986-11-28	1993-04-13	Glaxo Group Limited	Tricyclic ketones useful as HT3 -receptor antagonists
GB8812002D0 (en) *	1988-05-20	1988-06-22	Glaxo Group Ltd	Chemical compounds
DE3822792C2 (de) *	1987-07-11	1997-11-27	Sandoz Ag	Neue Verwendung von 5HT¶3¶-Antagonisten
US5360800A (en) *	1987-09-03	1994-11-01	Glaxo Group Limited	Tetrahydro-1H-pyrido[4,3-b]indol-1-one derivatives
GB8720693D0 (en) *	1987-09-03	1987-10-07	Glaxo Group Ltd	Chemical compounds
US4939144A (en) *	1987-10-22	1990-07-03	Glaxo Group Limited	Tricyclic ketone derivatives as 5-HT antagonists
US5116984A (en) *	1988-04-07	1992-05-26	Glaxo Group Limited	Imidazole derivatives
DK185489A (da) *	1988-04-22	1989-10-23	Duphar Int Res	Imidazolylmethyl-cycloalkanoebaaindoloner, deres fremstilling og anvendelse
JPH0256485A (ja) *	1988-04-27	1990-02-26	Glaxo Group Ltd	ラクタム誘導体
GB8812636D0 (en) *	1988-05-27	1988-06-29	Glaxo Group Ltd	Chemical compounds
EP0350129A1 (en) *	1988-07-07	1990-01-10	Duphar International Research B.V	New annelated indoleketones with an imidazolylalkyl substituent
NO169714C (no) *	1988-08-02	1992-07-29	Glaxo Group Ltd	Analogifremgangsmaate for fremstilling av terapeutisk aktive laktamderivater
HU207078B (en) *	1988-08-02	1993-03-01	Glaxo Group Ltd	Process for producing lactam derivatives and pharmaceutical compositions comprising such compounds
US5008272A (en) *	1988-08-15	1991-04-16	Glaxo Group Limited	Lactam derivatives
US4997831A (en) *	1988-09-01	1991-03-05	Glaxo Group Limited	Lactam derivatives
GB8820653D0 (en) *	1988-09-01	1988-10-05	Glaxo Group Ltd	Medicaments
GB8820651D0 (en) *	1988-09-01	1988-10-05	Glaxo Group Ltd	Medicaments
GB8820650D0 (en) *	1988-09-01	1988-10-05	Glaxo Group Ltd	Medicaments
AU627221B2 (en) *	1988-09-27	1992-08-20	Fujisawa Pharmaceutical Co., Ltd.	Pyridoindole derivatives and processes for preparation thereof
GB8823980D0 (en) *	1988-10-13	1988-11-23	Glaxo Group Ltd	Chemical compounds
US5223625A (en) *	1988-12-22	1993-06-29	Duphar International Research B.V.	Annelated indolo [3,2,-C]lactams
HU204049B (en) *	1989-02-28	1991-11-28	Glaxo Group Ltd	Process for producing lactam derivatives and pharmaceutical compositions comprising same
GB8904551D0 (en) *	1989-02-28	1989-04-12	Glaxo Group Ltd	Chemical compounds
GB8904552D0 (en)	1989-02-28	1989-04-12	Glaxo Group Ltd	Chemical process
AU631632B2 (en)	1989-04-21	1992-12-03	Novartis Ag	Therapeutic use of 5-ht3 receptor antagonists
GB8928208D0 (en) *	1989-12-13	1990-02-14	Glaxo Group Ltd	Medicaments
HU211081B (en) *	1990-12-18	1995-10-30	Sandoz Ag	Process for producing indole derivatives as serotonin antagonists and pharmaceutical compositions containing the same
KR100368895B1 (ko) *	2000-03-30	2003-01-24	하나제약 주식회사	1,2,3,9-테트라하이드로-9-메틸-3-[(2-메틸-1ｈ-이미다졸-1-일)메틸]-4ｈ-카바졸-4-온의 제조방법
ATE356623T1 (de)	2002-01-18	2007-04-15	Aryx Therapeutics	5-ht3-rezeptorantagonisten und verwendungsverfahren
PL2432467T3 (pl)	2009-05-20	2018-07-31	INSERM (Institut National de la Santé et de la Recherche Médicale)	Zastosowanie antagonistów receptora 5-ht3 serotoniny w leczeniu zaburzeń przedsionkowych ze zmianami chorobowymi
ES2432618T3 (es)	2009-05-20	2013-12-04	Inserm (Institut National De La Santé Et De La Recherche Medicale)	Antagonistas del receptor 5-HT3 de serotonina para usar en el tratamiento o prevención de una patología del oído interno con déficit vestibular

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3740404A (en) *	1969-05-09	1973-06-19	American Cyanamid Co	Piperidinomethylenedihydrocarbazolones
US3634420A (en) *	1969-05-09	1972-01-11	American Cyanamid Co	3(morpholinomethyl)-2 3-dihydro-carbazol-4(1h)-ones
GB1365296A (en) *	1970-10-30	1974-08-29	Unilever Ltd	Dentifrice compositions
US4176230A (en) *	1977-08-04	1979-11-27	Hoffmann-La Roche Inc.	5-(6-Alkylindol-3-ylmethylene)-1,3-dimethyl-2-(methylimino)-4-imidazolidinones
MC1286A1 (fr) *	1978-11-01	1980-07-22	Wellcome Found	Preparation de composes heterocycliques utilisables en pharmacie et de medicaments contenant ces composes
DK151884C (da) *	1979-03-07	1988-06-13	Pfizer	Analogifremgangsmaade til fremstilling af 3-(1-imidazolylalkyl)indolderivater eller farmaceutisk acceptable syreadditionssalte deraf
US4695578A (en) *	1984-01-25	1987-09-22	Glaxo Group Limited	1,2,3,9-tetrahydro-3-imidazol-1-ylmethyl-4H-carbazol-4-ones, composition containing them, and method of using them to treat neuronal 5HT function disturbances
IL74165A (en) *	1984-01-25	1988-11-15	Glaxo Group Ltd	1,2,3,9-tetrahydro-3-(1h-imidazole-1-yl methyl)-4h-carbazol-4-one compounds,their preparation and pharmaceutical compositions containing them
EP0191562B1 (en) *	1985-01-23	1991-07-10	Glaxo Group Limited	Tetrahydrocarbazolone derivatives
GB8518745D0 (en) *	1985-07-24	1985-08-29	Glaxo Group Ltd	Heterocyclic compounds
GB8518743D0 (en) *	1985-07-24	1985-08-29	Glaxo Group Ltd	Heterocyclic compounds
GB8518741D0 (en) *	1985-07-24	1985-08-29	Glaxo Group Ltd	Process

1987
- 1987-11-26 GR GR871809A patent/GR871809B/el unknown
- 1987-11-27 BE BE8701353A patent/BE1001004A4/fr not_active IP Right Cessation
- 1987-11-27 NL NL8702851A patent/NL8702851A/nl not_active Application Discontinuation
- 1987-11-27 DE DE19873740352 patent/DE3740352A1/de not_active Ceased
- 1987-11-27 US US07/126,202 patent/US4822881A/en not_active Expired - Fee Related
- 1987-11-27 GB GB8727835A patent/GB2202530B/en not_active Expired - Fee Related
- 1987-11-27 FR FR878716488A patent/FR2611366B1/fr not_active Expired - Fee Related
- 1987-11-27 IE IE323287A patent/IE61510B1/en not_active IP Right Cessation
- 1987-11-27 NO NO874959A patent/NO172581C/no unknown
- 1987-11-27 IT IT8748642A patent/IT1211936B/it active
- 1987-11-27 AU AU81845/87A patent/AU605805B2/en not_active Ceased
- 1987-11-27 NZ NZ222725A patent/NZ222725A/xx unknown
- 1987-11-27 DK DK624887A patent/DK169675B1/da active
- 1987-11-27 SE SE8704746A patent/SE467255B/sv not_active IP Right Cessation
- 1987-11-27 ES ES8703405A patent/ES2008360A6/es not_active Expired
- 1987-11-27 AT AT0312487A patent/AT396933B/de not_active IP Right Cessation
- 1987-11-27 FI FI875235A patent/FI92062C/sv not_active IP Right Cessation
- 1987-11-27 CA CA000552963A patent/CA1326032C/en not_active Expired - Fee Related
- 1987-11-27 CH CH4614/87A patent/CH676120A5/fr not_active IP Right Cessation
- 1987-11-27 PH PH36132A patent/PH30436A/en unknown
- 1987-11-27 IL IL84635A patent/IL84635A/xx not_active IP Right Cessation
1991
- 1991-06-18 SG SG46591A patent/SG46591G/en unknown
- 1991-07-04 HK HK515/91A patent/HK51591A/xx not_active IP Right Cessation
- 1991-12-23 CZ CS914045A patent/CZ404591A3/cs unknown

Also Published As

Publication number	Publication date
PH30436A (en)	1997-05-09
CH676120A5 (sv)	1990-12-14
GB8727835D0 (en)	1987-12-31
AU605805B2 (en)	1991-01-24
IT1211936B (it)	1989-11-08
DK624887D0 (da)	1987-11-27
GB2202530B (en)	1990-04-18
NO172581C (no)	1993-08-11
SE8704746L (sv)	1988-05-29
FI875235A7 (sv)	1988-05-29
IE61510B1 (en)	1994-11-16
AT396933B (de)	1993-12-27
US4822881A (en)	1989-04-18
IT8748642A0 (it)	1987-11-27
DK169675B1 (da)	1995-01-09
IE873232L (en)	1988-05-28
ATA312487A (de)	1993-05-15
DE3740352A1 (de)	1988-06-09
NO172581B (no)	1993-05-03
IL84635A0 (en)	1988-04-29
GR871809B (en)	1988-03-07
HK51591A (en)	1991-07-12
NO874959L (no)	1988-05-30
DK624887A (da)	1988-05-29
BE1001004A4 (fr)	1989-06-06
NL8702851A (nl)	1988-06-16
ES2008360A6 (es)	1989-07-16
IL84635A (en)	1993-01-31
SE467255B (sv)	1992-06-22
NO874959D0 (no)	1987-11-27
FI92062B (sv)	1994-06-15
CA1326032C (en)	1994-01-11
SG46591G (en)	1991-07-26
FR2611366A1 (fr)	1988-09-02
FI92062C (sv)	1994-09-26
GB2202530A (en)	1988-09-28
AU8184587A (en)	1988-06-02
CZ404591A3 (en)	1993-08-11
NZ222725A (en)	1990-08-28
FR2611366B1 (fr)	1990-03-16
FI875235A0 (sv)	1987-11-27

Publication	Publication Date	Title
SE8704746D0 (sv)	1987-11-27	Tricykliska ketoner
EA199700156A1 (ru)	1997-12-30	Производные индола как антагонисты рецептора 5-нт
ES8801247A1 (es)	1987-12-16	Un procedimiento para la preparacion de nuevos derivados de carbazolona
FI931370A0 (fi)	1993-03-26	Kvaeve innehaollande analoger av icke-aromatiska heterocykliska foereningar med en fusionerad ring
DE3684195D1 (de)	1992-04-16	Substituierte imidazolylmethyltetrahydrocarbazolone.
ES2060655T3 (es)	1994-12-01	Derivados de lactamas.
DE3685471D1 (de)	1992-07-02	Tetrahydrocarbazolonderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen.
ES533338A0 (es)	1985-08-01	Derivados de la 2-pirimidinil-1-piperazina
NO964236D0 (no)	1996-10-04	Anvendelse av serotonin-antagonister (5HT3) for behandling av fibromyalgi
UA27467C2 (uk)	2000-09-15	ПОХІДНІ ІНДОЛУ ЯК 5-НТ<sub>1</sub> АГОНІСТИ ТА ПРОМІЖНІ СПОЛУКИ
EP0266899A3 (en)	1989-09-27	Indole derivatives
EP0339959A3 (en)	1991-03-20	Lactam derivatives
NO871861D0 (no)	1987-05-05	Fremgangsmaate for fremstilling av nye dopamin beta-hydroxylase inhibitorer.
ES2000936A6 (es)	1988-04-01	Un procedimiento para la preparacion de 3-imidazolin -metiltetrahidrocarbazolonas.
EP0356098A3 (en)	1990-07-25	Lactam derivatives
IE892999L (en)	1990-03-27	Pyridoindole derivatives and processes for preparation¹thereof
MX9700080A (es)	1997-04-30	Derivados de aril y heteroaril alcoxinaftaleno.
ES2143630T3 (es)	2000-05-16	Derivados azabicicloalquilos de imidazo(1,5-a)indol-3-ona utilizados como antagonistas de 5ht3.
DE3872722D1 (de)	1992-08-20	Indol-derivate.
EA199900043A1 (ru)	1999-06-24	ПРОИЗВОДНЫЕ ПИРИДИЛКАРБАМОИЛИНДОЛИНОВ В КАЧЕСТВЕ АНТАГОНИСТОВ 5-НТ2с-РЕЦЕПТОРОВ
YU51599A (sh)	2001-03-07	POSTUPAK I INTERMEDIJERI ZA β3-ADRENERGIČNI RECEPTORSKI AGONIST
DK245789A (da)	1989-11-21	Tricycliske ketoner
DK0521766T3 (da)	1995-02-20	Hidtil ukendt fremgangsmåde til syntese af enantiomerer af 3-aminochromanderivater
EG16489A (en)	1988-01-31	Process for the preparation of accridanone derivatives

Legal Events

Date	Code	Title	Description
1995-01-31	NAL	Patent in force	Ref document number: 8704746-0 Format of ref document f/p: F
1999-08-02	NUG	Patent has lapsed	Ref document number: 8704746-0 Format of ref document f/p: F

Date

Code

Title

Description

1995-01-31

NAL

Patent in force

Ref document number: 8704746-0

Format of ref document f/p: F

1999-08-02

NUG

Patent has lapsed