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ITMI20032059A1 - Processo per la preparazione di doxifluridina. - Google Patents

Processo per la preparazione di doxifluridina.

Info

Publication number
ITMI20032059A1
ITMI20032059A1 IT002059A ITMI20032059A ITMI20032059A1 IT MI20032059 A1 ITMI20032059 A1 IT MI20032059A1 IT 002059 A IT002059 A IT 002059A IT MI20032059 A ITMI20032059 A IT MI20032059A IT MI20032059 A1 ITMI20032059 A1 IT MI20032059A1
Authority
IT
Italy
Prior art keywords
doxifluridine
preparation
Prior art date
Application number
IT002059A
Other languages
English (en)
Inventor
Giorgio Bertolini
Sara Maculan
Original Assignee
Clariant Lsm Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Clariant Lsm Italia Spa filed Critical Clariant Lsm Italia Spa
Priority to IT002059A priority Critical patent/ITMI20032059A1/it
Priority to JP2006536208A priority patent/JP2007509128A/ja
Priority to PCT/IB2004/003448 priority patent/WO2005040184A1/en
Priority to US10/576,598 priority patent/US20070073050A1/en
Priority to KR1020067007581A priority patent/KR20060110867A/ko
Priority to EP04791727A priority patent/EP1678192A1/en
Publication of ITMI20032059A1 publication Critical patent/ITMI20032059A1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT002059A 2003-10-22 2003-10-22 Processo per la preparazione di doxifluridina. ITMI20032059A1 (it)

Priority Applications (6)

Application Number Priority Date Filing Date Title
IT002059A ITMI20032059A1 (it) 2003-10-22 2003-10-22 Processo per la preparazione di doxifluridina.
JP2006536208A JP2007509128A (ja) 2003-10-22 2004-10-21 ドキシフルリジンの製造方法
PCT/IB2004/003448 WO2005040184A1 (en) 2003-10-22 2004-10-21 Process for the preparation of doxifluridine
US10/576,598 US20070073050A1 (en) 2003-10-22 2004-10-21 Process for the preparation of doxifluridine
KR1020067007581A KR20060110867A (ko) 2003-10-22 2004-10-21 독시플루리딘의 제조 방법
EP04791727A EP1678192A1 (en) 2003-10-22 2004-10-21 Process for the preparation of doxifluridine

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT002059A ITMI20032059A1 (it) 2003-10-22 2003-10-22 Processo per la preparazione di doxifluridina.

Publications (1)

Publication Number Publication Date
ITMI20032059A1 true ITMI20032059A1 (it) 2005-04-23

Family

ID=34509454

Family Applications (1)

Application Number Title Priority Date Filing Date
IT002059A ITMI20032059A1 (it) 2003-10-22 2003-10-22 Processo per la preparazione di doxifluridina.

Country Status (6)

Country Link
US (1) US20070073050A1 (it)
EP (1) EP1678192A1 (it)
JP (1) JP2007509128A (it)
KR (1) KR20060110867A (it)
IT (1) ITMI20032059A1 (it)
WO (1) WO2005040184A1 (it)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2210895A1 (en) 2009-01-27 2010-07-28 F. Hoffmann-La Roche AG Process for the recovery of beta-Acetylfuranoside
CN108117574A (zh) * 2017-12-27 2018-06-05 连云港笃翔化工有限公司 一种去氧氟尿苷的合成方法
CN108558960A (zh) * 2018-05-16 2018-09-21 新乡拓新药业股份有限公司 一种1,2,3-三-O-乙酰基-5-脱氧-β-D-核糖的制备方法
KR102704255B1 (ko) * 2021-04-02 2024-09-06 주식회사 경보제약 독시플루리딘의 제조 방법

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1135258A (en) * 1979-06-15 1982-11-09 Richard D'souza Process for the preparation of 5'deoxy-5-fluorouridine
US4330729A (en) * 1980-07-30 1982-05-18 General Electric Company Locking support arrangement for a flexible sound-generating diaphragm

Also Published As

Publication number Publication date
JP2007509128A (ja) 2007-04-12
WO2005040184A1 (en) 2005-05-06
EP1678192A1 (en) 2006-07-12
KR20060110867A (ko) 2006-10-25
US20070073050A1 (en) 2007-03-29

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