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RU2004139022A - Фармацевтические препараты для орального употребления, содержащие заполненные биологически активными веществами ионообменные смолы, а также структурно-вязкие агенты гелеобразования в качестве загустителей - Google Patents

Фармацевтические препараты для орального употребления, содержащие заполненные биологически активными веществами ионообменные смолы, а также структурно-вязкие агенты гелеобразования в качестве загустителей Download PDF

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Publication number
RU2004139022A
RU2004139022A RU2004139022/15A RU2004139022A RU2004139022A RU 2004139022 A RU2004139022 A RU 2004139022A RU 2004139022/15 A RU2004139022/15 A RU 2004139022/15A RU 2004139022 A RU2004139022 A RU 2004139022A RU 2004139022 A RU2004139022 A RU 2004139022A
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RU
Russia
Prior art keywords
biologically active
pharmaceutical preparation
ion exchanger
preparation according
agents
Prior art date
Application number
RU2004139022/15A
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English (en)
Other versions
RU2380091C2 (ru
Inventor
Дирк МЕРТИН (DE)
Дирк Мертин
Маркус ЭДИНГЛО (DE)
Маркус Эдингло
Герт ДАУБЕ (DE)
Герт Даубе
Original Assignee
Байер ХельсКер АГ (DE)
Байер ХельсКер АГ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Байер ХельсКер АГ (DE), Байер ХельсКер АГ filed Critical Байер ХельсКер АГ (DE)
Publication of RU2004139022A publication Critical patent/RU2004139022A/ru
Application granted granted Critical
Publication of RU2380091C2 publication Critical patent/RU2380091C2/ru

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/58Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. poly[meth]acrylate, polyacrylamide, polystyrene, polyvinylpyrrolidone, polyvinylalcohol or polystyrene sulfonic acid resin
    • A61K47/585Ion exchange resins, e.g. polystyrene sulfonic acid resin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dispersion Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Cosmetics (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Claims (10)

1. Фармацевтический препарат, содержащий одно или несколько связанных с ионитом биологически активных веществ, отличающийся тем, что наполненный ионит диспергирован в среде-носителе, содержащей один или несколько структурно-вязких агентов гелеобразования.
2. Фармацевтический препарат по п.1, отличающийся тем, что в качестве структурно-вязкого агента гелеобразования он содержит полиакриловую кислоту, ксантан, микрокристаллическую целлюлозу, простой эфир целлюлозы, бентонит, высокодисперсный диоксид кремния или смесь указанных агентов гелеобразования.
3. Фармацевтический препарат по п.1, отличающийся тем, что ионит является кислым ионитом.
4. Фармацевтический препарат по п.1, отличающийся тем, что среда-носитель содержит воду.
5. Фармацевтический препарат по п.1, отличающийся тем, что биологически активным веществом, связанным с ионитом, является хинолоновый антибиотик.
6. Фармацевтический препарат по п.1, отличающийся тем, что биологически активным веществом, связанным с ионитом, является прадофлоксацин.
7. Фармацевтический препарат по п.1, отличающийся тем, что биологически активным веществом, связанным с ионитом, является энрофлоксацин.
8. Фармацевтический препарат по п.1, отличающийся тем, что биологически активным веществом, связанным с ионитом, является флупиртин.
9. Применение фармацевтических препаратов по п.1 для орального применения.
10. Применение структурно-вязких агентов гелеобразования для улучшения свойств жидких суспензий, предназначенных для использования в качестве орально применяемых лекарственных средств для животных.
RU2004139022/15A 2002-05-31 2003-05-19 Фармацевтические препараты для орального употребления, содержащие заполненные биологически активными веществами ионообменные смолы, а также структурно-вязкие агенты гелеобразования в качестве загустителей RU2380091C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10224086.8 2002-05-31
DE10224086A DE10224086A1 (de) 2002-05-31 2002-05-31 Pharmazeutische Zubereitungen zur oralen Anwendung enthaltend wirkstoffbeladene Ionentauscherharze sowie strukturviskose Gelbildner als Verdicker

Publications (2)

Publication Number Publication Date
RU2004139022A true RU2004139022A (ru) 2005-07-10
RU2380091C2 RU2380091C2 (ru) 2010-01-27

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
RU2004139022/15A RU2380091C2 (ru) 2002-05-31 2003-05-19 Фармацевтические препараты для орального употребления, содержащие заполненные биологически активными веществами ионообменные смолы, а также структурно-вязкие агенты гелеобразования в качестве загустителей

Country Status (27)

Country Link
US (1) US8545829B2 (ru)
EP (1) EP1513500B1 (ru)
JP (2) JP5350574B2 (ru)
KR (3) KR20120123607A (ru)
CN (1) CN1671361B (ru)
AR (2) AR039861A1 (ru)
AT (1) ATE421317T1 (ru)
AU (1) AU2003242545B2 (ru)
BR (2) BR0311511A (ru)
CA (1) CA2487648C (ru)
CR (1) CR7598A (ru)
DE (2) DE10224086A1 (ru)
DK (1) DK1513500T3 (ru)
ES (1) ES2319115T3 (ru)
HR (1) HRP20041219B1 (ru)
IL (2) IL165322A0 (ru)
MX (1) MXPA04011820A (ru)
MY (1) MY140953A (ru)
NO (1) NO333939B1 (ru)
PL (1) PL207269B1 (ru)
PT (1) PT1513500E (ru)
RU (1) RU2380091C2 (ru)
SI (1) SI1513500T1 (ru)
TW (1) TWI333422B (ru)
UA (1) UA84270C2 (ru)
WO (1) WO2003101422A2 (ru)
ZA (1) ZA200409616B (ru)

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CN103349659A (zh) * 2006-09-26 2013-10-16 塔罗制药北美有限公司 液体药物组合物以及应用
DE102006049520A1 (de) 2006-10-20 2008-04-24 Bayer Healthcare Ag Verfahren zur Herstellung von Pradofloxacin
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US20090247575A1 (en) * 2008-03-26 2009-10-01 Taro Pharmaceuticals North America, Inc. Stabilizing lipid compositions for oral pharmaceutical agents
PL2544532T3 (pl) 2010-03-12 2017-08-31 Monsanto Technology Llc Agrochemiczne kompozycje żelowe
ES2588008T3 (es) * 2010-05-19 2016-10-28 Astellas Pharma Inc. Composición farmacéutica que contiene solifenacina
EP2768488A4 (en) 2011-10-19 2015-04-15 Rp Scherer Technologies Llc TWO-PHASE PHARMACEUTICAL DELIVERY SYSTEM
FR2998305B1 (fr) * 2012-11-22 2015-02-20 Henkel Ag & Co Kgaa Substances actives contenant des groupes sulfonates ameliorant la puissance de lavage primaire
KR101697095B1 (ko) * 2015-09-30 2017-01-18 주식회사 포스코 더스트 막힘을 방지할 수 있는 배가스 청정 라인의 실탱크
CN111989314B (zh) 2018-04-25 2024-04-30 拜耳动物保健有限责任公司 喹诺酮甲酸酯水解的方法
CN114249749B (zh) * 2022-01-08 2024-03-22 天象生物药业邢台有限责任公司 一种马波沙星甲酸盐的转化方法

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Also Published As

Publication number Publication date
CN1671361B (zh) 2010-05-12
NO20045700L (no) 2004-12-29
WO2003101422A3 (de) 2004-12-09
US20060177414A1 (en) 2006-08-10
EP1513500B1 (de) 2009-01-21
MY140953A (en) 2010-02-12
BR0311511A (pt) 2005-02-22
PL373456A1 (en) 2005-08-22
NO333939B1 (no) 2013-10-28
PT1513500E (pt) 2009-04-02
JP2011012087A (ja) 2011-01-20
SI1513500T1 (sl) 2009-06-30
JP2006503806A (ja) 2006-02-02
BRPI0311511A (ru) 2005-02-22
CA2487648A1 (en) 2003-12-11
HRP20041219A2 (en) 2006-02-28
UA84270C2 (ru) 2008-10-10
IL165322A (en) 2015-11-30
ES2319115T3 (es) 2009-05-04
BRPI0311511A8 (pt) 2017-07-11
CA2487648C (en) 2012-03-13
EP1513500A2 (de) 2005-03-16
MXPA04011820A (es) 2005-03-31
JP5350574B2 (ja) 2013-11-27
CR7598A (es) 2008-07-31
KR101258373B1 (ko) 2013-04-30
RU2380091C2 (ru) 2010-01-27
KR20050010015A (ko) 2005-01-26
WO2003101422A2 (de) 2003-12-11
BRPI0311511B1 (pt) 2018-07-10
TWI333422B (en) 2010-11-21
TW200406230A (en) 2004-05-01
AU2003242545B2 (en) 2010-02-18
HRP20041219B1 (hr) 2013-05-31
DK1513500T3 (da) 2009-05-11
ATE421317T1 (de) 2009-02-15
IL165322A0 (en) 2006-01-15
CN1671361A (zh) 2005-09-21
AU2003242545A1 (en) 2003-12-19
PL207269B1 (pl) 2010-11-30
ZA200409616B (en) 2006-05-31
DE10224086A1 (de) 2003-12-11
KR20120123607A (ko) 2012-11-08
HK1083200A1 (en) 2006-06-30
AR039861A1 (es) 2005-03-02
DE50311123D1 (de) 2009-03-12
KR20120006092A (ko) 2012-01-17
AR105798A2 (es) 2017-11-08
US8545829B2 (en) 2013-10-01

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