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PL1697326T3 - Krystaliczna postać chinoliny i sposób jej wytwarzania - Google Patents

Krystaliczna postać chinoliny i sposób jej wytwarzania

Info

Publication number
PL1697326T3
PL1697326T3 PL04807807T PL04807807T PL1697326T3 PL 1697326 T3 PL1697326 T3 PL 1697326T3 PL 04807807 T PL04807807 T PL 04807807T PL 04807807 T PL04807807 T PL 04807807T PL 1697326 T3 PL1697326 T3 PL 1697326T3
Authority
PL
Poland
Prior art keywords
crystal form
production
quinoline compound
stability
drug substance
Prior art date
Application number
PL04807807T
Other languages
English (en)
Inventor
Yoshio Ohara
Yasutaka Takada
Hiroo Matsumoto
Akihiro Yoshida
Original Assignee
Nissan Chemical Ind Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34736450&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL1697326(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Nissan Chemical Ind Ltd filed Critical Nissan Chemical Ind Ltd
Publication of PL1697326T3 publication Critical patent/PL1697326T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14Radicals substituted by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL04807807T 2003-12-26 2004-12-17 Krystaliczna postać chinoliny i sposób jej wytwarzania PL1697326T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2003431788 2003-12-26
PCT/JP2004/019451 WO2005063711A1 (en) 2003-12-26 2004-12-17 Crystal form of quinoline compound and process for its production
EP04807807A EP1697326B1 (en) 2003-12-26 2004-12-17 Crystal form of quinoline compound and process for its production

Publications (1)

Publication Number Publication Date
PL1697326T3 true PL1697326T3 (pl) 2011-12-30

Family

ID=34736450

Family Applications (1)

Application Number Title Priority Date Filing Date
PL04807807T PL1697326T3 (pl) 2003-12-26 2004-12-17 Krystaliczna postać chinoliny i sposób jej wytwarzania

Country Status (21)

Country Link
US (19) US20070112024A1 (pl)
EP (1) EP1697326B1 (pl)
JP (7) JP5186108B2 (pl)
KR (11) KR20070001910A (pl)
CN (2) CN102321019B (pl)
AT (1) ATE518835T1 (pl)
AU (2) AU2004309241A1 (pl)
CA (1) CA2551050C (pl)
CY (1) CY1112464T1 (pl)
DK (1) DK1697326T3 (pl)
ES (1) ES2367172T3 (pl)
IL (1) IL176470A (pl)
MX (1) MX338019B (pl)
NZ (1) NZ548041A (pl)
PL (1) PL1697326T3 (pl)
PT (1) PT1697326E (pl)
RU (1) RU2370489C2 (pl)
SI (1) SI1697326T1 (pl)
TW (1) TWI328006B (pl)
WO (1) WO2005063711A1 (pl)
ZA (1) ZA200605658B (pl)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2513837A1 (en) 2003-02-12 2004-08-26 Paul Adriaan Van Der Schaaf Crystalline forms of pitavastatin calcium
TWI328006B (en) 2003-12-26 2010-08-01 Nissan Chemical Ind Ltd Crystal form of quinoline compound and process for its production
US7801272B2 (en) * 2007-09-28 2010-09-21 Rigaku Corporation X-ray diffraction apparatus and X-ray diffraction method
WO2011089623A2 (en) * 2010-01-20 2011-07-28 Cadila Healthcare Limited Process for preparing pitavastatin and pharmaceutically acceptable salts thereof
KR101158517B1 (ko) 2010-04-29 2012-06-21 동방에프티엘(주) 고 순도 피타바스타틴 칼슘염 결정형 a의 제조방법
WO2012025939A1 (en) 2010-08-25 2012-03-01 Cadila Healthcare Limited Pitavastatin calcium and process for its preparation
EP3178812A1 (en) 2010-11-12 2017-06-14 Hetero Research Foundation Novel polymorphs of pitavastatin calcium
RU2452939C1 (ru) * 2011-01-18 2012-06-10 Закрытое акционерное общество "Научные приборы" Рентгенодифракционный способ идентификации партий фармацевтической продукции
ITMI20111475A1 (it) * 2011-08-02 2013-02-03 Dipharma Francis Srl Forme cristalline di pitavastatina sale di calcio
PT2751081T (pt) * 2011-09-12 2017-04-04 D O O Farma Grs Forma polimórfica de pitavastatina cálcica
WO2013098773A1 (en) * 2011-12-28 2013-07-04 Dr. Reddy's Laboratories Limited Crystalline forms of pitavastatin calcium
US20150164809A1 (en) * 2012-08-08 2015-06-18 Kowa Company, Ltd. Medicine
IN2015DN03012A (pl) * 2012-09-27 2015-10-02 Nissan Chemical Ind Ltd
JP2014034574A (ja) * 2013-01-25 2014-02-24 Kowa Company Ltd 医薬
BR112015022849B1 (pt) 2013-03-15 2020-02-18 Asieris Pharmaceutical Technologies Co., Ltd. Sais de adição de base de nitroxolina, usos e processo para preparação dos mesmos, bem como seu cristal, composição farmacêutica e processo para preparação da mesma
CN105213319A (zh) * 2015-09-17 2016-01-06 青岛华之草医药科技有限公司 一种降血脂药物匹伐他汀钙组合物干混悬剂
JP2016222714A (ja) * 2016-09-20 2016-12-28 興和株式会社 医薬
WO2021181360A1 (en) * 2020-03-13 2021-09-16 Cadila Healthcare Limited Novel salts of quinolone compounds
KR20230159487A (ko) * 2021-03-19 2023-11-21 자이두스 라이프사이언시즈 리미티드 고체 형태의 퀴놀론 화합물 및 이의 제조 방법

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3175944A (en) * 1956-06-18 1965-03-30 Upjohn Co Dihydronovobiocin and derivatives thereof
IL63968A (en) 1980-10-01 1985-10-31 Glaxo Group Ltd Form 2 ranitidine hydrochloride,its preparation and pharmaceutical compositions containing it
GB8320521D0 (en) * 1983-07-29 1983-09-01 Glaxo Group Ltd Chemical process
JPS61171460A (ja) * 1985-01-23 1986-08-02 Dainippon Pharmaceut Co Ltd 塩酸メクロフエノキサ−ト1型結晶の製造法
JP2569746B2 (ja) * 1987-08-20 1997-01-08 日産化学工業株式会社 キノリン系メバロノラクトン類
JP2877366B2 (ja) 1988-08-25 1999-03-31 協和醗酵工業株式会社 結晶状l−アスコルビン酸−2−リン酸ナトリウム塩の製造法
JP3528186B2 (ja) * 1991-06-24 2004-05-17 日産化学工業株式会社 光学活性キノリンメバロン酸のジアステレオマー塩
JPH0613526A (ja) 1992-06-25 1994-01-21 Seiko Epson Corp 半導体装置用リードフレーム及びその製造方法
JP2575590B2 (ja) * 1992-07-31 1997-01-29 塩野義製薬株式会社 トリアゾリルチオメチルチオセファロスポリン塩酸塩およびその水和物結晶ならびにそれらの製法
FR2694558B1 (fr) 1992-08-05 1994-10-28 Sanofi Elf Monohydrate du sel disodique de l'acide 4-chlorophénylthiométhylène bisphosphonique, sa préparation, les compositions pharmaceutiques en contenant.
DE4235133A1 (de) 1992-10-19 1994-04-21 Bayer Ag Kristallines (R)-(-)-2-Cycloheptyl-N-methylsulfonyl-[4-(2-chinolinyl-methoxy)-phenyl]-acetamid
JP3623531B2 (ja) 1993-06-07 2005-02-23 ビーエーエスエフ アクチェンゲゼルシャフト 結晶質l−アスコルビン酸−2−燐酸エステルマグネシウム塩の製造法
JP3558684B2 (ja) * 1994-06-28 2004-08-25 塩野義製薬株式会社 ピロリジルチオカルバペネム誘導体の乾燥方法
CZ20012357A3 (cs) * 1999-01-14 2001-09-12 Nissan Chemical Industries, Ltd. Způsob přípravy chinolinkarbaldehydu
CA2450820C (en) * 2001-08-16 2011-03-15 Teva Pharmaceutical Industries Ltd. Processes for preparing calcium salt forms of statins
US6835838B2 (en) 2002-01-28 2004-12-28 Novartis Ag Process for the manufacture of organic compounds
CN1305853C (zh) * 2002-01-31 2007-03-21 诺瓦提斯公司 Hmg辅酶a还原酶抑制剂的制备方法
US6869970B2 (en) * 2002-02-04 2005-03-22 Novartis Ag Crystalline salt forms of valsartan
CA2482937A1 (en) * 2002-04-17 2003-10-23 Yamanouchi Pharmaceutical Co., Ltd. A novel crystal of anhydride of a quinoxalinedione derivative
CA2513837A1 (en) * 2003-02-12 2004-08-26 Paul Adriaan Van Der Schaaf Crystalline forms of pitavastatin calcium
TWI328006B (en) * 2003-12-26 2010-08-01 Nissan Chemical Ind Ltd Crystal form of quinoline compound and process for its production

Also Published As

Publication number Publication date
RU2006127044A (ru) 2008-02-10
AU2011213742A1 (en) 2011-09-08
US20150158816A1 (en) 2015-06-11
KR20160075844A (ko) 2016-06-29
US20230322679A1 (en) 2023-10-12
US20170226061A1 (en) 2017-08-10
US20110082298A1 (en) 2011-04-07
KR20170010111A (ko) 2017-01-25
US20190152916A1 (en) 2019-05-23
ATE518835T1 (de) 2011-08-15
CN102321019A (zh) 2012-01-18
CA2551050C (en) 2020-06-02
SI1697326T1 (sl) 2011-11-30
JP2018052988A (ja) 2018-04-05
JP2007516952A (ja) 2007-06-28
KR20200015826A (ko) 2020-02-12
EP1697326A1 (en) 2006-09-06
AU2004309241A1 (en) 2005-07-14
JP2016029102A (ja) 2016-03-03
US20090176987A1 (en) 2009-07-09
MX338019B (es) 2016-03-29
CA2551050A1 (en) 2005-07-14
JP2013136640A (ja) 2013-07-11
US20140206719A1 (en) 2014-07-24
HK1095328A1 (en) 2007-05-04
US20140058109A1 (en) 2014-02-27
US20110319624A1 (en) 2011-12-29
KR20110017936A (ko) 2011-02-22
AU2011213742C1 (en) 2017-04-06
US20130204000A1 (en) 2013-08-08
CN102321019B (zh) 2016-06-08
KR20190083674A (ko) 2019-07-12
US20240294476A1 (en) 2024-09-05
KR20130014643A (ko) 2013-02-07
JP2012072175A (ja) 2012-04-12
IL176470A0 (en) 2006-10-05
ES2367172T3 (es) 2011-10-31
AU2011213742B2 (en) 2014-05-15
WO2005063711A1 (en) 2005-07-14
DK1697326T3 (da) 2011-09-19
US20180297956A1 (en) 2018-10-18
KR20170098976A (ko) 2017-08-30
US20120245200A1 (en) 2012-09-27
KR20200130510A (ko) 2020-11-18
IL176470A (en) 2011-10-31
JP2017061536A (ja) 2017-03-30
JP5267643B2 (ja) 2013-08-21
US20200216395A1 (en) 2020-07-09
US20220177433A1 (en) 2022-06-09
JP2014205719A (ja) 2014-10-30
KR20070001910A (ko) 2007-01-04
US20180072676A1 (en) 2018-03-15
TW200530186A (en) 2005-09-16
RU2370489C2 (ru) 2009-10-20
TWI328006B (en) 2010-08-01
US20190367458A1 (en) 2019-12-05
CN1898211A (zh) 2007-01-17
KR20180132973A (ko) 2018-12-12
ZA200605658B (en) 2007-11-28
NZ548041A (en) 2010-04-30
KR20180040732A (ko) 2018-04-20
EP1697326B1 (en) 2011-08-03
US20070112024A1 (en) 2007-05-17
CY1112464T1 (el) 2015-12-09
PT1697326E (pt) 2011-09-12
JP5186108B2 (ja) 2013-04-17
US20210053923A1 (en) 2021-02-25

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