PT2925757T - Compostos e composições para o tratamento de doenças parasitárias - Google Patents
Compostos e composições para o tratamento de doenças parasitáriasInfo
- Publication number
- PT2925757T PT2925757T PT137959771T PT13795977T PT2925757T PT 2925757 T PT2925757 T PT 2925757T PT 137959771 T PT137959771 T PT 137959771T PT 13795977 T PT13795977 T PT 13795977T PT 2925757 T PT2925757 T PT 2925757T
- Authority
- PT
- Portugal
- Prior art keywords
- compositions
- compounds
- treatment
- parasitic diseases
- parasitic
- Prior art date
Links
- 208000030852 Parasitic disease Diseases 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261728018P | 2012-11-19 | 2012-11-19 | |
| US201361847860P | 2013-07-18 | 2013-07-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT2925757T true PT2925757T (pt) | 2018-01-09 |
Family
ID=49667630
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT137959771T PT2925757T (pt) | 2012-11-19 | 2013-11-18 | Compostos e composições para o tratamento de doenças parasitárias |
Country Status (19)
| Country | Link |
|---|---|
| US (3) | US9556169B2 (pt) |
| EP (1) | EP2925757B1 (pt) |
| JP (1) | JP6298472B2 (pt) |
| CN (1) | CN105164124B (pt) |
| AR (1) | AR093532A1 (pt) |
| CY (1) | CY1119727T1 (pt) |
| DK (1) | DK2925757T3 (pt) |
| ES (1) | ES2655030T3 (pt) |
| HR (1) | HRP20171998T1 (pt) |
| HU (1) | HUE037600T2 (pt) |
| LT (1) | LT2925757T (pt) |
| ME (1) | ME03042B (pt) |
| PL (1) | PL2925757T3 (pt) |
| PT (1) | PT2925757T (pt) |
| RS (1) | RS56720B1 (pt) |
| SI (1) | SI2925757T1 (pt) |
| TW (1) | TWI600654B (pt) |
| UY (1) | UY35146A (pt) |
| WO (1) | WO2014078802A1 (pt) |
Families Citing this family (28)
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|---|---|---|---|---|
| MA41338B1 (fr) * | 2015-01-16 | 2019-07-31 | Hoffmann La Roche | Composés de pyrazine pour le traitement de maladies infectieuses |
| CA3012107A1 (en) | 2016-01-21 | 2017-07-27 | Novartis Ag | Compounds and compositions for the treatment of cryptosporidiosis |
| TWI679197B (zh) * | 2016-05-05 | 2019-12-11 | 瑞士商伊蘭科動物健康公司 | 雜芳基-1,2,4-三唑及雜芳基-三唑化合物 |
| WO2018011163A1 (en) * | 2016-07-14 | 2018-01-18 | F. Hoffmann-La Roche Ag | 6,7-dihydro-4h-pyrazolo[1,5-a]pyrazine and 6,7-dihydro-4h-triazolo[1,5-a]pyrazine compounds for the treatment of infectious diseases |
| BR112019007594A2 (pt) * | 2016-10-13 | 2019-07-02 | Loyola University Of Chicago | método para bloquear a transmissão do parasita da malária |
| MA52337A (fr) | 2017-03-01 | 2021-03-03 | Anacor Pharmaceuticals Inc | Nouveaux analogues d'oxaborole et utilisations de ces derniers |
| ES2966369T3 (es) * | 2017-03-20 | 2024-04-22 | Broad Inst Inc | Compuestos y métodos para el tratamiento de enfermedades parasitarias |
| EP3601233B1 (en) | 2017-03-27 | 2024-08-14 | Hydro-Québec | Salts for use in electrolyte compositions or as electrode additives |
| CN107037148B (zh) * | 2017-04-07 | 2019-11-19 | 上海药明康德新药开发有限公司 | 卤泛曲林的高效液相检测方法 |
| JOP20190278A1 (ar) | 2017-05-31 | 2019-11-28 | Novartis Ag | مركبات 5، 6-ثنائية الحلقة مندمجة وتركيبات لعلاج الأمراض الطفيلية |
| US11628593B2 (en) | 2017-10-02 | 2023-04-18 | Dal-Tile, Llc | Method for manufacturing an engineered stone and an engineered stone |
| PE20211275A1 (es) * | 2018-07-09 | 2021-07-19 | Boehringer Ingelheim Animal Health Usa Inc | Compuestos heterociclicos antihelminticos |
| GB201811695D0 (en) * | 2018-07-17 | 2018-08-29 | Salvensis | Compounds for use in the treatment of fascioliasis |
| AR117788A1 (es) * | 2019-01-14 | 2021-08-25 | Pi Industries Ltd | Compuestos de fenilamidina 3-sustituida, preparación y uso |
| KR20220002890A (ko) | 2019-03-19 | 2022-01-07 | 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 | 구충성 아자-벤조티오펜 및 아자-벤조푸란 화합물 |
| EP3980414A1 (en) * | 2019-06-07 | 2022-04-13 | Elanco Tiergesundheit AG | Bicyclic derivatives for treating endoparasites |
| RU2019123849A (ru) * | 2019-07-29 | 2021-02-01 | Дзе Брихэм Энд Уимен`З Хоспитал, Инк. | Ингибиторы фактора ингибирования миграции макрофагов |
| MX2022015038A (es) | 2020-05-29 | 2023-01-04 | Boehringer Ingelheim Animal Health Usa Inc | Compuestos heterociclicos como anthelminticos. |
| WO2023275590A1 (en) | 2021-06-29 | 2023-01-05 | Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. | Detection of phosphoinositides in blood cells as a biomarker for alpha synuclein associated pathologies and a method of treatment of parkinson's disease and the related neurodegenerations |
| EP4413000A1 (en) | 2021-10-04 | 2024-08-14 | FoRx Therapeutics AG | N,n-dimethyl-4-(7-(n-(1-methylcyclopropyl)sulfamoyl)-imidazo[1,5-a]pyridin-5-yl)piperazine-1-carboxamide derivatives and the corresponding pyrazolo[1,5-a]pyridine derivatives as parg inhibitors for the treatment of cancer |
| PE20250675A1 (es) | 2021-11-01 | 2025-03-04 | Boehringer Ingelheim Vetmedica Gmbh | Compuestos de pirrolopiridazina como antihelminticos |
| CA3181279A1 (en) * | 2022-03-24 | 2023-09-24 | Bloom Energy Corporation | Fuel cell stack assembly including heat sink inserts |
| US12338188B2 (en) | 2022-06-30 | 2025-06-24 | Dal-Tile, Llc | Method for manufacturing a decorative element comprising an engineered stone and a decorative element comprising an engineered stone |
| US12358305B2 (en) | 2022-06-30 | 2025-07-15 | Dal-Tile, Llc | Method for manufacturing a decorative element comprising an engineered stone and a decorative element comprising an engineered stone |
| WO2024006974A2 (en) * | 2022-07-01 | 2024-01-04 | The Scripps Research Institute | Antimalarial compounds |
| US20240124450A1 (en) | 2022-09-21 | 2024-04-18 | Pfizer Inc. | Novel SIK Inhibitors |
| WO2024196989A1 (en) * | 2023-03-20 | 2024-09-26 | University Of Central Florida Research Foundation, Inc. | Anti-malarial therapy |
| AR132354A1 (es) * | 2023-04-13 | 2025-06-18 | Syngenta Crop Protection Ag | Derivados de pirazolo[1,5-a]piridina |
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-
2013
- 2013-11-18 ES ES13795977.1T patent/ES2655030T3/es active Active
- 2013-11-18 WO PCT/US2013/070601 patent/WO2014078802A1/en not_active Ceased
- 2013-11-18 SI SI201330889T patent/SI2925757T1/en unknown
- 2013-11-18 HR HRP20171998TT patent/HRP20171998T1/hr unknown
- 2013-11-18 ME MEP-2017-266A patent/ME03042B/me unknown
- 2013-11-18 US US14/443,609 patent/US9556169B2/en not_active Expired - Fee Related
- 2013-11-18 RS RS20171296A patent/RS56720B1/sr unknown
- 2013-11-18 PT PT137959771T patent/PT2925757T/pt unknown
- 2013-11-18 DK DK13795977.1T patent/DK2925757T3/en active
- 2013-11-18 EP EP13795977.1A patent/EP2925757B1/en active Active
- 2013-11-18 CN CN201380070822.0A patent/CN105164124B/zh not_active Expired - Fee Related
- 2013-11-18 TW TW102141950A patent/TWI600654B/zh not_active IP Right Cessation
- 2013-11-18 HU HUE13795977A patent/HUE037600T2/hu unknown
- 2013-11-18 JP JP2015542882A patent/JP6298472B2/ja not_active Expired - Fee Related
- 2013-11-18 LT LTEP13795977.1T patent/LT2925757T/lt unknown
- 2013-11-18 PL PL13795977T patent/PL2925757T3/pl unknown
- 2013-11-19 UY UY0001035146A patent/UY35146A/es unknown
- 2013-11-19 AR ARP130104250A patent/AR093532A1/es unknown
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2016
- 2016-07-26 US US15/220,149 patent/US9926314B2/en not_active Expired - Fee Related
-
2018
- 2018-01-03 CY CY20181100008T patent/CY1119727T1/el unknown
- 2018-02-06 US US15/889,578 patent/US20180230145A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US9926314B2 (en) | 2018-03-27 |
| SI2925757T1 (en) | 2018-01-31 |
| PL2925757T3 (pl) | 2018-06-29 |
| US20150344471A1 (en) | 2015-12-03 |
| US9556169B2 (en) | 2017-01-31 |
| HRP20171998T1 (hr) | 2018-02-09 |
| JP6298472B2 (ja) | 2018-03-20 |
| DK2925757T3 (en) | 2018-01-15 |
| JP2016505529A (ja) | 2016-02-25 |
| UY35146A (es) | 2014-06-30 |
| TW201429967A (zh) | 2014-08-01 |
| EP2925757B1 (en) | 2017-10-04 |
| AR093532A1 (es) | 2015-06-10 |
| CN105164124A (zh) | 2015-12-16 |
| EP2925757A1 (en) | 2015-10-07 |
| LT2925757T (lt) | 2017-12-27 |
| ME03042B (me) | 2018-10-20 |
| US20180230145A1 (en) | 2018-08-16 |
| WO2014078802A1 (en) | 2014-05-22 |
| TWI600654B (zh) | 2017-10-01 |
| CY1119727T1 (el) | 2018-06-27 |
| CN105164124B (zh) | 2017-03-15 |
| US20160333012A1 (en) | 2016-11-17 |
| HUE037600T2 (hu) | 2018-09-28 |
| RS56720B1 (sr) | 2018-03-30 |
| ES2655030T3 (es) | 2018-02-16 |
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