RU2003119067A - METHOD FOR PRODUCING BETULIN ACID - Google Patents
METHOD FOR PRODUCING BETULIN ACID Download PDFInfo
- Publication number
- RU2003119067A RU2003119067A RU2003119067/04A RU2003119067A RU2003119067A RU 2003119067 A RU2003119067 A RU 2003119067A RU 2003119067/04 A RU2003119067/04 A RU 2003119067/04A RU 2003119067 A RU2003119067 A RU 2003119067A RU 2003119067 A RU2003119067 A RU 2003119067A
- Authority
- RU
- Russia
- Prior art keywords
- acid
- producing
- producing betulin
- betulin acid
- sodium borohydride
- Prior art date
Links
- JYDNKGUBLIKNAM-UHFFFAOYSA-N Oxyallobutulin Natural products C1CC(=O)C(C)(C)C2CCC3(C)C4(C)CCC5(CO)CCC(C(=C)C)C5C4CCC3C21C JYDNKGUBLIKNAM-UHFFFAOYSA-N 0.000 title claims 2
- FVWJYYTZTCVBKE-ROUWMTJPSA-N betulin Chemical compound C1C[C@H](O)C(C)(C)[C@@H]2CC[C@@]3(C)[C@]4(C)CC[C@@]5(CO)CC[C@@H](C(=C)C)[C@@H]5[C@H]4CC[C@@H]3[C@]21C FVWJYYTZTCVBKE-ROUWMTJPSA-N 0.000 title claims 2
- MVIRREHRVZLANQ-UHFFFAOYSA-N betulin Natural products CC(=O)OC1CCC2(C)C(CCC3(C)C2CC=C4C5C(CCC5(CO)CCC34C)C(=C)C)C1(C)C MVIRREHRVZLANQ-UHFFFAOYSA-N 0.000 title claims 2
- 239000002253 acid Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- QGJZLNKBHJESQX-UHFFFAOYSA-N 3-Epi-Betulin-Saeure Natural products C1CC(O)C(C)(C)C2CCC3(C)C4(C)CCC5(C(O)=O)CCC(C(=C)C)C5C4CCC3C21C QGJZLNKBHJESQX-UHFFFAOYSA-N 0.000 claims 3
- CLOUCVRNYSHRCF-UHFFFAOYSA-N 3beta-Hydroxy-20(29)-Lupen-3,27-oic acid Natural products C1CC(O)C(C)(C)C2CCC3(C)C4(C(O)=O)CCC5(C)CCC(C(=C)C)C5C4CCC3C21C CLOUCVRNYSHRCF-UHFFFAOYSA-N 0.000 claims 3
- QTBSBXVTEAMEQO-UHFFFAOYSA-N Acetic acid Chemical compound CC(O)=O QTBSBXVTEAMEQO-UHFFFAOYSA-N 0.000 claims 3
- DIZWSDNSTNAYHK-XGWVBXMLSA-N Betulinic acid Natural products CC(=C)[C@@H]1C[C@H]([C@H]2CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)C(=O)O DIZWSDNSTNAYHK-XGWVBXMLSA-N 0.000 claims 3
- QGJZLNKBHJESQX-FZFNOLFKSA-N betulinic acid Chemical compound C1C[C@H](O)C(C)(C)[C@@H]2CC[C@@]3(C)[C@]4(C)CC[C@@]5(C(O)=O)CC[C@@H](C(=C)C)[C@@H]5[C@H]4CC[C@@H]3[C@]21C QGJZLNKBHJESQX-FZFNOLFKSA-N 0.000 claims 3
- PZXJOHSZQAEJFE-UHFFFAOYSA-N dihydrobetulinic acid Natural products C1CC(O)C(C)(C)C2CCC3(C)C4(C)CCC5(C(O)=O)CCC(C(C)C)C5C4CCC3C21C PZXJOHSZQAEJFE-UHFFFAOYSA-N 0.000 claims 3
- MQYXUWHLBZFQQO-UHFFFAOYSA-N nepehinol Natural products C1CC(O)C(C)(C)C2CCC3(C)C4(C)CCC5(C)CCC(C(=C)C)C5C4CCC3C21C MQYXUWHLBZFQQO-UHFFFAOYSA-N 0.000 claims 3
- SLJTWDNVZKIDAU-SVAFSPIFSA-N Betulonic acid Chemical compound C1CC(=O)C(C)(C)[C@@H]2CC[C@@]3(C)[C@]4(C)CC[C@@]5(C(O)=O)CC[C@@H](C(=C)C)[C@@H]5[C@H]4CC[C@@H]3[C@]21C SLJTWDNVZKIDAU-SVAFSPIFSA-N 0.000 claims 2
- SLJTWDNVZKIDAU-CKURCAGRSA-N Betulonic acid Natural products CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@@H](CC[C@@H]4[C@@]5(C)CCC(=O)C(C)(C)[C@@H]5CC[C@@]34C)[C@@H]12)C(=O)O SLJTWDNVZKIDAU-CKURCAGRSA-N 0.000 claims 2
- 229910000033 sodium borohydride Inorganic materials 0.000 claims 2
- 239000012279 sodium borohydride Substances 0.000 claims 2
- WGLPBDUCMAPZCE-UHFFFAOYSA-N Trioxochromium Chemical compound O=[Cr](=O)=O WGLPBDUCMAPZCE-UHFFFAOYSA-N 0.000 claims 1
- 229910000423 chromium oxide Inorganic materials 0.000 claims 1
- 230000001590 oxidative effect Effects 0.000 claims 1
- 159000000000 sodium salts Chemical class 0.000 claims 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims 1
Landscapes
- Steroid Compounds (AREA)
Claims (1)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2003119067/04A RU2246500C1 (en) | 2003-06-24 | 2003-06-24 | Method for preparing betulinic acid |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2003119067/04A RU2246500C1 (en) | 2003-06-24 | 2003-06-24 | Method for preparing betulinic acid |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2003119067A true RU2003119067A (en) | 2005-01-10 |
| RU2246500C1 RU2246500C1 (en) | 2005-02-20 |
Family
ID=34881398
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2003119067/04A RU2246500C1 (en) | 2003-06-24 | 2003-06-24 | Method for preparing betulinic acid |
Country Status (1)
| Country | Link |
|---|---|
| RU (1) | RU2246500C1 (en) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2013038314A1 (en) * | 2011-09-12 | 2013-03-21 | Stora Enso Oyj | Method for preparation of betulinic acid |
| CN107573397A (en) * | 2017-09-13 | 2018-01-12 | 江苏耐雀生物工程技术有限公司 | A kind of method for preparing betulic acid |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2428426C1 (en) * | 2010-03-11 | 2011-09-10 | Нина Борисовна Мельникова | Method for obtaining betulinic acid |
| RU2458933C1 (en) * | 2011-05-10 | 2012-08-20 | Государственное образовательное учреждение высшего профессионального образования "Нижегородская государственная медицинская академия" Министерства здравоохранения и социального развития Российской Федерации (ГОУ ВПО НижГМА Минздравсоцразвития России) | Method for producing betulinic acid |
| RU2463041C1 (en) * | 2011-05-10 | 2012-10-10 | Государственное образовательное учреждение высшего профессионального образования "Нижегородская государственная медицинская академия" Министерства здравоохранения и социального развития Российской Федерации (ГОУ ВПО НижГМА Минздравсоцразвития России) | Method of obtaining betulinic acid |
| RU2565773C1 (en) * | 2014-10-20 | 2015-10-20 | Федеральное государственное бюджетное учреждение науки Институт органической химии Уфимского научного центра Российской академии наук (ИОХ УНЦ РАН) | Method for producing betulinic acid |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6232481B1 (en) * | 2000-01-11 | 2001-05-15 | Regents Of The University Of Minnesota | Method for manufacturing betulinic acid |
| RU2190622C1 (en) * | 2001-12-26 | 2002-10-10 | Рощин Виктор Иванович | Method of synthesis of betulinic acid |
-
2003
- 2003-06-24 RU RU2003119067/04A patent/RU2246500C1/en not_active IP Right Cessation
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2013038314A1 (en) * | 2011-09-12 | 2013-03-21 | Stora Enso Oyj | Method for preparation of betulinic acid |
| CN107573397A (en) * | 2017-09-13 | 2018-01-12 | 江苏耐雀生物工程技术有限公司 | A kind of method for preparing betulic acid |
| CN107573397B (en) * | 2017-09-13 | 2019-07-30 | 江苏耐雀生物工程技术有限公司 | A method of preparing betulic acid |
Also Published As
| Publication number | Publication date |
|---|---|
| RU2246500C1 (en) | 2005-02-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20070625 |