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PL1778686T3 - Pochodne triazolopirydynylosulfanylowe jako inhibitory kinazy MAP P38 - Google Patents

Pochodne triazolopirydynylosulfanylowe jako inhibitory kinazy MAP P38

Info

Publication number
PL1778686T3
PL1778686T3 PL05772546T PL05772546T PL1778686T3 PL 1778686 T3 PL1778686 T3 PL 1778686T3 PL 05772546 T PL05772546 T PL 05772546T PL 05772546 T PL05772546 T PL 05772546T PL 1778686 T3 PL1778686 T3 PL 1778686T3
Authority
PL
Poland
Prior art keywords
kinase inhibitors
map kinase
triazolopyridinylsulfanyl
derivatives
triazolopyridinylsulfanyl derivatives
Prior art date
Application number
PL05772546T
Other languages
English (en)
Inventor
John Paul Mathias
David Simon Millan
Russell Andrew Lewthwaite
Christopher Phillips
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0418015A external-priority patent/GB0418015D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of PL1778686T3 publication Critical patent/PL1778686T3/pl

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    • C07—ORGANIC CHEMISTRY
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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PL05772546T 2004-08-12 2005-08-09 Pochodne triazolopirydynylosulfanylowe jako inhibitory kinazy MAP P38 PL1778686T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0418015A GB0418015D0 (en) 2004-08-12 2004-08-12 New compounds
US69155905P 2005-06-17 2005-06-17
EP05772546A EP1778686B9 (en) 2004-08-12 2005-08-09 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors
PCT/IB2005/002574 WO2006018718A2 (en) 2004-08-12 2005-08-09 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors

Publications (1)

Publication Number Publication Date
PL1778686T3 true PL1778686T3 (pl) 2009-04-30

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
PL05772546T PL1778686T3 (pl) 2004-08-12 2005-08-09 Pochodne triazolopirydynylosulfanylowe jako inhibitory kinazy MAP P38

Country Status (34)

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US (2) US7511057B2 (pl)
EP (1) EP1778686B9 (pl)
JP (1) JP4084836B2 (pl)
AP (1) AP2326A (pl)
AR (1) AR050692A1 (pl)
AT (1) ATE412652T1 (pl)
AU (1) AU2005273612B2 (pl)
BR (1) BRPI0514255A (pl)
CA (1) CA2576297C (pl)
CR (1) CR8918A (pl)
CU (1) CU23497A3 (pl)
CY (1) CY1108788T1 (pl)
DE (1) DE602005010714D1 (pl)
DK (1) DK1778686T3 (pl)
EA (1) EA012119B1 (pl)
EC (1) ECSP077232A (pl)
ES (1) ES2314690T3 (pl)
GE (1) GEP20104973B (pl)
GT (1) GT200500218A (pl)
HN (1) HN2005000418A (pl)
HR (1) HRP20080608T3 (pl)
IL (1) IL181047A (pl)
MA (1) MA28798B1 (pl)
MX (1) MX2007001759A (pl)
MY (1) MY140021A (pl)
NL (1) NL1029726C2 (pl)
NO (1) NO339320B1 (pl)
NZ (1) NZ552868A (pl)
PL (1) PL1778686T3 (pl)
PT (1) PT1778686E (pl)
SI (1) SI1778686T1 (pl)
SV (1) SV2006002193A (pl)
TN (1) TNSN07050A1 (pl)
WO (1) WO2006018718A2 (pl)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7579360B2 (en) * 2005-06-09 2009-08-25 Bristol-Myers Squibb Company Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors
US7572807B2 (en) * 2005-06-09 2009-08-11 Bristol-Myers Squibb Company Heteroaryl 11-beta-hydroxysteroid dehydrogenase type I inhibitors
EP1984363A1 (en) * 2006-02-09 2008-10-29 Pfizer Limited Triazolopyridine compounds
JP5244369B2 (ja) * 2006-11-10 2013-07-24 富士フイルム株式会社 ５−アミノピラゾール誘導体の製造方法、アゾ色素
EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
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