FR2840303B1 - Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile - Google Patents
Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophileInfo
- Publication number
- FR2840303B1 FR2840303B1 FR0206717A FR0206717A FR2840303B1 FR 2840303 B1 FR2840303 B1 FR 2840303B1 FR 0206717 A FR0206717 A FR 0206717A FR 0206717 A FR0206717 A FR 0206717A FR 2840303 B1 FR2840303 B1 FR 2840303B1
- Authority
- FR
- France
- Prior art keywords
- vinylation
- arylation
- alkylation
- nucleophilic compound
- nucleophilic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 230000029936 alkylation Effects 0.000 title 1
- 238000005804 alkylation reaction Methods 0.000 title 1
- 238000006254 arylation reaction Methods 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 230000000269 nucleophilic effect Effects 0.000 title 1
- 238000006886 vinylation reaction Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
- C07D213/53—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/06—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Priority Applications (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/159,829 US7202367B2 (en) | 2002-05-31 | 2002-05-31 | Process for arylating or vinylating or alkynating a nucleophilic compound |
| FR0206717A FR2840303B1 (fr) | 2002-05-31 | 2002-05-31 | Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile |
| EP03756038A EP1509502A1 (fr) | 2002-05-31 | 2003-06-02 | Procede de formation d une liaison carbone-carbone ou carbone-heteroatome |
| CNA038166712A CN1668595A (zh) | 2002-05-31 | 2003-06-02 | 形成碳－碳或碳－杂原子键的方法 |
| US10/515,856 US20050234239A1 (en) | 2002-03-31 | 2003-06-02 | Method of forming a carbon-carbon or carbon-heteroatom linkage |
| CA002487475A CA2487475A1 (fr) | 2002-05-31 | 2003-06-02 | Procede de formation d'une liaison carbone-carbone ou carbone-heteroatome |
| PCT/FR2003/001647 WO2003101966A1 (fr) | 2002-05-31 | 2003-06-02 | Procede de formation d'une liaison carbone-carbone ou carbone-heteroatome |
| JP2004509659A JP2006501159A (ja) | 2002-05-31 | 2003-06-02 | 炭素−炭素結合又は炭素−ヘテロ原子結合の形成方法 |
| AU2003255620A AU2003255620A1 (en) | 2002-05-31 | 2003-06-02 | Method of forming a carbon-carbon or carbon-heteroatom linkage |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/159,829 US7202367B2 (en) | 2002-05-31 | 2002-05-31 | Process for arylating or vinylating or alkynating a nucleophilic compound |
| FR0206717A FR2840303B1 (fr) | 2002-05-31 | 2002-05-31 | Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2840303A1 FR2840303A1 (fr) | 2003-12-05 |
| FR2840303B1 true FR2840303B1 (fr) | 2005-07-15 |
Family
ID=32232264
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR0206717A Expired - Fee Related FR2840303B1 (fr) | 2002-03-31 | 2002-05-31 | Procede d'arylation ou de vinylation ou d'alcylynation d'un compose nucleophile |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US7202367B2 (fr) |
| FR (1) | FR2840303B1 (fr) |
| WO (1) | WO2003101966A1 (fr) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102004039280A1 (de) * | 2004-08-13 | 2006-02-23 | Merck Patent Gmbh | 1,5-Diphenyl-pyrazole |
| SA06270147B1 (ar) | 2005-06-09 | 2009-12-22 | نوفارتيس ايه جي | عملية لتخليق 5-(مثيل–1h–إيميدازول–1-يل )–3-(ثلاثي فلـورو مثيل)–بنزامـين |
| GT200600207A (es) * | 2005-06-09 | 2007-01-15 | Novartis Ag | Proceso para la síntesis de compuestos orgánicos |
| JP2006342127A (ja) * | 2005-06-10 | 2006-12-21 | Koei Chem Co Ltd | アリールピラゾール類の製造法 |
| US9162953B2 (en) * | 2006-07-05 | 2015-10-20 | Centre Nationale De Recherche Scientifique | Iron-copper co-catalyzed process for carbon-carbon or carbon-heteroatom bonding |
| US8034815B2 (en) | 2007-01-11 | 2011-10-11 | Critical Outcome Technologies, Inc. | Compounds and method for treatment of cancer |
| FR2915200B1 (fr) | 2007-04-20 | 2009-07-03 | Centre Nat Rech Scient | Procede de preparation de ligands de type phosphines butadieniques,leurs complexes avec le cuivre,et leurs applications en catalyse |
| FR2921659B1 (fr) * | 2007-09-28 | 2013-01-18 | Centre Nat Rech Scient | Utilisation de complexes cuivre/phosphines cyclovinyliques comme catalyseurs d'arylation |
| US9272274B2 (en) | 2007-12-06 | 2016-03-01 | Centre National De La Recherche Scientifique (C.N.R.S.) | Catalytic system for cross-coupling reactions |
| CA2710039C (fr) | 2007-12-26 | 2018-07-03 | Critical Outcome Technologies, Inc. | Semicarbazones, thiosemicarnazones et composes associes, et methodes de traitement du cancer |
| EP2318406B1 (fr) | 2008-07-17 | 2016-01-27 | Critical Outcome Technologies, Inc. | Composés inhibiteurs et procédés de traitement du cancer |
| MX2011006425A (es) | 2008-12-24 | 2011-07-20 | Syngenta Ltd | Metodos para la preparacion de fungicidas. |
| CA2999435A1 (fr) | 2010-04-01 | 2011-10-06 | Critical Outcome Technologies Inc. | Composes et methodes pour le traitement du vih |
| MA34957B1 (fr) | 2011-02-23 | 2014-03-01 | Lupin Ltd | Derives heteroaryle a titre modulateurs des nachr alpha 7 |
| EP2822946A1 (fr) | 2012-03-06 | 2015-01-14 | Lupin Limited | Dérivés de thiazole en tant que modulateurs de nachr alpha 7 |
| WO2014060381A1 (fr) | 2012-10-18 | 2014-04-24 | Bayer Cropscience Ag | Composés hétérocycliques pour la lutte contre les nuisibles |
| US20150284380A1 (en) | 2012-10-31 | 2015-10-08 | Bayer Cropscience Ag | Novel heterocyclic compounds as pest control agents |
| US9231217B2 (en) * | 2013-11-28 | 2016-01-05 | Semiconductor Energy Laboratory Co., Ltd. | Synthesis method of organometallic complex, synthesis method of pyrazine derivative, 5,6-diaryl-2-pyrazyl triflate, light-emitting element, light-emitting device, electronic device, and lighting device |
| ES2941857T3 (es) | 2018-04-12 | 2023-05-26 | Bayer Ag | Derivados de N-(ciclopropilmetil)-5-(metilsulfonil)-n-{1-[1-(pirimidin-2-il)-1h-1,2,4-triazol-5-il]etil}benzamida y los correspondientes derivados de piridina-carboxamida como plaguicidas |
| CN112645909B (zh) * | 2021-01-25 | 2024-09-27 | 苏州大学 | 一种合成α-苄基苯并呋喃类化合物的方法 |
| CN114149364A (zh) * | 2021-12-21 | 2022-03-08 | 无锡捷化医药科技有限公司 | 一种n-(6-甲氧基吡啶-3-基)-3-甲基吡啶-2-磺酰胺的制备方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2272813B1 (fr) * | 2001-04-24 | 2016-11-16 | Massachusetts Institute of Technology (MIT) | Formation de liaisons carbone-oxygène catalysée au cuivre |
-
2002
- 2002-05-31 FR FR0206717A patent/FR2840303B1/fr not_active Expired - Fee Related
- 2002-05-31 US US10/159,829 patent/US7202367B2/en not_active Expired - Fee Related
-
2003
- 2003-06-02 WO PCT/FR2003/001647 patent/WO2003101966A1/fr not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003101966A1 (fr) | 2003-12-11 |
| US20030236413A1 (en) | 2003-12-25 |
| FR2840303A1 (fr) | 2003-12-05 |
| US7202367B2 (en) | 2007-04-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |
Effective date: 20080131 |