PL2668163T3 - Sposób wytwarzania 6-podstawionych 4-amino-3-chloro-5-fluoro-pikolinianów - Google Patents

Sposób wytwarzania 6-podstawionych 4-amino-3-chloro-5-fluoro-pikolinianów

Info

Publication number: PL2668163T3
Authority: PL; Poland
Prior art keywords: picolinates; fluoro; chloro; amino; substituted
Prior art date: 2011-01-25

Application number

PL12739865T

Other languages

English (en)

Inventor

Kim E Arndt

James M Renga

Yuanming Zhu

Gregory T Whiteker

Christian T Lowe

Original Assignee

Dow Agrosciences Llc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2011-01-25

Filing date

2012-01-24

Publication date

2017-10-31

2012-01-24 Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc

2017-10-31 Publication of PL2668163T3 publication Critical patent/PL2668163T3/pl

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/84—Nitriles
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/803—Processes of preparation
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Dentistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Plant Pathology (AREA)
General Health & Medical Sciences (AREA)
Wood Science & Technology (AREA)
Zoology (AREA)
Environmental Sciences (AREA)
Pest Control & Pesticides (AREA)
Agronomy & Crop Science (AREA)
Pyridine Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

PL12739865T 2011-01-25 2012-01-24 Sposób wytwarzania 6-podstawionych 4-amino-3-chloro-5-fluoro-pikolinianów PL2668163T3 (pl)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US201161435966P	2011-01-25	2011-01-25
PCT/US2012/022285 WO2012103041A2 (en)	2011-01-25	2012-01-24	Process for the preparation of 4-amino-3-chloro-5-fluoro-6-(substituted) picolinates
EP12739865.9A EP2668163B1 (en)	2011-01-25	2012-01-24	Process for the preparation of 6-substituted 4-amino-3-chloro-5-fluoro-picolinates

Publications (1)

Publication Number	Publication Date
PL2668163T3 true PL2668163T3 (pl)	2017-10-31

Family

ID=46544648

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL12739865T PL2668163T3 (pl)	2011-01-25	2012-01-24	Sposób wytwarzania 6-podstawionych 4-amino-3-chloro-5-fluoro-pikolinianów

Country Status (20)

Country	Link
US (3)	US20120190857A1 (pl)
EP (1)	EP2668163B1 (pl)
JP (1)	JP5739018B2 (pl)
KR (1)	KR101537879B1 (pl)
CN (2)	CN104788368B (pl)
AR (1)	AR085022A1 (pl)
AU (1)	AU2012209277B2 (pl)
BR (2)	BR112013019025A2 (pl)
CA (1)	CA2825475C (pl)
CO (1)	CO6731125A2 (pl)
HK (2)	HK1199245A1 (pl)
IL (1)	IL227646A (pl)
MX (1)	MX342328B (pl)
PL (1)	PL2668163T3 (pl)
RU (1)	RU2545021C1 (pl)
SG (1)	SG192093A1 (pl)
TW (1)	TWI592401B (pl)
UA (1)	UA106945C2 (pl)
WO (1)	WO2012103041A2 (pl)
ZA (1)	ZA201305577B (pl)

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* Cited by examiner, † Cited by third party
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TWI592401B (zh)	2011-01-25	2017-07-21	陶氏農業科學公司	用於製備４－胺基－３－氯－５－氟－６－（經取代的）吡啶甲酸酯的方法（一）
US9113629B2 (en)	2013-03-15	2015-08-25	Dow Agrosciences Llc	4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides
JP6543241B2 (ja)	2013-03-15	2019-07-10	ダウアグロサイエンシィズエルエルシー	４−アミノ−６−（複素環式）ピコリネートおよび６−アミノ−２−（複素環式）ピリミジン−４−カルボキシレートならびに除草剤としてのそれらの使用
WO2014150809A1 (en)	2013-03-15	2014-09-25	Dow Agrosciences Llc	Novel 4-aminopyridine and 6-aminopyrimidine carboxylates as herbicides
US9637505B2 (en)	2013-03-15	2017-05-02	Dow Agrosciences Llc	4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides
BR102014028162A2 (pt)	2013-11-12	2015-09-08	Dow Agrosciences Llc	processo para fluoração de compostos
TW201609651A (zh)	2013-11-12	2016-03-16	陶氏農業科學公司	用於氟化化合物之過程（一）
BR102014028164A2 (pt) *	2013-11-12	2015-09-08	Dow Agrosciences Llc	processo para fluoração de compostos
TWI726900B (zh)	2015-08-04	2021-05-11	美商陶氏農業科學公司	用於氟化化合物之過程
CN109415319A (zh) *	2016-05-19	2019-03-01	美国陶氏益农公司	通过直接苏楚基偶联合成芳基羧酸酯
CN107954925A (zh) *	2016-10-18	2018-04-24	内蒙古佳瑞米精细化工有限公司	一种2,3-二氯-5-三氟甲基吡啶前杂的去除方法
CN113015721B (zh)	2018-09-19	2025-07-25	科迪华农业科技有限责任公司	毒莠定卤素类似物的制备
BR112022018513A2 (pt)	2020-03-18	2022-11-01	Corteva Agriscience Llc	Síntese melhorada de 6-aril-4-aminopicolinatos
CN115279737A (zh) *	2020-03-18	2022-11-01	科迪华农业科技有限责任公司	4-氨基-6-(杂环)吡啶甲酸酯的改进合成

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US3285925A (en) *	1962-03-06	1966-11-15	Dow Chemical Co	Amino-trichloropicolinic acid compounds
US3803159A (en) *	1967-12-26	1974-04-09	Dow Chemical Co	Fluorine containing cyanopyridines
US3629424A (en) *	1967-12-26	1971-12-21	Dow Chemical Co	Cyanofluoropyridines and fungicidal compositions and methods for using the same
US4336384A (en) *	1981-04-23	1982-06-22	The Dow Chemical Company	Preparation of 4-amino-3,5,6-trichloropicolinic acid
US5807804A (en) *	1996-02-22	1998-09-15	American Cyanamid Company	Substituted pyridine herbicidal agents
FR2803592A1 (fr) *	2000-01-06	2001-07-13	Aventis Cropscience Sa	Nouveaux derives de l'acide 3-hydroxypicolinique, leur procede de preparation et compositions fongicides les contenant.
US6297197B1 (en)	2000-01-14	2001-10-02	Dow Agrosciences Llc	4-aminopicolinates and their use as herbicides
EP1246802B1 (en) *	2000-01-14	2007-03-14	Dow Agrosciences LLC	4-aminopicolinates and their use as herbicides
AR037228A1 (es)	2001-07-30	2004-11-03	Dow Agrosciences Llc	Compuestos del acido 6-(aril o heteroaril)-4-aminopicolinico, composicion herbicida que los comprende y metodo para controlar vegetacion no deseada
UA82358C2 (uk) *	2003-04-02	2008-04-10	Дау Агросайенсиз Ллс	6-алкіл або алкеніл-4-амінопіколінати гербіцидна композиція, спосіб боротьби з небажаною рослинністю
US7314849B2 (en)	2006-01-13	2008-01-01	Dow Agrosciences Llc	6-(poly-substituted aryl)-4-aminopicolinates and their use as herbicides
ES2410504T3 (es) *	2007-10-02	2013-07-02	Dow Agrosciences, Llc	Ácidos 4-amino-picolínicos sustituidos y su uso como herbicidas
US8252938B2 (en) *	2009-06-08	2012-08-28	Dow Agrosciences, Llc.	Process for the preparation of 6-(aryl)-4-aminopicolinates
GB0910766D0 (en) *	2009-06-22	2009-08-05	Syngenta Ltd	Chemical compounds
GB201008290D0 (en) *	2010-05-18	2010-06-30	Syngenta Ltd	Chemical compounds
TWI592401B (zh)	2011-01-25	2017-07-21	陶氏農業科學公司	用於製備４－胺基－３－氯－５－氟－６－（經取代的）吡啶甲酸酯的方法（一）

2012
- 2012-01-20 TW TW101102582A patent/TWI592401B/zh not_active IP Right Cessation
- 2012-01-24 BR BR112013019025A patent/BR112013019025A2/pt not_active Application Discontinuation
- 2012-01-24 HK HK14112715.3A patent/HK1199245A1/xx unknown
- 2012-01-24 JP JP2013551275A patent/JP5739018B2/ja not_active Expired - Fee Related
- 2012-01-24 CA CA2825475A patent/CA2825475C/en not_active Expired - Fee Related
- 2012-01-24 WO PCT/US2012/022285 patent/WO2012103041A2/en not_active Ceased
- 2012-01-24 CN CN201510105205.0A patent/CN104788368B/zh not_active Expired - Fee Related
- 2012-01-24 US US13/356,669 patent/US20120190857A1/en not_active Abandoned
- 2012-01-24 MX MX2013008603A patent/MX342328B/es active IP Right Grant
- 2012-01-24 KR KR1020137021995A patent/KR101537879B1/ko not_active Expired - Fee Related
- 2012-01-24 SG SG2013056023A patent/SG192093A1/en unknown
- 2012-01-24 PL PL12739865T patent/PL2668163T3/pl unknown
- 2012-01-24 BR BRBR102012001636-2A patent/BR102012001636A2/pt not_active Application Discontinuation
- 2012-01-24 AR ARP120100234A patent/AR085022A1/es unknown
- 2012-01-24 RU RU2013139300/04A patent/RU2545021C1/ru not_active IP Right Cessation
- 2012-01-24 EP EP12739865.9A patent/EP2668163B1/en not_active Not-in-force
- 2012-01-24 UA UAA201310403A patent/UA106945C2/uk unknown
- 2012-01-24 AU AU2012209277A patent/AU2012209277B2/en not_active Ceased
- 2012-01-24 CN CN201280014336.2A patent/CN103874685B/zh not_active Expired - Fee Related
2013
- 2013-07-23 ZA ZA2013/05577A patent/ZA201305577B/en unknown
- 2013-07-24 IL IL227646A patent/IL227646A/en active IP Right Grant
- 2013-07-24 CO CO13175298A patent/CO6731125A2/es unknown
2014
- 2014-02-04 US US14/171,791 patent/US9067890B2/en not_active Expired - Fee Related
- 2014-12-18 HK HK16100734.3A patent/HK1213875A1/zh unknown
2015
- 2015-06-09 US US14/734,347 patent/US9452984B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
UA106945C2 (uk)	2014-10-27
ZA201305577B (en)	2014-09-25
JP5739018B2 (ja)	2015-06-24
EP2668163B1 (en)	2017-05-10
AU2012209277B2 (en)	2015-09-17
KR101537879B1 (ko)	2015-07-17
CO6731125A2 (es)	2013-08-15
TWI592401B (zh)	2017-07-21
IL227646A (en)	2016-10-31
EP2668163A4 (en)	2015-03-11
US9452984B2 (en)	2016-09-27
RU2013139300A (ru)	2015-04-10
MX2013008603A (es)	2013-08-12
US9067890B2 (en)	2015-06-30
BR112013019025A2 (pt)	2016-07-12
CA2825475A1 (en)	2012-08-02
MX342328B (es)	2016-09-22
US20140142317A1 (en)	2014-05-22
HK1213875A1 (zh)	2016-07-15
IL227646A0 (en)	2013-09-30
BR102012001636A2 (pt)	2015-07-28
AR085022A1 (es)	2013-08-07
TW201309649A (zh)	2013-03-01
EP2668163A2 (en)	2013-12-04
HK1199245A1 (en)	2015-06-26
SG192093A1 (en)	2013-08-30
CA2825475C (en)	2017-08-22
WO2012103041A2 (en)	2012-08-02
RU2545021C1 (ru)	2015-03-27
CN104788368A (zh)	2015-07-22
CN103874685A (zh)	2014-06-18
WO2012103041A3 (en)	2014-05-01
CN104788368B (zh)	2017-09-26
JP2014515725A (ja)	2014-07-03
CN103874685B (zh)	2016-02-03
KR20130121950A (ko)	2013-11-06
US20150274669A1 (en)	2015-10-01
US20120190857A1 (en)	2012-07-26

Publication	Publication Date	Title
IL227648A0 (en)	2013-09-30	Process for preparing 4-amino-5-fluoro-3-halo-6-(converted) picolinates
ZA201305972B (en)	2014-04-30	Method for the preparation of biphephos
PL2668163T3 (pl)	2017-10-31	Sposób wytwarzania 6-podstawionych 4-amino-3-chloro-5-fluoro-pikolinianów
ZA201305582B (en)	2014-09-25	Process for the preparation of 4-amino-5-fluoro-3-halo-6-(sunstituted)picolinates
SG11201400939YA (en)	2014-07-30	Process for the preparation of methoxymelonal
IL232418A (en)	2016-10-31	Process for preparation of cell-c-aryl glucosides
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ZA201405824B (en)	2015-11-25	Process for the preparation of substituted phenylpropanones
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HUP1200675A2 (en)	2014-05-28	Process for the preparation of pyrimidinyl-piperazines