[go: up one dir, main page]

IT201700025273A1 - Co-cristalli di vinpocetina e loro processo di preparazione - Google Patents

Co-cristalli di vinpocetina e loro processo di preparazione

Info

Publication number
IT201700025273A1
IT201700025273A1 IT102017000025273A IT201700025273A IT201700025273A1 IT 201700025273 A1 IT201700025273 A1 IT 201700025273A1 IT 102017000025273 A IT102017000025273 A IT 102017000025273A IT 201700025273 A IT201700025273 A IT 201700025273A IT 201700025273 A1 IT201700025273 A1 IT 201700025273A1
Authority
IT
Italy
Prior art keywords
vinpocetin
crystals
preparation process
preparation
Prior art date
Application number
IT102017000025273A
Other languages
English (en)
Italian (it)
Inventor
Barbara Pacchetti
Andrea Mereu
Giuseppe Paladino
Original Assignee
Linnea Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Linnea Sa filed Critical Linnea Sa
Priority to IT102017000025273A priority Critical patent/IT201700025273A1/it
Priority to PCT/EP2018/055314 priority patent/WO2018162393A1/fr
Publication of IT201700025273A1 publication Critical patent/IT201700025273A1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D461/00Heterocyclic compounds containing indolo [3,2,1-d,e] pyrido [3,2,1,j] [1,5]-naphthyridine ring systems, e.g. vincamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/05Phenols
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/475Quinolines; Isoquinolines having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IT102017000025273A 2017-03-07 2017-03-07 Co-cristalli di vinpocetina e loro processo di preparazione IT201700025273A1 (it)

Priority Applications (2)

Application Number Priority Date Filing Date Title
IT102017000025273A IT201700025273A1 (it) 2017-03-07 2017-03-07 Co-cristalli di vinpocetina e loro processo di preparazione
PCT/EP2018/055314 WO2018162393A1 (fr) 2017-03-07 2018-03-05 Co-cristaux de vinpocétine et leur procédé de préparation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT102017000025273A IT201700025273A1 (it) 2017-03-07 2017-03-07 Co-cristalli di vinpocetina e loro processo di preparazione

Publications (1)

Publication Number Publication Date
IT201700025273A1 true IT201700025273A1 (it) 2018-09-07

Family

ID=59409630

Family Applications (1)

Application Number Title Priority Date Filing Date
IT102017000025273A IT201700025273A1 (it) 2017-03-07 2017-03-07 Co-cristalli di vinpocetina e loro processo di preparazione

Country Status (2)

Country Link
IT (1) IT201700025273A1 (fr)
WO (1) WO2018162393A1 (fr)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0154756A1 (fr) * 1984-02-29 1985-09-18 Covex (S.A.) Citrate de vinpocetine et son procédé de préparation
EP0689844A1 (fr) * 1994-06-23 1996-01-03 Tecnimede-Sociedade Tecnico-Medicinal, S.A. Complexes de vinpocetine avec cyclodextrines, procédé pour leur préparation et compositions pharmaceutiques les contenant

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0154756A1 (fr) * 1984-02-29 1985-09-18 Covex (S.A.) Citrate de vinpocetine et son procédé de préparation
EP0689844A1 (fr) * 1994-06-23 1996-01-03 Tecnimede-Sociedade Tecnico-Medicinal, S.A. Complexes de vinpocetine avec cyclodextrines, procédé pour leur préparation et compositions pharmaceutiques les contenant

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
DRITAN HASA ET AL: "Enhanced Oral Bioavailability of Vinpocetine Through Mechanochemical Salt Formation: Physico-Chemical Characterization andStudies", PHARMACEUTICAL RESEARCH, KLUWER ACADEMIC PUBLISHERS-PLENUM PUBLISHERS, NL, vol. 28, no. 8, 19 March 2011 (2011-03-19), pages 1870 - 1883, XP019921751, ISSN: 1573-904X, DOI: 10.1007/S11095-011-0415-8 *

Also Published As

Publication number Publication date
WO2018162393A1 (fr) 2018-09-13

Similar Documents

Publication Publication Date Title
IL290809A (en) Tau-protein targeting protacs and associated methods of use
HUE046756T2 (hu) Benzoxazepin-oxazolidinon vegyületek és azok alkalmazási módszerei
PL3507418T3 (pl) Sposoby biopochodnej derywatyzacji powierzchni celulozowych
MA46481A (fr) Compositions d'oligonucléotides et méthodes associées
HUE052373T2 (hu) Szubsztituált krománok és alkalmazási eljárások
PT3319952T (pt) Processo de produção de canabidiol e delta-9-tetrahidrocanabinol
PT3368534T (pt) Ditosilato de valbenazina e polimorfos do mesmo
PT3548033T (pt) Compostos e respectivos métodos de utilização
HUE054874T2 (hu) Magas elaszticitású hialuronán készítmények és alkalmazási eljárások
HUE050124T2 (hu) Eljárás biopolimerek dezacetilezésére
HUE055199T2 (hu) Oxiszterolok és alkalmazási eljárásaik
LT3652491T (lt) Produkto liofilizavimo būdas
IL256322B (en) Improved formulations of deferasirox and methods of making the same
HUE046509T2 (hu) Új vegyület és eljárás
IL285784A (en) Graphene and the production of graphene
EP3565542A4 (fr) Formes polymorphes de rad1901-2hcl
EP3366001A4 (fr) Cryptage et décryptage de langage postscript
DK3453721T3 (da) Process of manufacture of annexin v
IL253889A0 (en) Detection of brain injury
HUE054093T2 (hu) Anti-HtrA1 antitestek és azok alkalmazási eljárásai
BR112017026560A2 (pt) processo para preparação de apremilast e seus intermediários.
PL3630738T3 (pl) Sposób wytwarzania ozanimodu
IL257764B (en) Methods for treatment of diseases
HUE049157T2 (hu) Intermedierek piridazinon herbicidek elõállítására és eljárás azok elõállítására
EP3328384A4 (fr) Traitement de la fibrose