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HN2002000319A - Benzamida, heteroarilamida y amidas inversas - Google Patents

Benzamida, heteroarilamida y amidas inversas

Info

Publication number
HN2002000319A
HN2002000319A HN2002000319A HN2002000319A HN2002000319A HN 2002000319 A HN2002000319 A HN 2002000319A HN 2002000319 A HN2002000319 A HN 2002000319A HN 2002000319 A HN2002000319 A HN 2002000319A HN 2002000319 A HN2002000319 A HN 2002000319A
Authority
HN
Honduras
Prior art keywords
heteroarilamida
benzamida
amidas
invested
preparation
Prior art date
Application number
HN2002000319A
Other languages
English (en)
Inventor
Allen Jacob Duplantier
Chakrapani Subramanyam
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HN2002000319A publication Critical patent/HN2002000319A/es

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D253/00Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/061,2,4-Triazines
    • C07D253/0651,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
    • C07D253/071,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D253/075Two hetero atoms, in positions 3 and 5
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    • C07ORGANIC CHEMISTRY
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    • C07D211/72Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62Oxygen or sulfur atoms
    • C07D213/63One oxygen atom
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    • C07D241/08Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
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    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
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Abstract

LA PRESENTE INVENCIÓN SE REFIERE A NUEVAS BENZAMIDAHETEROARILAMIDA Y AMIDA INVERSA, A PROCESOS PARA SU PREPARACION, A INTERMEDIOS UTILES EN SU PREPARACIÓN A COMPOSICIONES FARMACEUTICAS QUE LAS CONTIENEN Y A SU USO EN TERAPIA.
HN2002000319A 2001-11-12 2002-11-11 Benzamida, heteroarilamida y amidas inversas HN2002000319A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US33678101P 2001-11-12 2001-11-12

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HN2002000319A true HN2002000319A (es) 2003-12-20

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HN2002000319A HN2002000319A (es) 2001-11-12 2002-11-11 Benzamida, heteroarilamida y amidas inversas

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EP (1) EP1448535B1 (es)
JP (1) JP4365218B2 (es)
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IL (1) IL161329A0 (es)
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Families Citing this family (74)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PA8557501A1 (es) * 2001-11-12 2003-06-30 Pfizer Prod Inc Benzamida, heteroarilamida y amidas inversas
PA8591801A1 (es) * 2002-12-31 2004-07-26 Pfizer Prod Inc Inhibidores benzamidicos del receptor p2x7.
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