SE8500965D0 - Mellanprodukter for framstellning av beta-laktamasinhibitorer - Google Patents

Mellanprodukter for framstellning av beta-laktamasinhibitorer

Info

Publication number: SE8500965D0
Authority: SE; Sweden
Prior art keywords: beta; alpha; lactama; intermediates; inhibitors
Prior art date: 1979-09-26

Application number

SE8500965A

Other languages

English (en)

Other versions

SE461528B (sv

Inventor

W E Barth

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-09-26

Filing date

1985-02-27

Publication date

1985-02-27

1985-02-27 Application filed by Pfizer filed Critical Pfizer

1985-02-27 Publication of SE8500965D0 publication Critical patent/SE8500965D0/sv

1990-02-26 Publication of SE461528B publication Critical patent/SE461528B/sv

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
- C07D499/32—Esters

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Saccharide Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

SE8500965A 1979-09-26 1985-02-27 Mellanprodukter foer framstaellning av acetoximetyl-penamfoereningar, som aer anvaendbara som -laktamasinhibitorer SE461528B (sv)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/079,127 US4256733A (en)	1979-09-26	1979-09-26	Acetoxymethyl penam compounds as β-lactamase inhibitors

Publications (2)

Publication Number	Publication Date
SE8500965D0 true SE8500965D0 (sv)	1985-02-27
SE461528B SE461528B (sv)	1990-02-26

Family

ID=22148609

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
SE8005714A SE449865B (sv)	1979-09-26	1980-08-13	Acetoximetyl-pencillansyra derivat och dess anvendning sasom beta-laktamasinhibitorer
SE8500965A SE461528B (sv)	1979-09-26	1985-02-27	Mellanprodukter foer framstaellning av acetoximetyl-penamfoereningar, som aer anvaendbara som -laktamasinhibitorer

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
SE8005714A SE449865B (sv)	1979-09-26	1980-08-13	Acetoximetyl-pencillansyra derivat och dess anvendning sasom beta-laktamasinhibitorer

Country Status (36)

Country	Link
US (1)	US4256733A (sv)
JP (1)	JPS6016958B2 (sv)
KR (1)	KR840000796B1 (sv)
AR (1)	AR224547A1 (sv)
AT (1)	AT366384B (sv)
AU (1)	AU517074B2 (sv)
BE (1)	BE885389A (sv)
CA (1)	CA1150242A (sv)
CH (1)	CH645646A5 (sv)
CS (1)	CS212284B2 (sv)
DD (1)	DD153123A5 (sv)
DE (1)	DE3035995C2 (sv)
DK (1)	DK404980A (sv)
EG (1)	EG14888A (sv)
ES (1)	ES8106528A1 (sv)
FI (2)	FI67552C (sv)
FR (1)	FR2465736A1 (sv)
GB (2)	GB2059420B (sv)
GR (1)	GR70065B (sv)
HU (1)	HU183212B (sv)
IE (2)	IE50506B1 (sv)
IL (1)	IL61117A (sv)
IN (1)	IN154557B (sv)
IT (1)	IT1132754B (sv)
LU (1)	LU82795A1 (sv)
MX (1)	MX6580E (sv)
NL (1)	NL185923C (sv)
NO (2)	NO160370C (sv)
NZ (1)	NZ195058A (sv)
PH (1)	PH15697A (sv)
PL (1)	PL126949B1 (sv)
PT (1)	PT71837B (sv)
SE (2)	SE449865B (sv)
SU (1)	SU959628A3 (sv)
YU (1)	YU41733B (sv)
ZA (1)	ZA805132B (sv)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4364957A (en) *	1979-09-26	1982-12-21	Pfizer Inc.	Bis-esters of alkanediols as antibacterial agents
US4511512A (en) *	1980-05-01	1985-04-16	Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Produktionsaktiensel skab)	Substantially pure dicyclohexyl ammonium 6-β-bromo-penicillanate
US4474698A (en) *	1980-12-11	1984-10-02	Pfizer Inc.	Process for preparing esters of penicillanic acid sulfone
US4361513A (en) *	1980-12-11	1982-11-30	Pfizer Inc.	Esters of penicillanic acid sulfone
US4558042A (en) *	1981-05-06	1985-12-10	Farmitalia Carlo Erba S.P.A.	β-Lactam-containing antibacterial agents and β-lactamase inhibitors
ZA826687B (en) *	1981-09-14	1983-07-27	Pfizer	Beta-lactamase inhibiting 2-beta-substituted-2-alpha-methyl 5(r)penam-3-alpha-carboxylic acid 1,1-dioxides and intermediates therefor
JPS58185589A (ja) *	1982-04-23	1983-10-29	Taiho Yakuhin Kogyo Kk	ペニシリン誘導体
JPS62198687A (ja) *	1986-02-27	1987-09-02	Taiho Yakuhin Kogyo Kk	２β−置換チオメチルペニシリン誘導体
US4861768A (en) *	1986-02-27	1989-08-29	Taiho Pharmaceutical Company, Limited	2 β-substituted thiomethylpenicillin derivatives and their preparation and use
SK63894A3 (en) *	1991-12-19	1995-03-08	Novo Nordisk As	Method of preparation of beta-lactam antibiotic
CN115385934A (zh) *	2022-10-26	2022-11-25	北京纳百生物科技有限公司	一种舒巴坦半抗原及其合成方法和应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE648188A (sv)	1963-05-29	1964-09-16
IN149747B (sv)	1977-06-07	1982-04-03	Pfizer

1979
- 1979-09-26 US US06/079,127 patent/US4256733A/en not_active Expired - Lifetime
1980
- 1980-08-13 SE SE8005714A patent/SE449865B/sv not_active IP Right Cessation
- 1980-08-20 ZA ZA00805132A patent/ZA805132B/xx unknown
- 1980-08-20 IN IN607/DEL/80A patent/IN154557B/en unknown
- 1980-09-19 HU HU802310A patent/HU183212B/hu unknown
- 1980-09-19 SU SU802983144A patent/SU959628A3/ru active
- 1980-09-22 CS CS806403A patent/CS212284B2/cs unknown
- 1980-09-22 PL PL1980226868A patent/PL126949B1/pl unknown
- 1980-09-23 CA CA000360886A patent/CA1150242A/en not_active Expired
- 1980-09-23 GR GR62939A patent/GR70065B/el unknown
- 1980-09-23 IL IL61117A patent/IL61117A/xx unknown
- 1980-09-23 EG EG584/80A patent/EG14888A/xx active
- 1980-09-23 AT AT0474680A patent/AT366384B/de not_active IP Right Cessation
- 1980-09-23 GB GB8030639A patent/GB2059420B/en not_active Expired
- 1980-09-24 MX MX809044U patent/MX6580E/es unknown
- 1980-09-24 PH PH24617A patent/PH15697A/en unknown
- 1980-09-24 KR KR1019800003721A patent/KR840000796B1/ko not_active Expired
- 1980-09-24 AR AR282629A patent/AR224547A1/es active
- 1980-09-24 LU LU82795A patent/LU82795A1/fr unknown
- 1980-09-24 DE DE3035995A patent/DE3035995C2/de not_active Expired
- 1980-09-25 BE BE0/202222A patent/BE885389A/fr not_active IP Right Cessation
- 1980-09-25 ES ES495354A patent/ES8106528A1/es not_active Expired
- 1980-09-25 NZ NZ195058A patent/NZ195058A/xx unknown
- 1980-09-25 NL NLAANVRAGE8005344,A patent/NL185923C/xx not_active IP Right Cessation
- 1980-09-25 IE IE1998/80A patent/IE50506B1/en not_active IP Right Cessation
- 1980-09-25 FI FI803028A patent/FI67552C/fi not_active IP Right Cessation
- 1980-09-25 IE IE1095/85A patent/IE50507B1/en unknown
- 1980-09-25 DD DD80224128A patent/DD153123A5/de unknown
- 1980-09-25 NO NO802836A patent/NO160370C/no unknown
- 1980-09-25 FR FR8020618A patent/FR2465736A1/fr active Granted
- 1980-09-25 AU AU62713/80A patent/AU517074B2/en not_active Ceased
- 1980-09-25 DK DK404980A patent/DK404980A/da not_active Application Discontinuation
- 1980-09-25 JP JP55133639A patent/JPS6016958B2/ja not_active Expired
- 1980-09-25 IT IT24920/80A patent/IT1132754B/it active
- 1980-09-25 CH CH719980A patent/CH645646A5/fr not_active IP Right Cessation
- 1980-09-25 PT PT71837A patent/PT71837B/pt unknown
- 1980-09-25 YU YU2449/80A patent/YU41733B/xx unknown
1983
- 1983-03-25 NO NO83831082A patent/NO160299C/no unknown
- 1983-07-22 GB GB08319784A patent/GB2125037B/en not_active Expired
1984
- 1984-01-30 FI FI840367A patent/FI67854C/fi not_active IP Right Cessation
1985
- 1985-02-27 SE SE8500965A patent/SE461528B/sv not_active IP Right Cessation

Also Published As

Publication number	Publication date
IE50506B1 (en)	1986-04-30
PT71837A (en)	1980-10-01
IE801095L (en)	1981-01-09
BE885389A (fr)	1981-03-25
PL226868A1 (sv)	1981-10-16
SU959628A3 (ru)	1982-09-15
NO802836L (no)	1981-03-27
AU6271380A (en)	1981-04-09
IN154557B (sv)	1984-11-10
GB2059420A (en)	1981-04-23
AT366384B (de)	1982-04-13
NL185923C (nl)	1990-08-16
NO160370B (no)	1989-01-02
GR70065B (sv)	1982-07-26
PL126949B1 (en)	1983-09-30
YU244980A (en)	1983-02-28
GB8319784D0 (en)	1983-08-24
JPS6016958B2 (ja)	1985-04-30
DD153123A5 (de)	1981-12-23
NZ195058A (en)	1982-12-07
JPS5657788A (en)	1981-05-20
HU183212B (en)	1984-04-28
IL61117A (en)	1983-10-31
PT71837B (en)	1981-07-09
FI67552C (fi)	1985-04-10
GB2059420B (en)	1984-03-14
FI67854C (fi)	1985-06-10
EG14888A (en)	1985-06-30
NL185923B (nl)	1990-03-16
IE50507B1 (en)	1986-04-30
FR2465736B1 (sv)	1982-04-30
DE3035995A1 (de)	1981-04-02
US4256733A (en)	1981-03-17
AR224547A1 (es)	1981-12-15
NO160370C (no)	1989-04-12
ATA474680A (de)	1981-08-15
FI67854B (fi)	1985-02-28
ES495354A0 (es)	1981-08-16
FI803028A7 (fi)	1981-03-27
LU82795A1 (fr)	1981-04-17
ZA805132B (en)	1981-12-30
CS212284B2 (en)	1982-03-26
PH15697A (en)	1983-03-14
NO831082L (no)	1981-03-27
ES8106528A1 (es)	1981-08-16
IL61117A0 (en)	1980-11-30
KR840000796B1 (ko)	1984-06-12
NO160299B (no)	1988-12-27
KR830003494A (ko)	1983-06-20
FI840367L (fi)	1984-01-30
SE449865B (sv)	1987-05-25
NO160299C (no)	1989-04-05
IT8024920A0 (it)	1980-09-25
MX6580E (es)	1985-07-24
YU41733B (en)	1987-12-31
SE461528B (sv)	1990-02-26
CH645646A5 (fr)	1984-10-15
FI67552B (fi)	1984-12-31
IE801998L (en)	1981-03-26
AU517074B2 (en)	1981-07-09
NL8005344A (nl)	1981-03-30
DE3035995C2 (de)	1985-01-10
SE8005714L (sv)	1981-03-27
GB2125037B (en)	1984-08-01
FI840367A0 (fi)	1984-01-30
GB2125037A (en)	1984-02-29
CA1150242A (en)	1983-07-19
FR2465736A1 (fr)	1981-03-27
IT1132754B (it)	1986-07-02
DK404980A (da)	1981-03-27

Publication	Publication Date	Title
SE8305916L (sv)	1983-10-27	Mellanprodukter for framstellning av penicillansyra-1,1-dioxider
AU6354880A (en)	1981-04-30	Derivatives of 6beta-hydroxyalkylpenicillanic acids as beta-lactamase inhibitors
ZA817696B (en)	1982-10-27	N-substituted omega-(2-oxo-4-imidazolin-1-yl)alcanoic acids,salts and esters thereof,process for producing the same and these active agents containing pharmaceutical compounds
SE8500965D0 (sv)	1985-02-27	Mellanprodukter for framstellning av beta-laktamasinhibitorer
IE780899L (en)	1978-11-05	Azetidinopyrrole derivatives
IL90056A (en)	1993-04-04	Topical pharmaceutical compositions containing 4-quinoline carboxylic acid derivatives
SE8404308D0 (sv)	1984-08-29	Polyprenylkarboxylsyraamider, forfarande for deras framstellning samt farmaceutiska kompositioner innehallande dessa foreningar
NZ201895A (en)	1985-03-20	2-beta-substituted-2-alpha-methyl-(5r)-penam-3-alpha-carboxylic acid 1,1-dioxides;intermediates and pharmaceutical compositions
SE7609495L (sv)	1977-02-28	N-tetrahydrofurfuryl-noroximorfon, dess syraadditionssalter, lekemedel innehallande dessa samt forfarande for framstellning derav
NO810758L (no)	1981-09-08	Fremgangsmaate for oekning av den orale absorpsjon av beta-lactamantibiotika
DE3062787D1 (en)	1983-05-19	Novel process for the preparation of 6-aminopenicillanic acid-1,1-dioxide and its salts
SE7906681L (sv)	1980-02-12	Ftalazonderivat
ES476259A1 (es)	1979-04-16	Un procedimiento para la preparacion de un compuesto.
GB2014574A (en)	1979-08-30	Lactam Compounds
FI830192A0 (fi)	1983-01-20	Foerfarande foer framstaellning av penicillinderivat

Legal Events

Date	Code	Title	Description
1995-01-31	NUG	Patent has lapsed	Ref document number: 8500965-2 Effective date: 19910131 Format of ref document f/p: F

Date

Code

Title

Description

1995-01-31

NUG

Patent has lapsed

Ref document number: 8500965-2

Effective date: 19910131

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