[go: up one dir, main page]

PE20061077A1 - Composicion farmaceutica que comprende 7-terbutoxi-imino-metil-camptotecina - Google Patents

Composicion farmaceutica que comprende 7-terbutoxi-imino-metil-camptotecina

Info

Publication number
PE20061077A1
PE20061077A1 PE2005001353A PE2005001353A PE20061077A1 PE 20061077 A1 PE20061077 A1 PE 20061077A1 PE 2005001353 A PE2005001353 A PE 2005001353A PE 2005001353 A PE2005001353 A PE 2005001353A PE 20061077 A1 PE20061077 A1 PE 20061077A1
Authority
PE
Peru
Prior art keywords
composition
weight
terbutoxi
camptotechin
imino
Prior art date
Application number
PE2005001353A
Other languages
English (en)
Inventor
Isabel Ottinger
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35691476&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20061077(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PE20061077A1 publication Critical patent/PE20061077A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61JCONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
    • A61J3/00Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00Preparations for use in therapy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA QUE COMPRENDE: A) UN PRINCIPIO ACTIVO TAL COMO 7-TERBUTOXI-IMINO-METIL-CAMPTOTECINA EN UNA CANTIDAD COMPRENDIDA ENTRE 0.05% A 20% EN PESO DE LA COMPOSICION; B) UN AGENTE LIPOFILICO TALES COMO MONOGLICERIDOS Y DIGLICERIDOS DE ACIDOS GRASOS DE 8 A 10 ATOMOS DE CARBONO, CITRATO DE TRIETILO, ENTRE OTROS; EN UNA CANTIDAD COMPRENDIDA ENTRE 5% A 85% EN PESO DE LA COMPOSICION; C) UN TENSOACTIVO A BASE DE ACEITE DE RICINO HIDROGENADO CON POLIETILENGLICOL EN UNA CANTIDAD COMPRENDIDA ENTRE 5% A 90% EN PESO DE LA COMPOSICION; D) UN COMPONENTE HIDROFILICO TALES COMO PROPILENGLICOL, PEG 400, LACTATO DE ETILO, ENTRE OTROS, EN UNA CANTIDAD COMPRENDIDA ENTRE 5% A 60% EN PESO DE LA COMPOSICION; E) UN COSOLVENTE EN UNA CANTIDAD COMPRENDIDA ENTRE 0 A 20% EN PESO DE LA COMPOSICION Y F) UNO O MAS ADITIVOS TALES COMO ANTIOXIDANTES, AGENTES ANTIMICROBIANOS, ESTABILIZANTES, ENTRE OTROS. TAMBIEN SE REFIERE A UN PROCESO DE PREPARACION. DICHA COMPOSICION ES UTIL EN EL TRATAMIENTO DE ENFERMEDADES PROLIFERATIVAS TAL COMO EL CANCER
PE2005001353A 2004-11-19 2005-11-17 Composicion farmaceutica que comprende 7-terbutoxi-imino-metil-camptotecina PE20061077A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US62975704P 2004-11-19 2004-11-19

Publications (1)

Publication Number Publication Date
PE20061077A1 true PE20061077A1 (es) 2006-11-13

Family

ID=35691476

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2005001353A PE20061077A1 (es) 2004-11-19 2005-11-17 Composicion farmaceutica que comprende 7-terbutoxi-imino-metil-camptotecina

Country Status (28)

Country Link
US (1) US8518961B2 (es)
EP (1) EP1814520B1 (es)
JP (1) JP4982378B2 (es)
KR (1) KR101283840B1 (es)
CN (1) CN101056619A (es)
AR (1) AR052033A1 (es)
AU (1) AU2005306018B2 (es)
BR (1) BRPI0518448A2 (es)
CA (1) CA2584343C (es)
DK (1) DK1814520T3 (es)
ES (1) ES2572133T3 (es)
GT (1) GT200500310A (es)
HR (1) HRP20160446T1 (es)
HU (1) HUE027135T2 (es)
IL (1) IL182703A (es)
MA (1) MA29076B1 (es)
MX (1) MX2007005897A (es)
MY (1) MY148647A (es)
NO (1) NO342592B1 (es)
NZ (1) NZ554551A (es)
PE (1) PE20061077A1 (es)
PL (1) PL1814520T3 (es)
RU (3) RU2007122470A (es)
SI (1) SI1814520T1 (es)
TN (1) TNSN07193A1 (es)
TW (1) TWI368521B (es)
WO (1) WO2006053755A1 (es)
ZA (1) ZA200703148B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GT200500310A (es) 2004-11-19 2006-06-19 Compuestos organicos
SA06270147B1 (ar) 2005-06-09 2009-12-22 نوفارتيس ايه جي عملية لتخليق 5-(مثيل–1h–إيميدازول–1-يل )–3-(ثلاثي فلـورو مثيل)–بنزامـين
ITRM20050418A1 (it) * 2005-08-04 2007-02-05 Sigma Tau Ind Farmaceuti Sistemi terapeutici a rilascio immediato per il migliorato assorbimento orale di 7-[(e)-t-butilossimminometil] camptotecina.
JP2009504616A (ja) * 2005-08-10 2009-02-05 ノバルティス アクチエンゲゼルシャフト トポイソメラーゼI阻害剤、7−tert−ブトキシイミノメチルカンプトテシンの微粒子組成物
WO2008055146A2 (en) * 2006-10-31 2008-05-08 Wyeth Formulations of phospholipase enzyme inhibitors
US20100070052A1 (en) * 2008-08-19 2010-03-18 Robb Fujioka System and method for providing applications and peripherals to a fixed price component-based computing platform
MX340819B (es) 2010-06-29 2016-07-26 Poniard Pharmaceuticals Inc * Formulacion oral de inhibidores de quinasa.
EP2588476A4 (en) 2010-06-30 2014-07-23 Verastem Inc SYNTHESIS AND USE OF KINASE INHIBITORS
US12226412B2 (en) 2012-05-25 2025-02-18 Corcept Therapeutics, Inc. Heteroaryl-ketone fused azadecalin glucocorticoid receptor modulators
US8859774B2 (en) 2012-05-25 2014-10-14 Corcept Therapeutics, Inc. Heteroaryl-ketone fused azadecalin glucocorticoid receptor modulators
MX2021007322A (es) * 2018-12-19 2021-07-07 Corcept Therapeutics Inc Formulaciones farmaceuticas que contienen relacorilant, un compuesto de azadecalina fusionado con heteroaril-cetona.
CA3229030A1 (en) * 2021-09-05 2023-03-09 Yi-Wen Chu Formulations with enhanced sn-38 solubility and oral absorption
EP4577191A1 (en) * 2022-08-24 2025-07-02 Lyotropic Delivery Systems Ltd. Oral delivery of active compounds for treating glycogen storage diseases
AU2023355849A1 (en) 2022-10-06 2025-04-03 Corcept Therapeutics Incorporated Formulations of glucocorticoid receptor modulators
IL320512A (en) 2022-10-28 2025-06-01 Corcept Therapeutics Inc Amyotrophic lateral sclerosis treatments using desocorilant

Family Cites Families (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9113872D0 (en) 1991-06-27 1991-08-14 Sandoz Ag Improvements in or relating to organic compounds
JPH08504811A (ja) 1992-12-24 1996-05-28 ヘマジェン/ピーエフシー フルオロカーボンのエマルジョン
TW406020B (en) 1993-09-29 2000-09-21 Bristol Myers Squibb Co Stabilized pharmaceutical composition and its method for preparation and stabilizing solvent
US5597829A (en) * 1994-05-09 1997-01-28 Bionumerik Pharmaceuticals, Inc. Lactone stable formulation of camptothecin and methods for uses thereof
US5726181A (en) * 1995-06-05 1998-03-10 Bionumerik Pharmaceuticals, Inc. Formulations and compositions of poorly water soluble camptothecin derivatives
US6458373B1 (en) 1997-01-07 2002-10-01 Sonus Pharmaceuticals, Inc. Emulsion vehicle for poorly soluble drugs
DK0999826T3 (da) 1997-07-29 2004-07-26 Upjohn Co Selv-emulgerende formulering til lipofile forbindelser
AR013261A1 (es) 1997-08-01 2000-12-13 Smithkline Beecham Corp Formulaciones farmaceuticas para analogos de camptotecina en capsula de gelatina
EP1075252A2 (en) 1998-05-07 2001-02-14 ELAN CORPORATION, Plc Solvent/cosolvent free microemulsion and emulsion preconcentrate drug delivery systems
US20030059465A1 (en) 1998-05-11 2003-03-27 Unger Evan C. Stabilized nanoparticle formulations of camptotheca derivatives
GB9903547D0 (en) 1999-02-16 1999-04-07 Novartis Ag Organic compounds
DE69901379T2 (de) * 1999-03-09 2002-11-07 Istituto Nazionale Per Lo Studio E La Cura Dei Tumori, Mailand/Milano Camptothecin-Derivate mit Antitumor-Wirkung
IT1306129B1 (it) * 1999-04-13 2001-05-30 Sigma Tau Ind Farmaceuti Esteri della l-carnitina o di alcanoil l-carnitine utilizzabili comelipidi cationici per l'immissione intracellulare di composti
CA2373994A1 (en) 1999-05-24 2000-11-30 Sonus Pharmaceuticals, Inc. Emulsion vehicle for poorly soluble drugs
GB9918885D0 (en) 1999-08-10 1999-10-13 Pharmacia & Upjohn Spa Pharmaceutical formulations in hydroxypropymethycellulose capsules
GB9925127D0 (en) 1999-10-22 1999-12-22 Pharmacia & Upjohn Spa Oral formulations for anti-tumor compounds
US20040009229A1 (en) * 2000-01-05 2004-01-15 Unger Evan Charles Stabilized nanoparticle formulations of camptotheca derivatives
GB0001928D0 (en) * 2000-01-27 2000-03-22 Novartis Ag Organic compounds
US20020150615A1 (en) * 2001-02-12 2002-10-17 Howard Sands Injectable pharmaceutical composition comprising microdroplets of a camptothecin
US6653319B1 (en) * 2001-08-10 2003-11-25 University Of Kentucky Research Foundation Pharmaceutical formulation for poorly water soluble camptothecin analogues
JP2005508354A (ja) 2001-10-15 2005-03-31 クリチテック インコーポレーテッド 水に溶けにくい薬物の送込み用組成物および方法並びに治療方法
US20060078618A1 (en) 2001-12-11 2006-04-13 Constantinides Panayiotis P Lipid particles and suspensions and uses thereof
JP2003267891A (ja) 2002-03-13 2003-09-25 Mitsubishi-Kagaku Foods Corp W/o/w型エマルション製剤
CZ294371B6 (cs) * 2002-06-10 2004-12-15 Pliva - Lachema, A. S. Stabilizovaná farmaceutická kompozice na bázi polyoxyethylovaného ricinového oleje a způsob její přípravy
EP1393719A1 (en) 2002-08-23 2004-03-03 Munich Biotech AG Camptothecin-carboxylate formulations
JP4426749B2 (ja) 2002-07-11 2010-03-03 株式会社産学連携機構九州 O/w型エマルション製剤
US20040171560A1 (en) * 2002-12-23 2004-09-02 Dabur Research Foundation Stabilized pharmaceutical composition
JP2006199590A (ja) * 2003-09-04 2006-08-03 Nano Career Kk 水溶性の塩基性薬物内包ナノ粒子含有組成物
KR20060110872A (ko) * 2003-10-29 2006-10-25 소너스파머슈티칼즈인코포레이티드 토코페롤 변성 치료제 약물 화합물
EP1706098A4 (en) * 2003-11-26 2012-08-15 Supernus Pharmaceuticals Inc MICELLAR SYSTEMS SUITABLE FOR THE DELIVERY OF LIPOPHILIC OR HYDROPHOBIC COMPOUNDS
WO2005060871A1 (en) 2003-12-17 2005-07-07 Bionumerik Pharmaceuticals, Inc. Pharmaceutical formulations of camptothecins and process for making same
GT200500310A (es) 2004-11-19 2006-06-19 Compuestos organicos

Also Published As

Publication number Publication date
MX2007005897A (es) 2007-06-19
RU2007122470A (ru) 2008-12-27
KR101283840B1 (ko) 2013-07-15
WO2006053755A1 (en) 2006-05-26
MY148647A (en) 2013-05-15
CA2584343A1 (en) 2006-05-26
SI1814520T1 (sl) 2016-06-30
NZ554551A (en) 2010-01-29
RU2015131700A (ru) 2017-02-02
NO342592B1 (no) 2018-06-18
AU2005306018A1 (en) 2006-05-26
NO20072258L (no) 2007-08-10
JP2008520606A (ja) 2008-06-19
ES2572133T3 (es) 2016-05-30
AU2005306018B2 (en) 2009-12-17
TWI368521B (en) 2012-07-21
TNSN07193A1 (en) 2008-11-21
CN101056619A (zh) 2007-10-17
DK1814520T3 (en) 2016-05-30
AR052033A1 (es) 2007-02-28
US20080125450A1 (en) 2008-05-29
EP1814520B1 (en) 2016-04-13
HRP20160446T1 (hr) 2016-05-20
PL1814520T3 (pl) 2016-08-31
ZA200703148B (en) 2008-09-25
RU2012120388A (ru) 2013-11-27
RU2620331C2 (ru) 2017-05-24
GT200500310A (es) 2006-06-19
MA29076B1 (fr) 2007-12-03
IL182703A (en) 2015-11-30
KR20070084357A (ko) 2007-08-24
TW200631606A (en) 2006-09-16
IL182703A0 (en) 2007-09-20
BRPI0518448A2 (pt) 2008-11-18
HUE027135T2 (en) 2016-08-29
CA2584343C (en) 2013-09-24
JP4982378B2 (ja) 2012-07-25
US8518961B2 (en) 2013-08-27
EP1814520A1 (en) 2007-08-08

Similar Documents

Publication Publication Date Title
PE20061077A1 (es) Composicion farmaceutica que comprende 7-terbutoxi-imino-metil-camptotecina
ES2524320T3 (es) Composición para la prevención o el tratamiento de enfermedad asociada con trombo o émbolo
PE20060464A1 (es) Composicion farmaceutica que comprende flibanserina para el tratamiento de trastornos sexuales
CY1120888T1 (el) Διαδερμικες φαρμακευτικες συνθεσεις περιλαμβανοντας ενεργους παραγοντες
AR073123A1 (es) Composicion farmaceutica que comprende un taxano sustancialmente amorfo para utilizarse en el tratamiento de la enfermedad neoplasica
AR052545A1 (es) Suspension no acuosa inyectable
SV2008003071A (es) Composiciones farmaceuticas de antagonistas del anticuerpo anti-cd40
HRP20220361T1 (hr) Postupak i sastav za liječenje očne hipertenzije i glaukoma
PE20130216A1 (es) Formulacion topica para un inhibidor de jak
PE20151425A1 (es) Formulaciones farmaceuticas muy concentradas que comprenden un anticuerpo anti-cd20
EA201170413A1 (ru) Составы с замедленным высвобождением, полученные с применением неводных носителей
CO6311006A2 (es) Composicion farmaceutica que comprende un agente que activa las celulas t regulatorias cd4+cd25+ efectiva a dosis altas
HUP0301405A2 (hu) Fokozott oldékonyságú gyógyhatású komponenseket tartalmazó készítmények
CO2021000174A2 (es) Composiciones tópicas para el alivio del dolor
MX349176B (es) Suministro transdermico de farmaco empleando un osmolito y un agente vasoactivo.
BR112015020707A2 (pt) formulações transdermicas
MX2024000828A (es) Formulaciones de parasiticida de isoxazolina y metodos para el tratamiento de la blefaritis.
MX393613B (es) Composiciones de gel para administracion transdermica para maximizar las concentraciones de farmaco en el estrato corneo y suero, y metodos de uso de las mismas.
MX2021016055A (es) Formulaciones y métodos de parasiticidas de isoxazolina para el tratamiento de la blefaritis.
PE20090387A1 (es) Formulacion de pasireotida
BRPI0418070A (pt) composição para cuidados pessoais, uso de uma uréia substituìda e método para reduzir a degradação da cor de uma composição para cuidados pessoais
ES2614481T3 (es) Composición para la administración de principios activos mediante dispositivos de implante
AR061269A1 (es) Composicion y metodo de revascularizacion para el tratamiento de enfermedades isquemicas usando eritropoyetina
CR20180014A (es) Composiciones de matriz polimérica tópicas que comprenden una alta concentración de hialuronato de sodio bio-fermentado y sus usos
MX2022013275A (es) Composicion conservadora/de cuidado personal sinergica con ester de poliglicerol.

Legal Events

Date Code Title Description
FC Refusal
FG Grant, registration
FD Application declared void or lapsed