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PA8531401A1 - SPIROPIRIMIDIN-2,4,6-TRIONA METALOPROTEINASE INHIBITORS - Google Patents

SPIROPIRIMIDIN-2,4,6-TRIONA METALOPROTEINASE INHIBITORS

Info

Publication number
PA8531401A1
PA8531401A1 PA20018531401A PA8531401A PA8531401A1 PA 8531401 A1 PA8531401 A1 PA 8531401A1 PA 20018531401 A PA20018531401 A PA 20018531401A PA 8531401 A PA8531401 A PA 8531401A PA 8531401 A1 PA8531401 A1 PA 8531401A1
Authority
PA
Panama
Prior art keywords
spiropirimidin
triona
inhibitors
metaloproteinase inhibitors
metaloproteinase
Prior art date
Application number
PA20018531401A
Other languages
Spanish (es)
Inventor
Mark Carl Noe
Brian Scott Bronk
Martin James Wythes
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PA8531401A1 publication Critical patent/PA8531401A1/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10—Spiro-condensed systems
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Abstract

LA PRESENTE INVENCION SE REFIERE A INHIBIDORES DE 5-ESPIROPIRIMIDIN-2,4,6-TRIONA, METALOPROTEINASAS DE FORMULA, EN LA QUE EL CITADO "A" ES UN ANILLO HETEROCICLICO DE 5 A 7 MIEMBROS COMO SE DEFINE EN LA MEMORIA DESCRIPTIVA, Y A COMPOSICIONES FARMACEUTICAS Y PROCEDIMIENTOS DE TRATAMIENTO DE LA INFLAMACION, EL CANCER Y OTRAS DOLENCIAS.THE PRESENT INVENTION REFERS TO INHIBITORS OF 5-SPIROPIRIMIDIN-2,4,6-TRIONA, METALOPROTEINASES OF FORMULA, IN WHICH THE CITED "A" IS A HETEROCICLICAL RING OF 5 TO 7 MEMBERS AS DEFINED IN THE DESCRIPTIVE MEMORY, AND PHARMACEUTICAL COMPOSITIONS AND PROCEDURES OF TREATMENT OF INFLAMMATION, CANCER AND OTHER DOLENCES.

PA20018531401A 2000-10-26 2001-10-26 SPIROPIRIMIDIN-2,4,6-TRIONA METALOPROTEINASE INHIBITORS PA8531401A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24338900P 2000-10-26 2000-10-26

Publications (1)

Publication Number Publication Date
PA8531401A1 true PA8531401A1 (en) 2003-06-30

Family

ID=22918584

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20018531401A PA8531401A1 (en) 2000-10-26 2001-10-26 SPIROPIRIMIDIN-2,4,6-TRIONA METALOPROTEINASE INHIBITORS

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Country Link
EP (1) EP1332146A2 (en)
JP (1) JP2004518635A (en)
KR (1) KR20040004412A (en)
CN (1) CN1501937A (en)
AP (1) AP2001002318A0 (en)
AR (1) AR035069A1 (en)
AU (1) AU2002210813A1 (en)
BG (1) BG107653A (en)
BR (1) BR0114913A (en)
CA (1) CA2425283A1 (en)
CZ (1) CZ20031083A3 (en)
EA (1) EA005762B1 (en)
EC (1) ECSP034567A (en)
EE (1) EE200300196A (en)
GT (1) GT200100213A (en)
HN (1) HN2001000244A (en)
HR (1) HRP20030332A2 (en)
HU (1) HUP0301577A3 (en)
IL (1) IL154948A0 (en)
IS (1) IS6762A (en)
MA (1) MA26957A1 (en)
MX (1) MXPA03003735A (en)
NO (1) NO20031853L (en)
OA (1) OA12529A (en)
PA (1) PA8531401A1 (en)
PE (1) PE20020589A1 (en)
PL (1) PL366201A1 (en)
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