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IL90892A0 - Rifapentine hydrohalides - Google Patents

Rifapentine hydrohalides

Info

Publication number
IL90892A0
IL90892A0 IL90892A IL9089289A IL90892A0 IL 90892 A0 IL90892 A0 IL 90892A0 IL 90892 A IL90892 A IL 90892A IL 9089289 A IL9089289 A IL 9089289A IL 90892 A0 IL90892 A0 IL 90892A0
Authority
IL
Israel
Prior art keywords
pct
rifapentine
sec
date
hydrohalides
Prior art date
Application number
IL90892A
Other languages
English (en)
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of IL90892A0 publication Critical patent/IL90892A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Dental Preparations (AREA)
  • Fats And Perfumes (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Liquid Crystal Substances (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
IL90892A 1988-07-13 1989-07-06 Rifapentine hydrohalides IL90892A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888816620A GB8816620D0 (en) 1988-07-13 1988-07-13 Rifapentine hydrohalides

Publications (1)

Publication Number Publication Date
IL90892A0 true IL90892A0 (en) 1990-02-09

Family

ID=10640347

Family Applications (1)

Application Number Title Priority Date Filing Date
IL90892A IL90892A0 (en) 1988-07-13 1989-07-06 Rifapentine hydrohalides

Country Status (20)

Country Link
US (1) US5306715A (xx)
EP (1) EP0440642B1 (xx)
JP (1) JP2716553B2 (xx)
KR (1) KR0135312B1 (xx)
CN (1) CN1039421A (xx)
AT (1) ATE111101T1 (xx)
AU (1) AU632754B2 (xx)
CA (1) CA1339215C (xx)
DE (1) DE68918107T2 (xx)
DK (1) DK173423B1 (xx)
ES (1) ES2018374A6 (xx)
GB (1) GB8816620D0 (xx)
GR (1) GR1002222B (xx)
HK (1) HK1005455A1 (xx)
HU (1) HU210716A9 (xx)
IE (1) IE65812B1 (xx)
IL (1) IL90892A0 (xx)
PT (1) PT91132B (xx)
WO (1) WO1990000553A1 (xx)
ZA (1) ZA894991B (xx)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI94339C (fi) 1989-07-21 1995-08-25 Warner Lambert Co Menetelmä farmaseuttisesti käyttökelpoisen /R-(R*,R*)/-2-(4-fluorifenyyli)- , -dihydroksi-5-(1-metyylietyyli)-3-fenyyli-4-/(fenyyliamino)karbonyyli/-1H-pyrroli-1-heptaanihapon ja sen farmaseuttisesti hyväksyttävien suolojen valmistamiseksi
DK0536197T3 (da) * 1990-06-29 1995-11-13 Lepetit Spa Ren, krystallinsk form af rifapentine
HRP20000162B1 (en) 2000-03-20 2004-06-30 Pliva D D Amorphous torasemide modification
JP4393098B2 (ja) * 2002-06-21 2010-01-06 独立行政法人科学技術振興機構 アンサマイシン系抗生物質の新規用途及び新規血管新生抑制物質のスクリーニング方法
EP1592668A1 (en) * 2003-02-12 2005-11-09 Ciba SC Holding AG Crystalline forms of pitavastatin calcium
ITMI20032144A1 (it) * 2003-11-07 2005-05-08 Alfa Wassermann Spa Forme polimorfe di rifaximina, processi per ottenerle e
ES2522895T3 (es) * 2005-03-03 2014-11-19 Alfa Wassermann S.P.A. Nuevas formas polimorfas de rifaximina, procedimientos para su producción y uso de las mismas en preparados medicinales
JP2007246514A (ja) * 2006-02-14 2007-09-27 Toyama Chem Co Ltd ピペラシリンナトリウムの新規な結晶
CN101611040A (zh) * 2007-01-31 2009-12-23 富山化学工业株式会社 哌拉西林钠的新颖结晶
IT1398550B1 (it) 2010-03-05 2013-03-01 Alfa Wassermann Spa Formulazioni comprendenti rifaximina utili per ottenere un effetto prolungato nel tempo
CA2861104A1 (en) * 2012-01-25 2013-08-01 Salix Pharmaceuticals, Ltd. Rifaximin derivative and uses thereof
ITBO20120368A1 (it) 2012-07-06 2014-01-07 Alfa Wassermann Spa Composizioni comprendenti rifaximina e amminoacidi, cristalli di rifaximina derivanti da tali composizioni e loro uso.
US20240199642A1 (en) * 2021-04-21 2024-06-20 Interquim S.A. De C.V. Method for obtaining rifapentine with a new crystalline form

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR208F (xx) * 1964-07-31
GB1478563A (en) * 1975-03-05 1977-07-06 Lepetit Spa Rifamycin derivatives
FR2309556A1 (fr) * 1975-04-29 1976-11-26 Aries Robert Aminoguanidines derivees de la rifamycine
US4876258A (en) * 1987-08-13 1989-10-24 Ciba-Geigy Corporation Biphenylyl compounds
KR890701591A (ko) * 1987-09-25 1989-12-21 베르너 발데그 4-(트리알킬벤질)-피페라지닐 화합물의 디아실 유도체

Also Published As

Publication number Publication date
KR900701798A (ko) 1990-12-04
PT91132A (pt) 1990-02-08
DK292590A (da) 1990-12-10
AU632754B2 (en) 1993-01-14
ZA894991B (en) 1990-08-29
GR1002222B (en) 1996-04-17
WO1990000553A1 (en) 1990-01-25
JP2716553B2 (ja) 1998-02-18
DK292590D0 (da) 1990-12-10
HK1005455A1 (en) 1999-01-08
DK173423B1 (da) 2000-10-09
IE65812B1 (en) 1995-11-15
ATE111101T1 (de) 1994-09-15
EP0440642A1 (en) 1991-08-14
KR0135312B1 (ko) 1998-04-23
DE68918107D1 (de) 1994-10-13
DE68918107T2 (de) 1995-01-26
AU3770289A (en) 1990-02-05
JPH03506025A (ja) 1991-12-26
CN1039421A (zh) 1990-02-07
HU210716A9 (en) 1995-06-28
GR890100448A (el) 1990-06-27
CA1339215C (en) 1997-08-05
EP0440642B1 (en) 1994-09-07
GB8816620D0 (en) 1988-08-17
ES2018374A6 (es) 1991-04-01
PT91132B (pt) 1994-12-30
US5306715A (en) 1994-04-26
IE892247L (en) 1990-01-13

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