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PE20070377A1 - Formulaciones liquidas para la administracion controlada de derivados de bencisoxazol - Google Patents

Formulaciones liquidas para la administracion controlada de derivados de bencisoxazol

Info

Publication number
PE20070377A1
PE20070377A1 PE2006000919A PE2006000919A PE20070377A1 PE 20070377 A1 PE20070377 A1 PE 20070377A1 PE 2006000919 A PE2006000919 A PE 2006000919A PE 2006000919 A PE2006000919 A PE 2006000919A PE 20070377 A1 PE20070377 A1 PE 20070377A1
Authority
PE
Peru
Prior art keywords
liquid formulations
controlled administration
liquid
benzisoxazole derivatives
derivative
Prior art date
Application number
PE2006000919A
Other languages
English (en)
Inventor
Noymi V Yam
Nipun Davar
Suneel K Gupta
Gayatri Sathyan
Original Assignee
Alza Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alza Corp filed Critical Alza Corp
Publication of PE20070377A1 publication Critical patent/PE20070377A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4891Coated capsules; Multilayered drug free capsule shells
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Psychiatry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

REFERIDA A UNA FORMA DE DOSIFICACION QUE COMPRENDE UNA ESTRUCTURA DE DOSIFICACION DE LIBERACION CONTROLADA Y UNA FORMULACION LIQUIDA CONTENIDA DENTRO DE LA ESTRUCTURA DE DOSIFICACION DE LIBERACION CONTROLADA, DONDE LA FORMULACION LIQUIDA COMPRENDE UN DERIVADO DE BENCISOXAZOL Y UN VEHICULO LIQUIDO. EL DERIVADO DE BENCISOXAZOL SE SELECCIONA DE PALIPERIDONA O RISPERIDONA Y SE ENCUENTRA EN UNA CANTIDAD DE ENTRE 0,1 MG A 20 MG; EL VEHICULO LIQUIDO COMPRENDE UN SOLVENTE LIPOFILICO, UN TENSOACTIVO O UN SOLVENTE HIDROFILICO. DICHA FORMA DE DOSIFICACION PRESENTA UNA BIODISPONIBILIDAD MEJORADA
PE2006000919A 2005-07-28 2006-07-31 Formulaciones liquidas para la administracion controlada de derivados de bencisoxazol PE20070377A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US70314305P 2005-07-28 2005-07-28

Publications (1)

Publication Number Publication Date
PE20070377A1 true PE20070377A1 (es) 2007-06-13

Family

ID=37450765

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2006000919A PE20070377A1 (es) 2005-07-28 2006-07-31 Formulaciones liquidas para la administracion controlada de derivados de bencisoxazol

Country Status (5)

Country Link
US (1) US20070026067A1 (es)
AR (1) AR055099A1 (es)
PE (1) PE20070377A1 (es)
UY (1) UY29701A1 (es)
WO (1) WO2007016388A2 (es)

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US20050208132A1 (en) * 2002-07-29 2005-09-22 Gayatri Sathyan Methods and dosage forms for reducing side effects of benzisozazole derivatives
HUE056937T2 (hu) 2006-02-03 2022-04-28 Opko Renal Llc A D-vitamin elégtelenség és hiány kezelése 25-hidroxivitamin D2-vel és 25-hidroxivitamin D3-mal
EP3357496B1 (en) 2006-06-21 2020-02-19 Opko Ireland Global Holdings, Ltd. Therapy using vitamin d repletion agent and vitamin d hormone replacement agent
CN104523707B (zh) 2007-04-25 2022-08-26 欧普科Ip 控股Ii 有限公司 包含维生素d化合物和蜡质载体的口服控释组合物
WO2009047644A2 (en) 2007-04-25 2009-04-16 Cytochroma Inc. Method of treating vitamin d insufficiency and deficiency
WO2008134523A1 (en) 2007-04-25 2008-11-06 Proventiv Therapeutics, Llc Method of safely and effectively treating and preventing secondary hyperparathyroidism in chronic kidney disease
KR101852042B1 (ko) 2008-04-02 2018-04-25 사이토크로마 인코포레이티드 비타민 d 결핍 및 관련 장애에 유용한 방법, 조성물, 용도 및 키트
EP2161019A1 (en) 2008-09-05 2010-03-10 KRKA, D.D., Novo Mesto Prolonged release multiparticulate pharmaceutical composition comprising paliperidone
CN101711752B (zh) * 2009-11-26 2011-09-21 中国科学院上海药物研究所 一种苯并异噁唑类衍生物的控释制剂及其制备方法
US9271939B2 (en) 2010-03-15 2016-03-01 Inventia Healthcare Private Limited Stabilized prolonged release pharmaceutical composition comprising atypical antipsychotic
WO2011123476A1 (en) 2010-03-29 2011-10-06 Cytochroma Inc. Methods and compositions for reducing parathyroid levels
KR101311920B1 (ko) 2010-12-21 2013-09-26 한국생명공학연구원 란타나이드 금속착체를 이용한 형광 나노입자 및 그 제조방법
KR101847947B1 (ko) 2013-03-15 2018-05-28 옵코 아이피 홀딩스 Ⅱ 인코포레이티드 안정화되고 변형된 비타민 d 방출 제형
US10220047B2 (en) 2014-08-07 2019-03-05 Opko Ireland Global Holdings, Ltd. Adjunctive therapy with 25-hydroxyvitamin D and articles therefor
EP3436026A1 (en) 2016-03-28 2019-02-06 OPKO Ireland Global Holdings, Ltd. Methods of vitamin d treatment
EP3466409B1 (en) * 2017-10-05 2023-06-07 Vianex S.A. Self-emulsifying compositions of weakly ionizable or non-ionizable active pharmaceutical ingredients

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Also Published As

Publication number Publication date
US20070026067A1 (en) 2007-02-01
AR055099A1 (es) 2007-08-08
UY29701A1 (es) 2006-12-29
WO2007016388A2 (en) 2007-02-08
WO2007016388A3 (en) 2007-08-16

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Legal Events

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FA Abandonment or withdrawal