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DK1697326T3 - Krystalform af en quinolinforbindelse og fremgangsmåde til fremstilling deraf - Google Patents

Krystalform af en quinolinforbindelse og fremgangsmåde til fremstilling deraf

Info

Publication number
DK1697326T3
DK1697326T3 DK04807807.5T DK04807807T DK1697326T3 DK 1697326 T3 DK1697326 T3 DK 1697326T3 DK 04807807 T DK04807807 T DK 04807807T DK 1697326 T3 DK1697326 T3 DK 1697326T3
Authority
DK
Denmark
Prior art keywords
crystal form
preparation
quinoline compound
stability
drug substance
Prior art date
Application number
DK04807807.5T
Other languages
English (en)
Inventor
Yoshio Ohara
Yasutaka Takada
Hiroo Matsumoto
Akihiro Yoshida
Original Assignee
Nissan Chemical Ind Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34736450&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1697326(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Nissan Chemical Ind Ltd filed Critical Nissan Chemical Ind Ltd
Application granted granted Critical
Publication of DK1697326T3 publication Critical patent/DK1697326T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14Radicals substituted by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK04807807.5T 2003-12-26 2004-12-17 Krystalform af en quinolinforbindelse og fremgangsmåde til fremstilling deraf DK1697326T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2003431788 2003-12-26
PCT/JP2004/019451 WO2005063711A1 (en) 2003-12-26 2004-12-17 Crystal form of quinoline compound and process for its production

Publications (1)

Publication Number Publication Date
DK1697326T3 true DK1697326T3 (da) 2011-09-19

Family

ID=34736450

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04807807.5T DK1697326T3 (da) 2003-12-26 2004-12-17 Krystalform af en quinolinforbindelse og fremgangsmåde til fremstilling deraf

Country Status (21)

Country Link
US (19) US20070112024A1 (da)
EP (1) EP1697326B1 (da)
JP (7) JP5186108B2 (da)
KR (11) KR20200015826A (da)
CN (2) CN1898211A (da)
AT (1) ATE518835T1 (da)
AU (2) AU2004309241A1 (da)
CA (1) CA2551050C (da)
CY (1) CY1112464T1 (da)
DK (1) DK1697326T3 (da)
ES (1) ES2367172T3 (da)
IL (1) IL176470A (da)
MX (1) MX338019B (da)
NZ (1) NZ548041A (da)
PL (1) PL1697326T3 (da)
PT (1) PT1697326E (da)
RU (1) RU2370489C2 (da)
SI (1) SI1697326T1 (da)
TW (1) TWI328006B (da)
WO (1) WO2005063711A1 (da)
ZA (1) ZA200605658B (da)

Families Citing this family (19)

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EP3299359A1 (en) 2003-02-12 2018-03-28 Nissan Chemical Industries, Ltd. Crystalline and amorphous forms of pitavastatin hemicalcium salt
TWI328006B (en) 2003-12-26 2010-08-01 Nissan Chemical Ind Ltd Crystal form of quinoline compound and process for its production
US7801272B2 (en) * 2007-09-28 2010-09-21 Rigaku Corporation X-ray diffraction apparatus and X-ray diffraction method
WO2011089623A2 (en) 2010-01-20 2011-07-28 Cadila Healthcare Limited Process for preparing pitavastatin and pharmaceutically acceptable salts thereof
KR101158517B1 (ko) 2010-04-29 2012-06-21 동방에프티엘(주) 고 순도 피타바스타틴 칼슘염 결정형 a의 제조방법
US9034901B2 (en) 2010-08-25 2015-05-19 Cadila Healthcare Limited Pitavastatin calcium and process for its preparation
EP2638013A4 (en) 2010-11-12 2014-03-26 Hetero Research Foundation NEW POLYMORPHS OF CALCIUM PIVASTATIN
RU2452939C1 (ru) * 2011-01-18 2012-06-10 Закрытое акционерное общество "Научные приборы" Рентгенодифракционный способ идентификации партий фармацевтической продукции
ITMI20111475A1 (it) * 2011-08-02 2013-02-03 Dipharma Francis Srl Forme cristalline di pitavastatina sale di calcio
ES2620968T3 (es) 2011-09-12 2017-06-30 Farma Grs, D.O.O. Forma polimórfica de pitavastatina cálcica
WO2013098773A1 (en) * 2011-12-28 2013-07-04 Dr. Reddy's Laboratories Limited Crystalline forms of pitavastatin calcium
KR101461841B1 (ko) 2012-08-08 2014-11-13 코와 가부시키가이샤 의약
IN2015DN03012A (da) * 2012-09-27 2015-10-02 Nissan Chemical Ind Ltd
JP2014034574A (ja) * 2013-01-25 2014-02-24 Kowa Company Ltd 医薬
BR112015022849B1 (pt) * 2013-03-15 2020-02-18 Asieris Pharmaceutical Technologies Co., Ltd. Sais de adição de base de nitroxolina, usos e processo para preparação dos mesmos, bem como seu cristal, composição farmacêutica e processo para preparação da mesma
CN105213319A (zh) * 2015-09-17 2016-01-06 青岛华之草医药科技有限公司 一种降血脂药物匹伐他汀钙组合物干混悬剂
JP2016222714A (ja) * 2016-09-20 2016-12-28 興和株式会社 医薬
WO2021181360A1 (en) * 2020-03-13 2021-09-16 Cadila Healthcare Limited Novel salts of quinolone compounds
US20240300899A1 (en) * 2021-03-19 2024-09-12 Zydus Lifesciences Limited A quinolone compound in solid forms and processes for the preparation thereof

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JPS61171460A (ja) * 1985-01-23 1986-08-02 Dainippon Pharmaceut Co Ltd 塩酸メクロフエノキサ−ト1型結晶の製造法
JP2569746B2 (ja) * 1987-08-20 1997-01-08 日産化学工業株式会社 キノリン系メバロノラクトン類
JP2877366B2 (ja) 1988-08-25 1999-03-31 協和醗酵工業株式会社 結晶状l−アスコルビン酸−2−リン酸ナトリウム塩の製造法
JP3528186B2 (ja) * 1991-06-24 2004-05-17 日産化学工業株式会社 光学活性キノリンメバロン酸のジアステレオマー塩
JPH0613526A (ja) 1992-06-25 1994-01-21 Seiko Epson Corp 半導体装置用リードフレーム及びその製造方法
JP2575590B2 (ja) * 1992-07-31 1997-01-29 塩野義製薬株式会社 トリアゾリルチオメチルチオセファロスポリン塩酸塩およびその水和物結晶ならびにそれらの製法
FR2694558B1 (fr) 1992-08-05 1994-10-28 Sanofi Elf Monohydrate du sel disodique de l'acide 4-chlorophénylthiométhylène bisphosphonique, sa préparation, les compositions pharmaceutiques en contenant.
DE4235133A1 (de) 1992-10-19 1994-04-21 Bayer Ag Kristallines (R)-(-)-2-Cycloheptyl-N-methylsulfonyl-[4-(2-chinolinyl-methoxy)-phenyl]-acetamid
JP3623531B2 (ja) 1993-06-07 2005-02-23 ビーエーエスエフ アクチェンゲゼルシャフト 結晶質l−アスコルビン酸−2−燐酸エステルマグネシウム塩の製造法
JP3558684B2 (ja) * 1994-06-28 2004-08-25 塩野義製薬株式会社 ピロリジルチオカルバペネム誘導体の乾燥方法
CZ20012357A3 (cs) * 1999-01-14 2001-09-12 Nissan Chemical Industries, Ltd. Způsob přípravy chinolinkarbaldehydu
IL160077A0 (en) * 2001-08-16 2004-06-20 Teva Pharma Processes for preparing calcium salt forms of statins
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DE60326819D1 (de) * 2002-01-31 2009-05-07 Novartis Ag Verfahren zur herstellung von inhibitoren der hmg-coa-reduktase
US6869970B2 (en) * 2002-02-04 2005-03-22 Novartis Ag Crystalline salt forms of valsartan
US20050130978A1 (en) * 2002-04-17 2005-06-16 Masamichi Yuda Novel crystal of quinoxalinedione derivative anhydride
EP3299359A1 (en) * 2003-02-12 2018-03-28 Nissan Chemical Industries, Ltd. Crystalline and amorphous forms of pitavastatin hemicalcium salt
TWI328006B (en) 2003-12-26 2010-08-01 Nissan Chemical Ind Ltd Crystal form of quinoline compound and process for its production

Also Published As

Publication number Publication date
AU2011213742A1 (en) 2011-09-08
KR20110017936A (ko) 2011-02-22
WO2005063711A1 (en) 2005-07-14
US20210053923A1 (en) 2021-02-25
KR20200130510A (ko) 2020-11-18
RU2370489C2 (ru) 2009-10-20
US20140058109A1 (en) 2014-02-27
US20220177433A1 (en) 2022-06-09
AU2011213742C1 (en) 2017-04-06
AU2011213742B2 (en) 2014-05-15
JP2007516952A (ja) 2007-06-28
TWI328006B (en) 2010-08-01
EP1697326B1 (en) 2011-08-03
US20090176987A1 (en) 2009-07-09
US20240294476A1 (en) 2024-09-05
PL1697326T3 (pl) 2011-12-30
US20170226061A1 (en) 2017-08-10
ZA200605658B (en) 2007-11-28
CN102321019B (zh) 2016-06-08
KR20200015826A (ko) 2020-02-12
JP5186108B2 (ja) 2013-04-17
EP1697326A1 (en) 2006-09-06
IL176470A (en) 2011-10-31
US20230322679A1 (en) 2023-10-12
JP2017061536A (ja) 2017-03-30
JP2018052988A (ja) 2018-04-05
KR20160075844A (ko) 2016-06-29
KR20190083674A (ko) 2019-07-12
JP2012072175A (ja) 2012-04-12
KR20180132973A (ko) 2018-12-12
CN1898211A (zh) 2007-01-17
TW200530186A (en) 2005-09-16
KR20170098976A (ko) 2017-08-30
JP2013136640A (ja) 2013-07-11
PT1697326E (pt) 2011-09-12
KR20180040732A (ko) 2018-04-20
US20120245200A1 (en) 2012-09-27
US20190367458A1 (en) 2019-12-05
US20140206719A1 (en) 2014-07-24
KR20170010111A (ko) 2017-01-25
US20110319624A1 (en) 2011-12-29
RU2006127044A (ru) 2008-02-10
KR20070001910A (ko) 2007-01-04
CA2551050A1 (en) 2005-07-14
JP2016029102A (ja) 2016-03-03
US20130204000A1 (en) 2013-08-08
KR20130014643A (ko) 2013-02-07
CY1112464T1 (el) 2015-12-09
HK1095328A1 (en) 2007-05-04
US20110082298A1 (en) 2011-04-07
US20070112024A1 (en) 2007-05-17
NZ548041A (en) 2010-04-30
ES2367172T3 (es) 2011-10-31
ATE518835T1 (de) 2011-08-15
JP5267643B2 (ja) 2013-08-21
IL176470A0 (en) 2006-10-05
US20150158816A1 (en) 2015-06-11
US20200216395A1 (en) 2020-07-09
US20190152916A1 (en) 2019-05-23
US20180072676A1 (en) 2018-03-15
JP2014205719A (ja) 2014-10-30
CN102321019A (zh) 2012-01-18
US20180297956A1 (en) 2018-10-18
CA2551050C (en) 2020-06-02
AU2004309241A1 (en) 2005-07-14
SI1697326T1 (sl) 2011-11-30
MX338019B (es) 2016-03-29

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